Dabrafenib Gene Set

Dataset LINCS KinomeScan Kinase Inhibitor Targets
Category physical interactions
Type small molecule
Description An organofluorine compound and antineoplastic agent, used as its mesylate salt in treatment of metastatic melanoma. (Chemical Entities of Biological Interest Ontology, CHEBI_75045)
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Genes

68 kinases inhibited by the Dabrafenib small molecule from the KinomeScan Kinase Inhibitor Targets dataset.

Symbol Name Standardized Value
PIK3C2B phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 beta 1.36211
CSK c-src tyrosine kinase 1.36211
BMPR1B bone morphogenetic protein receptor, type IB 1.36211
CDK3 cyclin-dependent kinase 3 1.35325
CDKL5 cyclin-dependent kinase-like 5 1.34449
MKNK2 MAP kinase interacting serine/threonine kinase 2 1.34449
ERBB3 erb-b2 receptor tyrosine kinase 3 1.34449
NEK6 NIMA-related kinase 6 1.34449
STK36 serine/threonine kinase 36 1.33582
CDK2 cyclin-dependent kinase 2 1.33582
ULK3 unc-51 like kinase 3 1.31878
LIMK1 LIM domain kinase 1 1.31878
SIK1 salt-inducible kinase 1 1.3104
PI4KB phosphatidylinositol 4-kinase, catalytic, beta 1.3104
CDKL2 cyclin-dependent kinase-like 2 (CDC2-related kinase) 1.3104
CIT citron rho-interacting serine/threonine kinase 1.30212
EPHB6 EPH receptor B6 1.28583
ZAK sterile alpha motif and leucine zipper containing kinase AZK 1.28583
HIPK1 homeodomain interacting protein kinase 1 1.28583
PTK6 protein tyrosine kinase 6 1.27782
TNK1 tyrosine kinase, non-receptor, 1 1.26209
HIPK3 homeodomain interacting protein kinase 3 1.23916
ULK2 unc-51 like autophagy activating kinase 2 1.23916
CAMK1D calcium/calmodulin-dependent protein kinase ID 1.23916
NEK7 NIMA-related kinase 7 1.23916
GAK cyclin G associated kinase 1.23916
DCLK2 doublecortin-like kinase 2 1.23916
LCK LCK proto-oncogene, Src family tyrosine kinase 1.22432
DCLK3 doublecortin-like kinase 3 1.22432
CSF1R colony stimulating factor 1 receptor 1.22432
TEK TEK tyrosine kinase, endothelial 1.19568
HIPK2 homeodomain interacting protein kinase 2 1.19568
CDK15 cyclin-dependent kinase 15 1.17508
RIPK2 receptor-interacting serine-threonine kinase 2 1.16838
HCK HCK proto-oncogene, Src family tyrosine kinase 1.15523
CDK5 cyclin-dependent kinase 5 1.15523
PAK3 p21 protein (Cdc42/Rac)-activated kinase 3 1.1424
BLK BLK proto-oncogene, Src family tyrosine kinase 1.1424
CDK8 cyclin-dependent kinase 8 1.12988
NEK9 NIMA-related kinase 9 1.12988
DCLK1 doublecortin-like kinase 1 1.12373
CDK7 cyclin-dependent kinase 7 1.11767
DDR1 discoidin domain receptor tyrosine kinase 1 1.08283
TGFBR2 transforming growth factor, beta receptor II (70/80kDa) 1.08283
SRC SRC proto-oncogene, non-receptor tyrosine kinase 1.07728
CDK14 cyclin-dependent kinase 14 1.05057
FRK fyn-related Src family tyrosine kinase 1.05057
ITK IL2-inducible T-cell kinase 1.04035
HIPK4 homeodomain interacting protein kinase 4 1.02553
BRSK2 BR serine/threonine kinase 2 0.993117
STK16 serine/threonine kinase 16 0.993117
PAK7 p21 protein (Cdc42/Rac)-activated kinase 7 0.993117
EPHA3 EPH receptor A3 0.984392
AURKB aurora kinase B 0.975893
LYN LYN proto-oncogene, Src family tyrosine kinase 0.955601
NEK2 NIMA-related kinase 2 0.944052
BMPR2 bone morphogenetic protein receptor, type II (serine/threonine kinase) 0.936602
BRSK1 BR serine/threonine kinase 1 0.936602
ACVR1 activin A receptor, type I 0.936602
CAMK1 calcium/calmodulin-dependent protein kinase I 0.889549
ABL2 ABL proto-oncogene 2, non-receptor tyrosine kinase 0.869001
MAP3K10 mitogen-activated protein kinase kinase kinase 10 0.860727
TAOK2 TAO kinase 2 0.860727
AXL AXL receptor tyrosine kinase 0.850157
FYN FYN proto-oncogene, Src family tyrosine kinase 0.850157
TNIK TRAF2 and NCK interacting kinase 0.850157
ULK1 unc-51 like autophagy activating kinase 1 0.850157
STK25 serine/threonine kinase 25 0.850157