Prestwick-642-2160 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the Prestwick-642-2160 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABLIM1 actin binding LIM protein 1
ACTA2 actin, alpha 2, smooth muscle, aorta
AKAP7 A kinase (PRKA) anchor protein 7
ALDH1L1 aldehyde dehydrogenase 1 family, member L1
ALS2CL ALS2 C-terminal like
APAF1 apoptotic peptidase activating factor 1
APP amyloid beta (A4) precursor protein
AQP1 aquaporin 1 (Colton blood group)
ARHGAP35 Rho GTPase activating protein 35
ATF7 activating transcription factor 7
ATP9B ATPase, class II, type 9B
AURKA aurora kinase A
BTN3A1 butyrophilin, subfamily 3, member A1
C1ORF68 chromosome 1 open reading frame 68
C7ORF69 chromosome 7 open reading frame 69
CACNA1I calcium channel, voltage-dependent, T type, alpha 1I subunit
CALML3 calmodulin-like 3
CAMK4 calcium/calmodulin-dependent protein kinase IV
CAMKK2 calcium/calmodulin-dependent protein kinase kinase 2, beta
CASZ1 castor zinc finger 1
CCNK cyclin K
CD93 CD93 molecule
CDRT1 CMT1A duplicated region transcript 1
CHRM3 cholinergic receptor, muscarinic 3
CLCN7 chloride channel, voltage-sensitive 7
COL19A1 collagen, type XIX, alpha 1
COL6A1 collagen, type VI, alpha 1
COPG2IT1 COPG2 imprinted transcript 1 (non-protein coding)
CROT carnitine O-octanoyltransferase
DHRS7 dehydrogenase/reductase (SDR family) member 7
DOCK6 dedicator of cytokinesis 6
DSCAM Down syndrome cell adhesion molecule
EFNA4 ephrin-A4
ERAP1 endoplasmic reticulum aminopeptidase 1
F5 coagulation factor V (proaccelerin, labile factor)
FER1L4 fer-1-like family member 4, pseudogene (functional)
FOXG1 forkhead box G1
FTCD formimidoyltransferase cyclodeaminase
GALC galactosylceramidase
GFOD2 glucose-fructose oxidoreductase domain containing 2
HSD11B1 hydroxysteroid (11-beta) dehydrogenase 1
IGHG1 immunoglobulin heavy constant gamma 1 (G1m marker)
IL6ST interleukin 6 signal transducer
IRX4 iroquois homeobox 4
ITPK1 inositol-tetrakisphosphate 1-kinase
KCTD2 potassium channel tetramerization domain containing 2
KIF13A kinesin family member 13A
KLHL36 kelch-like family member 36
LAMP1 lysosomal-associated membrane protein 1
LCN2 lipocalin 2
LHB luteinizing hormone beta polypeptide
LILRA2 leukocyte immunoglobulin-like receptor, subfamily A (with TM domain), member 2
MAP4 microtubule-associated protein 4
MBOAT2 membrane bound O-acyltransferase domain containing 2
MUC8 mucin 8
NCAM1 neural cell adhesion molecule 1
NCLN nicalin
NDUFA2 NADH dehydrogenase (ubiquinone) 1 alpha subcomplex, 2, 8kDa
NEK11 NIMA-related kinase 11
NEURL1 neuralized E3 ubiquitin protein ligase 1
NFKBIB nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, beta
NQO1 NAD(P)H dehydrogenase, quinone 1
NR2E3 nuclear receptor subfamily 2, group E, member 3
OR1D2 olfactory receptor, family 1, subfamily D, member 2
OR7E24 olfactory receptor, family 7, subfamily E, member 24
PAPPA pregnancy-associated plasma protein A, pappalysin 1
PARVB parvin, beta
PATZ1 POZ (BTB) and AT hook containing zinc finger 1
PCDH12 protocadherin 12
PI4K2A phosphatidylinositol 4-kinase type 2 alpha
PLCD1 phospholipase C, delta 1
PLSCR3 phospholipid scramblase 3
PNLIPRP1 pancreatic lipase-related protein 1
POLR2L polymerase (RNA) II (DNA directed) polypeptide L, 7.6kDa
PPARD peroxisome proliferator-activated receptor delta
PQLC2 PQ loop repeat containing 2
PRKAR2A protein kinase, cAMP-dependent, regulatory, type II, alpha
PRKCQ protein kinase C, theta
PYCRL pyrroline-5-carboxylate reductase-like
RECQL5 RecQ protein-like 5
RUSC2 RUN and SH3 domain containing 2
S1PR4 sphingosine-1-phosphate receptor 4
SEC14L5 SEC14-like 5 (S. cerevisiae)
SEMA4G sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4G
SLC17A7 solute carrier family 17 (vesicular glutamate transporter), member 7
SLC1A7 solute carrier family 1 (glutamate transporter), member 7
SLCO2B1 solute carrier organic anion transporter family, member 2B1
SORBS3 sorbin and SH3 domain containing 3
SPAG8 sperm associated antigen 8
SPTBN1 spectrin, beta, non-erythrocytic 1
ST7L suppression of tumorigenicity 7 like
TMPRSS6 transmembrane protease, serine 6
TRGV5 T cell receptor gamma variable 5
TSTA3 tissue specific transplantation antigen P35B
UBE2I ubiquitin-conjugating enzyme E2I
WFDC8 WAP four-disulfide core domain 8
XYLB xylulokinase homolog (H. influenzae)
ZNF747 zinc finger protein 747

decreased expression

Symbol Name
ACOX2 acyl-CoA oxidase 2, branched chain
ALDH1B1 aldehyde dehydrogenase 1 family, member B1
AMIGO2 adhesion molecule with Ig-like domain 2
AP5S1 adaptor-related protein complex 5, sigma 1 subunit
APBB1IP amyloid beta (A4) precursor protein-binding, family B, member 1 interacting protein
APOL6 apolipoprotein L, 6
AXIN1 axin 1
C1ORF56 chromosome 1 open reading frame 56
C5 complement component 5
C5ORF45 chromosome 5 open reading frame 45
C6ORF47 chromosome 6 open reading frame 47
C9ORF3 chromosome 9 open reading frame 3
CAMKMT calmodulin-lysine N-methyltransferase
CAND2 cullin-associated and neddylation-dissociated 2 (putative)
CCDC85C coiled-coil domain containing 85C
CDH10 cadherin 10, type 2 (T2-cadherin)
CEL carboxyl ester lipase
CENPT centromere protein T
CLCN2 chloride channel, voltage-sensitive 2
CLN6 ceroid-lipofuscinosis, neuronal 6, late infantile, variant
CNTN1 contactin 1
DDN dendrin
DOC2A double C2-like domains, alpha
ELMO3 engulfment and cell motility 3
EXOSC1 exosome component 1
FAM188A family with sequence similarity 188, member A
FBRS fibrosin
FDXR ferredoxin reductase
FMOD fibromodulin
GABRB2 gamma-aminobutyric acid (GABA) A receptor, beta 2
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GATA6 GATA binding protein 6
GRIP2 glutamate receptor interacting protein 2
GSR glutathione reductase
GSTA3 glutathione S-transferase alpha 3
GSTT1 glutathione S-transferase theta 1
GTF2A1 general transcription factor IIA, 1, 19/37kDa
GTF3C5 general transcription factor IIIC, polypeptide 5, 63kDa
HIST1H1T histone cluster 1, H1t
HNRNPA3P1 heterogeneous nuclear ribonucleoprotein A3 pseudogene 1
HOXA5 homeobox A5
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IFIT2 interferon-induced protein with tetratricopeptide repeats 2
IGF2BP2 insulin-like growth factor 2 mRNA binding protein 2
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
IL22 interleukin 22
ITGAX integrin, alpha X (complement component 3 receptor 4 subunit)
ITPKB inositol-trisphosphate 3-kinase B
KIAA0754 KIAA0754
KRT8P12 keratin 8 pseudogene 12
LIME1 Lck interacting transmembrane adaptor 1
LOC100287590 uncharacterized LOC100287590
LRRK1 leucine-rich repeat kinase 1
LTC4S leukotriene C4 synthase
MAPK3 mitogen-activated protein kinase 3
MEFV Mediterranean fever
MYL5 myosin, light chain 5, regulatory
MYO1E myosin IE
NECAB3 N-terminal EF-hand calcium binding protein 3
OASL 2'-5'-oligoadenylate synthetase-like
OVGP1 oviductal glycoprotein 1, 120kDa
PAFAH1B2 platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (30kDa)
PARG poly (ADP-ribose) glycohydrolase
PARP12 poly (ADP-ribose) polymerase family, member 12
PDLIM2 PDZ and LIM domain 2 (mystique)
PECR peroxisomal trans-2-enoyl-CoA reductase
PGGT1B protein geranylgeranyltransferase type I, beta subunit
PIM1 Pim-1 proto-oncogene, serine/threonine kinase
PMP22 peripheral myelin protein 22
POLL polymerase (DNA directed), lambda
PPFIA4 protein tyrosine phosphatase, receptor type, f polypeptide (PTPRF), interacting protein (liprin), alpha 4
PRAMEF11 PRAME family member 11
PRSS53 protease, serine, 53
R3HCC1L R3H domain and coiled-coil containing 1-like
RAB33A RAB33A, member RAS oncogene family
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RASAL1 RAS protein activator like 1 (GAP1 like)
RNF2 ring finger protein 2
RPA4 replication protein A4, 30kDa
RRAS related RAS viral (r-ras) oncogene homolog
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC2A8 solute carrier family 2 (facilitated glucose transporter), member 8
SLITRK5 SLIT and NTRK-like family, member 5
SULT1B1 sulfotransferase family, cytosolic, 1B, member 1
SV2A synaptic vesicle glycoprotein 2A
TCTN1 tectonic family member 1
TET3 tet methylcytosine dioxygenase 3
THEM6 thioesterase superfamily member 6
TICAM1 toll-like receptor adaptor molecule 1
TNFRSF14 tumor necrosis factor receptor superfamily, member 14
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
UNC119 unc-119 homolog (C. elegans)
UPB1 ureidopropionase, beta
XAB2 XPA binding protein 2
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZNF185 zinc finger protein 185 (LIM domain)
ZNF444 zinc finger protein 444
ZNF749 zinc finger protein 749
ZW10 zw10 kinetochore protein