Prestwick-664-6033 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the Prestwick-664-6033 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
APLP1 amyloid beta (A4) precursor-like protein 1
BCAM basal cell adhesion molecule (Lutheran blood group)
BFSP2 beaded filament structural protein 2, phakinin
BIN1 bridging integrator 1
C2ORF72 chromosome 2 open reading frame 72
CACNG1 calcium channel, voltage-dependent, gamma subunit 1
CCDC64 coiled-coil domain containing 64
CCPG1 cell cycle progression 1
CD48 CD48 molecule
CDK14 cyclin-dependent kinase 14
CELP carboxyl ester lipase pseudogene
CEND1 cell cycle exit and neuronal differentiation 1
CFAP45 cilia and flagella associated protein 45
CHST2 carbohydrate (N-acetylglucosamine-6-O) sulfotransferase 2
CNN1 calponin 1, basic, smooth muscle
CNTNAP2 contactin associated protein-like 2
COL6A1 collagen, type VI, alpha 1
CSN3 casein kappa
CTSE cathepsin E
DMBT1 deleted in malignant brain tumors 1
DMPK dystrophia myotonica-protein kinase
DOK4 docking protein 4
ECE1 endothelin converting enzyme 1
ECEL1 endothelin converting enzyme-like 1
EDA ectodysplasin A
EIF4EBP2 eukaryotic translation initiation factor 4E binding protein 2
EPHB2 EPH receptor B2
F12 coagulation factor XII (Hageman factor)
FCAR Fc fragment of IgA receptor
FGF22 fibroblast growth factor 22
FMO5 flavin containing monooxygenase 5
GAL galanin/GMAP prepropeptide
GJB1 gap junction protein, beta 1, 32kDa
GPD1 glycerol-3-phosphate dehydrogenase 1 (soluble)
GPR85 G protein-coupled receptor 85
GTDC1 glycosyltransferase-like domain containing 1
HIST1H3I histone cluster 1, H3i
HNRNPDL heterogeneous nuclear ribonucleoprotein D-like
HPCAL4 hippocalcin like 4
IFNB1 interferon, beta 1, fibroblast
IL1RN interleukin 1 receptor antagonist
IPW imprinted in Prader-Willi syndrome (non-protein coding)
KCNK10 potassium channel, two pore domain subfamily K, member 10
KDM5B lysine (K)-specific demethylase 5B
KIAA0125 KIAA0125
KIR2DL1 killer cell immunoglobulin-like receptor, two domains, long cytoplasmic tail, 1
KIR2DS1 killer cell immunoglobulin-like receptor, two domains, short cytoplasmic tail, 1
KLHL20 kelch-like family member 20
LAT2 linker for activation of T cells family, member 2
LILRB3 leukocyte immunoglobulin-like receptor, subfamily B (with TM and ITIM domains), member 3
MED16 mediator complex subunit 16
MFAP5 microfibrillar associated protein 5
MKRN3 makorin ring finger protein 3
MLNR motilin receptor
MRPS12 mitochondrial ribosomal protein S12
MYL10 myosin, light chain 10, regulatory
MYL3 myosin, light chain 3, alkali; ventricular, skeletal, slow
NR2F1 nuclear receptor subfamily 2, group F, member 1
NRG2 neuregulin 2
PCDH1 protocadherin 1
PCM1 pericentriolar material 1
PLA2G4C phospholipase A2, group IVC (cytosolic, calcium-independent)
PMFBP1 polyamine modulated factor 1 binding protein 1
PNMAL1 paraneoplastic Ma antigen family-like 1
PQBP1 polyglutamine binding protein 1
PRSS3 protease, serine, 3
PVR poliovirus receptor
PYY2 peptide YY, 2 (pseudogene)
RAP2B RAP2B, member of RAS oncogene family
RASA3 RAS p21 protein activator 3
RASSF9 Ras association (RalGDS/AF-6) domain family (N-terminal) member 9
RFPL3 ret finger protein-like 3
RGS12 regulator of G-protein signaling 12
RGS14 regulator of G-protein signaling 14
RGS4 regulator of G-protein signaling 4
RUSC2 RUN and SH3 domain containing 2
S100A8 S100 calcium binding protein A8
S100A9 S100 calcium binding protein A9
SAMD9 sterile alpha motif domain containing 9
SERPINB5 serpin peptidase inhibitor, clade B (ovalbumin), member 5
SLC16A3 solute carrier family 16 (monocarboxylate transporter), member 3
SLC1A2 solute carrier family 1 (glial high affinity glutamate transporter), member 2
SLC22A7 solute carrier family 22 (organic anion transporter), member 7
SLC4A4 solute carrier family 4 (sodium bicarbonate cotransporter), member 4
SLC52A1 solute carrier family 52 (riboflavin transporter), member 1
SNCA synuclein, alpha (non A4 component of amyloid precursor)
SNTA1 syntrophin, alpha 1
SOGA1 suppressor of glucose, autophagy associated 1
SP100 SP100 nuclear antigen
SPHK2 sphingosine kinase 2
TAOK2 TAO kinase 2
TBX2 T-box 2
TGM1 transglutaminase 1
THPO thrombopoietin
TRD T cell receptor delta locus
TRIM22 tripartite motif containing 22
VIPR2 vasoactive intestinal peptide receptor 2
ZNF112 zinc finger protein 112
ZNF589 zinc finger protein 589

decreased expression

Symbol Name
AKR1B1 aldo-keto reductase family 1, member B1 (aldose reductase)
ANP32A-IT1 ANP32A intronic transcript 1
AOC2 amine oxidase, copper containing 2 (retina-specific)
APBB3 amyloid beta (A4) precursor protein-binding, family B, member 3
ASAP3 ArfGAP with SH3 domain, ankyrin repeat and PH domain 3
ATG10 autophagy related 10
AUTS2 autism susceptibility candidate 2
BMP4 bone morphogenetic protein 4
C1ORF159 chromosome 1 open reading frame 159
C5AR2 complement component 5a receptor 2
CACNA1H calcium channel, voltage-dependent, T type, alpha 1H subunit
CAPG capping protein (actin filament), gelsolin-like
CCDC85C coiled-coil domain containing 85C
CD8A CD8a molecule
CDH10 cadherin 10, type 2 (T2-cadherin)
CHRNB2 cholinergic receptor, nicotinic, beta 2 (neuronal)
CLDN17 claudin 17
CLIP4 CAP-GLY domain containing linker protein family, member 4
COPZ2 coatomer protein complex, subunit zeta 2
CPB1 carboxypeptidase B1 (tissue)
CTSF cathepsin F
CUZD1 CUB and zona pellucida-like domains 1
CYP2B7P cytochrome P450, family 2, subfamily B, polypeptide 7, pseudogene
DNM3 dynamin 3
EHMT1 euchromatic histone-lysine N-methyltransferase 1
EN2 engrailed homeobox 2
EPHX2 epoxide hydrolase 2, cytoplasmic
EXD3 exonuclease 3'-5' domain containing 3
F3 coagulation factor III (thromboplastin, tissue factor)
FAM110B family with sequence similarity 110, member B
FAM131A family with sequence similarity 131, member A
FAM188A family with sequence similarity 188, member A
FAM53B family with sequence similarity 53, member B
FBXW4P1 F-box and WD repeat domain containing 4 pseudogene 1
FGL1 fibrinogen-like 1
GDAP2 ganglioside induced differentiation associated protein 2
GEMIN8 gem (nuclear organelle) associated protein 8
GNL1 guanine nucleotide binding protein-like 1
GPX2 glutathione peroxidase 2
GSTA4 glutathione S-transferase alpha 4
HDAC5 histone deacetylase 5
HIST1H2AJ histone cluster 1, H2aj
HOXC5 homeobox C5
IL22 interleukin 22
INPP1 inositol polyphosphate-1-phosphatase
INPP5J inositol polyphosphate-5-phosphatase J
IQCG IQ motif containing G
IQSEC2 IQ motif and Sec7 domain 2
IRF2BP1 interferon regulatory factor 2 binding protein 1
KIAA0754 KIAA0754
LMX1B LIM homeobox transcription factor 1, beta
MMP3 matrix metallopeptidase 3
MORN1 MORN repeat containing 1
MUC3A mucin 3A, cell surface associated
NDE1 nudE neurodevelopment protein 1
NDOR1 NADPH dependent diflavin oxidoreductase 1
NPIPB3 nuclear pore complex interacting protein family, member B3
OLFML2A olfactomedin-like 2A
ONECUT2 one cut homeobox 2
PACS1 phosphofurin acidic cluster sorting protein 1
PADI1 peptidyl arginine deiminase, type I
PDGFRL platelet-derived growth factor receptor-like
PER3 period circadian clock 3
PGPEP1 pyroglutamyl-peptidase I
PLA2G3 phospholipase A2, group III
PMCH pro-melanin-concentrating hormone
POM121 POM121 transmembrane nucleoporin
PRRG4 proline rich Gla (G-carboxyglutamic acid) 4 (transmembrane)
QSER1 glutamine and serine rich 1
RASSF2 Ras association (RalGDS/AF-6) domain family member 2
RGS2 regulator of G-protein signaling 2
RNF122 ring finger protein 122
RNF208 ring finger protein 208
S100A2 S100 calcium binding protein A2
SALL2 spalt-like transcription factor 2
SLC12A6 solute carrier family 12 (potassium/chloride transporter), member 6
SLC12A9 solute carrier family 12, member 9
SLC17A5 solute carrier family 17 (acidic sugar transporter), member 5
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SP1 Sp1 transcription factor
STARD13 StAR-related lipid transfer (START) domain containing 13
STRA6 stimulated by retinoic acid 6
SYT17 synaptotagmin XVII
TBC1D17 TBC1 domain family, member 17
TMEM242 transmembrane protein 242
TMEM53 transmembrane protein 53
TOM1 target of myb1 (chicken)
TSPYL2 TSPY-like 2
VASH2 vasohibin 2
ZNF211 zinc finger protein 211
ZNF212 zinc finger protein 212
ZNF219 zinc finger protein 219
ZNF282 zinc finger protein 282
ZNF362 zinc finger protein 362
ZNF428 zinc finger protein 428
ZNF532 zinc finger protein 532
ZNF573 zinc finger protein 573
ZNF580 zinc finger protein 580
ZNF862 zinc finger protein 862