CRCGN012_HEPG2_24H:E21 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description telone ii 10.05 um perturbation at 24 h in HEPG2 (Carcinogenome)
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Genes

99 genes differentially expressed following the CRCGN012_HEPG2_24H:E21 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
E2F2 E2F transcription factor 2 7.38596
PPARG peroxisome proliferator-activated receptor gamma 5.41584
PFKL phosphofructokinase, liver 4.91723
ADRB2 adrenoceptor beta 2, surface 4.1977
CHMP6 charged multivesicular body protein 6 4.10962
NFATC4 nuclear factor of activated T-cells, cytoplasmic, calcineurin-dependent 4 4.07786
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 4.04656
IKBKE inhibitor of kappa light polypeptide gene enhancer in B-cells, kinase epsilon 3.92219
BACE2 beta-site APP-cleaving enzyme 2 3.86976
P4HTM prolyl 4-hydroxylase, transmembrane (endoplasmic reticulum) 3.84605
SRC SRC proto-oncogene, non-receptor tyrosine kinase 3.71888
MAST2 microtubule associated serine/threonine kinase 2 3.66945
CSK c-src tyrosine kinase 3.50169
PHKG2 phosphorylase kinase, gamma 2 (testis) 3.45249
SNAP25 synaptosomal-associated protein, 25kDa 3.41005
MOK MOK protein kinase 3.39355
MNAT1 MNAT CDK-activating kinase assembly factor 1 3.28542
LPAR2 lysophosphatidic acid receptor 2 3.09872
PWP2 PWP2 periodic tryptophan protein homolog (yeast) 3.08611
DYNLT3 dynein, light chain, Tctex-type 3 3.05446
HOXA10 homeobox A10 3.0327
CXCR4 chemokine (C-X-C motif) receptor 4 2.96612
NOTCH1 notch 1 2.96134
PAX1 paired box 1 2.85319
ADGRE5 adhesion G protein-coupled receptor E5 2.7794
RPP38 ribonuclease P/MRP 38kDa subunit 2.73372
UBQLN2 ubiquilin 2 2.63097
RELB v-rel avian reticuloendotheliosis viral oncogene homolog B 2.5654
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5 2.53606
MYO1F myosin IF 2.50526
GATD3 glutamine amidotransferase class 1 domain containing 3 2.50417
NPFFR1 neuropeptide FF receptor 1 2.44696
APBA1 amyloid beta (A4) precursor protein-binding, family A, member 1 2.42679
UPK2 uroplakin 2 2.39801
PLS1 plastin 1 2.37871
DCUN1D4 DCN1, defective in cullin neddylation 1, domain containing 4 2.32756
APLP1 amyloid beta (A4) precursor-like protein 1 2.28677
CCNF cyclin F 2.25281
GPER1 G protein-coupled estrogen receptor 1 2.24752
HOXA10-HOXA9 HOXA10-HOXA9 readthrough 2.23243
KLRC4-KLRK1 KLRC4-KLRK1 readthrough 2.21828
CLIP2 CAP-GLY domain containing linker protein 2 2.21519
B3GAT1 beta-1,3-glucuronyltransferase 1 2.20497
WNT3 wingless-type MMTV integration site family, member 3 2.18827
CSDC2 cold shock domain containing C2, RNA binding 2.18327
TMEM50B transmembrane protein 50B 2.16903
POMT2 protein-O-mannosyltransferase 2 2.15814
CT55 cancer/testis antigen 55 2.15276
MAP7 microtubule-associated protein 7 2.14055
OLIG2 oligodendrocyte lineage transcription factor 2 2.13681
SLC5A5 solute carrier family 5 (sodium/iodide cotransporter), member 5 2.13377
KCNAB3 potassium channel, voltage gated subfamily A regulatory beta subunit 3 2.1123
TMEM161A transmembrane protein 161A 2.11055
ATP1A3 ATPase, Na+/K+ transporting, alpha 3 polypeptide 2.11048
MAP3K20 mitogen-activated protein kinase kinase kinase 20 2.10947
CD207 CD207 molecule, langerin 2.09205
TIAM1 T-cell lymphoma invasion and metastasis 1 2.08565
MAPK4 mitogen-activated protein kinase 4 2.07778
TRPM2 transient receptor potential cation channel, subfamily M, member 2 2.06683
STK10 serine/threonine kinase 10 2.06519
OVOL3 ovo-like zinc finger 3 2.06373
ZBTB25 zinc finger and BTB domain containing 25 2.04821
TRAPPC10 trafficking protein particle complex 10 2.04167
IHH indian hedgehog 2.03613
ATAD3A ATPase family, AAA domain containing 3A 2.03066
SH2B2 SH2B adaptor protein 2 2.02908
PCBP4 poly(rC) binding protein 4 2.02739
LOC102723996 ICOS ligand 2.02543
OMG oligodendrocyte myelin glycoprotein 2.00281
RAX retina and anterior neural fold homeobox 2.00181

decreased expression

Symbol Name Standardized Value
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2 -6.25868
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -6.2367
KDM3A lysine (K)-specific demethylase 3A -5.90917
SLC7A5 solute carrier family 7 (amino acid transporter light chain, L system), member 5 -5.00071
PCNA proliferating cell nuclear antigen -4.38021
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1 -4.03041
EGF epidermal growth factor -3.98858
ZDHHC6 zinc finger, DHHC-type containing 6 -3.83113
UGDH UDP-glucose 6-dehydrogenase -3.69325
TARBP1 TAR (HIV-1) RNA binding protein 1 -3.39309
ADI1 acireductone dioxygenase 1 -3.36079
CD320 CD320 molecule -3.17175
CNDP2 CNDP dipeptidase 2 (metallopeptidase M20 family) -3.07593
LDHD lactate dehydrogenase D -3.01812
CCNB2 cyclin B2 -2.91264
HACD3 3-hydroxyacyl-CoA dehydratase 3 -2.74028
DNM1L dynamin 1-like -2.68162
ITGB1BP1 integrin beta 1 binding protein 1 -2.66688
PCK2 phosphoenolpyruvate carboxykinase 2 (mitochondrial) -2.64802
MRPS2 mitochondrial ribosomal protein S2 -2.64769
MAPK13 mitogen-activated protein kinase 13 -2.5195
DNAJB6 DnaJ (Hsp40) homolog, subfamily B, member 6 -2.51108
GNAS GNAS complex locus -2.48205
LYPLA1 lysophospholipase I -2.24233
SLC35F2 solute carrier family 35, member F2 -2.18895
WASHC4 WASH complex subunit 4 -2.13405
G0S2 G0/G1 switch 2 -2.04687
TERF2IP telomeric repeat binding factor 2, interacting protein -2.03962
MAP4K4 mitogen-activated protein kinase kinase kinase kinase 4 -2.00654