Cilostazol_LS 180 Gene Set

Dataset Tahoe Therapeutics Tahoe 100M Perturbation Atlas
Category transcriptomics
Type cell type
Description Cilostazol perturbation in LS 180 cell line (Tahoe Therapeutics)
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Genes

200 genes differentially expressed following the Cilostazol_LS 180 drug perturbation from the Tahoe Therapeutics Tahoe 100M Perturbation Atlas dataset.

increased expression

Symbol Name Standardized Value
PTMA prothymosin, alpha 0.178505
VEGFA vascular endothelial growth factor A 0.164051
CEMIP cell migration inducing protein, hyaluronan binding 0.104762
ONECUT3 one cut homeobox 3 0.100753
TPT1 tumor protein, translationally-controlled 1 0.0959773
FAM13A family with sequence similarity 13, member A 0.0781194
TNFRSF10B tumor necrosis factor receptor superfamily, member 10b 0.0722228
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase 0.0682531
ANKRD11 ankyrin repeat domain 11 0.0675253
TNS4 tensin 4 0.0623633
EPCAM epithelial cell adhesion molecule 0.0617917
PRRC2C proline-rich coiled-coil 2C 0.0601609
RBM39 RNA binding motif protein 39 0.057523
MYH9 myosin, heavy chain 9, non-muscle 0.0572008
PPP2R2A protein phosphatase 2, regulatory subunit B, alpha 0.0550712
EEF1A1 eukaryotic translation elongation factor 1 alpha 1 0.052329
H1-0 H1.0 linker histone 0.0519441
RNF43 ring finger protein 43 0.0513983
EREG epiregulin 0.0487204
KRT8 keratin 8, type II 0.0468684
SREBF2 sterol regulatory element binding transcription factor 2 0.0463924
ACTN4 actinin, alpha 4 0.0460857
NDRG1 N-myc downstream regulated 1 0.0457335
FLNB filamin B, beta 0.0451935
KRT18 keratin 18, type I 0.0451688
HNRNPH1 heterogeneous nuclear ribonucleoprotein H1 (H) 0.0443654
KDM3A lysine (K)-specific demethylase 3A 0.0436121
ANXA2 annexin A2 0.0426231
SYNCRIP synaptotagmin binding, cytoplasmic RNA interacting protein 0.042597
OGA O-GlcNAcase 0.0415695
PRSS3 protease, serine, 3 0.0403266
ITGB1 integrin, beta 1 (fibronectin receptor, beta polypeptide, antigen CD29 includes MDF2, MSK12) 0.0393996
PLAUR plasminogen activator, urokinase receptor 0.0385943
DSCAM Down syndrome cell adhesion molecule 0.0371973
SHB Src homology 2 domain containing adaptor protein B 0.0371496
LAMB3 laminin, beta 3 0.037119
CTBP2 C-terminal binding protein 2 0.0367652
ETS2 v-ets avian erythroblastosis virus E26 oncogene homolog 2 0.0365844
AFDN afadin, adherens junction formation factor 0.0359059
RNF145 ring finger protein 145 0.0358948
PNISR PNN-interacting serine/arginine-rich protein 0.0358116
NCOR1 nuclear receptor corepressor 1 0.0346042
ANXA11 annexin A11 0.033944
TMSB10 thymosin beta 10 0.0337632
EPHA2 EPH receptor A2 0.0337201
EEF2 eukaryotic translation elongation factor 2 0.0331163
SRRM2 serine/arginine repetitive matrix 2 0.0329428
CDH17 cadherin 17, LI cadherin (liver-intestine) 0.0327909
RHPN2 rhophilin, Rho GTPase binding protein 2 0.0325686
CTNND1 catenin (cadherin-associated protein), delta 1 0.0322545
LUC7L3 LUC7-like 3 (S. cerevisiae) 0.0315537
EIF4B eukaryotic translation initiation factor 4B 0.0308196
MINK1 misshapen-like kinase 1 0.0302866
HSD17B12 hydroxysteroid (17-beta) dehydrogenase 12 0.0301098
MATR3 matrin 3 0.0299116
SLC20A1 solute carrier family 20 (phosphate transporter), member 1 0.0294494
TAF1D TATA box binding protein (TBP)-associated factor, RNA polymerase I, D, 41kDa 0.0292571
AREG amphiregulin 0.0292549
ABHD17C abhydrolase domain containing 17C 0.0289327
ARHGEF10L Rho guanine nucleotide exchange factor (GEF) 10-like 0.0289192
EIF3A eukaryotic translation initiation factor 3, subunit A 0.0288595
PRAG1 PEAK1 related, kinase-activating pseudokinase 1 0.0286213
CALM2 calmodulin 2 (phosphorylase kinase, delta) 0.0283577
UBE2D3 ubiquitin-conjugating enzyme E2D 3 0.0282663
LAMC2 laminin, gamma 2 0.02805
HNRNPU heterogeneous nuclear ribonucleoprotein U (scaffold attachment factor A) 0.0280088
IER3 immediate early response 3 0.0279573
GAK cyclin G associated kinase 0.0279205
LOC102724023 ES1 protein homolog, mitochondrial 0.0278063
NKD1 naked cuticle homolog 1 (Drosophila) 0.0275838
EWSR1 EWS RNA-binding protein 1 0.0275147
NAMPT nicotinamide phosphoribosyltransferase 0.0272004
HNRNPAB heterogeneous nuclear ribonucleoprotein A/B 0.0270993
MYL12B myosin, light chain 12B, regulatory 0.0269792
B4GALT5 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 5 0.0269509
KCNK1 potassium channel, two pore domain subfamily K, member 1 0.0267814
RAD21 RAD21 homolog (S. pombe) 0.0266853
RPL34 ribosomal protein L34 0.0265842
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11 0.0259148
CTNNB1 catenin (cadherin-associated protein), beta 1, 88kDa 0.0258275
NECTIN2 nectin cell adhesion molecule 2 0.0258264
ZNF292 zinc finger protein 292 0.0258122
PPP6R3 protein phosphatase 6, regulatory subunit 3 0.0256894
TANC1 tetratricopeptide repeat, ankyrin repeat and coiled-coil containing 1 0.0256007
NUCKS1 nuclear casein kinase and cyclin-dependent kinase substrate 1 0.0255669
PLEC plectin 0.0255339
KLF6 Kruppel-like factor 6 0.0254969
MACF1 microtubule-actin crosslinking factor 1 0.0254676
PUM1 pumilio RNA-binding family member 1 0.0254477
ZFAND3 zinc finger, AN1-type domain 3 0.0250787
THOC2 THO complex 2 0.0249926
VDR vitamin D (1,25- dihydroxyvitamin D3) receptor 0.0249859
FOXJ3 forkhead box J3 0.0247442
SPRED2 sprouty-related, EVH1 domain containing 2 0.024661
EIF4H eukaryotic translation initiation factor 4H 0.0245899
GPHN gephyrin 0.0245023
DDX5 DEAD (Asp-Glu-Ala-Asp) box helicase 5 0.0243524
SERPINB1 serpin peptidase inhibitor, clade B (ovalbumin), member 1 0.0243448
RPS3 ribosomal protein S3 0.0239399
SCD stearoyl-CoA desaturase (delta-9-desaturase) 0.0239352

decreased expression

Symbol Name Standardized Value
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1 -0.221106
GAPDH glyceraldehyde-3-phosphate dehydrogenase -0.14355
PHLDA1 pleckstrin homology-like domain, family A, member 1 -0.0966528
SLC12A2 solute carrier family 12 (sodium/potassium/chloride transporter), member 2 -0.0863624
PTPRK protein tyrosine phosphatase, receptor type, K -0.0773458
PDIA3 protein disulfide isomerase family A, member 3 -0.066438
ZSWIM6 zinc finger, SWIM-type containing 6 -0.0636655
HSP90AA1 heat shock protein 90kDa alpha (cytosolic), class A member 1 -0.0627551
POTEF POTE ankyrin domain family, member F -0.0575828
MUC6 mucin 6, oligomeric mucus/gel-forming -0.0569949
EXT1 exostosin glycosyltransferase 1 -0.05452
MYO1E myosin IE -0.0535871
MUC5AC mucin 5AC, oligomeric mucus/gel-forming -0.0512009
MUC17 mucin 17, cell surface associated -0.0505431
HSP90AB1 heat shock protein 90kDa alpha (cytosolic), class B member 1 -0.0483592
MBNL1 muscleblind-like splicing regulator 1 -0.0476074
GMDS GDP-mannose 4,6-dehydratase -0.0472244
ALCAM activated leukocyte cell adhesion molecule -0.0452068
LOC112694756 uncharaterized LOC112694756 -0.0447007
EGFR epidermal growth factor receptor -0.0437007
RNF217 ring finger protein 217 -0.0436269
P4HB prolyl 4-hydroxylase, beta polypeptide -0.0426776
ATP1B1 ATPase, Na+/K+ transporting, beta 1 polypeptide -0.041029
HSPD1 heat shock 60kDa protein 1 (chaperonin) -0.040468
GREB1L growth regulation by estrogen in breast cancer-like -0.0399529
PSD3 pleckstrin and Sec7 domain containing 3 -0.0398065
PDE4D phosphodiesterase 4D, cAMP-specific -0.0396334
CCSER1 coiled-coil serine-rich protein 1 -0.0394261
MARCHF3 membrane associated ring-CH-type finger 3 -0.0392167
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) -0.038918
SLC38A2 solute carrier family 38, member 2 -0.0387114
NPSR1 neuropeptide S receptor 1 -0.0386113
TPM4 tropomyosin 4 -0.0383125
ASPH aspartate beta-hydroxylase -0.0372145
RPS6 ribosomal protein S6 -0.0371454
NAB1 NGFI-A binding protein 1 (EGR1 binding protein 1) -0.0371086
PTEN phosphatase and tensin homolog -0.0362078
CANX calnexin -0.0359912
PPP3CA protein phosphatase 3, catalytic subunit, alpha isozyme -0.0358013
GLS2 glutaminase 2 (liver, mitochondrial) -0.0354023
SLC5A3 solute carrier family 5 (sodium/myo-inositol cotransporter), member 3 -0.0346947
PARD3B par-3 family cell polarity regulator beta -0.0346181
PITPNC1 phosphatidylinositol transfer protein, cytoplasmic 1 -0.0344172
ZBTB20 zinc finger and BTB domain containing 20 -0.0335407
MRPS6 mitochondrial ribosomal protein S6 -0.0335328
MAML3 mastermind-like 3 (Drosophila) -0.0334866
SLC35F3 solute carrier family 35, member F3 -0.0330968
PKM pyruvate kinase, muscle -0.0329491
LMO7 LIM domain 7 -0.0328642
NALF1 NALCN channel auxiliary factor 1 -0.0327187
PABPC1 poly(A) binding protein, cytoplasmic 1 -0.03263
MT2A metallothionein 2A -0.0321996
PTPRB protein tyrosine phosphatase, receptor type, B -0.0321554
BCAT1 branched chain amino-acid transaminase 1, cytosolic -0.0320755
HMGA1 high mobility group AT-hook 1 -0.0318524
LGALS3 lectin, galactoside-binding, soluble, 3 -0.0317674
CLOCK clock circadian regulator -0.0290738
PATJ PATJ crumbs cell polarity complex component -0.0290615
GRIN2B glutamate receptor, ionotropic, N-methyl D-aspartate 2B -0.0290424
SLCO1B3-SLCO1B7 SLCO1B3-SLCO1B7 readthrough -0.0281732
MBNL2 muscleblind-like splicing regulator 2 -0.0279385
SVIL supervillin -0.0277919
ATP2B1 ATPase, Ca++ transporting, plasma membrane 1 -0.0274276
FTH1 ferritin, heavy polypeptide 1 -0.0273548
AGR2 anterior gradient 2 -0.0272582
RTN3 reticulon 3 -0.0266876
RPS25 ribosomal protein S25 -0.0264567
KTN1 kinectin 1 (kinesin receptor) -0.0264324
FBXO11 F-box protein 11 -0.0257515
LGR4 leucine-rich repeat containing G protein-coupled receptor 4 -0.0257179
RPS8 ribosomal protein S8 -0.0249928
GBE1 glucan (1,4-alpha-), branching enzyme 1 -0.0246937
AFF1 AF4/FMR2 family, member 1 -0.0246888
LDHA lactate dehydrogenase A -0.024577
UNC13B unc-13 homolog B (C. elegans) -0.0245258
RPL21 ribosomal protein L21 -0.0244726
RPS12 ribosomal protein S12 -0.0242932
INTS6 integrator complex subunit 6 -0.0238731
PRG2 proteoglycan 2, bone marrow (natural killer cell activator, eosinophil granule major basic protein) -0.0237093
PALLD palladin, cytoskeletal associated protein -0.0236885
ARHGAP6 Rho GTPase activating protein 6 -0.0236554
DSTN destrin (actin depolymerizing factor) -0.0236406
RPS23 ribosomal protein S23 -0.0231395
GOLGB1 golgin B1 -0.0229833
TRAM1 translocation associated membrane protein 1 -0.0226237
YBX1 Y box binding protein 1 -0.0222516
ARIH1 ariadne RBR E3 ubiquitin protein ligase 1 -0.022192
CATSPERB catsper channel auxiliary subunit beta -0.0221525
CRIM1 cysteine rich transmembrane BMP regulator 1 (chordin-like) -0.0220486
AKAP13 A kinase (PRKA) anchor protein 13 -0.0218003
MBD5 methyl-CpG binding domain protein 5 -0.0217339
RAPGEF2 Rap guanine nucleotide exchange factor (GEF) 2 -0.0215135
SPDYA speedy/RINGO cell cycle regulator family member A -0.0214056
EHBP1 EH domain binding protein 1 -0.0213767
MT1E metallothionein 1E -0.021316
HERC4 HECT and RLD domain containing E3 ubiquitin protein ligase 4 -0.0212907
NFAT5 nuclear factor of activated T-cells 5, tonicity-responsive -0.0211916
SPTAN1 spectrin, alpha, non-erythrocytic 1 -0.0211814
FOSB FBJ murine osteosarcoma viral oncogene homolog B -0.0209599
TTC3 tetratricopeptide repeat domain 3 -0.0206986