CRCGN017_MCF10A.TP53.M_24H:P06 Gene Set

Dataset Carcinogenome Chemical Perturbation Carcinogenicity Signatures
Category transcriptomics
Type small molecule perturbation
Description reserpine 11.25 um perturbation at 24 h in MCF10A.TP53.M (Carcinogenome)
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Genes

119 genes differentially expressed following the CRCGN017_MCF10A.TP53.M_24H:P06 small molecule perturbation from the Carcinogenome Chemical Perturbation Carcinogenicity Signatures dataset.

increased expression

Symbol Name Standardized Value
CASP2 caspase 2, apoptosis-related cysteine peptidase 6.67781
STK10 serine/threonine kinase 10 4.27878
MMP2 matrix metallopeptidase 2 3.79541
SSR3 signal sequence receptor, gamma (translocon-associated protein gamma) 3.78765
EIF2S3 eukaryotic translation initiation factor 2, subunit 3 gamma, 52kDa 3.60313
ZNF652 zinc finger protein 652 3.28687
MB myoglobin 3.17293
SPDEF SAM pointed domain containing ETS transcription factor 3.14109
CXCR4 chemokine (C-X-C motif) receptor 4 3.13824
MTA2 metastasis associated 1 family, member 2 3.12113
MPC2 mitochondrial pyruvate carrier 2 3.12038
ADGRE5 adhesion G protein-coupled receptor E5 3.10954
MDM4 MDM4, p53 regulator 3.05836
ABCB6 ATP-binding cassette, sub-family B (MDR/TAP), member 6 (Langereis blood group) 2.94592
COMP cartilage oligomeric matrix protein 2.89976
LAP3 leucine aminopeptidase 3 2.87365
CHN1 chimerin 1 2.85282
STRN3 striatin, calmodulin binding protein 3 2.73173
EGLN3 egl-9 family hypoxia-inducible factor 3 2.70224
PALMD palmdelphin 2.66317
RNF125 ring finger protein 125, E3 ubiquitin protein ligase 2.65245
HNRNPL heterogeneous nuclear ribonucleoprotein L 2.64845
RBP4 retinol binding protein 4, plasma 2.64318
ADO 2-aminoethanethiol (cysteamine) dioxygenase 2.63041
HMGCR 3-hydroxy-3-methylglutaryl-CoA reductase 2.60825
MOSPD1 motile sperm domain containing 1 2.58315
RAB21 RAB21, member RAS oncogene family 2.56694
LDAF1 lipid droplet assembly factor 1 2.54715
RBBP5 retinoblastoma binding protein 5 2.5153
KLHL9 kelch-like family member 9 2.50448
REL v-rel avian reticuloendotheliosis viral oncogene homolog 2.46265
NIT1 nitrilase 1 2.44722
MYBPC2 myosin binding protein C, fast type 2.4338
CERK ceramide kinase 2.41441
CEPT1 choline/ethanolamine phosphotransferase 1 2.38826
ADGRG1 adhesion G protein-coupled receptor G1 2.37891
KLHL21 kelch-like family member 21 2.37824
ITGB1BP2 integrin beta 1 binding protein (melusin) 2 2.3615
IFI6 interferon, alpha-inducible protein 6 2.34948
PLEKHA2 pleckstrin homology domain containing, family A (phosphoinositide binding specific) member 2 2.34689
HSPB3 heat shock 27kDa protein 3 2.30435
HNRNPH1 heterogeneous nuclear ribonucleoprotein H1 (H) 2.29868
GNL3L guanine nucleotide binding protein-like 3 (nucleolar)-like 2.29493
TPD52L2 tumor protein D52-like 2 2.26894
MTCL1 microtubule crosslinking factor 1 2.25482
MFAP5 microfibrillar associated protein 5 2.24346
PTPRS protein tyrosine phosphatase, receptor type, S 2.23198
PRPF39 pre-mRNA processing factor 39 2.19581
KLRC4 killer cell lectin-like receptor subfamily C, member 4 2.19187
RGCC regulator of cell cycle 2.18471
ZNF587B zinc finger protein 587B 2.17873
NUTF2 nuclear transport factor 2 2.17
NOPCHAP1 NOP protein chaperone 1 2.16205
PLN phospholamban 2.15996
EIF5AL1 eukaryotic translation initiation factor 5A-like 1 2.15531
TMPRSS3 transmembrane protease, serine 3 2.15362
THRAP3 thyroid hormone receptor associated protein 3 2.15311
DNAJA2 DnaJ (Hsp40) homolog, subfamily A, member 2 2.14953
DNAJC17 DnaJ (Hsp40) homolog, subfamily C, member 17 2.14394
GNLY granulysin 2.12385
SLC27A6 solute carrier family 27 (fatty acid transporter), member 6 2.12306
CHST4 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 4 2.10213
NCR3 natural cytotoxicity triggering receptor 3 2.09291
SLC10A2 solute carrier family 10 (sodium/bile acid cotransporter), member 2 2.07764
TESK1 testis-specific kinase 1 2.07247
ANXA4 annexin A4 2.06308
STAP1 signal transducing adaptor family member 1 2.06209
KIR3DL1 killer cell immunoglobulin-like receptor, three domains, long cytoplasmic tail, 1 2.04798
WDR91 WD repeat domain 91 2.04695
ZNF701 zinc finger protein 701 2.04591
TNNI2 troponin I type 2 (skeletal, fast) 2.04402
ANGPTL2 angiopoietin-like 2 2.04365
ZNF224 zinc finger protein 224 2.04241
HSPA6 heat shock 70kDa protein 6 (HSP70B') 2.04086
ZNF221 zinc finger protein 221 2.0366
ALDH1B1 aldehyde dehydrogenase 1 family, member B1 2.02881
FRAS1 Fraser extracellular matrix complex subunit 1 2.02555
PLA2R1 phospholipase A2 receptor 1, 180kDa 2.02202
PGPEP1 pyroglutamyl-peptidase I 2.0212
ZNF692 zinc finger protein 692 2.02078
U2AF2 U2 small nuclear RNA auxiliary factor 2 2.01511
PDGFRB platelet-derived growth factor receptor, beta polypeptide 2.0118

decreased expression

Symbol Name Standardized Value
BASP1 brain abundant, membrane attached signal protein 1 -5.47771
KIF14 kinesin family member 14 -4.63203
CDK4 cyclin-dependent kinase 4 -4.34734
COTL1 coactosin-like F-actin binding protein 1 -3.346
CAB39 calcium binding protein 39 -3.30735
TM9SF2 transmembrane 9 superfamily member 2 -3.11299
EBNA1BP2 EBNA1 binding protein 2 -2.92021
TRAPPC3 trafficking protein particle complex 3 -2.79207
AXIN1 axin 1 -2.72786
UBE2C ubiquitin-conjugating enzyme E2C -2.6992
PSMC4 proteasome (prosome, macropain) 26S subunit, ATPase, 4 -2.48248
NME2 NME/NM23 nucleoside diphosphate kinase 2 -2.48207
ERAL1 Era-like 12S mitochondrial rRNA chaperone 1 -2.47306
PCCB propionyl CoA carboxylase, beta polypeptide -2.43061
NIT2 nitrilase family, member 2 -2.42967
HMG20B high mobility group 20B -2.38512
MSMO1 methylsterol monooxygenase 1 -2.37213
RAD51C RAD51 paralog C -2.31391
PSRC1 proline/serine-rich coiled-coil 1 -2.28021
GRWD1 glutamate-rich WD repeat containing 1 -2.27805
NME4 NME/NM23 nucleoside diphosphate kinase 4 -2.27762
EIF2B3 eukaryotic translation initiation factor 2B, subunit 3 gamma, 58kDa -2.27253
NDUFS5 NADH dehydrogenase (ubiquinone) Fe-S protein 5, 15kDa (NADH-coenzyme Q reductase) -2.25743
POLR3K polymerase (RNA) III (DNA directed) polypeptide K, 12.3 kDa -2.19172
ELAC2 elaC ribonuclease Z 2 -2.18495
GNG5 guanine nucleotide binding protein (G protein), gamma 5 -2.16939
EXOSC9 exosome component 9 -2.16764
SORBS3 sorbin and SH3 domain containing 3 -2.1312
UQCRH ubiquinol-cytochrome c reductase hinge protein -2.11262
TOMM34 translocase of outer mitochondrial membrane 34 -2.07971
PSMG1 proteasome (prosome, macropain) assembly chaperone 1 -2.06872
RPN1 ribophorin I -2.06702
SUPT5H suppressor of Ty 5 homolog (S. cerevisiae) -2.06194
MRPL18 mitochondrial ribosomal protein L18 -2.05343
SNRNP25 small nuclear ribonucleoprotein 25kDa (U11/U12) -2.02018
ATP5PD ATP synthase peripheral stalk subunit d -2.015
FNDC4 fibronectin type III domain containing 4 -2.00992