Prestwick-1085-5774 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the Prestwick-1085-5774 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADAM22 ADAM metallopeptidase domain 22
ADRBK2 adrenergic, beta, receptor kinase 2
ALOX5AP arachidonate 5-lipoxygenase-activating protein
ALPK1 alpha-kinase 1
ARHGEF15 Rho guanine nucleotide exchange factor (GEF) 15
ARTN artemin
ATP6V0A1 ATPase, H+ transporting, lysosomal V0 subunit a1
C1ORF54 chromosome 1 open reading frame 54
C1S complement component 1, s subcomponent
C6 complement component 6
C9ORF9 chromosome 9 open reading frame 9
CD40 CD40 molecule, TNF receptor superfamily member 5
CEACAM7 carcinoembryonic antigen-related cell adhesion molecule 7
CHRNA4 cholinergic receptor, nicotinic, alpha 4 (neuronal)
CHST5 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 5
CLCN7 chloride channel, voltage-sensitive 7
CNR2 cannabinoid receptor 2 (macrophage)
CPB2 carboxypeptidase B2 (plasma)
CPN2 carboxypeptidase N, polypeptide 2
CSDC2 cold shock domain containing C2, RNA binding
DAGLA diacylglycerol lipase, alpha
EDA ectodysplasin A
EPB41L5 erythrocyte membrane protein band 4.1 like 5
FAM63A family with sequence similarity 63, member A
FBXL18 F-box and leucine-rich repeat protein 18
FCAR Fc fragment of IgA receptor
FCN2 ficolin (collagen/fibrinogen domain containing lectin) 2
FGB fibrinogen beta chain
FLT4 fms-related tyrosine kinase 4
FMNL1 formin-like 1
FUT7 fucosyltransferase 7 (alpha (1,3) fucosyltransferase)
GATM glycine amidinotransferase (L-arginine:glycine amidinotransferase)
GFOD2 glucose-fructose oxidoreductase domain containing 2
GNRH2 gonadotropin-releasing hormone 2
GRIK5 glutamate receptor, ionotropic, kainate 5
GUSBP3 glucuronidase, beta pseudogene 3
HECW1 HECT, C2 and WW domain containing E3 ubiquitin protein ligase 1
HGF hepatocyte growth factor (hepapoietin A; scatter factor)
HOMER3 homer scaffolding protein 3
HOXB7 homeobox B7
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
INADL InaD-like (Drosophila)
KCNE4 potassium channel, voltage gated subfamily E regulatory beta subunit 4
KIAA0125 KIAA0125
KIAA0319L KIAA0319-like
KLF4 Kruppel-like factor 4 (gut)
KMT2A lysine (K)-specific methyltransferase 2A
KRT85 keratin 85, type II
LOC647070 uncharacterized LOC647070
MED25 mediator complex subunit 25
MRPS18C mitochondrial ribosomal protein S18C
MS4A1 membrane-spanning 4-domains, subfamily A, member 1
MSI1 musashi RNA-binding protein 1
NFKBIL1 nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor-like 1
NRCAM neuronal cell adhesion molecule
OBSL1 obscurin-like 1
OR7A10 olfactory receptor, family 7, subfamily A, member 10
PAIP2B poly(A) binding protein interacting protein 2B
PCDHB13 protocadherin beta 13
PFKFB4 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 4
PGK2 phosphoglycerate kinase 2
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PKNOX1 PBX/knotted 1 homeobox 1
PLK4 polo-like kinase 4
PML promyelocytic leukemia
PPIAL4A peptidylprolyl isomerase A (cyclophilin A)-like 4A
PRKACA protein kinase, cAMP-dependent, catalytic, alpha
RAB6B RAB6B, member RAS oncogene family
RDX radixin
REPS1 RALBP1 associated Eps domain containing 1
RUNX1T1 runt-related transcription factor 1; translocated to, 1 (cyclin D-related)
S1PR1 sphingosine-1-phosphate receptor 1
SCN11A sodium channel, voltage gated, type XI alpha subunit
SCN1B sodium channel, voltage gated, type I beta subunit
SFTPB surfactant protein B
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC25A21 solute carrier family 25 (mitochondrial oxoadipate carrier), member 21
SLCO4C1 solute carrier organic anion transporter family, member 4C1
SMARCD1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 1
SRCAP Snf2-related CREBBP activator protein
ST18 suppression of tumorigenicity 18, zinc finger
TAGLN3 transgelin 3
TAPBP TAP binding protein (tapasin)
TAS2R4 taste receptor, type 2, member 4
TBX1 T-box 1
TFCP2L1 transcription factor CP2-like 1
TMEM206 transmembrane protein 206
TNFRSF13B tumor necrosis factor receptor superfamily, member 13B
TNIK TRAF2 and NCK interacting kinase
TPM1 tropomyosin 1 (alpha)
TRIM29 tripartite motif containing 29
TRIM31 tripartite motif containing 31
ULBP1 UL16 binding protein 1
USP2 ubiquitin specific peptidase 2
VNN1 vanin 1
VWA5A von Willebrand factor A domain containing 5A
WIZ widely interspaced zinc finger motifs
XIAP X-linked inhibitor of apoptosis, E3 ubiquitin protein ligase

decreased expression

Symbol Name
ADCY6 adenylate cyclase 6
ADTRP androgen-dependent TFPI-regulating protein
APBB3 amyloid beta (A4) precursor protein-binding, family B, member 3
ARHGEF1 Rho guanine nucleotide exchange factor (GEF) 1
ARHGEF28 Rho guanine nucleotide exchange factor (GEF) 28
B3GALT4 UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 4
BCL9 B-cell CLL/lymphoma 9
BEND5 BEN domain containing 5
BET1L Bet1 golgi vesicular membrane trafficking protein-like
C17ORF53 chromosome 17 open reading frame 53
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
C1RL complement component 1, r subcomponent-like
C5ORF45 chromosome 5 open reading frame 45
C7ORF43 chromosome 7 open reading frame 43
CBX4 chromobox homolog 4
CENPJ centromere protein J
CHMP6 charged multivesicular body protein 6
CLCA1 chloride channel accessory 1
CLUHP3 clustered mitochondria (cluA/CLU1) homolog pseudogene 3
CNIH3 cornichon family AMPA receptor auxiliary protein 3
COBL cordon-bleu WH2 repeat protein
CUL9 cullin 9
DCAF4 DDB1 and CUL4 associated factor 4
DNAJC28 DnaJ (Hsp40) homolog, subfamily C, member 28
DNAL4 dynein, axonemal, light chain 4
ELOVL4 ELOVL fatty acid elongase 4
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM120C family with sequence similarity 120C
FAM184A family with sequence similarity 184, member A
FAM86C1 family with sequence similarity 86, member C1
FAT4 FAT atypical cadherin 4
FBRS fibrosin
FKBP10 FK506 binding protein 10, 65 kDa
FLVCR2 feline leukemia virus subgroup C cellular receptor family, member 2
GABBR1 gamma-aminobutyric acid (GABA) B receptor, 1
GALNT14 polypeptide N-acetylgalactosaminyltransferase 14
GALT galactose-1-phosphate uridylyltransferase
GAN gigaxonin
GIT1 G protein-coupled receptor kinase interacting ArfGAP 1
GMEB1 glucocorticoid modulatory element binding protein 1
GNG4 guanine nucleotide binding protein (G protein), gamma 4
GPR19 G protein-coupled receptor 19
GRAMD4 GRAM domain containing 4
HIST1H1D histone cluster 1, H1d
HIST1H2BJ histone cluster 1, H2bj
HIST1H3C histone cluster 1, H3c
HOXC10 homeobox C10
IL2 interleukin 2
INO80D INO80 complex subunit D
ITK IL2-inducible T-cell kinase
JAM3 junctional adhesion molecule 3
KDM4D lysine (K)-specific demethylase 4D
KRT9 keratin 9, type I
LINS lines homolog (Drosophila)
LSM14B LSM14B, SCD6 homolog B (S. cerevisiae)
MAST3 microtubule associated serine/threonine kinase 3
MDFI MyoD family inhibitor
MXRA8 matrix-remodelling associated 8
MYL5 myosin, light chain 5, regulatory
NARFL nuclear prelamin A recognition factor-like
NBEAL2 neurobeachin-like 2
NKX3-2 NK3 homeobox 2
NT5M 5',3'-nucleotidase, mitochondrial
PHKG2 phosphorylase kinase, gamma 2 (testis)
PLEKHO1 pleckstrin homology domain containing, family O member 1
PLSCR4 phospholipid scramblase 4
PLXNB3 plexin B3
PTPRH protein tyrosine phosphatase, receptor type, H
RAB3A RAB3A, member RAS oncogene family
RGCC regulator of cell cycle
RHOBTB2 Rho-related BTB domain containing 2
RNF126P1 ring finger protein 126 pseudogene 1
RPL23AP32 ribosomal protein L23a pseudogene 32
RRNAD1 ribosomal RNA adenine dimethylase domain containing 1
RUFY2 RUN and FYVE domain containing 2
SARS2 seryl-tRNA synthetase 2, mitochondrial
SLC25A10 solute carrier family 25 (mitochondrial carrier; dicarboxylate transporter), member 10
SLC4A8 solute carrier family 4, sodium bicarbonate cotransporter, member 8
SPEG SPEG complex locus
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2
TBP TATA box binding protein
TCTN2 tectonic family member 2
TEAD3 TEA domain family member 3
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
TRIM25 tripartite motif containing 25
TRIM66 tripartite motif containing 66
TSC22D4 TSC22 domain family, member 4
TTLL7 tubulin tyrosine ligase-like family member 7
TUBA4B tubulin, alpha 4b
WDR33 WD repeat domain 33
WNT10B wingless-type MMTV integration site family, member 10B
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZNF211 zinc finger protein 211
ZNF286A zinc finger protein 286A
ZNF358 zinc finger protein 358
ZNF480 zinc finger protein 480
ZNF76 zinc finger protein 76
ZNF768 zinc finger protein 768