Entecavir (monohydrate)_H4 Gene Set

Dataset Tahoe Therapeutics Tahoe 100M Perturbation Atlas
Category transcriptomics
Type cell type
Description Entecavir (monohydrate) perturbation in H4 cell line (Tahoe Therapeutics)
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Genes

200 genes differentially expressed following the Entecavir (monohydrate)_H4 drug perturbation from the Tahoe Therapeutics Tahoe 100M Perturbation Atlas dataset.

increased expression

Symbol Name Standardized Value
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase 0.0922776
FAM13A family with sequence similarity 13, member A 0.0860138
GBE1 glucan (1,4-alpha-), branching enzyme 1 0.0844086
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) 0.0836818
SDK1 sidekick cell adhesion molecule 1 0.0805334
FNDC3B fibronectin type III domain containing 3B 0.0666425
ERO1A endoplasmic reticulum oxidoreductase 1 alpha 0.0610738
PIK3C2A phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 alpha 0.0577839
RBPJ recombination signal binding protein for immunoglobulin kappa J region 0.0575022
MYOF myoferlin 0.0557644
HELZ helicase with zinc finger 0.0541179
FHIP1A FHF complex subunit HOOK interacting protein 1A 0.0508414
RAB1A RAB1A, member RAS oncogene family 0.049833
SLC2A3 solute carrier family 2 (facilitated glucose transporter), member 3 0.0475112
MEF2A myocyte enhancer factor 2A 0.0467347
PLOD2 procollagen-lysine, 2-oxoglutarate 5-dioxygenase 2 0.0439711
SRP54 signal recognition particle 54kDa 0.0434275
WSB1 WD repeat and SOCS box containing 1 0.0430436
P4HB prolyl 4-hydroxylase, beta polypeptide 0.0422602
CALR calreticulin 0.0420356
HILPDA hypoxia inducible lipid droplet-associated 0.0410947
PRELID2 PRELI domain containing 2 0.0406873
ELL2 elongation factor, RNA polymerase II, 2 0.0406849
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1 0.0403531
GNPDA1 glucosamine-6-phosphate deaminase 1 0.0395792
PDIA3 protein disulfide isomerase family A, member 3 0.0391556
NDRG1 N-myc downstream regulated 1 0.038777
ADM adrenomedullin 0.0387617
P4HA1 prolyl 4-hydroxylase, alpha polypeptide I 0.0387117
ERRFI1 ERBB receptor feedback inhibitor 1 0.038655
KMT2C lysine (K)-specific methyltransferase 2C 0.0384464
HERC3 HECT and RLD domain containing E3 ubiquitin protein ligase 3 0.0374102
PCBP2 poly(rC) binding protein 2 0.0369234
SETD5 SET domain containing 5 0.0367632
TBC1D23 TBC1 domain family, member 23 0.0366652
UBA6 ubiquitin-like modifier activating enzyme 6 0.0365409
KCNMA1 potassium channel, calcium activated large conductance subfamily M alpha, member 1 0.0364233
COPA coatomer protein complex, subunit alpha 0.036317
RTN4 reticulon 4 0.0361276
SLC2A1 solute carrier family 2 (facilitated glucose transporter), member 1 0.0361032
MSN moesin 0.0359853
TRA2A transformer 2 alpha homolog (Drosophila) 0.0353501
ADAM17 ADAM metallopeptidase domain 17 0.0353104
ENO2 enolase 2 (gamma, neuronal) 0.0341733
USP3 ubiquitin specific peptidase 3 0.0334464
SEC24A SEC24 family member A 0.033118
TIMP3 TIMP metallopeptidase inhibitor 3 0.0321404
ATP13A3 ATPase type 13A3 0.0320678
DGKD diacylglycerol kinase, delta 130kDa 0.0320236
HIP1 huntingtin interacting protein 1 0.0318705
CNOT2 CCR4-NOT transcription complex, subunit 2 0.0317042
NBAS neuroblastoma amplified sequence 0.0314382
ESYT2 extended synaptotagmin-like protein 2 0.0314
TNFRSF10B tumor necrosis factor receptor superfamily, member 10b 0.0312075
MARCHF6 membrane associated ring-CH-type finger 6 0.0310787
RNF220 ring finger protein 220 0.0308941
TFG TRK-fused gene 0.0308507
SEC31A SEC31 homolog A (S. cerevisiae) 0.0304838
GFPT1 glutamine--fructose-6-phosphate transaminase 1 0.0301683
ZNF292 zinc finger protein 292 0.0300878
INSIG2 insulin induced gene 2 0.0298414
AFF4 AF4/FMR2 family, member 4 0.0296431
FNIP1 folliculin interacting protein 1 0.0288911
JARID2 jumonji, AT rich interactive domain 2 0.0285274
TTC3 tetratricopeptide repeat domain 3 0.0284862
USP37 ubiquitin specific peptidase 37 0.0280153
GPRC5A G protein-coupled receptor, class C, group 5, member A 0.0278908
SPARC secreted protein, acidic, cysteine-rich (osteonectin) 0.0276279
CDK19 cyclin-dependent kinase 19 0.0274111
ABCA1 ATP-binding cassette, sub-family A (ABC1), member 1 0.0273878
HOOK2 hook microtubule-tethering protein 2 0.0272138
PCBP3 poly(rC) binding protein 3 0.0271358
LRRFIP1 leucine rich repeat (in FLII) interacting protein 1 0.0271304
SCFD1 sec1 family domain containing 1 0.0271285
ACBD3 acyl-CoA binding domain containing 3 0.0266967
CCNL1 cyclin L1 0.026688
ZNF395 zinc finger protein 395 0.0264965
GOLGB1 golgin B1 0.0263167
CANX calnexin 0.0263048
RB1CC1 RB1-inducible coiled-coil 1 0.0262936
PFKFB4 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 4 0.0260986
YEATS2 YEATS domain containing 2 0.0260599
EGLN3 egl-9 family hypoxia-inducible factor 3 0.0259261
NUP58 nucleoporin 58 0.0258529
MXI1 MAX interactor 1, dimerization protein 0.0258468
CNOT1 CCR4-NOT transcription complex, subunit 1 0.0258449
CD109 CD109 molecule 0.0256555
C1D C1D nuclear receptor corepressor 0.0256028
MAGT1 magnesium transporter 1 0.0255994
PKM pyruvate kinase, muscle 0.0255318
PDK3 pyruvate dehydrogenase kinase, isozyme 3 0.0253378
RELCH RAB11 binding and LisH domain, coiled-coil and HEAT repeat containing 0.0247934
MYH9 myosin, heavy chain 9, non-muscle 0.0246699
KPNA4 karyopherin alpha 4 (importin alpha 3) 0.0244705
CHD1 chromodomain helicase DNA binding protein 1 0.0242214
VMP1 vacuole membrane protein 1 0.0242104
LCOR ligand dependent nuclear receptor corepressor 0.0239936
USP9X ubiquitin specific peptidase 9, X-linked 0.0238074
RICTOR RPTOR independent companion of MTOR, complex 2 0.0237653
EIF2AK3 eukaryotic translation initiation factor 2-alpha kinase 3 0.0237471

decreased expression

Symbol Name Standardized Value
NALF1 NALCN channel auxiliary factor 1 -0.179342
GAPDH glyceraldehyde-3-phosphate dehydrogenase -0.139274
CXCL8 chemokine (C-X-C motif) ligand 8 -0.122393
VIM vimentin -0.10541
ITGA2 integrin, alpha 2 (CD49B, alpha 2 subunit of VLA-2 receptor) -0.103731
MT2A metallothionein 2A -0.0985484
TMSB10 thymosin beta 10 -0.0980696
KYNU kynureninase -0.0951034
CD44 CD44 molecule (Indian blood group) -0.0768951
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11 -0.0743238
FTL ferritin, light polypeptide -0.0667605
EXT1 exostosin glycosyltransferase 1 -0.0549267
SEMA5A sema domain, seven thrombospondin repeats (type 1 and type 1-like), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 5A -0.0527566
NAV3 neuron navigator 3 -0.0489586
PTPRG protein tyrosine phosphatase, receptor type, G -0.046807
PDE4D phosphodiesterase 4D, cAMP-specific -0.0466661
NLGN1 neuroligin 1 -0.0456892
FN1 fibronectin 1 -0.0437954
OSMR oncostatin M receptor -0.0405559
COL6A3 collagen, type VI, alpha 3 -0.0398922
ANTXR2 anthrax toxin receptor 2 -0.0397623
HDAC9 histone deacetylase 9 -0.0385697
DST dystonin -0.0376767
INHBA inhibin, beta A -0.0361835
MAP1B microtubule-associated protein 1B -0.0358445
TMSB4X thymosin beta 4, X-linked -0.0348672
KCNQ5 potassium channel, voltage gated KQT-like subfamily Q, member 5 -0.0336038
NAV1 neuron navigator 1 -0.0330249
TNNC1 troponin C type 1 (slow) -0.0328666
RPS19 ribosomal protein S19 -0.032138
YBX1 Y box binding protein 1 -0.0310927
FBXL17 F-box and leucine-rich repeat protein 17 -0.0310381
LYPD6B LY6/PLAUR domain containing 6B -0.0307642
SH3KBP1 SH3-domain kinase binding protein 1 -0.0303048
DTNA dystrobrevin, alpha -0.0294225
RPL35A ribosomal protein L35a -0.0281835
SEC61G Sec61 gamma subunit -0.0281294
IGFBP3 insulin-like growth factor binding protein 3 -0.0280733
TEAD1 TEA domain family member 1 (SV40 transcriptional enhancer factor) -0.0280486
TENM3 teneurin transmembrane protein 3 -0.0276427
SIPA1L1 signal-induced proliferation-associated 1 like 1 -0.0275793
TPTE transmembrane phosphatase with tensin homology -0.0272083
UBE2K ubiquitin-conjugating enzyme E2K -0.0271307
EHBP1 EH domain binding protein 1 -0.0268969
CALD1 caldesmon 1 -0.0268084
OR51B5 olfactory receptor, family 51, subfamily B, member 5 -0.02671
TNS3 tensin 3 -0.0264639
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1 -0.0263902
AK1 adenylate kinase 1 -0.0263849
ACTN4 actinin, alpha 4 -0.0263245
MT1X metallothionein 1X -0.0261039
FSTL1 follistatin-like 1 -0.0258609
CALM1 calmodulin 1 (phosphorylase kinase, delta) -0.0258497
LGALS1 lectin, galactoside-binding, soluble, 1 -0.0254552
CDK6 cyclin-dependent kinase 6 -0.0251389
VEGFC vascular endothelial growth factor C -0.0251373
RPL32 ribosomal protein L32 -0.0250275
SRGAP1 SLIT-ROBO Rho GTPase activating protein 1 -0.0250195
RPS4X ribosomal protein S4, X-linked -0.0249007
FAF1 Fas (TNFRSF6) associated factor 1 -0.0247067
ZC3HAV1 zinc finger CCCH-type, antiviral 1 -0.0243786
HIBADH 3-hydroxyisobutyrate dehydrogenase -0.0240407
EGR1 early growth response 1 -0.023801
DCBLD2 discoidin, CUB and LCCL domain containing 2 -0.0236435
IGFBP5 insulin-like growth factor binding protein 5 -0.0234269
SCMH1 sex comb on midleg homolog 1 (Drosophila) -0.0231581
PAPPA2 pappalysin 2 -0.0230676
MYLK myosin light chain kinase -0.0230203
ATXN10 ataxin 10 -0.0230008
AOPEP aminopeptidase O (putative) -0.0229437
HSPD1 heat shock 60kDa protein 1 (chaperonin) -0.0224626
BICD1 bicaudal D homolog 1 (Drosophila) -0.022135
CLMP CXADR-like membrane protein -0.0219959
ETV6 ets variant 6 -0.0219379
PHF14 PHD finger protein 14 -0.0217319
ASPH aspartate beta-hydroxylase -0.0215077
RPL36 ribosomal protein L36 -0.0213401
RPL34 ribosomal protein L34 -0.0212185
CCND1 cyclin D1 -0.021184
CREB5 cAMP responsive element binding protein 5 -0.0211267
TXNRD1 thioredoxin reductase 1 -0.0211027
SBF2 SET binding factor 2 -0.0210935
ARHGAP24 Rho GTPase activating protein 24 -0.02083
GNB1 guanine nucleotide binding protein (G protein), beta polypeptide 1 -0.0204858
RACK1 receptor for activated C kinase 1 -0.0204319
LAMB1 laminin, beta 1 -0.0203044
NAALADL2 N-acetylated alpha-linked acidic dipeptidase-like 2 -0.020197
MICAL2 microtubule associated monooxygenase, calponin and LIM domain containing 2 -0.0201953
ANKRD11 ankyrin repeat domain 11 -0.0200615
SEMA3A sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3A -0.0198558
ENO1 enolase 1, (alpha) -0.0197373
RPL12 ribosomal protein L12 -0.0195673
NEDD4 neural precursor cell expressed, developmentally down-regulated 4, E3 ubiquitin protein ligase -0.0194677
HLCS holocarboxylase synthetase (biotin-(proprionyl-CoA-carboxylase (ATP-hydrolysing)) ligase) -0.0191759
MYO9A myosin IXA -0.0191322
TUBB tubulin, beta class I -0.0190457
PARP14 poly (ADP-ribose) polymerase family, member 14 -0.019032
GLIS3 GLIS family zinc finger 3 -0.0189981
RPLP1 ribosomal protein, large, P1 -0.0186787
ASTN2 astrotactin 2 -0.0186711