BICUCULLINE Gene Set

Dataset DGIdb Drug Targets 2026
Category physical interactions
Type drug
Description Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated from Dicentra cucullaria, Adlumia fungosa, Fumariaceae, and several Corydalis species. (Chemical Entities of Biological Interest Ontology, CHEBI_3092)
External Link https://dgidb.org/results?searchType=drug&searchTerms=BICUCULLINE
Similar Terms
Downloads & Tools

Genes

7 interacting proteins for the BICUCULLINE drug from theDGIdb Drug Targets 2026 dataset.

Symbol Name Standardized Value
KCNN1 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 1 0.343714
GABRA1 gamma-aminobutyric acid (GABA) A receptor, alpha 1 0.173169
GABRA4 gamma-aminobutyric acid (GABA) A receptor, alpha 4 0.0763809
GABRA6 gamma-aminobutyric acid (GABA) A receptor, alpha 6 0.0706702
GABRA3 gamma-aminobutyric acid (GABA) A receptor, alpha 3 0.0635438
GABRA5 gamma-aminobutyric acid (GABA) A receptor, alpha 5 0.0619813
GABRA2 gamma-aminobutyric acid (GABA) A receptor, alpha 2 0.0619813