CRCGN008_HEPG2_24H:G04 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description tetracycline 5.03 um perturbation at 24 h in HEPG2 (Carcinogenome)
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Genes

212 genes differentially expressed following the CRCGN008_HEPG2_24H:G04 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 10.0
RPP38 ribonuclease P/MRP 38kDa subunit 5.3104
UBQLN2 ubiquilin 2 4.90535
PPARG peroxisome proliferator-activated receptor gamma 4.76405
NOTCH1 notch 1 4.57475
NUDT9 nudix (nucleoside diphosphate linked moiety X)-type motif 9 4.2519
KCNK1 potassium channel, two pore domain subfamily K, member 1 4.02535
VAV3 vav 3 guanine nucleotide exchange factor 3.72857
EGF epidermal growth factor 3.61055
DDIT4 DNA-damage-inducible transcript 4 3.31105
CDC45 cell division cycle 45 3.25015
GPATCH8 G patch domain containing 8 3.23172
NOSIP nitric oxide synthase interacting protein 3.1914
PCK2 phosphoenolpyruvate carboxykinase 2 (mitochondrial) 3.16115
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2 3.03953
MTHFD2 methylenetetrahydrofolate dehydrogenase (NADP+ dependent) 2, methenyltetrahydrofolate cyclohydrolase 3.02985
ADAT1 adenosine deaminase, tRNA-specific 1 2.7115
ARID4B AT rich interactive domain 4B (RBP1-like) 2.4134
AARS1 alanyl-tRNA synthetase 1 2.39225
MMP1 matrix metallopeptidase 1 2.3169
CYCS cytochrome c, somatic 2.2678
CCP110 centriolar coiled coil protein 110kDa 2.26665
CPSF7 cleavage and polyadenylation specific factor 7, 59kDa 2.15965
TMEM33 transmembrane protein 33 2.15485
ZNF518A zinc finger protein 518A 2.15415
EI24 etoposide induced 2.4 2.11795
ANO1 anoctamin 1, calcium activated chloride channel 2.1034
PHGDH phosphoglycerate dehydrogenase 2.0841
RPS6KA1 ribosomal protein S6 kinase, 90kDa, polypeptide 1 2.0578
GOLGA4 golgin A4 2.00915

decreased expression

Symbol Name Standardized Value
NUP85 nucleoporin 85kDa -5.36455
PCNA proliferating cell nuclear antigen -4.77245
CHMP4B charged multivesicular body protein 4B -4.7165
MAPK13 mitogen-activated protein kinase 13 -4.6386
NRIP1 nuclear receptor interacting protein 1 -4.36067
PSMD2 proteasome (prosome, macropain) 26S subunit, non-ATPase, 2 -4.12595
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma -3.67415
ZNF586 zinc finger protein 586 -3.25695
GNAS GNAS complex locus -3.14856
HSPA8 heat shock 70kDa protein 8 -3.14723
RNF167 ring finger protein 167 -3.10005
FGF23 fibroblast growth factor 23 -2.97195
DRD1 dopamine receptor D1 -2.79935
RIT2 Ras-like without CAAX 2 -2.78365
ZFR2 zinc finger RNA binding protein 2 -2.7815
DDX3Y DEAD (Asp-Glu-Ala-Asp) box helicase 3, Y-linked -2.76175
AKAP5 A kinase (PRKA) anchor protein 5 -2.7499
DEFB126 defensin, beta 126 -2.73625
OTUD7B OTU deubiquitinase 7B -2.66825
LIN7B lin-7 homolog B (C. elegans) -2.63475
ULBP1 UL16 binding protein 1 -2.5879
EXT1 exostosin glycosyltransferase 1 -2.57315
MEP1B meprin A, beta -2.5473
H3-4 H3.4 histone, cluster member -2.5441
KCNA10 potassium channel, voltage gated shaker related subfamily A, member 10 -2.54365
SLC8A2 solute carrier family 8 (sodium/calcium exchanger), member 2 -2.5422
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2 -2.52055
GABRA3 gamma-aminobutyric acid (GABA) A receptor, alpha 3 -2.5111
TRHR thyrotropin-releasing hormone receptor -2.51015
GPR75 G protein-coupled receptor 75 -2.5003
CBX8 chromobox homolog 8 -2.4773
ACAA1 acetyl-CoA acyltransferase 1 -2.4592
CDHR2 cadherin-related family member 2 -2.45845
ZNF250 zinc finger protein 250 -2.45685
BRINP1 bone morphogenetic protein/retinoic acid inducible neural-specific 1 -2.43485
ARMCX4 armadillo repeat containing, X-linked 4 -2.42105
RGS9BP regulator of G protein signaling 9 binding protein -2.409
SCAI suppressor of cancer cell invasion -2.3983
PCDHB12 protocadherin beta 12 -2.3955
ZNF613 zinc finger protein 613 -2.3934
PACC1 proton activated chloride channel 1 -2.3913
ZNF415 zinc finger protein 415 -2.3883
OR1E2 olfactory receptor, family 1, subfamily E, member 2 -2.36745
CHIA chitinase, acidic -2.3626
IL3 interleukin 3 -2.35965
ZNF221 zinc finger protein 221 -2.33725
HEYL hes-related family bHLH transcription factor with YRPW motif-like -2.3329
RBM34 RNA binding motif protein 34 -2.32822
TAS2R16 taste receptor, type 2, member 16 -2.30945
ZIC4 Zic family member 4 -2.3034
NRSN2 neurensin 2 -2.30275
TRPC4 transient receptor potential cation channel, subfamily C, member 4 -2.29395
GRIA4 glutamate receptor, ionotropic, AMPA 4 -2.2913
GRM5 glutamate receptor, metabotropic 5 -2.28997
FIG4 FIG4 phosphoinositide 5-phosphatase -2.2858
GUCA1ANB-GUCA1A GUCA1ANB-GUCA1A readthrough -2.28335
GRIA1 glutamate receptor, ionotropic, AMPA 1 -2.28155
WRNIP1 Werner helicase interacting protein 1 -2.2741
HUNK hormonally up-regulated Neu-associated kinase -2.2505
ZNF660-ZNF197 ZNF660-ZNF197 readthrough -2.2487
SLC1A6 solute carrier family 1 (high affinity aspartate/glutamate transporter), member 6 -2.24815
ADRA2B adrenoceptor alpha 2B -2.2431
NLGN1 neuroligin 1 -2.2407
ZNF606 zinc finger protein 606 -2.23935
SLC52A1 solute carrier family 52 (riboflavin transporter), member 1 -2.2366
LRAT lecithin retinol acyltransferase (phosphatidylcholine--retinol O-acyltransferase) -2.2361
OR2B6 olfactory receptor, family 2, subfamily B, member 6 -2.2318
S100G S100 calcium binding protein G -2.2305
MKRN3 makorin ring finger protein 3 -2.2279
MAP1LC3C microtubule-associated protein 1 light chain 3 gamma -2.22295
ZNF334 zinc finger protein 334 -2.22285
S1PR2 sphingosine-1-phosphate receptor 2 -2.21375
AMELX amelogenin, X-linked -2.20845
PNOC prepronociceptin -2.20765
SYP synaptophysin -2.20725
NDUFAF5 NADH dehydrogenase (ubiquinone) complex I, assembly factor 5 -2.20365
HTR2C 5-hydroxytryptamine (serotonin) receptor 2C, G protein-coupled -2.20155
SUMO4 small ubiquitin-like modifier 4 -2.19715
KIR2DS4 killer cell immunoglobulin-like receptor, two domains, short cytoplasmic tail, 4 -2.19558
ZBTB38 zinc finger and BTB domain containing 38 -2.1921
SLC17A1 solute carrier family 17 (organic anion transporter), member 1 -2.1886
TACR3 tachykinin receptor 3 -2.18545
GRM7 glutamate receptor, metabotropic 7 -2.17567
MAP4K1 mitogen-activated protein kinase kinase kinase kinase 1 -2.17502
LDHC lactate dehydrogenase C -2.1724
DNAJC15 DnaJ (Hsp40) homolog, subfamily C, member 15 -2.1709
CMTM6 CKLF-like MARVEL transmembrane domain containing 6 -2.1695
ELL2 elongation factor, RNA polymerase II, 2 -2.1691
PSG5 pregnancy specific beta-1-glycoprotein 5 -2.16735
ACTG1 actin gamma 1 -2.16693
LMAN1L lectin, mannose-binding, 1 like -2.16545
SSTR1 somatostatin receptor 1 -2.1602
CHRNA10 cholinergic receptor, nicotinic, alpha 10 (neuronal) -2.15915
GRIK1 glutamate receptor, ionotropic, kainate 1 -2.15755
ZNF274 zinc finger protein 274 -2.1573
LSM5 LSM5 homolog, U6 small nuclear RNA associated (S. cerevisiae) -2.15462
ZNF813 zinc finger protein 813 -2.15255
OR2F1 olfactory receptor, family 2, subfamily F, member 1 (gene/pseudogene) -2.14595
HOPX HOP homeobox -2.1459
HTR3B 5-hydroxytryptamine (serotonin) receptor 3B, ionotropic -2.14475
GLRA1 glycine receptor, alpha 1 -2.14075
BPY2B basic charge, Y-linked, 2B -2.13965
H2AP H2A.P histone -2.13955
DDX25 DEAD (Asp-Glu-Ala-Asp) box helicase 25 -2.13775
ATP5F1E ATP synthase F1 subunit epsilon -2.13635
KCNK2 potassium channel, two pore domain subfamily K, member 2 -2.1337
ADCYAP1R1 adenylate cyclase activating polypeptide 1 (pituitary) receptor type I -2.1326
KCNAB1 potassium channel, voltage gated subfamily A regulatory beta subunit 1 -2.13194
LRP1B low density lipoprotein receptor-related protein 1B -2.13185
CD52 CD52 molecule -2.12918
TBL1XR1 transducin (beta)-like 1 X-linked receptor 1 -2.1272
SNTG1 syntrophin, gamma 1 -2.12395
HSPB7 heat shock 27kDa protein family, member 7 (cardiovascular) -2.1223
RBP3 retinol binding protein 3, interstitial -2.12225
TAS2R7 taste receptor, type 2, member 7 -2.1212
MAGEB3 melanoma antigen family B3 -2.1205
LOC102725023 killer cell immunoglobulin-like receptor 2DS3 allele 0020101 -2.11225
MTNR1B melatonin receptor 1B -2.1116
ZNF585B zinc finger protein 585B -2.10805
SORCS3 sortilin-related VPS10 domain containing receptor 3 -2.1026
FGF22 fibroblast growth factor 22 -2.1017
ACTL6B actin-like 6B -2.0996
AZGP1 alpha-2-glycoprotein 1, zinc-binding -2.0988
TBX4 T-box 4 -2.0977
ZNF223 zinc finger protein 223 -2.0953
RNF17 ring finger protein 17 -2.09123
B4GALNT1 beta-1,4-N-acetyl-galactosaminyl transferase 1 -2.0906
KIR3DL1 killer cell immunoglobulin-like receptor, three domains, long cytoplasmic tail, 1 -2.08973
ACE angiotensin I converting enzyme -2.08655
DNAJB6 DnaJ (Hsp40) homolog, subfamily B, member 6 -2.08655
DLK2 delta-like 2 homolog (Drosophila) -2.08305
RND1 Rho family GTPase 1 -2.0789
NEUROD6 neuronal differentiation 6 -2.0756
IFNA2 interferon, alpha 2 -2.07475
FOXD3 forkhead box D3 -2.0709
KCTD2 potassium channel tetramerization domain containing 2 -2.07033
KRTAP1-3 keratin associated protein 1-3 -2.0694
FGF14 fibroblast growth factor 14 -2.06765
IFNA16 interferon, alpha 16 -2.0667
SLITRK2 SLIT and NTRK-like family, member 2 -2.06565
ARMCX6 armadillo repeat containing, X-linked 6 -2.0645
KHDRBS2 KH domain containing, RNA binding, signal transduction associated 2 -2.06335
ASIC2 acid sensing (proton gated) ion channel 2 -2.06095
HABP4 hyaluronan binding protein 4 -2.05675
SCN8A sodium channel, voltage gated, type VIII alpha subunit -2.0557
GPR15 G protein-coupled receptor 15 -2.0542
CHFR checkpoint with forkhead and ring finger domains, E3 ubiquitin protein ligase -2.05385
OR5I1 olfactory receptor, family 5, subfamily I, member 1 -2.0535
TBC1D22B TBC1 domain family, member 22B -2.05095
PARK7 parkinson protein 7 -2.05065
FAM246A family with sequence similarity 246 member A -2.0458
TAS2R8 taste receptor, type 2, member 8 -2.04255
CRX cone-rod homeobox -2.0406
SPINT4 serine peptidase inhibitor, Kunitz type 4 -2.03935
SAGE1 sarcoma antigen 1 -2.0392
SAMD14 sterile alpha motif domain containing 14 -2.03855
FOXN1 forkhead box N1 -2.0362
ELOA2 elongin A2 -2.035
SCG3 secretogranin III -2.0309
KCNJ4 potassium channel, inwardly rectifying subfamily J, member 4 -2.02997
GPR50 G protein-coupled receptor 50 -2.0292
ZNF208 zinc finger protein 208 -2.02765
PRSS50 protease, serine, 50 -2.0273
MEPE matrix extracellular phosphoglycoprotein -2.0267
TLX1 T-cell leukemia homeobox 1 -2.02555
GRM8 glutamate receptor, metabotropic 8 -2.02533
CADM3 cell adhesion molecule 3 -2.02443
PTPRN protein tyrosine phosphatase, receptor type, N -2.0219
GRM6 glutamate receptor, metabotropic 6 -2.0211
ANKS1B ankyrin repeat and sterile alpha motif domain containing 1B -2.01915
OR1E1 olfactory receptor, family 1, subfamily E, member 1 -2.01865
NTN3 netrin 3 -2.0153
HIGD1B HIG1 hypoxia inducible domain family, member 1B -2.01465
CD58 CD58 molecule -2.00997
KCNA4 potassium channel, voltage gated shaker related subfamily A, member 4 -2.00915
SLC34A2 solute carrier family 34 (type II sodium/phosphate cotransporter), member 2 -2.00825
ALDOC aldolase C, fructose-bisphosphate -2.00765
CRISP1 cysteine-rich secretory protein 1 -2.00662
GGA3 golgi-associated, gamma adaptin ear containing, ARF binding protein 3 -2.00502
TSKS testis-specific serine kinase substrate -2.00475
BRDT bromodomain, testis-specific -2.0036
AIG1 androgen-induced 1 -2.00135