CRCGN014_HEPG2_3H:C06 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description caprolactam 40.0 um perturbation at 3 h in HEPG2 (Carcinogenome)
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Genes

186 genes differentially expressed following the CRCGN014_HEPG2_3H:C06 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
CIAO3 cytosolic iron-sulfur assembly component 3 5.65195
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 5.42431
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5 5.25546
CCL2 chemokine (C-C motif) ligand 2 5.15179
DIPK1A divergent protein kinase domain 1A 5.05564
TERT telomerase reverse transcriptase 4.93721
PPP1R13B protein phosphatase 1, regulatory subunit 13B 4.64562
CXCL2 chemokine (C-X-C motif) ligand 2 4.39277
ADGRE5 adhesion G protein-coupled receptor E5 4.36904
HOXA10 homeobox A10 4.15659
CASP2 caspase 2, apoptosis-related cysteine peptidase 4.05581
SLC27A3 solute carrier family 27 (fatty acid transporter), member 3 4.05431
NOTCH1 notch 1 3.99109
KCNK1 potassium channel, two pore domain subfamily K, member 1 3.80214
PLSCR3 phospholipid scramblase 3 3.7539
CLPX caseinolytic mitochondrial matrix peptidase chaperone subunit 3.74651
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha 3.7143
CCNA1 cyclin A1 3.61901
IGFBP3 insulin-like growth factor binding protein 3 3.57682
SHB Src homology 2 domain containing adaptor protein B 3.30789
PTK2 protein tyrosine kinase 2 3.2236
GNGT1 guanine nucleotide binding protein (G protein), gamma transducing activity polypeptide 1 3.21619
CYCS cytochrome c, somatic 3.0912
NUDT9 nudix (nucleoside diphosphate linked moiety X)-type motif 9 2.88337
ANO1 anoctamin 1, calcium activated chloride channel 2.83609
MEST mesoderm specific transcript 2.80106
KIFBP kinesin family binding protein 2.79261
LPAR3 lysophosphatidic acid receptor 3 2.73138
ADAMTS20 ADAM metallopeptidase with thrombospondin type 1 motif, 20 2.6981
RPS6KA1 ribosomal protein S6 kinase, 90kDa, polypeptide 1 2.63837
AGTR2 angiotensin II receptor, type 2 2.60816
JCAD junctional cadherin 5 associated 2.56827
GTPBP10 GTP-binding protein 10 (putative) 2.55113
SLC25A30 solute carrier family 25, member 30 2.54185
EPHA3 EPH receptor A3 2.53277
MAGEB3 melanoma antigen family B3 2.52912
ATP1B4 ATPase, Na+/K+ transporting, beta 4 polypeptide 2.52238
RIPPLY2-CYB5R4 RIPPLY2-CYB5R4 readthrough 2.49883
PLA2G2F phospholipase A2, group IIF 2.49213
PRDM9 PR domain containing 9 2.48679
PSORS1C1 psoriasis susceptibility 1 candidate 1 2.44781
CFAP43 cilia and flagella associated protein 43 2.44039
RAD21L1 RAD21-like 1 (S. pombe) 2.4317
TLL1 tolloid-like 1 2.41443
COLEC10 collectin sub-family member 10 (C-type lectin) 2.41218
MAGEB4 melanoma antigen family B4 2.4061
ZFY zinc finger protein, Y-linked 2.40341
MYEF2 myelin expression factor 2 2.38827
NOX3 NADPH oxidase 3 2.38288
LTB lymphotoxin beta (TNF superfamily, member 3) 2.37893
SHC1 SHC (Src homology 2 domain containing) transforming protein 1 2.37405
IFNA8 interferon, alpha 8 2.37237
PPARGC1B peroxisome proliferator-activated receptor gamma, coactivator 1 beta 2.3669
TEX12 testis expressed 12 2.36267
NDUFAF5 NADH dehydrogenase (ubiquinone) complex I, assembly factor 5 2.3603
ZNF493 zinc finger protein 493 2.35012
IFNA16 interferon, alpha 16 2.3354
OR2B2 olfactory receptor, family 2, subfamily B, member 2 2.32279
PAPOLB poly(A) polymerase beta (testis specific) 2.31595
POU6F2 POU class 6 homeobox 2 2.31042
ZNF234 zinc finger protein 234 2.30888
PPEF2 protein phosphatase, EF-hand calcium binding domain 2 2.30791
TAF13 TAF13 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 18kDa 2.29936
TEX15 testis expressed 15 2.28956
KCNA4 potassium channel, voltage gated shaker related subfamily A, member 4 2.27908
LEFTY1 left-right determination factor 1 2.26664
P2RX3 purinergic receptor P2X, ligand gated ion channel, 3 2.26604
ZNF157 zinc finger protein 157 2.25745
LHCGR luteinizing hormone/choriogonadotropin receptor 2.25476
VHL von Hippel-Lindau tumor suppressor, E3 ubiquitin protein ligase 2.25391
THNSL1 threonine synthase-like 1 (S. cerevisiae) 2.25272
CCR6 chemokine (C-C motif) receptor 6 2.25268
OR2B6 olfactory receptor, family 2, subfamily B, member 6 2.25025
FAM13C family with sequence similarity 13, member C 2.24309
PBOV1 prostate and breast cancer overexpressed 1 2.23574
DLK2 delta-like 2 homolog (Drosophila) 2.22609
CCDC144A coiled-coil domain containing 144A 2.22439
TAS2R9 taste receptor, type 2, member 9 2.22119
SLC30A4 solute carrier family 30 (zinc transporter), member 4 2.22055
IMPG2 interphotoreceptor matrix proteoglycan 2 2.21719
ZNF80 zinc finger protein 80 2.21185
ARSL arylsulfatase L 2.21109
RNF32 ring finger protein 32 2.21046
OR3A2 olfactory receptor, family 3, subfamily A, member 2 2.20604
GPR85 G protein-coupled receptor 85 2.19723
ACOXL acyl-CoA oxidase-like 2.19561
AGBL3 ATP/GTP binding protein-like 3 2.19387
PTTG2 pituitary tumor-transforming 2 2.19345
PCLO piccolo presynaptic cytomatrix protein 2.18635
MLNR motilin receptor 2.18557
DHRS3 dehydrogenase/reductase (SDR family) member 3 2.18469
IFT54 intraflagellar transport 54 2.18375
PCDHGA11 protocadherin gamma subfamily A, 11 2.17824
GNRH1 gonadotropin-releasing hormone 1 (luteinizing-releasing hormone) 2.17231
ZNF471 zinc finger protein 471 2.168
AMOT angiomotin 2.16669
CNTN5 contactin 5 2.166
MLF2 myeloid leukemia factor 2 2.16337
SPACA1 sperm acrosome associated 1 2.1564
FOXD2 forkhead box D2 2.15627
RAVER2 ribonucleoprotein, PTB-binding 2 2.14865
PURG purine-rich element binding protein G 2.1472
ZNF674 zinc finger protein 674 2.14378
OR2W1 olfactory receptor, family 2, subfamily W, member 1 2.13956
FAM131B family with sequence similarity 131, member B 2.13503
KIRREL1 kirre like nephrin family adhesion molecule 1 2.13347
TRIM49B tripartite motif containing 49B 2.133
ADRA1A adrenoceptor alpha 1A 2.1296
DGKE diacylglycerol kinase, epsilon 64kDa 2.1292
SPRYD7 SPRY domain containing 7 2.12741
MCF2L2 MCF.2 cell line derived transforming sequence-like 2 2.12518
BTC betacellulin 2.11995
PRAME preferentially expressed antigen in melanoma 2.11803
AP4E1 adaptor-related protein complex 4, epsilon 1 subunit 2.11268
PDE6C phosphodiesterase 6C, cGMP-specific, cone, alpha prime 2.11032
RAB31 RAB31, member RAS oncogene family 2.10834
STON1-GTF2A1L STON1-GTF2A1L readthrough 2.10674
RFPL1 ret finger protein-like 1 2.10359
GALR1 galanin receptor 1 2.09808
GHRH growth hormone releasing hormone 2.09384
FOXE3 forkhead box E3 2.09213
IFNAR1 interferon (alpha, beta and omega) receptor 1 2.08521
PPARA peroxisome proliferator-activated receptor alpha 2.08472
SMAGP small cell adhesion glycoprotein 2.0809
ZNF81 zinc finger protein 81 2.08058
IFNA5 interferon, alpha 5 2.07894
KNL1 kinetochore scaffold 1 2.07797
VAMP5 vesicle-associated membrane protein 5 2.07667
MTMR7 myotubularin related protein 7 2.07618
LMOD1 leiomodin 1 (smooth muscle) 2.07584
GPR18 G protein-coupled receptor 18 2.0719
NPVF neuropeptide VF precursor 2.07017
POU1F1 POU class 1 homeobox 1 2.06927
GLRA3 glycine receptor, alpha 3 2.06526
CPAMD8 C3 and PZP-like, alpha-2-macroglobulin domain containing 8 2.06242
LPA lipoprotein, Lp(a) 2.06139
CHRNB4 cholinergic receptor, nicotinic, beta 4 (neuronal) 2.05925
ELP5 elongator acetyltransferase complex subunit 5 2.05872
GNRHR gonadotropin-releasing hormone receptor 2.05196
DNAJC28 DnaJ (Hsp40) homolog, subfamily C, member 28 2.05134
IMPG1 interphotoreceptor matrix proteoglycan 1 2.05024
ZNF492 zinc finger protein 492 2.04908
MSH4 mutS homolog 4 2.04806
FCN2 ficolin (collagen/fibrinogen domain containing lectin) 2 2.04548
OR7E24 olfactory receptor, family 7, subfamily E, member 24 2.04089
TEX13A testis expressed 13A 2.03824
CNTNAP3B contactin associated protein-like 3B 2.03644
LAMB4 laminin, beta 4 2.03419
IL26 interleukin 26 2.03139
NCR3 natural cytotoxicity triggering receptor 3 2.02936
GCM2 glial cells missing homolog 2 (Drosophila) 2.02738
CRYGA crystallin, gamma A 2.02727
SLC6A16 solute carrier family 6, member 16 2.01979
ADAM18 ADAM metallopeptidase domain 18 2.01536
RRH retinal pigment epithelium-derived rhodopsin homolog 2.012

decreased expression

Symbol Name Standardized Value
UGDH UDP-glucose 6-dehydrogenase -5.1652
SLC35F2 solute carrier family 35, member F2 -5.04608
ZNF586 zinc finger protein 586 -4.98901
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -4.94069
CDC25B cell division cycle 25B -4.22675
CCNB2 cyclin B2 -4.04775
SNX11 sorting nexin 11 -3.67308
HMGCS1 3-hydroxy-3-methylglutaryl-CoA synthase 1 (soluble) -3.61613
TLR4 toll-like receptor 4 -3.43647
GLOD4 glyoxalase domain containing 4 -3.27037
LOC124907782 dual specificity protein phosphatase 22 -3.16963
DNTTIP2 deoxynucleotidyltransferase, terminal, interacting protein 2 -3.13329
PARP2 poly (ADP-ribose) polymerase 2 -3.12189
HAT1 histone acetyltransferase 1 -3.08663
PIK3R4 phosphoinositide-3-kinase, regulatory subunit 4 -2.84677
MAPK13 mitogen-activated protein kinase 13 -2.63156
SLC25A13 solute carrier family 25 (aspartate/glutamate carrier), member 13 -2.59788
HMG20B high mobility group 20B -2.55864
NLRP4 NLR family, pyrin domain containing 4 -2.40056
ITFG1 integrin alpha FG-GAP repeat containing 1 -2.39542
NAV3 neuron navigator 3 -2.21788
LMO4 LIM domain only 4 -2.20308
TBC1D10C TBC1 domain family, member 10C -2.20139
SNF8 SNF8, ESCRT-II complex subunit -2.2011
TP53BP2 tumor protein p53 binding protein 2 -2.17106
RBM14-RBM4 RBM14-RBM4 readthrough -2.12896
ALG9 ALG9, alpha-1,2-mannosyltransferase -2.11653
CETN3 centrin, EF-hand protein, 3 -2.10266
FUT8 fucosyltransferase 8 (alpha (1,6) fucosyltransferase) -2.07219
WDR7 WD repeat domain 7 -2.06848
DHX29 DEAH (Asp-Glu-Ala-His) box polypeptide 29 -2.03722