BREXANOLONE Gene Set

Dataset DGIdb Drug Targets 2026
Category physical interactions
Type drug
External Link https://dgidb.org/results?searchType=drug&searchTerms=BREXANOLONE
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Genes

16 interacting proteins for the BREXANOLONE drug from theDGIdb Drug Targets 2026 dataset.

Symbol Name Standardized Value
GABRD gamma-aminobutyric acid (GABA) A receptor, delta 0.0797169
GABRA1 gamma-aminobutyric acid (GABA) A receptor, alpha 1 0.0757614
GABRG2 gamma-aminobutyric acid (GABA) A receptor, gamma 2 0.0751875
GABRB2 gamma-aminobutyric acid (GABA) A receptor, beta 2 0.0727088
GABRG3 gamma-aminobutyric acid (GABA) A receptor, gamma 3 0.0719185
GABRA4 gamma-aminobutyric acid (GABA) A receptor, alpha 4 0.0668333
GABRA6 gamma-aminobutyric acid (GABA) A receptor, alpha 6 0.0618364
GABRA3 gamma-aminobutyric acid (GABA) A receptor, alpha 3 0.0556008
GABRA2 gamma-aminobutyric acid (GABA) A receptor, alpha 2 0.0542336
GABRA5 gamma-aminobutyric acid (GABA) A receptor, alpha 5 0.0542336
GABRQ gamma-aminobutyric acid (GABA) A receptor, theta 0.0424135
GABRG1 gamma-aminobutyric acid (GABA) A receptor, gamma 1 0.0403445
GABRE gamma-aminobutyric acid (GABA) A receptor, epsilon 0.0403445
GABRB3 gamma-aminobutyric acid (GABA) A receptor, beta 3 0.0389206
GABRB1 gamma-aminobutyric acid (GABA) A receptor, beta 1 0.038468
GABRP gamma-aminobutyric acid (GABA) A receptor, pi 0.0371713