CRCGN008_HEPG2_24H:G12 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description methoxychlor 1.25 um perturbation at 24 h in HEPG2 (Carcinogenome)
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Genes

87 genes differentially expressed following the CRCGN008_HEPG2_24H:G12 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
PPP1R13B protein phosphatase 1, regulatory subunit 13B 5.4611
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5 5.43155
NUDT9 nudix (nucleoside diphosphate linked moiety X)-type motif 9 5.21595
CHMP6 charged multivesicular body protein 6 5.092
PPARG peroxisome proliferator-activated receptor gamma 4.85795
BACE2 beta-site APP-cleaving enzyme 2 4.75235
STK10 serine/threonine kinase 10 4.66447
LYN LYN proto-oncogene, Src family tyrosine kinase 4.6491
CIAO3 cytosolic iron-sulfur assembly component 3 4.599
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5 4.56725
GPER1 G protein-coupled estrogen receptor 1 3.79043
MAP3K4 mitogen-activated protein kinase kinase kinase 4 3.73925
CEP57 centrosomal protein 57kDa 3.65088
CASP2 caspase 2, apoptosis-related cysteine peptidase 3.64631
CDCA4 cell division cycle associated 4 3.57265
LPAR2 lysophosphatidic acid receptor 2 3.44325
GSTZ1 glutathione S-transferase zeta 1 3.38395
IKBKE inhibitor of kappa light polypeptide gene enhancer in B-cells, kinase epsilon 2.89372
GRWD1 glutamate-rich WD repeat containing 1 2.7513
KIF20A kinesin family member 20A 2.7023
GZMH granzyme H (cathepsin G-like 2, protein h-CCPX) 2.6799
FCGR3B Fc fragment of IgG, low affinity IIIb, receptor (CD16b) 2.5051
MMS19 MMS19 nucleotide excision repair homolog (S. cerevisiae) 2.48625
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3 2.44135
WNT6 wingless-type MMTV integration site family, member 6 2.38775
PDE6G phosphodiesterase 6G, cGMP-specific, rod, gamma 2.3401
SORBS3 sorbin and SH3 domain containing 3 2.32603
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2 2.31961
UPK2 uroplakin 2 2.31225
MTERF3 mitochondrial transcription termination factor 3 2.2714
AMHR2 anti-Mullerian hormone receptor, type II 2.2575
TESC tescalcin 2.23505
HOOK2 hook microtubule-tethering protein 2 2.22795
KREMEN2 kringle containing transmembrane protein 2 2.21825
WDR25 WD repeat domain 25 2.2072
SYNGR3 synaptogyrin 3 2.19965
TMEM121 transmembrane protein 121 2.1803
CETP cholesteryl ester transfer protein, plasma 2.16825
TP53 tumor protein p53 2.1675
PEAK1 pseudopodium-enriched atypical kinase 1 2.15425
SYT17 synaptotagmin XVII 2.1511
BTK Bruton agammaglobulinemia tyrosine kinase 2.1496
TBP TATA box binding protein 2.13875
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1 2.1365
QSER1 glutamine and serine rich 1 2.1338
WDTC1 WD and tetratricopeptide repeats 1 2.10245
FIS1 fission 1 (mitochondrial outer membrane) homolog (S. cerevisiae) 2.0909
RXRG retinoid X receptor, gamma 2.0848
LOC124905743 low affinity immunoglobulin gamma Fc region receptor III-B 2.06415
N4BP3 NEDD4 binding protein 3 2.0515
GRIN2D glutamate receptor, ionotropic, N-methyl D-aspartate 2D 2.04895
TRPV4 transient receptor potential cation channel, subfamily V, member 4 2.01195
VSIG4 V-set and immunoglobulin domain containing 4 2.00745
ZFPM1 zinc finger protein, FOG family member 1 2.0044

decreased expression

Symbol Name Standardized Value
CD320 CD320 molecule -6.5438
HMG20B high mobility group 20B -6.39145
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2 -6.23925
DHRS7 dehydrogenase/reductase (SDR family) member 7 -5.9426
SLC7A5 solute carrier family 7 (amino acid transporter light chain, L system), member 5 -5.2978
ZMIZ1 zinc finger, MIZ-type containing 1 -4.93905
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -4.83225
TRIB3 tribbles pseudokinase 3 -4.7646
CDC20 cell division cycle 20 -4.6933
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1 -4.6202
FASTKD5 FAST kinase domains 5 -4.28715
NRIP1 nuclear receptor interacting protein 1 -4.23723
ALDH1A1 aldehyde dehydrogenase 1 family, member A1 -4.12405
CCNB1 cyclin B1 -4.11465
HLA-DMA major histocompatibility complex, class II, DM alpha -3.7998
CCNB2 cyclin B2 -3.63295
FGFR4 fibroblast growth factor receptor 4 -3.34838
PRPF4 pre-mRNA processing factor 4 -3.18103
LSM5 LSM5 homolog, U6 small nuclear RNA associated (S. cerevisiae) -2.9057
WASHC4 WASH complex subunit 4 -2.85662
CHIC2 cysteine-rich hydrophobic domain 2 -2.7421
ZW10 zw10 kinetochore protein -2.63485
TXNDC9 thioredoxin domain containing 9 -2.55748
OXA1L oxidase (cytochrome c) assembly 1-like -2.4344
GGCT gamma-glutamylcyclotransferase -2.384
COPS7A COP9 signalosome subunit 7A -2.3604
SCGB1D2 secretoglobin, family 1D, member 2 -2.16295
COL4A5 collagen, type IV, alpha 5 -2.1233
MOB3B MOB kinase activator 3B -2.08825
DAZAP1 DAZ associated protein 1 -2.081
ADCY7 adenylate cyclase 7 -2.058
TTBK2 tau tubulin kinase 2 -2.0234
HNRNPH2 heterogeneous nuclear ribonucleoprotein H2 (H') -2.00465