CRCGN015_MCF10A.WT.HP_24H:M19 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description mestranol 97.87 um perturbation at 24 h in MCF10A.WT.HP (Carcinogenome)
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Genes

271 genes differentially expressed following the CRCGN015_MCF10A.WT.HP_24H:M19 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
FKBP14 FK506 binding protein 14, 22 kDa 4.97201
METRN meteorin, glial cell differentiation regulator 4.9538
BZW2 basic leucine zipper and W2 domains 2 4.80248
CXCR4 chemokine (C-X-C motif) receptor 4 4.7946
HBA1 hemoglobin, alpha 1 4.73175
GATA3 GATA binding protein 3 3.98734
EMSY EMSY transcriptional repressor, BRCA2 interacting 3.57277
GRB10 growth factor receptor-bound protein 10 3.52871
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2 3.32927
AXIN1 axin 1 3.0709
SUV39H2 suppressor of variegation 3-9 homolog 2 (Drosophila) 3.05741
WIF1 WNT inhibitory factor 1 2.99983
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1 2.97315
TAF13 TAF13 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 18kDa 2.85431
FZD7 frizzled class receptor 7 2.84265
TNFSF15 tumor necrosis factor (ligand) superfamily, member 15 2.73476
CDK14 cyclin-dependent kinase 14 2.65555
GPRC5B G protein-coupled receptor, class C, group 5, member B 2.65525
CACNA2D3 calcium channel, voltage-dependent, alpha 2/delta subunit 3 2.63271
FAM204A family with sequence similarity 204, member A 2.62708
NDUFAF7 NADH dehydrogenase (ubiquinone) complex I, assembly factor 7 2.60862
DHDDS dehydrodolichyl diphosphate synthase 2.60222
TNMD tenomodulin 2.58867
CDH10 cadherin 10, type 2 (T2-cadherin) 2.58529
ATAD5 ATPase family, AAA domain containing 5 2.54609
CTAGE1 cutaneous T-cell lymphoma-associated antigen 1 2.53023
FGD6 FYVE, RhoGEF and PH domain containing 6 2.51977
DMTF1 cyclin D binding myb-like transcription factor 1 2.51949
PPEF2 protein phosphatase, EF-hand calcium binding domain 2 2.5076
PPP1R1A protein phosphatase 1, regulatory (inhibitor) subunit 1A 2.50747
CDC37L1 cell division cycle 37-like 1 2.50129
SCAI suppressor of cancer cell invasion 2.49138
PPP4R4 protein phosphatase 4, regulatory subunit 4 2.48191
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase 2.46266
SEMA3E sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3E 2.45566
LCOR ligand dependent nuclear receptor corepressor 2.45424
CRISP1 cysteine-rich secretory protein 1 2.44048
VEZT vezatin, adherens junctions transmembrane protein 2.44043
SYF2 SYF2 pre-mRNA-splicing factor 2.4357
ZNF460 zinc finger protein 460 2.43236
LIN28A lin-28 homolog A (C. elegans) 2.43081
TMOD2 tropomodulin 2 (neuronal) 2.4174
KCNJ3 potassium channel, inwardly rectifying subfamily J, member 3 2.40884
GJD3 gap junction protein, delta 3, 31.9kDa 2.40692
ANKRD10 ankyrin repeat domain 10 2.40556
RSF1 remodeling and spacing factor 1 2.40442
LRRTM4 leucine rich repeat transmembrane neuronal 4 2.40338
RAD54L RAD54-like (S. cerevisiae) 2.40262
STON1-GTF2A1L STON1-GTF2A1L readthrough 2.38687
ERC1 ELKS/RAB6-interacting/CAST family member 1 2.38233
CNTN6 contactin 6 2.37784
CLSTN2 calsyntenin 2 2.37376
ERBB4 erb-b2 receptor tyrosine kinase 4 2.3676
EDDM3A epididymal protein 3A 2.36695
CD1D CD1d molecule 2.34717
KCNV2 potassium channel, voltage gated modifier subfamily V, member 2 2.34607
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1 2.34417
GP6 glycoprotein VI (platelet) 2.34008
TMEM19 transmembrane protein 19 2.33613
RASSF9 Ras association (RalGDS/AF-6) domain family (N-terminal) member 9 2.3259
CEP152 centrosomal protein 152kDa 2.31668
THAP9 THAP domain containing 9 2.30811
SNRPB2 small nuclear ribonucleoprotein polypeptide B 2.3048
PIWIL1 piwi-like RNA-mediated gene silencing 1 2.30474
DGKE diacylglycerol kinase, epsilon 64kDa 2.29937
ZNF329 zinc finger protein 329 2.29855
MCF2L2 MCF.2 cell line derived transforming sequence-like 2 2.296
WDHD1 WD repeat and HMG-box DNA binding protein 1 2.29412
S1PR2 sphingosine-1-phosphate receptor 2 2.29356
DIAPH3 diaphanous-related formin 3 2.27829
HTR2A 5-hydroxytryptamine (serotonin) receptor 2A, G protein-coupled 2.27442
ADAM7 ADAM metallopeptidase domain 7 2.27383
CNKSR2 connector enhancer of kinase suppressor of Ras 2 2.26909
TAS2R8 taste receptor, type 2, member 8 2.26796
NPY1R neuropeptide Y receptor Y1 2.24904
MCPH1 microcephalin 1 2.24649
AOC2 amine oxidase, copper containing 2 (retina-specific) 2.24469
PCDHGA8 protocadherin gamma subfamily A, 8 2.24076
SLC25A31 solute carrier family 25 (mitochondrial carrier; adenine nucleotide translocator), member 31 2.23654
SIM1 single-minded family bHLH transcription factor 1 2.22617
LOC100996750 keratin-associated protein 4-7 2.22386
CATSPERG catsper channel auxiliary subunit gamma 2.22141
CFAP43 cilia and flagella associated protein 43 2.21564
NMBR neuromedin B receptor 2.21434
CDH20 cadherin 20, type 2 2.21425
CRYBA1 crystallin, beta A1 2.21402
CCDC144A coiled-coil domain containing 144A 2.21305
PKD2L2 polycystic kidney disease 2-like 2 2.21084
OMD osteomodulin 2.20593
TRMT9B tRNA methyltransferase 9B (putative) 2.20557
LRP1B low density lipoprotein receptor-related protein 1B 2.20225
FRS3 fibroblast growth factor receptor substrate 3 2.19785
IFNA5 interferon, alpha 5 2.19778
AUNIP aurora kinase A and ninein interacting protein 2.19672
ZNF37A zinc finger protein 37A 2.19452
SLCO5A1 solute carrier organic anion transporter family, member 5A1 2.19377
ZNF391 zinc finger protein 391 2.19309
KCND2 potassium channel, voltage gated Shal related subfamily D, member 2 2.19163
SCHIP1 schwannomin interacting protein 1 2.1903
JADE3 jade family PHD finger 3 2.18612
SERPINB10 serpin peptidase inhibitor, clade B (ovalbumin), member 10 2.18379
OLR1 oxidized low density lipoprotein (lectin-like) receptor 1 2.18036
LDHAL6B lactate dehydrogenase A-like 6B 2.17928
DCC DCC netrin 1 receptor 2.17683
NSUN7 NOP2/Sun domain family, member 7 2.17347
SNRK SNF related kinase 2.17048
NPY5R neuropeptide Y receptor Y5 2.16928
NOL4 nucleolar protein 4 2.16801
CPA1 carboxypeptidase A1 (pancreatic) 2.16568
PURG purine-rich element binding protein G 2.16536
ADGB androglobin 2.16493
EDDM3B epididymal protein 3B 2.16279
KIAA0319 KIAA0319 2.1626
KRT35 keratin 35, type I 2.1601
RASAL2 RAS protein activator like 2 2.15605
SPINT4 serine peptidase inhibitor, Kunitz type 4 2.1524
SLC35F5 solute carrier family 35, member F5 2.15156
IL4 interleukin 4 2.15052
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase 2.14377
GLRA3 glycine receptor, alpha 3 2.14338
ARSJ arylsulfatase family, member J 2.1374
KMT2D lysine (K)-specific methyltransferase 2D 2.13627
RAG1 recombination activating gene 1 2.13515
SPATA31C1 SPATA31 subfamily C, member 1 2.1351
SPATA6L spermatogenesis associated 6-like 2.13211
ANKRD34C ankyrin repeat domain 34C 2.13047
CENPQ centromere protein Q 2.12815
ZNF780B zinc finger protein 780B 2.12716
ZNF225 zinc finger protein 225 2.12538
PRRG2 proline rich Gla (G-carboxyglutamic acid) 2 2.12452
OR2J3 olfactory receptor, family 2, subfamily J, member 3 2.12212
UTF1 undifferentiated embryonic cell transcription factor 1 2.11938
ITGB6 integrin, beta 6 2.11891
LRRC1 leucine rich repeat containing 1 2.1177
ZNF749 zinc finger protein 749 2.11621
ACOXL acyl-CoA oxidase-like 2.11455
HID1 HID1 domain containing 2.11401
ARHGDIB Rho GDP dissociation inhibitor (GDI) beta 2.11093
INHBE inhibin, beta E 2.10925
ZNF549 zinc finger protein 549 2.10701
MBTD1 mbt domain containing 1 2.10677
GRM5 glutamate receptor, metabotropic 5 2.10557
CCDC30 coiled-coil domain containing 30 2.1046
SPO11 SPO11 meiotic protein covalently bound to DSB 2.10384
BTC betacellulin 2.10344
ATP1B4 ATPase, Na+/K+ transporting, beta 4 polypeptide 2.10162
CCDC82 coiled-coil domain containing 82 2.10111
HTN3 histatin 3 2.0936
SCN11A sodium channel, voltage gated, type XI alpha subunit 2.09162
KIF24 kinesin family member 24 2.09019
PARK7 parkinson protein 7 2.09011
PCDH11X protocadherin 11 X-linked 2.0894
MTMR7 myotubularin related protein 7 2.08822
MMP25 matrix metallopeptidase 25 2.08449
RBMXL2 RNA binding motif protein, X-linked-like 2 2.08439
GTPBP10 GTP-binding protein 10 (putative) 2.08432
IL37 interleukin 37 2.08411
GNRH1 gonadotropin-releasing hormone 1 (luteinizing-releasing hormone) 2.08178
ZNF814 zinc finger protein 814 2.07863
KCNJ13 potassium channel, inwardly rectifying subfamily J, member 13 2.07285
OPRPN opiorphin prepropeptide 2.07051
MAGEB4 melanoma antigen family B4 2.07017
RYR2 ryanodine receptor 2 (cardiac) 2.06773
TEX12 testis expressed 12 2.06755
NPHP1 nephronophthisis 1 (juvenile) 2.06733
BLTP3B bridge-like lipid transfer protein family member 3B 2.06659
ZNF492 zinc finger protein 492 2.06654
TSBP1 testis expressed basic protein 1 2.06571
KERA keratocan 2.06459
ELSPBP1 epididymal sperm binding protein 1 2.06359
MMRN2 multimerin 2 2.06054
AGBL3 ATP/GTP binding protein-like 3 2.06006
XPNPEP2 X-prolyl aminopeptidase (aminopeptidase P) 2, membrane-bound 2.05923
MTRF1L mitochondrial translational release factor 1-like 2.05747
EPPK1 epiplakin 1 2.05627
GRIN2B glutamate receptor, ionotropic, N-methyl D-aspartate 2B 2.05594
LRAT lecithin retinol acyltransferase (phosphatidylcholine--retinol O-acyltransferase) 2.05212
GNAT2 guanine nucleotide binding protein (G protein), alpha transducing activity polypeptide 2 2.05211
KIT v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog 2.05169
HTN1 histatin 1 2.05007
MAGEL2 melanoma antigen family L2 2.04906
GCM2 glial cells missing homolog 2 (Drosophila) 2.04869
CHRM2 cholinergic receptor, muscarinic 2 2.04746
PKN1 protein kinase N1 2.04664
SLC5A4 solute carrier family 5 (glucose activated ion channel), member 4 2.04502
TLR1 toll-like receptor 1 2.04476
SCARF1 scavenger receptor class F, member 1 2.04284
ZFP69B ZFP69 zinc finger protein B 2.04195
LIAS lipoic acid synthetase 2.03946
LGALS12 lectin, galactoside-binding, soluble, 12 2.03797
ZNF426 zinc finger protein 426 2.03719
CCDC121 coiled-coil domain containing 121 2.03688
CRISP2 cysteine-rich secretory protein 2 2.03489
EGR4 early growth response 4 2.03471
PCDHGB5 protocadherin gamma subfamily B, 5 2.03399
ATP10D ATPase, class V, type 10D 2.03228
QPCTL glutaminyl-peptide cyclotransferase-like 2.03134
SEPTIN10 septin 10 2.03111
OGFRL1 opioid growth factor receptor-like 1 2.03079
TLR6 toll-like receptor 6 2.03038
LGR4 leucine-rich repeat containing G protein-coupled receptor 4 2.02874
UVRAG UV radiation resistance associated 2.02836
KNL1 kinetochore scaffold 1 2.02736
FAM135A family with sequence similarity 135, member A 2.02551
KLF8 Kruppel-like factor 8 2.02537
PLCL1 phospholipase C-like 1 2.02503
SOX11 SRY (sex determining region Y)-box 11 2.02497
KLHL11 kelch-like family member 11 2.02378
GPR85 G protein-coupled receptor 85 2.02377
SPOCK3 sparc/osteonectin, cwcv and kazal-like domains proteoglycan (testican) 3 2.02342
NDST3 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 3 2.02307
CHRNB4 cholinergic receptor, nicotinic, beta 4 (neuronal) 2.02126
CBX2 chromobox homolog 2 2.02111
KCNJ9 potassium channel, inwardly rectifying subfamily J, member 9 2.02104
CFAP68 cilia and flagella associated protein 68 2.01917
CEP97 centrosomal protein 97kDa 2.01866
DIXDC1 DIX domain containing 1 2.01854
FAM13C family with sequence similarity 13, member C 2.01802
PDPN podoplanin 2.01658
SMPDL3B sphingomyelin phosphodiesterase, acid-like 3B 2.01535
CYLC2 cylicin, basic protein of sperm head cytoskeleton 2 2.01508
GABRA4 gamma-aminobutyric acid (GABA) A receptor, alpha 4 2.01484
NANOG Nanog homeobox 2.0144
ELOA2 elongin A2 2.01378
CDH8 cadherin 8, type 2 2.0136
MTUS2 microtubule associated tumor suppressor candidate 2 2.01269
LOC100996709 ADP-ribosylation factor-like protein 17 2.01252
DNAJC5 DnaJ (Hsp40) homolog, subfamily C, member 5 2.01184
SMR3B submaxillary gland androgen regulated protein 3B 2.01137
MKNK1 MAP kinase interacting serine/threonine kinase 1 2.01107
OR1D4 olfactory receptor, family 1, subfamily D, member 4 (gene/pseudogene) 2.00948
GAD2 glutamate decarboxylase 2 (pancreatic islets and brain, 65kDa) 2.00816
ZNF81 zinc finger protein 81 2.00783
SMR3A submaxillary gland androgen regulated protein 3A 2.00715
HSD3B2 hydroxy-delta-5-steroid dehydrogenase, 3 beta- and steroid delta-isomerase 2 2.00533
GSG1 germ cell associated 1 2.00354
GABRB1 gamma-aminobutyric acid (GABA) A receptor, beta 1 2.00071

decreased expression

Symbol Name Standardized Value
CCNB1 cyclin B1 -9.54884
TARBP1 TAR (HIV-1) RNA binding protein 1 -5.49533
CCDC86 coiled-coil domain containing 86 -5.35807
BASP1 brain abundant, membrane attached signal protein 1 -4.91015
PPP2R5E protein phosphatase 2, regulatory subunit B', epsilon isoform -4.552
GDF15 growth differentiation factor 15 -4.04338
LOC112694756 uncharaterized LOC112694756 -3.78789
CD320 CD320 molecule -3.22058
PTCD1 pentatricopeptide repeat domain 1 -3.12917
ALDOC aldolase C, fructose-bisphosphate -3.09808
PCCB propionyl CoA carboxylase, beta polypeptide -2.58435
CPSF4 cleavage and polyadenylation specific factor 4, 30kDa -2.55717
DROSHA drosha, ribonuclease type III -2.43714
CCL21 chemokine (C-C motif) ligand 21 -2.40253
HTRA1 HtrA serine peptidase 1 -2.36801
UBE2S ubiquitin-conjugating enzyme E2S -2.33766
RAB1B RAB1B, member RAS oncogene family -2.32151
KMT5B lysine methyltransferase 5B -2.31851
TMEM260 transmembrane protein 260 -2.31599
FABP5 fatty acid binding protein 5 (psoriasis-associated) -2.30505
HERC6 HECT and RLD domain containing E3 ubiquitin protein ligase family member 6 -2.29771
IRF7 interferon regulatory factor 7 -2.1685
EIF4EBP3 eukaryotic translation initiation factor 4E binding protein 3 -2.16797
PTTG1 pituitary tumor-transforming 1 -2.12816
RABGGTA Rab geranylgeranyltransferase, alpha subunit -2.11929
DCPS decapping enzyme, scavenger -2.1166
TSPAN3 tetraspanin 3 -2.10819
CREG1 cellular repressor of E1A-stimulated genes 1 -2.10617
PFN2 profilin 2 -2.06699
TXNDC5 thioredoxin domain containing 5 (endoplasmic reticulum) -2.05667
CASC3 cancer susceptibility candidate 3 -2.05496
MYLIP myosin regulatory light chain interacting protein -2.02507
SCYL3 SCY1-like 3 (S. cerevisiae) -2.01764
CLTC clathrin, heavy chain (Hc) -2.00104