Pasireotide (acetate)_J82 Gene Set

Dataset Tahoe Therapeutics Tahoe 100M Perturbation Atlas
Category transcriptomics
Type cell type
Description Pasireotide (acetate) perturbation in J82 cell line (Tahoe Therapeutics)
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Genes

200 genes differentially expressed following the Pasireotide (acetate)_J82 drug perturbation from the Tahoe Therapeutics Tahoe 100M Perturbation Atlas dataset.

increased expression

Symbol Name Standardized Value
MYH9 myosin, heavy chain 9, non-muscle 0.137957
MT2A metallothionein 2A 0.106578
IGFBP3 insulin-like growth factor binding protein 3 0.0988964
AKAP12 A kinase (PRKA) anchor protein 12 0.0978836
INTS6 integrator complex subunit 6 0.096957
ERBIN erbb2 interacting protein 0.0924249
DST dystonin 0.0885537
NAV2 neuron navigator 2 0.0874262
ASPH aspartate beta-hydroxylase 0.0866691
AHNAK AHNAK nucleoprotein 0.083568
PLOD2 procollagen-lysine, 2-oxoglutarate 5-dioxygenase 2 0.0827694
SERPINE1 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 1 0.0806736
RPS6 ribosomal protein S6 0.0787091
NEDD4L neural precursor cell expressed, developmentally down-regulated 4-like, E3 ubiquitin protein ligase 0.0727446
HNRNPA2B1 heterogeneous nuclear ribonucleoprotein A2/B1 0.0630513
ZSWIM6 zinc finger, SWIM-type containing 6 0.0603722
UACA uveal autoantigen with coiled-coil domains and ankyrin repeats 0.0587226
MKI67 marker of proliferation Ki-67 0.058188
PICALM phosphatidylinositol binding clathrin assembly protein 0.058027
MSN moesin 0.0538957
KTN1 kinectin 1 (kinesin receptor) 0.0510838
ANKRD11 ankyrin repeat domain 11 0.0507156
ASAP1 ArfGAP with SH3 domain, ankyrin repeat and PH domain 1 0.0506482
MACF1 microtubule-actin crosslinking factor 1 0.0497436
GLS2 glutaminase 2 (liver, mitochondrial) 0.0475713
HIVEP2 human immunodeficiency virus type I enhancer binding protein 2 0.0455292
SMURF2 SMAD specific E3 ubiquitin protein ligase 2 0.0454439
GOLGA4 golgin A4 0.0437518
CENPF centromere protein F, 350/400kDa 0.0433588
TPM3 tropomyosin 3 0.0428701
TLE4 transducin-like enhancer of split 4 0.0428483
YBX1 Y box binding protein 1 0.0428118
PALM2AKAP2 PALM2 and AKAP2 fusion 0.0415329
PPP1R15A protein phosphatase 1, regulatory subunit 15A 0.0408377
TMSB10 thymosin beta 10 0.0405285
NPM1 nucleophosmin (nucleolar phosphoprotein B23, numatrin) 0.0399655
SPTAN1 spectrin, alpha, non-erythrocytic 1 0.0395358
FNIP1 folliculin interacting protein 1 0.0395276
ABTB2 ankyrin repeat and BTB (POZ) domain containing 2 0.0385951
CRIM1 cysteine rich transmembrane BMP regulator 1 (chordin-like) 0.0381432
TRIO trio Rho guanine nucleotide exchange factor 0.0369334
BASP1 brain abundant, membrane attached signal protein 1 0.0369196
PRELID2 PRELI domain containing 2 0.0362773
GOLGB1 golgin B1 0.0361152
SLIT2 slit homolog 2 (Drosophila) 0.0354578
CORO1C coronin, actin binding protein, 1C 0.03541
PTK2 protein tyrosine kinase 2 0.0350909
NSD2 nuclear receptor binding SET domain protein 2 0.0350556
SPTBN1 spectrin, beta, non-erythrocytic 1 0.035004
APLP2 amyloid beta (A4) precursor-like protein 2 0.0349351
EEF1A1 eukaryotic translation elongation factor 1 alpha 1 0.0347896
HSPH1 heat shock 105kDa/110kDa protein 1 0.0347522
MAP4K4 mitogen-activated protein kinase kinase kinase kinase 4 0.0346981
LPP LIM domain containing preferred translocation partner in lipoma 0.0342202
PDLIM5 PDZ and LIM domain 5 0.0338933
HSP90AA1 heat shock protein 90kDa alpha (cytosolic), class A member 1 0.0337304
DYNC1H1 dynein, cytoplasmic 1, heavy chain 1 0.0337006
VEGFA vascular endothelial growth factor A 0.0336953
PABPC1 poly(A) binding protein, cytoplasmic 1 0.0333882
CTBP2 C-terminal binding protein 2 0.0332085
DOCK5 dedicator of cytokinesis 5 0.0331147
RPLP2 ribosomal protein, large, P2 0.03148
ACTN1 actinin, alpha 1 0.0314713
RPL23 ribosomal protein L23 0.031451
SMYD3 SET and MYND domain containing 3 0.0311846
BRD2 bromodomain containing 2 0.0310157
ATXN1 ataxin 1 0.0309886
AGAP1 ArfGAP with GTPase domain, ankyrin repeat and PH domain 1 0.0308817
SMC4 structural maintenance of chromosomes 4 0.0306617
KPNA4 karyopherin alpha 4 (importin alpha 3) 0.0305995
STC2 stanniocalcin 2 0.0305643
SH3RF1 SH3 domain containing ring finger 1 0.0304768
PRRC2C proline-rich coiled-coil 2C 0.0303856
HERC4 HECT and RLD domain containing E3 ubiquitin protein ligase 4 0.0303303
HNRNPUL2 heterogeneous nuclear ribonucleoprotein U-like 2 0.0301616
LAMC1 laminin, gamma 1 (formerly LAMB2) 0.030145
ASH1L ash1 (absent, small, or homeotic)-like (Drosophila) 0.0301106
NDRG1 N-myc downstream regulated 1 0.0300916
CLIC4 chloride intracellular channel 4 0.0300835
RPL19 ribosomal protein L19 0.0297869
TPX2 TPX2, microtubule-associated 0.0289885
PKM pyruvate kinase, muscle 0.0289146
ATRX alpha thalassemia/mental retardation syndrome X-linked 0.0287988
HSP90AB1 heat shock protein 90kDa alpha (cytosolic), class B member 1 0.0285654
EPB41L2 erythrocyte membrane protein band 4.1-like 2 0.0284814
HSPA8 heat shock 70kDa protein 8 0.0284412
SAMD4A sterile alpha motif domain containing 4A 0.0284119
MT1X metallothionein 1X 0.0280963
PPP6R3 protein phosphatase 6, regulatory subunit 3 0.0280585
DIAPH3 diaphanous-related formin 3 0.0280317
UBE2E2 ubiquitin-conjugating enzyme E2E 2 0.0277504
RPL35A ribosomal protein L35a 0.0277158
MAP4 microtubule-associated protein 4 0.0271828
MBNL1 muscleblind-like splicing regulator 1 0.0270542
RALY RALY heterogeneous nuclear ribonucleoprotein 0.0269478
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase 0.0267435
GBE1 glucan (1,4-alpha-), branching enzyme 1 0.0266256
WNT5B wingless-type MMTV integration site family, member 5B 0.0265796
CALD1 caldesmon 1 0.0265105
AFF1 AF4/FMR2 family, member 1 0.0263856

decreased expression

Symbol Name Standardized Value
CD44 CD44 molecule (Indian blood group) -0.0781774
NAMPT nicotinamide phosphoribosyltransferase -0.0746193
SLC12A8 solute carrier family 12, member 8 -0.0738863
F3 coagulation factor III (thromboplastin, tissue factor) -0.064413
ABI3BP ABI family, member 3 (NESH) binding protein -0.0587589
FN1 fibronectin 1 -0.0555247
CXCL8 chemokine (C-X-C motif) ligand 8 -0.0471176
HLA-B major histocompatibility complex, class I, B -0.0453657
GLIS3 GLIS family zinc finger 3 -0.0409015
NFKBIZ nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, zeta -0.0403607
FTH1 ferritin, heavy polypeptide 1 -0.0382108
LOC112694756 uncharaterized LOC112694756 -0.03301
PHLDB2 pleckstrin homology-like domain, family B, member 2 -0.0323316
OSMR oncostatin M receptor -0.0319835
TNFAIP3 tumor necrosis factor, alpha-induced protein 3 -0.0311103
POSTN periostin, osteoblast specific factor -0.0299324
ATP13A3 ATPase type 13A3 -0.0294202
NALF1 NALCN channel auxiliary factor 1 -0.0292489
TUBB tubulin, beta class I -0.028164
VDAC1 voltage-dependent anion channel 1 -0.0273902
HEG1 heart development protein with EGF-like domains 1 -0.0264033
CTSD cathepsin D -0.0258946
TMSB4X thymosin beta 4, X-linked -0.0257987
IGFBP5 insulin-like growth factor binding protein 5 -0.0252904
TXNRD1 thioredoxin reductase 1 -0.0248631
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) -0.0245182
RBMS3 RNA binding motif, single stranded interacting protein 3 -0.0239623
SCD stearoyl-CoA desaturase (delta-9-desaturase) -0.0238675
ADM adrenomedullin -0.0236252
ARF4 ADP-ribosylation factor 4 -0.0232958
BZW1 basic leucine zipper and W2 domains 1 -0.0219298
SOD2 superoxide dismutase 2, mitochondrial -0.0215918
TUBA1C tubulin, alpha 1c -0.0209929
KPNB1 karyopherin (importin) beta 1 -0.020392
SLC25A36 solute carrier family 25 (pyrimidine nucleotide carrier), member 36 -0.0202378
KLF7 Kruppel-like factor 7 (ubiquitous) -0.0201112
GAPDH glyceraldehyde-3-phosphate dehydrogenase -0.0198091
S100A6 S100 calcium binding protein A6 -0.019445
SULF1 sulfatase 1 -0.0193478
RHOBTB3 Rho-related BTB domain containing 3 -0.0193438
TUBA1B tubulin, alpha 1b -0.0189908
ANXA1 annexin A1 -0.0188961
HLA-C major histocompatibility complex, class I, C -0.018838
ARFGEF2 ADP-ribosylation factor guanine nucleotide-exchange factor 2 (brefeldin A-inhibited) -0.0183842
LOX lysyl oxidase -0.0181876
LDHA lactate dehydrogenase A -0.018031
NPEPPS aminopeptidase puromycin sensitive -0.0175834
GOLT1B golgi transport 1B -0.0172179
AFAP1 actin filament associated protein 1 -0.0169859
ANKRD28 ankyrin repeat domain 28 -0.0169717
COLEC10 collectin sub-family member 10 (C-type lectin) -0.01654
WDR45B WD repeat domain 45B -0.0164906
TANC2 tetratricopeptide repeat, ankyrin repeat and coiled-coil containing 2 -0.0163377
FSTL1 follistatin-like 1 -0.0163296
FTL ferritin, light polypeptide -0.0161274
TMEM41B transmembrane protein 41B -0.0160689
TFPI tissue factor pathway inhibitor (lipoprotein-associated coagulation inhibitor) -0.0159418
RNF144B ring finger protein 144B -0.0159351
ERO1A endoplasmic reticulum oxidoreductase 1 alpha -0.0158015
HLA-E major histocompatibility complex, class I, E -0.0157367
LMAN1 lectin, mannose-binding, 1 -0.01562
ARF1 ADP-ribosylation factor 1 -0.0155454
DPYD dihydropyrimidine dehydrogenase -0.0151952
OLR1 oxidized low density lipoprotein (lectin-like) receptor 1 -0.0148185
SEPTIN7 septin 7 -0.0147696
UBA6 ubiquitin-like modifier activating enzyme 6 -0.0146003
CAPZA1 capping protein (actin filament) muscle Z-line, alpha 1 -0.0141709
ZEB2 zinc finger E-box binding homeobox 2 -0.0141614
B4GALT5 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 5 -0.014042
PJA2 praja ring finger 2, E3 ubiquitin protein ligase -0.0140322
IER3 immediate early response 3 -0.0139791
TMEM178B transmembrane protein 178B -0.0138913
HIF1A hypoxia inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) -0.0138575
PLIN2 perilipin 2 -0.0137023
CSE1L CSE1 chromosome segregation 1-like (yeast) -0.0132923
PPME1 protein phosphatase methylesterase 1 -0.0132072
ANAPC5 anaphase promoting complex subunit 5 -0.0131915
LAMP1 lysosomal-associated membrane protein 1 -0.0131878
SLC9A8 solute carrier family 9, subfamily A (NHE8, cation proton antiporter 8), member 8 -0.0130802
CMPK1 cytidine monophosphate (UMP-CMP) kinase 1, cytosolic -0.0130135
DLG1 discs, large homolog 1 (Drosophila) -0.0127995
IL1RAP interleukin 1 receptor accessory protein -0.0127764
PGK1 phosphoglycerate kinase 1 -0.0127733
SRP54 signal recognition particle 54kDa -0.0127267
PNRC1 proline-rich nuclear receptor coactivator 1 -0.0126682
TRAM2 translocation associated membrane protein 2 -0.0124038
TIMP3 TIMP metallopeptidase inhibitor 3 -0.0124028
POLE3 polymerase (DNA directed), epsilon 3, accessory subunit -0.0123942
GNS glucosamine (N-acetyl)-6-sulfatase -0.0123173
ICAM1 intercellular adhesion molecule 1 -0.0121931
TFG TRK-fused gene -0.0121779
SURF4 surfeit 4 -0.0121356
DAB2 Dab, mitogen-responsive phosphoprotein, homolog 2 (Drosophila) -0.0120378
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1 -0.0120287
NUP155 nucleoporin 155kDa -0.0117387
PSG9 pregnancy specific beta-1-glycoprotein 9 -0.0117134
IRF2BP2 interferon regulatory factor 2 binding protein 2 -0.0115389
SEC24A SEC24 family member A -0.0115295
IL6 interleukin 6 -0.0115168
UFM1 ubiquitin-fold modifier 1 -0.0114668