Drug ADME Gene Set

Dataset Reactome Pathways 2024
Category structural or functional annotations
Type pathway
External Link https://reactome.org/PathwayBrowser/#/R-HSA-9748784
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Genes

108 proteins participating in the Drug ADME pathway from the Reactome Pathways 2024 dataset.

Symbol Name
ABCB1 ATP-binding cassette, sub-family B (MDR/TAP), member 1
ABCC1 ATP-binding cassette, sub-family C (CFTR/MRP), member 1
ABCC2 ATP-binding cassette, sub-family C (CFTR/MRP), member 2
ABCC3 ATP-binding cassette, sub-family C (CFTR/MRP), member 3
ABCC4 ATP-binding cassette, sub-family C (CFTR/MRP), member 4
ABCC5 ATP-binding cassette, sub-family C (CFTR/MRP), member 5
ABCG2 ATP-binding cassette, sub-family G (WHITE), member 2 (Junior blood group)
ACSM2A acyl-CoA synthetase medium-chain family member 2A
ACSM2B acyl-CoA synthetase medium-chain family member 2B
ACSM4 acyl-CoA synthetase medium-chain family member 4
ACSM5 acyl-CoA synthetase medium-chain family member 5
ACY1 aminoacylase 1
ADA adenosine deaminase
ADAL adenosine deaminase-like
ADH1A alcohol dehydrogenase 1A (class I), alpha polypeptide
ADK adenosine kinase
AKR1C1 aldo-keto reductase family 1, member C1
ALB albumin
BCHE butyrylcholinesterase
BSG basigin (Ok blood group)
CES1 carboxylesterase 1
CES2 carboxylesterase 2
CNDP2 CNDP dipeptidase 2 (metallopeptidase M20 family)
CYP2C19 cytochrome P450, family 2, subfamily C, polypeptide 19
CYP2C8 cytochrome P450, family 2, subfamily C, polypeptide 8
CYP2C9 cytochrome P450, family 2, subfamily C, polypeptide 9
CYP2D6 cytochrome P450, family 2, subfamily D, polypeptide 6
CYP2E1 cytochrome P450, family 2, subfamily E, polypeptide 1
CYP3A4 cytochrome P450, family 3, subfamily A, polypeptide 4
GGT1 gamma-glutamyltransferase 1
GGT5 gamma-glutamyltransferase 5
GGT6 gamma-glutamyltransferase 6
GGT7 gamma-glutamyltransferase 7
GLYAT glycine-N-acyltransferase
GLYATL1 glycine-N-acyltransferase-like 1
GLYATL2 glycine-N-acyltransferase-like 2
GLYATL3 glycine-N-acyltransferase-like 3
GMPS guanine monphosphate synthase
GSTA1 glutathione S-transferase alpha 1
GSTA2 glutathione S-transferase alpha 2
GSTM1 glutathione S-transferase mu 1
GSTP1 glutathione S-transferase pi 1
GSTT1 glutathione S-transferase theta 1
GUK1 guanylate kinase 1
HPRT1 hypoxanthine phosphoribosyltransferase 1
HSD11B1 hydroxysteroid (11-beta) dehydrogenase 1
HSD11B2 hydroxysteroid (11-beta) dehydrogenase 2
IMPDH1 IMP (inosine 5'-monophosphate) dehydrogenase 1
IMPDH2 IMP (inosine 5'-monophosphate) dehydrogenase 2
ITPA inosine triphosphatase (nucleoside triphosphate pyrophosphatase)
NAT1 N-acetyltransferase 1 (arylamine N-acetyltransferase)
NAT2 N-acetyltransferase 2 (arylamine N-acetyltransferase)
NME1 NME/NM23 nucleoside diphosphate kinase 1
NME2 NME/NM23 nucleoside diphosphate kinase 2
NT5C2 5'-nucleotidase, cytosolic II
NUDT15 nudix (nucleoside diphosphate linked moiety X)-type motif 15
PCK1 phosphoenolpyruvate carboxykinase 1 (soluble)
PNP purine nucleoside phosphorylase
PON1 paraoxonase 1
PON3 paraoxonase 3
RAC1 ras-related C3 botulinum toxin substrate 1 (rho family, small GTP binding protein Rac1)
SERPINA6 serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 6
SLC16A1 solute carrier family 16 (monocarboxylate transporter), member 1
SLC22A1 solute carrier family 22 (organic cation transporter), member 1
SLC22A2 solute carrier family 22 (organic cation transporter), member 2
SLC22A3 solute carrier family 22 (organic cation transporter), member 3
SLC22A7 solute carrier family 22 (organic anion transporter), member 7
SLC22A8 solute carrier family 22 (organic anion transporter), member 8
SLC28A2 solute carrier family 28 (concentrative nucleoside transporter), member 2
SLC28A3 solute carrier family 28 (concentrative nucleoside transporter), member 3
SLC29A1 solute carrier family 29 (equilibrative nucleoside transporter), member 1
SLC29A2 solute carrier family 29 (equilibrative nucleoside transporter), member 2
SLC29A3 solute carrier family 29 (equilibrative nucleoside transporter), member 3
SLCO1A2 solute carrier organic anion transporter family, member 1A2
SLCO1B1 solute carrier organic anion transporter family, member 1B1
SLCO1B3 solute carrier organic anion transporter family, member 1B3
SLCO2B1 solute carrier organic anion transporter family, member 2B1
SULT1A1 sulfotransferase family, cytosolic, 1A, phenol-preferring, member 1
SULT1A3 sulfotransferase family, cytosolic, 1A, phenol-preferring, member 3
SULT1A4 sulfotransferase family, cytosolic, 1A, phenol-preferring, member 4
SULT1C4 sulfotransferase family, cytosolic, 1C, member 4
SULT1E1 sulfotransferase family 1E, estrogen-preferring, member 1
SULT2A1 sulfotransferase family, cytosolic, 2A, dehydroepiandrosterone (DHEA)-preferring, member 1
TPMT thiopurine S-methyltransferase
UGT1A1 UDP glucuronosyltransferase 1 family, polypeptide A1
UGT1A10 UDP glucuronosyltransferase 1 family, polypeptide A10
UGT1A3 UDP glucuronosyltransferase 1 family, polypeptide A3
UGT1A4 UDP glucuronosyltransferase 1 family, polypeptide A4
UGT1A5 UDP glucuronosyltransferase 1 family, polypeptide A5
UGT1A6 UDP glucuronosyltransferase 1 family, polypeptide A6
UGT1A7 UDP glucuronosyltransferase 1 family, polypeptide A7
UGT1A8 UDP glucuronosyltransferase 1 family, polypeptide A8
UGT1A9 UDP glucuronosyltransferase 1 family, polypeptide A9
UGT2A1 UDP glucuronosyltransferase 2 family, polypeptide A1, complex locus
UGT2A3 UDP glucuronosyltransferase 2 family, polypeptide A3
UGT2B10 UDP glucuronosyltransferase 2 family, polypeptide B10
UGT2B11 UDP glucuronosyltransferase 2 family, polypeptide B11
UGT2B15 UDP glucuronosyltransferase 2 family, polypeptide B15
UGT2B17 UDP glucuronosyltransferase 2 family, polypeptide B17
UGT2B28 UDP glucuronosyltransferase 2 family, polypeptide B28
UGT2B4 UDP glucuronosyltransferase 2 family, polypeptide B4
UGT2B7 UDP glucuronosyltransferase 2 family, polypeptide B7
UGT3A1 UDP glycosyltransferase 3 family, polypeptide A1
UGT3A2 UDP glycosyltransferase 3 family, polypeptide A2
VAV1 vav 1 guanine nucleotide exchange factor
VAV2 vav 2 guanine nucleotide exchange factor
VAV3 vav 3 guanine nucleotide exchange factor
XDH xanthine dehydrogenase