PNU-0230031-4291 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the PNU-0230031-4291 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACAN aggrecan
ACVR1B activin A receptor, type IB
ADAP1 ArfGAP with dual PH domains 1
AKAP8L A kinase (PRKA) anchor protein 8-like
ANGPTL2 angiopoietin-like 2
ARHGEF17 Rho guanine nucleotide exchange factor (GEF) 17
ARID4B AT rich interactive domain 4B (RBP1-like)
ASTN1 astrotactin 1
ATP6AP2 ATPase, H+ transporting, lysosomal accessory protein 2
ATXN7L3B ataxin 7-like 3B
BAGE B melanoma antigen
C14ORF93 chromosome 14 open reading frame 93
CASP2 caspase 2, apoptosis-related cysteine peptidase
CEACAM3 carcinoembryonic antigen-related cell adhesion molecule 3
CHST5 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 5
CLDN8 claudin 8
CSF1R colony stimulating factor 1 receptor
CTNNA3 catenin (cadherin-associated protein), alpha 3
CTNND2 catenin (cadherin-associated protein), delta 2
CTNS cystinosin, lysosomal cystine transporter
CYP2C19 cytochrome P450, family 2, subfamily C, polypeptide 19
CYP4F2 cytochrome P450, family 4, subfamily F, polypeptide 2
DEFA4 defensin, alpha 4, corticostatin
DKFZP434C153 DKFZP434C153 protein
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha
DSC2 desmocollin 2
EDN1 endothelin 1
EPHA5 EPH receptor A5
EPN1 epsin 1
ERN2 endoplasmic reticulum to nucleus signaling 2
ERP44 endoplasmic reticulum protein 44
FUT6 fucosyltransferase 6 (alpha (1,3) fucosyltransferase)
GPR22 G protein-coupled receptor 22
GTF2A1 general transcription factor IIA, 1, 19/37kDa
HIPK2 homeodomain interacting protein kinase 2
HIST1H1E histone cluster 1, H1e
HIST1H4C histone cluster 1, H4c
HNRNPU heterogeneous nuclear ribonucleoprotein U (scaffold attachment factor A)
HNRNPUL2 heterogeneous nuclear ribonucleoprotein U-like 2
HOOK1 hook microtubule-tethering protein 1
HOXB7 homeobox B7
HRG histidine-rich glycoprotein
HRH4 histamine receptor H4
IL1RN interleukin 1 receptor antagonist
KAT6A K(lysine) acetyltransferase 6A
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KIAA0100 KIAA0100
KMT2A lysine (K)-specific methyltransferase 2A
LARP4B La ribonucleoprotein domain family, member 4B
LPP LIM domain containing preferred translocation partner in lipoma
LRP2BP LRP2 binding protein
LRRC48 leucine rich repeat containing 48
MBNL2 muscleblind-like splicing regulator 2
MDM4 MDM4, p53 regulator
MET MET proto-oncogene, receptor tyrosine kinase
NKTR natural killer cell triggering receptor
NPY4R neuropeptide Y receptor Y4
NTF3 neurotrophin 3
OR1D2 olfactory receptor, family 1, subfamily D, member 2
PDE2A phosphodiesterase 2A, cGMP-stimulated
PHEX phosphate regulating endopeptidase homolog, X-linked
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PKNOX2 PBX/knotted 1 homeobox 2
PKP3 plakophilin 3
PKP4 plakophilin 4
PLAA phospholipase A2-activating protein
PPARA peroxisome proliferator-activated receptor alpha
PRDM1 PR domain containing 1, with ZNF domain
PRELP proline/arginine-rich end leucine-rich repeat protein
PRKAB2 protein kinase, AMP-activated, beta 2 non-catalytic subunit
PRKCE protein kinase C, epsilon
PRR14L proline rich 14-like
PVT1 Pvt1 oncogene (non-protein coding)
RAP1GAP RAP1 GTPase activating protein
RDH16 retinol dehydrogenase 16 (all-trans)
RIMS3 regulating synaptic membrane exocytosis 3
RNGTT RNA guanylyltransferase and 5'-phosphatase
RUNDC3B RUN domain containing 3B
SCD stearoyl-CoA desaturase (delta-9-desaturase)
SLC15A1 solute carrier family 15 (oligopeptide transporter), member 1
SLC16A6 solute carrier family 16, member 6
SLC9A7 solute carrier family 9, subfamily A (NHE7, cation proton antiporter 7), member 7
SNCA synuclein, alpha (non A4 component of amyloid precursor)
SSX3 synovial sarcoma, X breakpoint 3
SUGP1 SURP and G patch domain containing 1
TAOK2 TAO kinase 2
TBC1D30 TBC1 domain family, member 30
TBL1Y transducin (beta)-like 1, Y-linked
TBRG4 transforming growth factor beta regulator 4
TEAD1 TEA domain family member 1 (SV40 transcriptional enhancer factor)
TFF3 trefoil factor 3 (intestinal)
THEMIS2 thymocyte selection associated family member 2
THTPA thiamine triphosphatase
VCL vinculin
WIZ widely interspaced zinc finger motifs
ZBTB33 zinc finger and BTB domain containing 33
ZDHHC17 zinc finger, DHHC-type containing 17
ZNF749 zinc finger protein 749

decreased expression

Symbol Name
ABHD4 abhydrolase domain containing 4
ACSS3 acyl-CoA synthetase short-chain family member 3
ALOX12P2 arachidonate 12-lipoxygenase pseudogene 2
ARHGEF16 Rho guanine nucleotide exchange factor (GEF) 16
ARMC4 armadillo repeat containing 4
ARMCX2 armadillo repeat containing, X-linked 2
ASIC3 acid sensing (proton gated) ion channel 3
AURKC aurora kinase C
C14ORF79 chromosome 14 open reading frame 79
CBL Cbl proto-oncogene, E3 ubiquitin protein ligase
CBX4 chromobox homolog 4
CBX8 chromobox homolog 8
CDKL3 cyclin-dependent kinase-like 3
CEP170B centrosomal protein 170B
CES3 carboxylesterase 3
CHRNA9 cholinergic receptor, nicotinic, alpha 9 (neuronal)
CINP cyclin-dependent kinase 2 interacting protein
CLDN1 claudin 1
CLEC16A C-type lectin domain family 16, member A
CORO1A coronin, actin binding protein, 1A
CRELD1 cysteine-rich with EGF-like domains 1
DHX57 DEAH (Asp-Glu-Ala-Asp/His) box polypeptide 57
DMBT1 deleted in malignant brain tumors 1
DNAJB2 DnaJ (Hsp40) homolog, subfamily B, member 2
EGLN3 egl-9 family hypoxia-inducible factor 3
ELP6 elongator acetyltransferase complex subunit 6
ENTPD5 ectonucleoside triphosphate diphosphohydrolase 5
FAM131B family with sequence similarity 131, member B
FGF23 fibroblast growth factor 23
GALNT14 polypeptide N-acetylgalactosaminyltransferase 14
GLS2 glutaminase 2 (liver, mitochondrial)
GMPR guanosine monophosphate reductase
GPR182 G protein-coupled receptor 182
GRINA glutamate receptor, ionotropic, N-methyl D-aspartate-associated protein 1 (glutamate binding)
HDAC7 histone deacetylase 7
HIST1H2AJ histone cluster 1, H2aj
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
HOXC13 homeobox C13
HYAL3 hyaluronoglucosaminidase 3
IRAK4 interleukin-1 receptor-associated kinase 4
JUNB jun B proto-oncogene
KDM8 lysine (K)-specific demethylase 8
KIAA1107 KIAA1107
KLHL25 kelch-like family member 25
KLHL36 kelch-like family member 36
KLRG1 killer cell lectin-like receptor subfamily G, member 1
LOC390998 ribosomal protein L10 pseudogene
LPAR6 lysophosphatidic acid receptor 6
LRP5 low density lipoprotein receptor-related protein 5
LRRC15 leucine rich repeat containing 15
LRRC61 leucine rich repeat containing 61
LRRK1 leucine-rich repeat kinase 1
LYPD3 LY6/PLAUR domain containing 3
MFGE8 milk fat globule-EGF factor 8 protein
MUC3B mucin 3B, cell surface associated
NABP2 nucleic acid binding protein 2
NXPH3 neurexophilin 3
OR2B6 olfactory receptor, family 2, subfamily B, member 6
OR3A3 olfactory receptor, family 3, subfamily A, member 3
PADI1 peptidyl arginine deiminase, type I
PALM paralemmin
PIM1 Pim-1 proto-oncogene, serine/threonine kinase
PLXNB3 plexin B3
PMPCA peptidase (mitochondrial processing) alpha
PODNL1 podocan-like 1
POLL polymerase (DNA directed), lambda
PREX2 phosphatidylinositol-3,4,5-trisphosphate-dependent Rac exchange factor 2
PRSS8 protease, serine, 8
PTPRS protein tyrosine phosphatase, receptor type, S
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RABL6 RAB, member RAS oncogene family-like 6
RUSC2 RUN and SH3 domain containing 2
SAMSN1 SAM domain, SH3 domain and nuclear localization signals 1
SCGB2A2 secretoglobin, family 2A, member 2
SCN1B sodium channel, voltage gated, type I beta subunit
SEC61A2 Sec61 alpha 2 subunit (S. cerevisiae)
SENP7 SUMO1/sentrin specific peptidase 7
SESN1 sestrin 1
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SLC12A8 solute carrier family 12, member 8
SMPD2 sphingomyelin phosphodiesterase 2, neutral membrane (neutral sphingomyelinase)
SOX21 SRY (sex determining region Y)-box 21
STAC SH3 and cysteine rich domain
STARD5 StAR-related lipid transfer (START) domain containing 5
TAF4B TAF4b RNA polymerase II, TATA box binding protein (TBP)-associated factor, 105kDa
TCEAL2 transcription elongation factor A (SII)-like 2
TENM1 teneurin transmembrane protein 1
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
TLN1 talin 1
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TNS2 tensin 2
TOR4A torsin family 4, member A
TSC22D4 TSC22 domain family, member 4
TUBA4B tubulin, alpha 4b
UNC119 unc-119 homolog (C. elegans)
URM1 ubiquitin related modifier 1
USP20 ubiquitin specific peptidase 20
WDR25 WD repeat domain 25
XAB2 XPA binding protein 2
ZYX zyxin