CRCGN008_HEPG2_24H:H07 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description tiabendazole 40.2 um perturbation at 24 h in HEPG2 (Carcinogenome)
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Genes

85 genes differentially expressed following the CRCGN008_HEPG2_24H:H07 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
CHN1 chimerin 1 7.02165
RPL39L ribosomal protein L39-like 6.1537
EPHB2 EPH receptor B2 5.69382
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5 5.36885
MYLK myosin light chain kinase 5.0192
GNAI1 guanine nucleotide binding protein (G protein), alpha inhibiting activity polypeptide 1 4.98905
INPP4B inositol polyphosphate-4-phosphatase, type II, 105kDa 4.81265
E2F2 E2F transcription factor 2 4.4933
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5 4.43385
NOTCH1 notch 1 4.27405
EAPP E2F-associated phosphoprotein 4.23845
DNAJB2 DnaJ (Hsp40) homolog, subfamily B, member 2 4.139
NMU neuromedin U 4.02685
ATP11B ATPase, class VI, type 11B 3.94195
STIMATE STIM activating enhancer 3.6132
P4HTM prolyl 4-hydroxylase, transmembrane (endoplasmic reticulum) 3.51905
HLA-DRA major histocompatibility complex, class II, DR alpha 3.51203
PEX11A peroxisomal biogenesis factor 11 alpha 3.499
CCDC85B coiled-coil domain containing 85B 3.381
SNAP25 synaptosomal-associated protein, 25kDa 3.3508
GNA15 guanine nucleotide binding protein (G protein), alpha 15 (Gq class) 3.3445
F3 coagulation factor III (thromboplastin, tissue factor) 2.71215
FXYD7 FXYD domain containing ion transport regulator 7 2.6733
JADE2 jade family PHD finger 2 2.6396
CEBPD CCAAT/enhancer binding protein (C/EBP), delta 2.6384
DEFA6 defensin, alpha 6, Paneth cell-specific 2.61555
PARL presenilin associated, rhomboid-like 2.52715
KIF20A kinesin family member 20A 2.49235
VWA1 von Willebrand factor A domain containing 1 2.47845
PIK3C2B phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 beta 2.4584
BPHL biphenyl hydrolase-like (serine hydrolase) 2.43795
VSNL1 visinin-like 1 2.42982
STRA6 stimulated by retinoic acid 6 2.4274
BTK Bruton agammaglobulinemia tyrosine kinase 2.3526
P2RY2 purinergic receptor P2Y, G-protein coupled, 2 2.33225
ALG9 ALG9, alpha-1,2-mannosyltransferase 2.28945
GALT galactose-1-phosphate uridylyltransferase 2.26825
CEP57 centrosomal protein 57kDa 2.2638
TGFB3 transforming growth factor, beta 3 2.2299
RNF186 ring finger protein 186 2.2269
HABP4 hyaluronan binding protein 4 2.2195
FAM168B family with sequence similarity 168, member B 2.15465
RGCC regulator of cell cycle 2.15275
ANO1 anoctamin 1, calcium activated chloride channel 2.1422
TNFRSF1B tumor necrosis factor receptor superfamily, member 1B 2.10435
SYNGR3 synaptogyrin 3 2.0606
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1 2.0569
EIF2B5 eukaryotic translation initiation factor 2B, subunit 5 epsilon, 82kDa 2.0565
THEM6 thioesterase superfamily member 6 2.0343
LRCH3 leucine-rich repeats and calponin homology (CH) domain containing 3 2.01705

decreased expression

Symbol Name Standardized Value
KDM3A lysine (K)-specific demethylase 3A -5.84225
ANKRD10 ankyrin repeat domain 10 -5.458
PCNA proliferating cell nuclear antigen -4.77245
TSPAN4 tetraspanin 4 -4.73425
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -4.62445
TM9SF3 transmembrane 9 superfamily member 3 -4.53755
SPAG4 sperm associated antigen 4 -4.32125
CDC20 cell division cycle 20 -4.2605
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma -4.1565
G3BP1 GTPase activating protein (SH3 domain) binding protein 1 -3.63153
CHIC2 cysteine-rich hydrophobic domain 2 -3.465
FGFR4 fibroblast growth factor receptor 4 -3.19497
ATF5 activating transcription factor 5 -2.94738
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3 -2.9265
HSPA8 heat shock 70kDa protein 8 -2.75777
FOS FBJ murine osteosarcoma viral oncogene homolog -2.7478
TENT4A terminal nucleotidyltransferase 4A -2.6418
DCK deoxycytidine kinase -2.594
PDIA5 protein disulfide isomerase family A, member 5 -2.44185
MAP1LC3B microtubule-associated protein 1 light chain 3 beta -2.3536
KRT18 keratin 18, type I -2.3279
MTHFD2L methylenetetrahydrofolate dehydrogenase (NADP+ dependent) 2-like -2.31075
ARPC5 actin related protein 2/3 complex, subunit 5, 16kDa -2.29995
FCHO1 FCH domain only 1 -2.26185
DRC9 dynein regulatory complex subunit 9 -2.18765
CLIC2 chloride intracellular channel 2 -2.17745
DPYSL2 dihydropyrimidinase-like 2 -2.16455
ARID5B AT rich interactive domain 5B (MRF1-like) -2.14615
DHRS7 dehydrogenase/reductase (SDR family) member 7 -2.13215
ABI1 abl-interactor 1 -2.12157
TPK1 thiamin pyrophosphokinase 1 -2.1124
HNMT histamine N-methyltransferase -2.08423
CDKN2AIP CDKN2A interacting protein -2.04995
GOLT1B golgi transport 1B -2.01755
BMP2 bone morphogenetic protein 2 -2.00612