50nM_dasatinib vs ctrl_K562 (Human) [19651622] Gene Set

Dataset SILAC Phosphoproteomics Signatures of Differentially Phosphorylated Proteins for Drugs
Category proteomics
Type drug perturbation
Description drug perturbation identified as [drug perturbation]_[cell line] ([organism]) [[publication PMID]] (SILAC Phosphoproteomics)
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Genes

125 proteins differentially phosphorylated following the 50nM_dasatinib vs ctrl_K562 (Human) [19651622] drug perturbation from the SILAC Phosphoproteomics Signatures of Differentially Phosphorylated Proteins for Drugs dataset.

increased phosphorylation

Symbol Name
AKAP11 A kinase (PRKA) anchor protein 11
BABAM1 BRISC and BRCA1 A complex member 1
C1ORF116 chromosome 1 open reading frame 116
CCDC132 coiled-coil domain containing 132
CEP170 centrosomal protein 170kDa
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DYNC1H1 dynein, cytoplasmic 1, heavy chain 1
EEF2K eukaryotic elongation factor 2 kinase
HDAC1 histone deacetylase 1
MAP1A microtubule-associated protein 1A
MARK4 MAP/microtubule affinity-regulating kinase 4
MFAP1 microfibrillar-associated protein 1
MIER1 mesoderm induction early response 1, transcriptional regulator
NAV1 neuron navigator 1
NIPBL Nipped-B homolog (Drosophila)
OSBPL8 oxysterol binding protein-like 8
PALLD palladin, cytoskeletal associated protein
PEX1 peroxisomal biogenesis factor 1
PHIP pleckstrin homology domain interacting protein
PNISR PNN-interacting serine/arginine-rich protein
PRPF4B pre-mRNA processing factor 4B
PTRH1 peptidyl-tRNA hydrolase 1 homolog (S. cerevisiae)
RNF220 ring finger protein 220
RPLP0 ribosomal protein, large, P0
SAFB scaffold attachment factor B
SEC16A SEC16 homolog A (S. cerevisiae)
SF3B1 splicing factor 3b, subunit 1, 155kDa
SLC4A7 solute carrier family 4, sodium bicarbonate cotransporter, member 7
SNRNP70 small nuclear ribonucleoprotein 70kDa (U1)
SRRM1 serine/arginine repetitive matrix 1
SRRM2 serine/arginine repetitive matrix 2
SRSF9 serine/arginine-rich splicing factor 9
SUGP2 SURP and G patch domain containing 2
SUGT1 SGT1, suppressor of G2 allele of SKP1 (S. cerevisiae)
TP53BP1 tumor protein p53 binding protein 1
VAMP8 vesicle-associated membrane protein 8
ZDHHC23 zinc finger, DHHC-type containing 23

decreased phosphorylation

Symbol Name
ABL1 ABL proto-oncogene 1, non-receptor tyrosine kinase
ADAM9 ADAM metallopeptidase domain 9
ADD2 adducin 2 (beta)
AGPAT9 1-acylglycerol-3-phosphate O-acyltransferase 9
ANKRD13D ankyrin repeat domain 13 family, member D
ARID3A AT rich interactive domain 3A (BRIGHT-like)
C10ORF71 chromosome 10 open reading frame 71
C11ORF84 chromosome 11 open reading frame 84
CACNA1D calcium channel, voltage-dependent, L type, alpha 1D subunit
CAPRIN1 cell cycle associated protein 1
CBFA2T3 core-binding factor, runt domain, alpha subunit 2; translocated to, 3
CCDC61 coiled-coil domain containing 61
CCDC88C coiled-coil domain containing 88C
CCDC9 coiled-coil domain containing 9
CENPA centromere protein A
CHD7 chromodomain helicase DNA binding protein 7
CSF1 colony stimulating factor 1 (macrophage)
DDX60 DEAD (Asp-Glu-Ala-Asp) box polypeptide 60
DHX29 DEAH (Asp-Glu-Ala-His) box polypeptide 29
DUT deoxyuridine triphosphatase
EBNA1BP2 EBNA1 binding protein 2
ERMAP erythroblast membrane-associated protein (Scianna blood group)
F2RL3 coagulation factor II (thrombin) receptor-like 3
GOLGA4 golgin A4
HECW2 HECT, C2 and WW domain containing E3 ubiquitin protein ligase 2
HEPH hephaestin
IFT46 intraflagellar transport 46
ILKAP integrin-linked kinase-associated serine/threonine phosphatase
L3MBTL2 l(3)mbt-like 2 (Drosophila)
LCP2 lymphocyte cytosolic protein 2 (SH2 domain containing leukocyte protein of 76kDa)
LENG1 leukocyte receptor cluster (LRC) member 1
MAPT microtubule-associated protein tau
MEF2C myocyte enhancer factor 2C
MTFR1 mitochondrial fission regulator 1
MYB v-myb avian myeloblastosis viral oncogene homolog
NBEAL2 neurobeachin-like 2
NUPL1 nucleoporin like 1
PAK1 p21 protein (Cdc42/Rac)-activated kinase 1
PAXIP1 PAX interacting (with transcription-activation domain) protein 1
PFKFB1 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 1
PITX1 paired-like homeodomain 1
PLD1 phospholipase D1, phosphatidylcholine-specific
PNKP polynucleotide kinase 3'-phosphatase
PPP1R14A protein phosphatase 1, regulatory (inhibitor) subunit 14A
PPP4R1 protein phosphatase 4, regulatory subunit 1
PRKCB protein kinase C, beta
PRMT5 protein arginine methyltransferase 5
PSMD2 proteasome (prosome, macropain) 26S subunit, non-ATPase, 2
PTTG2 pituitary tumor-transforming 2
RAD9A RAD9 homolog A (S. pombe)
RBMY1A1 RNA binding motif protein, Y-linked, family 1, member A1
RCSD1 RCSD domain containing 1
REPIN1 replication initiator 1
RER1 retention in endoplasmic reticulum sorting receptor 1
RET ret proto-oncogene
RPUSD2 RNA pseudouridylate synthase domain containing 2
RUNX1 runt-related transcription factor 1
SAMD1 sterile alpha motif domain containing 1
SAMSN1 SAM domain, SH3 domain and nuclear localization signals 1
SCML2 sex comb on midleg-like 2 (Drosophila)
SH2B3 SH2B adaptor protein 3
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SPAG7 sperm associated antigen 7
SSBP4 single stranded DNA binding protein 4
STK26 serine/threonine protein kinase 26
TACC1 transforming, acidic coiled-coil containing protein 1
TAL1 T-cell acute lymphocytic leukemia 1
TBC1D14 TBC1 domain family, member 14
TCF12 transcription factor 12
TNFRSF17 tumor necrosis factor receptor superfamily, member 17
TNIK TRAF2 and NCK interacting kinase
TNK1 tyrosine kinase, non-receptor, 1
TNKS2 tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase 2
TNRC6A trinucleotide repeat containing 6A
TOMM22 translocase of outer mitochondrial membrane 22 homolog (yeast)
TOR1AIP2 torsin A interacting protein 2
TRPS1 trichorhinophalangeal syndrome I
TTC25 tetratricopeptide repeat domain 25
UNG uracil-DNA glycosylase
VEGFA vascular endothelial growth factor A
WNK4 WNK lysine deficient protein kinase 4
YES1 YES proto-oncogene 1, Src family tyrosine kinase
YRDC yrdC N(6)-threonylcarbamoyltransferase domain containing
ZC3H18-AS1 ZC3H18 antisense RNA 1 (head to head)
ZFP36L2 ZFP36 ring finger protein-like 2
ZFP91 ZFP91 zinc finger protein
ZFYVE16 zinc finger, FYVE domain containing 16
ZNF768 zinc finger protein 768