AZD 5438 Gene Set

Dataset LINCS KinomeScan Kinase Inhibitor Targets
Category physical interactions
Type small molecule
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Genes

88 kinases inhibited by the AZD 5438 small molecule from the KinomeScan Kinase Inhibitor Targets dataset.

Symbol Name Standardized Value
CSNK1E casein kinase 1, epsilon 1.36211
CSNK2A2 casein kinase 2, alpha prime polypeptide 1.36211
CDK2 cyclin-dependent kinase 2 1.36211
STK17A serine/threonine kinase 17a 1.36211
GSK3B glycogen synthase kinase 3 beta 1.35325
CDKL2 cyclin-dependent kinase-like 2 (CDC2-related kinase) 1.35325
BMPR2 bone morphogenetic protein receptor, type II (serine/threonine kinase) 1.35325
STK16 serine/threonine kinase 16 1.35325
TLK2 tousled-like kinase 2 1.35325
CSNK1A1L casein kinase 1, alpha 1-like 1.35325
BMPR1B bone morphogenetic protein receptor, type IB 1.35325
GSK3A glycogen synthase kinase 3 alpha 1.34449
BMP2K BMP2 inducible kinase 1.34449
CDK17 cyclin-dependent kinase 17 1.34449
CDK3 cyclin-dependent kinase 3 1.34449
AURKA aurora kinase A 1.34449
STK3 serine/threonine kinase 3 1.34449
TLK1 tousled-like kinase 1 1.34449
CHUK conserved helix-loop-helix ubiquitous kinase 1.34449
IRAK1 interleukin-1 receptor-associated kinase 1 1.34449
EPHB6 EPH receptor B6 1.33582
CSNK1D casein kinase 1, delta 1.33582
MAPK7 mitogen-activated protein kinase 7 1.32726
CSNK2A1 casein kinase 2, alpha 1 polypeptide 1.31878
CDKL3 cyclin-dependent kinase-like 3 1.31878
MAK male germ cell-associated kinase 1.3104
CDK5 cyclin-dependent kinase 5 1.30212
TAOK1 TAO kinase 1 1.30212
ICK intestinal cell (MAK-like) kinase 1.29393
PI4KB phosphatidylinositol 4-kinase, catalytic, beta 1.27782
TGFBR2 transforming growth factor, beta receptor II (70/80kDa) 1.26991
CDK18 cyclin-dependent kinase 18 1.26991
GRK4 G protein-coupled receptor kinase 4 1.25436
CLK2 CDC-like kinase 2 1.25436
CDKL5 cyclin-dependent kinase-like 5 1.25436
HIPK1 homeodomain interacting protein kinase 1 1.23916
CDK9 cyclin-dependent kinase 9 1.2317
NUAK2 NUAK family, SNF1-like kinase, 2 1.22432
HIPK2 homeodomain interacting protein kinase 2 1.21703
CLK4 CDC-like kinase 4 1.21703
MAP3K3 mitogen-activated protein kinase kinase kinase 3 1.20983
MAP3K9 mitogen-activated protein kinase kinase kinase 9 1.20983
CLK1 CDC-like kinase 1 1.20983
HIPK3 homeodomain interacting protein kinase 3 1.20983
IKBKB inhibitor of kappa light polypeptide gene enhancer in B-cells, kinase beta 1.20271
RIPK4 receptor-interacting serine-threonine kinase 4 1.19568
DYRK1B dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1B 1.19568
DCLK3 doublecortin-like kinase 3 1.18186
TAOK3 TAO kinase 3 1.18186
RIPK1 receptor (TNFRSF)-interacting serine-threonine kinase 1 1.18186
STK36 serine/threonine kinase 36 1.17508
CIT citron rho-interacting serine/threonine kinase 1.1424
ACVR1 activin A receptor, type I 1.1424
MAP4K2 mitogen-activated protein kinase kinase kinase kinase 2 1.11767
CDK14 cyclin-dependent kinase 14 1.11767
RIOK2 RIO kinase 2 1.11767
CLK3 CDC-like kinase 3 1.11167
AURKC aurora kinase C 1.10576
TTK TTK protein kinase 1.09415
AAK1 AP2 associated kinase 1 1.09415
NUAK1 NUAK family, SNF1-like kinase, 1 1.08283
DYRK2 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 2 1.08283
CSNK1G3 casein kinase 1, gamma 3 1.05577
PKN2 protein kinase N2 1.05057
IRAK3 interleukin-1 receptor-associated kinase 3 1.04543
ROCK2 Rho-associated, coiled-coil containing protein kinase 2 1.03041
AURKB aurora kinase B 1.02071
GAK cyclin G associated kinase 1.02071
CDK15 cyclin-dependent kinase 15 1.02071
ULK3 unc-51 like kinase 3 1.01596
RIOK1 RIO kinase 1 1.01127
SRPK3 SRSF protein kinase 3 0.993117
TNIK TRAF2 and NCK interacting kinase 0.993117
PIP5K1A phosphatidylinositol-4-phosphate 5-kinase, type I, alpha 0.975893
EPHA3 EPH receptor A3 0.967615
STK24 serine/threonine kinase 24 0.963557
MYLK4 myosin light chain kinase family, member 4 0.955601
MINK1 misshapen-like kinase 1 0.947851
DDR1 discoidin domain receptor tyrosine kinase 1 0.944052
NTRK2 neurotrophic tyrosine kinase, receptor, type 2 0.936602
STK25 serine/threonine kinase 25 0.929345
MERTK MER proto-oncogene, tyrosine kinase 0.922275
PIP4K2B phosphatidylinositol-5-phosphate 4-kinase, type II, beta 0.91201
MAP3K11 mitogen-activated protein kinase kinase kinase 11 0.908676
STK26 serine/threonine protein kinase 26 0.866209
HIPK4 homeodomain interacting protein kinase 4 0.863451
ROCK1 Rho-associated, coiled-coil containing protein kinase 1 0.860727
CAMKK2 calcium/calmodulin-dependent protein kinase kinase 2, beta 0.852752