CRCGN014_HEPG2_3H:K16 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description retrorsine 19.35 um perturbation at 3 h in HEPG2 (Carcinogenome)
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Genes

72 genes differentially expressed following the CRCGN014_HEPG2_3H:K16 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
P4HTM prolyl 4-hydroxylase, transmembrane (endoplasmic reticulum) 6.1968
GATA3 GATA binding protein 3 5.69518
JADE2 jade family PHD finger 2 4.40887
C2CD2 C2 calcium-dependent domain containing 2 4.17791
CSK c-src tyrosine kinase 3.87355
IKZF1 IKAROS family zinc finger 1 (Ikaros) 3.61053
DRAP1 DR1-associated protein 1 (negative cofactor 2 alpha) 3.36907
E2F2 E2F transcription factor 2 3.34179
KIT v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog 3.31492
CRTAP cartilage associated protein 3.30684
RSF1 remodeling and spacing factor 1 3.21192
KLHL21 kelch-like family member 21 3.19366
BAX BCL2-associated X protein 3.18121
PPARG peroxisome proliferator-activated receptor gamma 3.16493
ABHD6 abhydrolase domain containing 6 3.05867
NR3C1 nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor) 3.01943
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5 3.01512
EMSY EMSY transcriptional repressor, BRCA2 interacting 2.9531
ADRB2 adrenoceptor beta 2, surface 2.9135
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5 2.85673
BACE2 beta-site APP-cleaving enzyme 2 2.71145
ALOX15 arachidonate 15-lipoxygenase 2.70443
DIPK1A divergent protein kinase domain 1A 2.67296
LOC122526780 uncharacterized LOC122526780 2.61118
STIMATE STIM activating enhancer 2.60586
STAP2 signal transducing adaptor family member 2 2.58768
SMARCD2 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 2 2.40815
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11 2.40796
PEX11A peroxisomal biogenesis factor 11 alpha 2.37979
IL12A interleukin 12A 2.35873
TFF1 trefoil factor 1 2.26886
ANO1 anoctamin 1, calcium activated chloride channel 2.24468
RPL39L ribosomal protein L39-like 2.19538
EGF epidermal growth factor 2.14599
STEAP1 six transmembrane epithelial antigen of the prostate 1 2.13711
GNAI2 guanine nucleotide binding protein (G protein), alpha inhibiting activity polypeptide 2 2.13305
RASSF1 Ras association (RalGDS/AF-6) domain family member 1 2.10319
GAN gigaxonin 2.07706
PGAM4 phosphoglycerate mutase family member 4 2.0692
SERPINE1 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 1 2.0686
LOXL1 lysyl oxidase-like 1 2.04605
HOXA10 homeobox A10 2.01996
SNAP25 synaptosomal-associated protein, 25kDa 2.01083

decreased expression

Symbol Name Standardized Value
CCNB2 cyclin B2 -10.0
OXA1L oxidase (cytochrome c) assembly 1-like -5.10842
CNDP2 CNDP dipeptidase 2 (metallopeptidase M20 family) -3.86636
DNAJA3 DnaJ (Hsp40) homolog, subfamily A, member 3 -3.80406
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma -3.68521
SLC7A5 solute carrier family 7 (amino acid transporter light chain, L system), member 5 -3.68494
LDHD lactate dehydrogenase D -3.52188
LSM5 LSM5 homolog, U6 small nuclear RNA associated (S. cerevisiae) -3.34584
PPP2R5E protein phosphatase 2, regulatory subunit B', epsilon isoform -3.32522
TARBP1 TAR (HIV-1) RNA binding protein 1 -3.27552
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2 -3.26544
ARID5B AT rich interactive domain 5B (MRF1-like) -3.06748
IARS2 isoleucyl-tRNA synthetase 2, mitochondrial -2.79874
CDC20 cell division cycle 20 -2.76232
SUPV3L1 suppressor of var1, 3-like 1 (S. cerevisiae) -2.58651
PCNA proliferating cell nuclear antigen -2.52885
WDR91 WD repeat domain 91 -2.45735
NRIP1 nuclear receptor interacting protein 1 -2.43415
TXNDC9 thioredoxin domain containing 9 -2.40119
YTHDF1 YTH N(6)-methyladenosine RNA binding protein 1 -2.38
LMO3 LIM domain only 3 (rhombotin-like 2) -2.31209
RAI14 retinoic acid induced 14 -2.20322
NHEJ1 nonhomologous end-joining factor 1 -2.19161
ZNF586 zinc finger protein 586 -2.17755
NGRN neugrin, neurite outgrowth associated -2.14888
TCFL5 transcription factor-like 5 (basic helix-loop-helix) -2.07326
ETHE1 ethylmalonic encephalopathy 1 -2.05613
HTRA1 HtrA serine peptidase 1 -2.03436
TDP2 tyrosyl-DNA phosphodiesterase 2 -2.01626