CRCGN013_HEPG2_24H:E17 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description methyl (z)-2-(dimethylamino)-n-((methylcarbamoyl)oxy)-2-oxoethanimidothioate 1.25 um perturbation at 24 h in HEPG2 (Carcinogenome)
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Genes

69 genes differentially expressed following the CRCGN013_HEPG2_24H:E17 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
NUDT9 nudix (nucleoside diphosphate linked moiety X)-type motif 9 6.82417
P4HTM prolyl 4-hydroxylase, transmembrane (endoplasmic reticulum) 6.33225
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 5.29166
CCNF cyclin F 4.27392
CCDC85B coiled-coil domain containing 85B 4.12405
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5 4.12158
EPHA3 EPH receptor A3 3.97839
RPP38 ribonuclease P/MRP 38kDa subunit 3.84573
AMDHD2 amidohydrolase domain containing 2 3.76394
MEF2C myocyte enhancer factor 2C 3.74866
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3 3.70389
CIAO3 cytosolic iron-sulfur assembly component 3 3.63261
PPARG peroxisome proliferator-activated receptor gamma 3.52594
PEX11A peroxisomal biogenesis factor 11 alpha 3.45646
CCL2 chemokine (C-C motif) ligand 2 3.29978
E2F2 E2F transcription factor 2 3.24069
MYLK myosin light chain kinase 3.16657
CCDC92 coiled-coil domain containing 92 3.09464
NFIL3 nuclear factor, interleukin 3 regulated 3.00891
CLPX caseinolytic mitochondrial matrix peptidase chaperone subunit 2.73535
GSTZ1 glutathione S-transferase zeta 1 2.65616
PLS1 plastin 1 2.55603
MMRN1 multimerin 1 2.50599
CYCS cytochrome c, somatic 2.41574
LCN2 lipocalin 2 2.4149
RERGL RERG/RAS-like 2.40026
ANKRD1 ankyrin repeat domain 1 (cardiac muscle) 2.39643
CHMP6 charged multivesicular body protein 6 2.334
PFKL phosphofructokinase, liver 2.33297
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18 2.31938
FZD7 frizzled class receptor 7 2.27782
CCDC186 coiled-coil domain containing 186 2.27256
TAF5L TAF5-like RNA polymerase II, p300/CBP-associated factor (PCAF)-associated factor, 65kDa 2.2396
TBXA2R thromboxane A2 receptor 2.22074
TNNT3 troponin T type 3 (skeletal, fast) 2.18772
RAPGEF1 Rap guanine nucleotide exchange factor (GEF) 1 2.18366
DUSP28 dual specificity phosphatase 28 2.11924
ADAT1 adenosine deaminase, tRNA-specific 1 2.07575
TPM3 tropomyosin 3 2.07511
CHMP1A charged multivesicular body protein 1A 2.04865
HLA-DMA major histocompatibility complex, class II, DM alpha 2.04489
CSRP3 cysteine and glycine-rich protein 3 (cardiac LIM protein) 2.03844
RBMXL2 RNA binding motif protein, X-linked-like 2 2.00944

decreased expression

Symbol Name Standardized Value
DNAJA3 DnaJ (Hsp40) homolog, subfamily A, member 3 -7.45468
CCNB2 cyclin B2 -4.87951
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma -4.49416
LDHD lactate dehydrogenase D -4.08981
DHRS7 dehydrogenase/reductase (SDR family) member 7 -3.97612
ANKRD10 ankyrin repeat domain 10 -3.83788
DSG2 desmoglein 2 -3.66308
OXA1L oxidase (cytochrome c) assembly 1-like -3.54575
ZNF586 zinc finger protein 586 -3.32162
ZMIZ1 zinc finger, MIZ-type containing 1 -3.21901
RFC2 replication factor C (activator 1) 2, 40kDa -3.13161
GALE UDP-galactose-4-epimerase -3.06443
HMG20B high mobility group 20B -3.00934
PPP2R3C protein phosphatase 2, regulatory subunit B'', gamma -2.99451
CHMP4B charged multivesicular body protein 4B -2.69026
FGFR4 fibroblast growth factor receptor 4 -2.68104
PPP2R5E protein phosphatase 2, regulatory subunit B', epsilon isoform -2.39589
CNDP2 CNDP dipeptidase 2 (metallopeptidase M20 family) -2.37149
HSD17B11 hydroxysteroid (17-beta) dehydrogenase 11 -2.34541
CDKN1B cyclin-dependent kinase inhibitor 1B (p27, Kip1) -2.29638
ANKRD27 ankyrin repeat domain 27 (VPS9 domain) -2.28349
PCNA proliferating cell nuclear antigen -2.2458
RGS20 regulator of G-protein signaling 20 -2.21639
VDAC1 voltage-dependent anion channel 1 -2.19683
CDC37 cell division cycle 37 -2.09852
ETFB electron-transfer-flavoprotein, beta polypeptide -2.01619