CRCGN009_HEPG2_24H:N02 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description theophylline 20.2 um perturbation at 24 h in HEPG2 (Carcinogenome)
Similar Terms
Downloads & Tools

Genes

90 genes differentially expressed following the CRCGN009_HEPG2_24H:N02 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
MEF2C myocyte enhancer factor 2C 6.63119
INPP4B inositol polyphosphate-4-phosphatase, type II, 105kDa 5.63875
MAMLD1 mastermind-like domain containing 1 5.45825
CLPX caseinolytic mitochondrial matrix peptidase chaperone subunit 5.22535
EPHA3 EPH receptor A3 4.96122
MAP7 microtubule-associated protein 7 3.97894
TIAM1 T-cell lymphoma invasion and metastasis 1 3.96851
CASP2 caspase 2, apoptosis-related cysteine peptidase 3.92534
C2CD2 C2 calcium-dependent domain containing 2 3.87001
RPL39L ribosomal protein L39-like 3.82806
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5 3.78108
EVL Enah/Vasp-like 3.74652
HLA-DMA major histocompatibility complex, class II, DM alpha 3.6036
KLHL9 kelch-like family member 9 3.56833
VAV3 vav 3 guanine nucleotide exchange factor 3.29862
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 3.08066
HERC6 HECT and RLD domain containing E3 ubiquitin protein ligase family member 6 2.99768
ATP11B ATPase, class VI, type 11B 2.97885
RPP38 ribonuclease P/MRP 38kDa subunit 2.91436
JADE2 jade family PHD finger 2 2.89732
KCNK1 potassium channel, two pore domain subfamily K, member 1 2.87696
IKZF1 IKAROS family zinc finger 1 (Ikaros) 2.77637
MYL1 myosin, light chain 1, alkali; skeletal, fast 2.77437
SYNGR3 synaptogyrin 3 2.66819
KLHL41 kelch-like family member 41 2.66724
CHMP6 charged multivesicular body protein 6 2.62076
TBC1D10C TBC1 domain family, member 10C 2.53574
MYBPH myosin binding protein H 2.51234
RRS1 RRS1 ribosome biogenesis regulator homolog (S. cerevisiae) 2.48164
CNPY3 canopy FGF signaling regulator 3 2.39118
SCRN1 secernin 1 2.33938
RYR3 ryanodine receptor 3 2.2793
ADRB2 adrenoceptor beta 2, surface 2.23554
TNNI1 troponin I type 1 (skeletal, slow) 2.23443
NUDT9 nudix (nucleoside diphosphate linked moiety X)-type motif 9 2.2221
MYL11 myosin light chain 11 2.16761
CHRNB3 cholinergic receptor, nicotinic, beta 3 (neuronal) 2.15919
CSRP3 cysteine and glycine-rich protein 3 (cardiac LIM protein) 2.13356
KRT36 keratin 36, type I 2.13201
TNNC2 troponin C type 2 (fast) 2.13048
APBB1IP amyloid beta (A4) precursor protein-binding, family B, member 1 interacting protein 2.11356
RYR1 ryanodine receptor 1 (skeletal) 2.0879
SYNPO2L synaptopodin 2-like 2.07005
KCNV2 potassium channel, voltage gated modifier subfamily V, member 2 2.0669
CD37 CD37 molecule 2.05535
TIMM22 translocase of inner mitochondrial membrane 22 homolog (yeast) 2.04405
MYL2 myosin, light chain 2, regulatory, cardiac, slow 2.04183
NR1H2 nuclear receptor subfamily 1, group H, member 2 2.03616
DCAF4 DDB1 and CUL4 associated factor 4 2.02878
IKBKE inhibitor of kappa light polypeptide gene enhancer in B-cells, kinase epsilon 2.02854
STXBP2 syntaxin binding protein 2 2.024
ENO3 enolase 3 (beta, muscle) 2.02076
MYOZ2 myozenin 2 2.01781
TANC2 tetratricopeptide repeat, ankyrin repeat and coiled-coil containing 2 2.01222

decreased expression

Symbol Name Standardized Value
VAT1 vesicle amine transport 1 -5.86739
CASP7 caspase 7, apoptosis-related cysteine peptidase -5.83302
PCNA proliferating cell nuclear antigen -5.64279
CDKN1B cyclin-dependent kinase inhibitor 1B (p27, Kip1) -4.63334
TARBP1 TAR (HIV-1) RNA binding protein 1 -4.35132
TLCD3A TLC domain containing 3A -4.036
ZMIZ1 zinc finger, MIZ-type containing 1 -3.59624
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1 -3.37412
CDC20 cell division cycle 20 -3.30774
PLEKHJ1 pleckstrin homology domain containing, family J member 1 -3.10562
LDHD lactate dehydrogenase D -3.02464
SNX11 sorting nexin 11 -2.94727
ITGB1BP1 integrin beta 1 binding protein 1 -2.79298
MRPS2 mitochondrial ribosomal protein S2 -2.78859
THAP11 THAP domain containing 11 -2.69421
ARID5B AT rich interactive domain 5B (MRF1-like) -2.68375
NR2F6 nuclear receptor subfamily 2, group F, member 6 -2.63784
NSDHL NAD(P) dependent steroid dehydrogenase-like -2.58926
ITFG1 integrin alpha FG-GAP repeat containing 1 -2.58303
CCNB2 cyclin B2 -2.55962
GOLT1B golgi transport 1B -2.53828
DERA deoxyribose-phosphate aldolase (putative) -2.51703
RGS2 regulator of G-protein signaling 2 -2.42716
MTA1 metastasis associated 1 -2.33331
ZDHHC6 zinc finger, DHHC-type containing 6 -2.25377
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -2.21388
FASTKD5 FAST kinase domains 5 -2.19065
FABP5 fatty acid binding protein 5 (psoriasis-associated) -2.17684
ADI1 acireductone dioxygenase 1 -2.17461
CCNB1 cyclin B1 -2.1341
ZW10 zw10 kinetochore protein -2.13318
REEP5 receptor accessory protein 5 -2.11576
NCOA6 nuclear receptor coactivator 6 -2.10431
DNAJA3 DnaJ (Hsp40) homolog, subfamily A, member 3 -2.05926
NT5DC2 5'-nucleotidase domain containing 2 -2.04392
NRIP1 nuclear receptor interacting protein 1 -2.04246