KIN001-220 Gene Set

Dataset LINCS KinomeScan Kinase Inhibitor Targets
Category physical interactions
Type small molecule
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Genes

48 kinases inhibited by the KIN001-220 small molecule from the KinomeScan Kinase Inhibitor Targets dataset.

Symbol Name Standardized Value
BMP2K BMP2 inducible kinase 1.36211
SLK STE20-like kinase 1.35325
RIOK3 RIO kinase 3 1.35325
AURKA aurora kinase A 1.32726
ADCK4 aarF domain containing kinase 4 1.32726
FLT3 fms-related tyrosine kinase 3 1.3104
AURKC aurora kinase C 1.26991
TNK1 tyrosine kinase, non-receptor, 1 1.26209
ULK3 unc-51 like kinase 3 1.24671
PIP4K2B phosphatidylinositol-5-phosphate 4-kinase, type II, beta 1.23916
STK16 serine/threonine kinase 16 1.23916
IRAK3 interleukin-1 receptor-associated kinase 3 1.22432
RET ret proto-oncogene 1.22432
SRPK1 SRSF protein kinase 1 1.21703
MERTK MER proto-oncogene, tyrosine kinase 1.20983
STK36 serine/threonine kinase 36 1.20271
AXL AXL receptor tyrosine kinase 1.20271
ACVR2A activin A receptor, type IIA 1.19568
TXK TXK tyrosine kinase 1.19568
HIPK4 homeodomain interacting protein kinase 4 1.18186
NEK7 NIMA-related kinase 7 1.16838
STK17A serine/threonine kinase 17a 1.16838
ZAK sterile alpha motif and leucine zipper containing kinase AZK 1.14877
HIPK1 homeodomain interacting protein kinase 1 1.12988
BMPR1B bone morphogenetic protein receptor, type IB 1.12373
DAPK1 death-associated protein kinase 1 1.09415
MAP3K11 mitogen-activated protein kinase kinase kinase 11 1.05057
CLK2 CDC-like kinase 2 1.03535
HIPK2 homeodomain interacting protein kinase 2 1.03041
DAPK3 death-associated protein kinase 3 1.02071
CAMK1D calcium/calmodulin-dependent protein kinase ID 1.00208
MKNK2 MAP kinase interacting serine/threonine kinase 2 1.00208
TBK1 TANK-binding kinase 1 1.00208
GAK cyclin G associated kinase 0.997567
CSF1R colony stimulating factor 1 receptor 0.963557
LCK LCK proto-oncogene, Src family tyrosine kinase 0.959553
AAK1 AP2 associated kinase 1 0.944052
MAP3K10 mitogen-activated protein kinase kinase kinase 10 0.936602
FLT4 fms-related tyrosine kinase 4 0.922275
SRPK3 SRSF protein kinase 3 0.915387
CSNK2A2 casein kinase 2, alpha prime polypeptide 0.915387
NEK5 NIMA-related kinase 5 0.91201
NEK6 NIMA-related kinase 6 0.895762
MET MET proto-oncogene, receptor tyrosine kinase 0.889549
GRK4 G protein-coupled receptor kinase 4 0.883492
LIMK1 LIM domain kinase 1 0.855378
TIE1 tyrosine kinase with immunoglobulin-like and EGF-like domains 1 0.850157
TNK2 tyrosine kinase, non-receptor, 2 0.850157