AG-013608-5904 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the AG-013608-5904 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCB9 ATP-binding cassette, sub-family B (MDR/TAP), member 9
ADGRA2 adhesion G protein-coupled receptor A2
ADGRB3 adhesion G protein-coupled receptor B3
ADTRP androgen-dependent TFPI-regulating protein
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2
ATP2B4 ATPase, Ca++ transporting, plasma membrane 4
BRF1 BRF1, RNA polymerase III transcription initiation factor 90 kDa subunit
BRINP2 bone morphogenetic protein/retinoic acid inducible neural-specific 2
C21ORF2 chromosome 21 open reading frame 2
CACNA1I calcium channel, voltage-dependent, T type, alpha 1I subunit
CALCR calcitonin receptor
CCR9 chemokine (C-C motif) receptor 9
CD1E CD1e molecule
CDH2 cadherin 2, type 1, N-cadherin (neuronal)
CEACAM1 carcinoembryonic antigen-related cell adhesion molecule 1 (biliary glycoprotein)
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CLDN17 claudin 17
COL4A3 collagen, type IV, alpha 3 (Goodpasture antigen)
CPNE7 copine VII
CSF1R colony stimulating factor 1 receptor
CYHR1 cysteine/histidine-rich 1
CYLD cylindromatosis (turban tumor syndrome)
DFNB31 deafness, autosomal recessive 31
DLC1 DLC1 Rho GTPase activating protein
DLL3 delta-like 3 (Drosophila)
DOCK3 dedicator of cytokinesis 3
DOK4 docking protein 4
EPS8L1 EPS8-like 1
FRMD4A FERM domain containing 4A
GPR6 G protein-coupled receptor 6
HLA-C major histocompatibility complex, class I, C
HOPX HOP homeobox
HRASLS2 HRAS-like suppressor 2
IL17RC interleukin 17 receptor C
INHBA inhibin, beta A
IQCC IQ motif containing C
KANK2 KN motif and ankyrin repeat domains 2
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KCNN4 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 4
KDR kinase insert domain receptor
KRT83 keratin 83, type II
LAT2 linker for activation of T cells family, member 2
LOXL3 lysyl oxidase-like 3
LRRC15 leucine rich repeat containing 15
MATN1 matrilin 1, cartilage matrix protein
MED16 mediator complex subunit 16
MGAT3 mannosyl (beta-1,4-)-glycoprotein beta-1,4-N-acetylglucosaminyltransferase
MRAS muscle RAS oncogene homolog
MRPL41 mitochondrial ribosomal protein L41
MTHFR methylenetetrahydrofolate reductase (NAD(P)H)
MVB12B multivesicular body subunit 12B
MYLK myosin light chain kinase
N4BP2L2-IT2 N4BPL2 intronic transcript 2
NAT6 N-acetyltransferase 6 (GCN5-related)
NDRG2 NDRG family member 2
NEDD4L neural precursor cell expressed, developmentally down-regulated 4-like, E3 ubiquitin protein ligase
NEIL1 nei endonuclease VIII-like 1 (E. coli)
NFKBIB nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, beta
NNMT nicotinamide N-methyltransferase
NSUN6 NOP2/Sun domain family, member 6
NUDC nudC nuclear distribution protein
PAK1 p21 protein (Cdc42/Rac)-activated kinase 1
PCDH1 protocadherin 1
PCSK1 proprotein convertase subtilisin/kexin type 1
PSG6 pregnancy specific beta-1-glycoprotein 6
PSMD9 proteasome (prosome, macropain) 26S subunit, non-ATPase, 9
RAB33A RAB33A, member RAS oncogene family
RARA retinoic acid receptor, alpha
RBMS2 RNA binding motif, single stranded interacting protein 2
RNF122 ring finger protein 122
RPS6KA2 ribosomal protein S6 kinase, 90kDa, polypeptide 2
RSG1 REM2 and RAB-like small GTPase 1
RUSC2 RUN and SH3 domain containing 2
RYR1 ryanodine receptor 1 (skeletal)
SEMA3F sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3F
SEMA6A sema domain, transmembrane domain (TM), and cytoplasmic domain, (semaphorin) 6A
SEMA7A semaphorin 7A, GPI membrane anchor (John Milton Hagen blood group)
SHANK2 SH3 and multiple ankyrin repeat domains 2
SIRT5 sirtuin 5
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMG5 SMG5 nonsense mediated mRNA decay factor
SOGA1 suppressor of glucose, autophagy associated 1
STK11 serine/threonine kinase 11
STOM stomatin
STX7 syntaxin 7
SYNE1 spectrin repeat containing, nuclear envelope 1
TIMP3 TIMP metallopeptidase inhibitor 3
TLE2 transducin-like enhancer of split 2
TMPRSS4 transmembrane protease, serine 4
TPMT thiopurine S-methyltransferase
TSC22D4 TSC22 domain family, member 4
URB1 URB1 ribosome biogenesis 1 homolog (S. cerevisiae)
VAMP1 vesicle-associated membrane protein 1 (synaptobrevin 1)
VWA5A von Willebrand factor A domain containing 5A
WAS Wiskott-Aldrich syndrome
ZNF493 zinc finger protein 493
ZNF589 zinc finger protein 589
ZNF646 zinc finger protein 646
ZSCAN2 zinc finger and SCAN domain containing 2

decreased expression

Symbol Name
A1CF APOBEC1 complementation factor
ABCC2 ATP-binding cassette, sub-family C (CFTR/MRP), member 2
ACAD10 acyl-CoA dehydrogenase family, member 10
ACTA1 actin, alpha 1, skeletal muscle
ACTN3 actinin, alpha 3 (gene/pseudogene)
AFF4 AF4/FMR2 family, member 4
AKT2 v-akt murine thymoma viral oncogene homolog 2
ALS2CL ALS2 C-terminal like
ARID5A AT rich interactive domain 5A (MRF1-like)
ARMC6 armadillo repeat containing 6
ASH1L ash1 (absent, small, or homeotic)-like (Drosophila)
AVPR1B arginine vasopressin receptor 1B
BCL2A1 BCL2-related protein A1
BMP15 bone morphogenetic protein 15
C10ORF95 chromosome 10 open reading frame 95
C1ORF54 chromosome 1 open reading frame 54
CASS4 Cas scaffolding protein family member 4
CCDC9 coiled-coil domain containing 9
CCKBR cholecystokinin B receptor
CD74 CD74 molecule, major histocompatibility complex, class II invariant chain
CETN1 centrin, EF-hand protein, 1
CHRNA6 cholinergic receptor, nicotinic, alpha 6 (neuronal)
CHRNB1 cholinergic receptor, nicotinic, beta 1 (muscle)
CLCA1 chloride channel accessory 1
CLCN6 chloride channel, voltage-sensitive 6
CLGN calmegin
COLGALT2 collagen beta(1-O)galactosyltransferase 2
CORT cortistatin
CXCR2 chemokine (C-X-C motif) receptor 2
DUOX2 dual oxidase 2
ELSPBP1 epididymal sperm binding protein 1
ENOX1 ecto-NOX disulfide-thiol exchanger 1
FANCE Fanconi anemia, complementation group E
FCGRT Fc fragment of IgG, receptor, transporter, alpha
FGR FGR proto-oncogene, Src family tyrosine kinase
FKBP10 FK506 binding protein 10, 65 kDa
FSTL3 follistatin-like 3 (secreted glycoprotein)
GABRA2 gamma-aminobutyric acid (GABA) A receptor, alpha 2
GIPR gastric inhibitory polypeptide receptor
GPX2 glutathione peroxidase 2
HOXA2 homeobox A2
HOXB2 homeobox B2
IDI2-AS1 IDI2 antisense RNA 1
IFNA14 interferon, alpha 14
IFNA16 interferon, alpha 16
IFT54 intraflagellar transport 54
IGKV3-20 immunoglobulin kappa variable 3-20
IL12RB2 interleukin 12 receptor, beta 2
INA internexin neuronal intermediate filament protein, alpha
ITIH2 inter-alpha-trypsin inhibitor heavy chain 2
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNA3 potassium channel, voltage gated shaker related subfamily A, member 3
KCNIP2 Kv channel interacting protein 2
KCNK10 potassium channel, two pore domain subfamily K, member 10
LGALS4 lectin, galactoside-binding, soluble, 4
LMAN1 lectin, mannose-binding, 1
LOC100286895 cell division cycle 27 homolog pseudogene
LPPR1 lipid phosphate phosphatase-related protein type 1
LRP4 low density lipoprotein receptor-related protein 4
MALL mal, T-cell differentiation protein-like
MANBA mannosidase, beta A, lysosomal
MAPK10 mitogen-activated protein kinase 10
MBNL3 muscleblind-like splicing regulator 3
MEFV Mediterranean fever
MRPS18C mitochondrial ribosomal protein S18C
MYO15A myosin XVA
NANOG Nanog homeobox
OSBP2 oxysterol binding protein 2
OVOL1 ovo-like zinc finger 1
PCDHGA10 protocadherin gamma subfamily A, 10
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PLAC4 placenta-specific 4
PLTP phospholipid transfer protein
PSG11 pregnancy specific beta-1-glycoprotein 11
RAB3D RAB3D, member RAS oncogene family
RAB40C RAB40C, member RAS oncogene family
RGS20 regulator of G-protein signaling 20
RND1 Rho family GTPase 1
S100A9 S100 calcium binding protein A9
S1PR2 sphingosine-1-phosphate receptor 2
SEMA6D sema domain, transmembrane domain (TM), and cytoplasmic domain, (semaphorin) 6D
SETBP1 SET binding protein 1
SIPA1 signal-induced proliferation-associated 1
SLAMF7 SLAM family member 7
SLFN12 schlafen family member 12
SULT4A1 sulfotransferase family 4A, member 1
TBL1Y transducin (beta)-like 1, Y-linked
TCEB3B transcription elongation factor B polypeptide 3B (elongin A2)
TDRD12 tudor domain containing 12
TEX14 testis expressed 14
TLR5 toll-like receptor 5
TM4SF4 transmembrane 4 L six family member 4
TMPRSS5 transmembrane protease, serine 5
TRIM25 tripartite motif containing 25
XDH xanthine dehydrogenase
ZBTB48 zinc finger and BTB domain containing 48
ZNF423 zinc finger protein 423
ZNF507 zinc finger protein 507