Clopidogrel_NCI-H2347 Gene Set

Dataset Tahoe Therapeutics Tahoe 100M Perturbation Atlas
Category transcriptomics
Type cell type
Description Clopidogrel perturbation in NCI-H2347 cell line (Tahoe Therapeutics)
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Genes

200 genes differentially expressed following the Clopidogrel_NCI-H2347 drug perturbation from the Tahoe Therapeutics Tahoe 100M Perturbation Atlas dataset.

increased expression

Symbol Name Standardized Value
TMSB4X thymosin beta 4, X-linked 0.0905594
TRIO trio Rho guanine nucleotide exchange factor 0.0851591
ASPH aspartate beta-hydroxylase 0.0734497
LMO7 LIM domain 7 0.0699608
FNDC3B fibronectin type III domain containing 3B 0.0696786
LPP LIM domain containing preferred translocation partner in lipoma 0.0640005
HNRNPH1 heterogeneous nuclear ribonucleoprotein H1 (H) 0.060317
DCBLD2 discoidin, CUB and LCCL domain containing 2 0.0542047
SAMD4A sterile alpha motif domain containing 4A 0.0540772
RAD21 RAD21 homolog (S. pombe) 0.0537664
EFNA5 ephrin-A5 0.0529435
PGK1 phosphoglycerate kinase 1 0.0507862
LAMC2 laminin, gamma 2 0.0504579
LAMB3 laminin, beta 3 0.0503981
NAMPT nicotinamide phosphoribosyltransferase 0.0470148
ITGA2 integrin, alpha 2 (CD49B, alpha 2 subunit of VLA-2 receptor) 0.046616
EXT1 exostosin glycosyltransferase 1 0.0445505
TPT1 tumor protein, translationally-controlled 1 0.0442822
NAV2 neuron navigator 2 0.0440649
YWHAZ tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein, zeta 0.0423489
BHLHE40 basic helix-loop-helix family, member e40 0.0419278
NPM1 nucleophosmin (nucleolar phosphoprotein B23, numatrin) 0.0412892
PJA2 praja ring finger 2, E3 ubiquitin protein ligase 0.0404969
LIMCH1 LIM and calponin homology domains 1 0.0402317
MBOAT2 membrane bound O-acyltransferase domain containing 2 0.0397142
HIF1A hypoxia inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) 0.0386942
PTK2 protein tyrosine kinase 2 0.0384902
KDM3A lysine (K)-specific demethylase 3A 0.0384868
HNRNPA2B1 heterogeneous nuclear ribonucleoprotein A2/B1 0.0372311
RPS24 ribosomal protein S24 0.0361616
ZNF292 zinc finger protein 292 0.0361521
CCND1 cyclin D1 0.034886
SQSTM1 sequestosome 1 0.034844
GRB10 growth factor receptor-bound protein 10 0.0347668
PLAU plasminogen activator, urokinase 0.0342313
HNRNPU heterogeneous nuclear ribonucleoprotein U (scaffold attachment factor A) 0.0341891
ARL6IP1 ADP-ribosylation factor-like 6 interacting protein 1 0.0337765
NPEPPS aminopeptidase puromycin sensitive 0.0335186
BZW1 basic leucine zipper and W2 domains 1 0.0332061
MARCHF6 membrane associated ring-CH-type finger 6 0.0330926
PARD3 par-3 family cell polarity regulator 0.0328866
ALCAM activated leukocyte cell adhesion molecule 0.0323757
RUNX1 runt-related transcription factor 1 0.0322938
RBM39 RNA binding motif protein 39 0.0316442
NAP1L1 nucleosome assembly protein 1-like 1 0.0307169
TOP2A topoisomerase (DNA) II alpha 170kDa 0.0306744
DDIT4 DNA-damage-inducible transcript 4 0.0303566
MYO6 myosin VI 0.0303356
KPNB1 karyopherin (importin) beta 1 0.0303164
ATP1B1 ATPase, Na+/K+ transporting, beta 1 polypeptide 0.0295879
CD2AP CD2-associated protein 0.0293111
MYH9 myosin, heavy chain 9, non-muscle 0.0287565
ITGB1 integrin, beta 1 (fibronectin receptor, beta polypeptide, antigen CD29 includes MDF2, MSK12) 0.0282168
SLC38A1 solute carrier family 38, member 1 0.0280102
CD46 CD46 molecule, complement regulatory protein 0.0279265
SEC31A SEC31 homolog A (S. cerevisiae) 0.0277505
HMGB2 high mobility group box 2 0.0271753
LMNA lamin A/C 0.0260491
DYRK1A dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A 0.0258342
WSB1 WD repeat and SOCS box containing 1 0.0256513
ARHGAP5 Rho GTPase activating protein 5 0.025599
ERBIN erbb2 interacting protein 0.0251945
FN1 fibronectin 1 0.0251123
ANXA2 annexin A2 0.0250506
MSMO1 methylsterol monooxygenase 1 0.0247001
EIF4G2 eukaryotic translation initiation factor 4 gamma, 2 0.0246732
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase 0.0246363
STRN3 striatin, calmodulin binding protein 3 0.0246138
MYL6 myosin, light chain 6, alkali, smooth muscle and non-muscle 0.0240546
PTPN12 protein tyrosine phosphatase, non-receptor type 12 0.0240423
FUT8 fucosyltransferase 8 (alpha (1,6) fucosyltransferase) 0.0239753
AFF4 AF4/FMR2 family, member 4 0.0237955
ATP11A ATPase, class VI, type 11A 0.0237925
DHX15 DEAH (Asp-Glu-Ala-His) box helicase 15 0.0237748
DSCAM Down syndrome cell adhesion molecule 0.0234363
CALM2 calmodulin 2 (phosphorylase kinase, delta) 0.0232161
ARID4B AT rich interactive domain 4B (RBP1-like) 0.0231869
KMT2C lysine (K)-specific methyltransferase 2C 0.0228625
AP3B1 adaptor-related protein complex 3, beta 1 subunit 0.0228486
OGA O-GlcNAcase 0.0224666
VCL vinculin 0.0221817
RPL35A ribosomal protein L35a 0.0221656
SPAG9 sperm associated antigen 9 0.021982
DDX5 DEAD (Asp-Glu-Ala-Asp) box helicase 5 0.0214016
FNIP1 folliculin interacting protein 1 0.0213793
PEG10 paternally expressed 10 0.0212814
CAVIN1 caveolae associated protein 1 0.0209695
ELL2 elongation factor, RNA polymerase II, 2 0.0209176
TAF1D TATA box binding protein (TBP)-associated factor, RNA polymerase I, D, 41kDa 0.0206806
SMG7 SMG7 nonsense mediated mRNA decay factor 0.020574
CLTC clathrin, heavy chain (Hc) 0.0205303
RAB11FIP1 RAB11 family interacting protein 1 (class I) 0.0204716
SLTM SAFB-like, transcription modulator 0.0203793
EIF3E eukaryotic translation initiation factor 3, subunit E 0.020273
DTNA dystrobrevin, alpha 0.0201978
ITCH itchy E3 ubiquitin protein ligase 0.0199542
RPS8 ribosomal protein S8 0.0198293
ARF1 ADP-ribosylation factor 1 0.01965
DST dystonin 0.0195843
ZBTB20 zinc finger and BTB domain containing 20 0.0195528

decreased expression

Symbol Name Standardized Value
GAPDH glyceraldehyde-3-phosphate dehydrogenase -0.322385
POTEF POTE ankyrin domain family, member F -0.191624
UBC ubiquitin C -0.157389
FTL ferritin, light polypeptide -0.107763
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1 -0.101259
ACTG1 actin gamma 1 -0.0700177
NDRG1 N-myc downstream regulated 1 -0.0638318
P4HB prolyl 4-hydroxylase, beta polypeptide -0.0626987
EEF2 eukaryotic translation elongation factor 2 -0.0603495
PABPC1 poly(A) binding protein, cytoplasmic 1 -0.0576038
FTH1 ferritin, heavy polypeptide 1 -0.0562981
TMSB10 thymosin beta 10 -0.047561
IGFBP3 insulin-like growth factor binding protein 3 -0.0461976
HMGA1 high mobility group AT-hook 1 -0.0459306
APLP2 amyloid beta (A4) precursor-like protein 2 -0.0433162
PCBP2 poly(rC) binding protein 2 -0.040463
LOC112694756 uncharaterized LOC112694756 -0.0402237
IFI27 interferon, alpha-inducible protein 27 -0.0401993
G0S2 G0/G1 switch 2 -0.0395733
RPL8 ribosomal protein L8 -0.0386956
PDIA4 protein disulfide isomerase family A, member 4 -0.0354969
RPS23 ribosomal protein S23 -0.0315627
PDIA3 protein disulfide isomerase family A, member 3 -0.0290227
ENO1 enolase 1, (alpha) -0.0244755
MDK midkine (neurite growth-promoting factor 2) -0.0222364
MT2A metallothionein 2A -0.022088
LY6E lymphocyte antigen 6 complex, locus E -0.0220679
IFITM3 interferon induced transmembrane protein 3 -0.0219391
TSC22D2 TSC22 domain family, member 2 -0.0216491
UPP1 uridine phosphorylase 1 -0.0215532
OAS3 2'-5'-oligoadenylate synthetase 3, 100kDa -0.0213836
RPS27A ribosomal protein S27a -0.0207376
VEGFA vascular endothelial growth factor A -0.0206259
RPL28 ribosomal protein L28 -0.0202024
FOSL1 FOS-like antigen 1 -0.0201829
IFI6 interferon, alpha-inducible protein 6 -0.0198897
PHLDA1 pleckstrin homology-like domain, family A, member 1 -0.0198808
TXNIP thioredoxin interacting protein -0.0194803
MAP4K5 mitogen-activated protein kinase kinase kinase kinase 5 -0.0192862
PPDPF pancreatic progenitor cell differentiation and proliferation factor -0.0191972
JUN jun proto-oncogene -0.0189205
EEF1G eukaryotic translation elongation factor 1 gamma -0.0189097
ENO2 enolase 2 (gamma, neuronal) -0.018571
EIF2AK2 eukaryotic translation initiation factor 2-alpha kinase 2 -0.0182148
EGR1 early growth response 1 -0.0180563
DDX24 DEAD (Asp-Glu-Ala-Asp) box helicase 24 -0.0176235
ASTN2 astrotactin 2 -0.0173432
RPS11 ribosomal protein S11 -0.0172428
BRD2 bromodomain containing 2 -0.0171323
HSPB1 heat shock 27kDa protein 1 -0.0169902
LAP3 leucine aminopeptidase 3 -0.0168187
EIF5 eukaryotic translation initiation factor 5 -0.0167253
RPS15 ribosomal protein S15 -0.0163803
RPL21 ribosomal protein L21 -0.016199
ATP5F1B ATP synthase F1 subunit beta -0.0161164
HNRNPDL heterogeneous nuclear ribonucleoprotein D-like -0.0157312
RPS10 ribosomal protein S10 -0.0156778
PARP14 poly (ADP-ribose) polymerase family, member 14 -0.0153069
MX1 MX dynamin-like GTPase 1 -0.015188
TAPBP TAP binding protein (tapasin) -0.0151257
RPS5 ribosomal protein S5 -0.0149251
LGALS3BP lectin, galactoside-binding, soluble, 3 binding protein -0.0148818
PKM pyruvate kinase, muscle -0.0148561
RPLP2 ribosomal protein, large, P2 -0.014776
HSP90AA1 heat shock protein 90kDa alpha (cytosolic), class A member 1 -0.0146161
HLA-B major histocompatibility complex, class I, B -0.0145266
MSN moesin -0.0144192
FXR1 fragile X mental retardation, autosomal homolog 1 -0.0143569
IFITM1 interferon induced transmembrane protein 1 -0.014352
LDHB lactate dehydrogenase B -0.0139111
PHLDA2 pleckstrin homology-like domain, family A, member 2 -0.0138288
MUC1 mucin 1, cell surface associated -0.0133519
SLC2A1 solute carrier family 2 (facilitated glucose transporter), member 1 -0.0130204
DDX60L DEAD (Asp-Glu-Ala-Asp) box polypeptide 60-like -0.0130181
HMGN2 high mobility group nucleosomal binding domain 2 -0.0129767
ERC2 ELKS/RAB6-interacting/CAST family member 2 -0.0128058
PDIA6 protein disulfide isomerase family A, member 6 -0.0127999
ZFP36L1 ZFP36 ring finger protein-like 1 -0.0127426
MXD1 MAX dimerization protein 1 -0.0121949
FOS FBJ murine osteosarcoma viral oncogene homolog -0.0117548
IFI16 interferon, gamma-inducible protein 16 -0.0115104
SLC34A2 solute carrier family 34 (type II sodium/phosphate cotransporter), member 2 -0.0114852
RPL15 ribosomal protein L15 -0.0114656
FOSB FBJ murine osteosarcoma viral oncogene homolog B -0.0114613
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) -0.0113513
RBCK1 RanBP-type and C3HC4-type zinc finger containing 1 -0.0112265
PPIB peptidylprolyl isomerase B (cyclophilin B) -0.0111558
CD44 CD44 molecule (Indian blood group) -0.0110728
SH3BGRL3 SH3 domain binding glutamate-rich protein like 3 -0.011006
CLDN4 claudin 4 -0.010977
RPS29 ribosomal protein S29 -0.0107953
HERC5 HECT and RLD domain containing E3 ubiquitin protein ligase 5 -0.0107782
HNRNPA1 heterogeneous nuclear ribonucleoprotein A1 -0.0106061
PFN1 profilin 1 -0.0106005
S100A10 S100 calcium binding protein A10 -0.0105507
GPRC5A G protein-coupled receptor, class C, group 5, member A -0.0098734
WASF2 WAS protein family, member 2 -0.009642
PPP1R13B protein phosphatase 1, regulatory subunit 13B -0.00956267
TFPI2 tissue factor pathway inhibitor 2 -0.00941054
ICAM1 intercellular adhesion molecule 1 -0.00934634