MG-262-7068 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the MG-262-7068 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADM adrenomedullin
ALDH2 aldehyde dehydrogenase 2 family (mitochondrial)
ALOXE3 arachidonate lipoxygenase 3
ARG2 arginase 2
ASNS asparagine synthetase (glutamine-hydrolyzing)
ATF3 activating transcription factor 3
BAG3 BCL2-associated athanogene 3
BID BH3 interacting domain death agonist
CASP7 caspase 7, apoptosis-related cysteine peptidase
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CHRNA5 cholinergic receptor, nicotinic, alpha 5 (neuronal)
CLK1 CDC-like kinase 1
CLU clusterin
CRYAB crystallin, alpha B
CSRP2 cysteine and glycine-rich protein 2
CTGF connective tissue growth factor
CXCL8 chemokine (C-X-C motif) ligand 8
CXCR4 chemokine (C-X-C motif) receptor 4
CYP39A1 cytochrome P450, family 39, subfamily A, polypeptide 1
DDIT3 DNA-damage-inducible transcript 3
DDIT4 DNA-damage-inducible transcript 4
DMRT1 doublesex and mab-3 related transcription factor 1
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
DST dystonin
DUSP1 dual specificity phosphatase 1
DUSP2 dual specificity phosphatase 2
FKBP4 FK506 binding protein 4, 59kDa
FOS FBJ murine osteosarcoma viral oncogene homolog
GABARAPL1 GABA(A) receptor-associated protein like 1
GADD45B growth arrest and DNA-damage-inducible, beta
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMGCS1 3-hydroxy-3-methylglutaryl-CoA synthase 1 (soluble)
HMOX1 heme oxygenase 1
HSPA1A heat shock 70kDa protein 1A
HSPA4 heat shock 70kDa protein 4
HSPA4L heat shock 70kDa protein 4-like
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPB1 heat shock 27kDa protein 1
HSPB8 heat shock 22kDa protein 8
HSPH1 heat shock 105kDa/110kDa protein 1
ICAM1 intercellular adhesion molecule 1
IER5 immediate early response 5
IL11 interleukin 11
IL17RB interleukin 17 receptor B
IL33R interleukin 33 receptor
IL7R interleukin 7 receptor
JUN jun proto-oncogene
KDM7A lysine (K)-specific demethylase 7A
KRT6A keratin 6A, type II
KRT6B keratin 6B, type II
LGSN lengsin, lens protein with glutamine synthetase domain
LIPG lipase, endothelial
MARS methionyl-tRNA synthetase
MBOAT7 membrane bound O-acyltransferase domain containing 7
MERTK MER proto-oncogene, tyrosine kinase
MICB MHC class I polypeptide-related sequence B
MLF1 myeloid leukemia factor 1
MRPL18 mitochondrial ribosomal protein L18
MSX1 msh homeobox 1
NEAT1 nuclear paraspeckle assembly transcript 1 (non-protein coding)
NKIRAS2 NFKB inhibitor interacting Ras-like 2
OSBPL3 oxysterol binding protein-like 3
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PGF placental growth factor
PLOD2 procollagen-lysine, 2-oxoglutarate 5-dioxygenase 2
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
PPARD peroxisome proliferator-activated receptor delta
PPP1R15A protein phosphatase 1, regulatory subunit 15A
PUS3 pseudouridylate synthase 3
RAI2 retinoic acid induced 2
RANGAP1 Ran GTPase activating protein 1
RFPL2 ret finger protein-like 2
RND1 Rho family GTPase 1
RNF6 ring finger protein (C3H2C3 type) 6
RUNX3 runt-related transcription factor 3
SAT1 spermidine/spermine N1-acetyltransferase 1
SCD stearoyl-CoA desaturase (delta-9-desaturase)
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SLC12A7 solute carrier family 12 (potassium/chloride transporter), member 7
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC3A2 solute carrier family 3 (amino acid transporter heavy chain), member 2
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SLC7A5 solute carrier family 7 (amino acid transporter light chain, L system), member 5
SQSTM1 sequestosome 1
STC2 stanniocalcin 2
TMEM2 transmembrane protein 2
TMEM97 transmembrane protein 97
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TRIM26 tripartite motif containing 26
TSPYL2 TSPY-like 2
UBB ubiquitin B
UBE2D1 ubiquitin-conjugating enzyme E2D 1
ULBP2 UL16 binding protein 2
USPL1 ubiquitin specific peptidase like 1
ZFYVE9 zinc finger, FYVE domain containing 9

decreased expression

Symbol Name
ABI3BP ABI family, member 3 (NESH) binding protein
ACTR3B ARP3 actin-related protein 3 homolog B (yeast)
ASTE1 asteroid homolog 1 (Drosophila)
BCAR3 breast cancer anti-estrogen resistance 3
BHLHE41 basic helix-loop-helix family, member e41
BNC2 basonuclin 2
C11ORF68 chromosome 11 open reading frame 68
C11ORF71 chromosome 11 open reading frame 71
C2CD2 C2 calcium-dependent domain containing 2
CBX7 chromobox homolog 7
CHST2 carbohydrate (N-acetylglucosamine-6-O) sulfotransferase 2
CLDN4 claudin 4
CTDSP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) small phosphatase 1
CXADR coxsackie virus and adenovirus receptor
DEAF1 DEAF1 transcription factor
DUSP4 dual specificity phosphatase 4
ERN2 endoplasmic reticulum to nucleus signaling 2
ESRP2 epithelial splicing regulatory protein 2
FAM105A family with sequence similarity 105, member A
FAM86B1 family with sequence similarity 86, member B1
FBXO5 F-box protein 5
FJX1 four jointed box 1 (Drosophila)
FOSL1 FOS-like antigen 1
FPGT fucose-1-phosphate guanylyltransferase
FZD8 frizzled class receptor 8
GALNT11 polypeptide N-acetylgalactosaminyltransferase 11
GNB1L guanine nucleotide binding protein (G protein), beta polypeptide 1-like
GRPR gastrin-releasing peptide receptor
GUCY1A3 guanylate cyclase 1, soluble, alpha 3
H1F0 H1 histone family, member 0
H1FX H1 histone family, member X
HAS2 hyaluronan synthase 2
HIST1H2AC histone cluster 1, H2ac
HK2 hexokinase 2
HMGA2 high mobility group AT-hook 2
HOXA10 homeobox A10
HOXA5 homeobox A5
HOXB13 homeobox B13
HPS6 Hermansky-Pudlak syndrome 6
IL33 interleukin 33
IMP3 IMP3, U3 small nucleolar ribonucleoprotein
INHBB inhibin, beta B
IRS1 insulin receptor substrate 1
KIF20A kinesin family member 20A
KIFC1 kinesin family member C1
KLF10 Kruppel-like factor 10
KRT15 keratin 15, type I
LIF leukemia inhibitory factor
LOC730101 uncharacterized LOC730101
LPAR6 lysophosphatidic acid receptor 6
MALL mal, T-cell differentiation protein-like
MCM3AP-AS1 MCM3AP antisense RNA 1
MNT MAX network transcriptional repressor
MOGS mannosyl-oligosaccharide glucosidase
MSL1 male-specific lethal 1 homolog (Drosophila)
NREP neuronal regeneration related protein
OSGEPL1 O-sialoglycoprotein endopeptidase-like 1
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
P3H4 prolyl 3-hydroxylase family member 4 (non-enzymatic)
PACSIN3 protein kinase C and casein kinase substrate in neurons 3
PALMD palmdelphin
PCYOX1L prenylcysteine oxidase 1 like
PEX11B peroxisomal biogenesis factor 11 beta
PHLDA1 pleckstrin homology-like domain, family A, member 1
PLAU plasminogen activator, urokinase
PLK1 polo-like kinase 1
PPAP2B phosphatidic acid phosphatase type 2B
PPM1H protein phosphatase, Mg2+/Mn2+ dependent, 1H
PRMT7 protein arginine methyltransferase 7
PSRC1 proline/serine-rich coiled-coil 1
PTGFR prostaglandin F receptor (FP)
PTK6 protein tyrosine kinase 6
PTX3 pentraxin 3, long
RANBP6 RAN binding protein 6
RHOBTB1 Rho-related BTB domain containing 1
RIN2 Ras and Rab interactor 2
RSAD1 radical S-adenosyl methionine domain containing 1
SAC3D1 SAC3 domain containing 1
SCO2 SCO2 cytochrome c oxidase assembly protein
SHROOM2 shroom family member 2
SOX9 SRY (sex determining region Y)-box 9
SPATA2L spermatogenesis associated 2-like
SPRY1 sprouty homolog 1, antagonist of FGF signaling (Drosophila)
SPRY2 sprouty homolog 2 (Drosophila)
ST3GAL1 ST3 beta-galactoside alpha-2,3-sialyltransferase 1
TENM4 teneurin transmembrane protein 4
TMEM187 transmembrane protein 187
TNRC6B trinucleotide repeat containing 6B
TNS3 tensin 3
TOP2A topoisomerase (DNA) II alpha 170kDa
TRIB2 tribbles pseudokinase 2
TRIOBP TRIO and F-actin binding protein
TSPAN15 tetraspanin 15
TUBGCP5 tubulin, gamma complex associated protein 5
ZBED8 zinc finger, BED-type containing 8
ZMYM3 zinc finger, MYM-type 3
ZNF248 zinc finger protein 248
ZNF302 zinc finger protein 302
ZNF33B zinc finger protein 33B
ZNF623 zinc finger protein 623