Prestwick-682-2819 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

200 genes differentially expressed following the Prestwick-682-2819 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACADS acyl-CoA dehydrogenase, C-2 to C-3 short chain
AKAP8L A kinase (PRKA) anchor protein 8-like
ALS2CL ALS2 C-terminal like
AMT aminomethyltransferase
ARHGDIB Rho GDP dissociation inhibitor (GDI) beta
ARTN artemin
ASIC4 acid sensing (proton gated) ion channel family member 4
B3GALT4 UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 4
BAIAP3 BAI1-associated protein 3
CAMK4 calcium/calmodulin-dependent protein kinase IV
CAPN5 calpain 5
CEP250 centrosomal protein 250kDa
CHRNA3 cholinergic receptor, nicotinic, alpha 3 (neuronal)
COL6A1 collagen, type VI, alpha 1
CORO7 coronin 7
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
CTIF CBP80/20-dependent translation initiation factor
CYHR1 cysteine/histidine-rich 1
DAPP1 dual adaptor of phosphotyrosine and 3-phosphoinositides
DICER1 dicer 1, ribonuclease type III
DKFZP434C153 DKFZP434C153 protein
DMTN dematin actin binding protein
EHMT2 euchromatic histone-lysine N-methyltransferase 2
EPHB2 EPH receptor B2
ERN2 endoplasmic reticulum to nucleus signaling 2
ETV5 ets variant 5
EYA3 EYA transcriptional coactivator and phosphatase 3
F13A1 coagulation factor XIII, A1 polypeptide
FAM46C family with sequence similarity 46, member C
FGFR4 fibroblast growth factor receptor 4
FXYD5 FXYD domain containing ion transport regulator 5
GLIPR1 GLI pathogenesis-related 1
GNAT2 guanine nucleotide binding protein (G protein), alpha transducing activity polypeptide 2
GPER1 G protein-coupled estrogen receptor 1
GTF2F1 general transcription factor IIF, polypeptide 1, 74kDa
H6PD hexose-6-phosphate dehydrogenase (glucose 1-dehydrogenase)
HADHA hydroxyacyl-CoA dehydrogenase/3-ketoacyl-CoA thiolase/enoyl-CoA hydratase (trifunctional protein), alpha subunit
HBEGF heparin-binding EGF-like growth factor
HCG4B HLA complex group 4B (non-protein coding)
HS3ST2 heparan sulfate (glucosamine) 3-O-sulfotransferase 2
IFNA17 interferon, alpha 17
IL1RAPL2 interleukin 1 receptor accessory protein-like 2
IL2RA interleukin 2 receptor, alpha
KATNB1 katanin p80 (WD repeat containing) subunit B 1
KIAA0319L KIAA0319-like
KIAA1109 KIAA1109
LENEP lens epithelial protein
LHX1 LIM homeobox 1
LIME1 Lck interacting transmembrane adaptor 1
LRRC37BP1 leucine rich repeat containing 37B pseudogene 1
MAGOH2P mago-nashi homolog 2, pseudogene
MAPK8 mitogen-activated protein kinase 8
MIER2 mesoderm induction early response 1, family member 2
MTA2 metastasis associated 1 family, member 2
MTHFR methylenetetrahydrofolate reductase (NAD(P)H)
MUC6 mucin 6, oligomeric mucus/gel-forming
NDUFAF5 NADH dehydrogenase (ubiquinone) complex I, assembly factor 5
NEUROD1 neuronal differentiation 1
NF1 neurofibromin 1
NOL10 nucleolar protein 10
NOTCH4 notch 4
NUP54 nucleoporin 54kDa
PADI3 peptidyl arginine deiminase, type III
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
POM121 POM121 transmembrane nucleoporin
POPDC3 popeye domain containing 3
PRDM2 PR domain containing 2, with ZNF domain
PSG6 pregnancy specific beta-1-glycoprotein 6
PTCH1 patched 1
PTGER2 prostaglandin E receptor 2 (subtype EP2), 53kDa
PVRL3 poliovirus receptor-related 3
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RAB6B RAB6B, member RAS oncogene family
RB1 retinoblastoma 1
RGS3 regulator of G-protein signaling 3
RNF19B ring finger protein 19B
RRP12 ribosomal RNA processing 12 homolog (S. cerevisiae)
SBNO2 strawberry notch homolog 2 (Drosophila)
SCAPER S-phase cyclin A-associated protein in the ER
SEMA3B sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3B
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SLC1A7 solute carrier family 1 (glutamate transporter), member 7
SLC43A1 solute carrier family 43 (amino acid system L transporter), member 1
SORBS3 sorbin and SH3 domain containing 3
STEAP4 STEAP family member 4
TBC1D17 TBC1 domain family, member 17
TBKBP1 TBK1 binding protein 1
TBX5 T-box 5
TEF thyrotrophic embryonic factor
TNFAIP3 tumor necrosis factor, alpha-induced protein 3
TNFRSF17 tumor necrosis factor receptor superfamily, member 17
TP53I11 tumor protein p53 inducible protein 11
UBXN6 UBX domain protein 6
WWP2 WW domain containing E3 ubiquitin protein ligase 2
XDH xanthine dehydrogenase
ZMAT4 zinc finger, matrin-type 4
ZNF224 zinc finger protein 224
ZNF230 zinc finger protein 230
ZNF37BP zinc finger protein 37B, pseudogene
ZNF444 zinc finger protein 444

decreased expression

Symbol Name
ABCA11P ATP-binding cassette, sub-family A (ABC1), member 11, pseudogene
ABCA7 ATP-binding cassette, sub-family A (ABC1), member 7
ADAM15 ADAM metallopeptidase domain 15
ADM adrenomedullin
AKAP5 A kinase (PRKA) anchor protein 5
ALPK1 alpha-kinase 1
APOLD1 apolipoprotein L domain containing 1
AUTS2 autism susceptibility candidate 2
BATF basic leucine zipper transcription factor, ATF-like
BMP10 bone morphogenetic protein 10
C1QB complement component 1, q subcomponent, B chain
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
C2ORF54 chromosome 2 open reading frame 54
CAMK1 calcium/calmodulin-dependent protein kinase I
CCDC130 coiled-coil domain containing 130
CDH10 cadherin 10, type 2 (T2-cadherin)
CENPO centromere protein O
CHMP6 charged multivesicular body protein 6
CLCN6 chloride channel, voltage-sensitive 6
CNTN1 contactin 1
COPZ2 coatomer protein complex, subunit zeta 2
CSTA cystatin A (stefin A)
CTRL chymotrypsin-like
DNM1 dynamin 1
DSCAM Down syndrome cell adhesion molecule
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
ERMAP erythroblast membrane-associated protein (Scianna blood group)
EXO5 exonuclease 5
GALNT12 polypeptide N-acetylgalactosaminyltransferase 12
GAMT guanidinoacetate N-methyltransferase
GAS2 growth arrest-specific 2
GLS2 glutaminase 2 (liver, mitochondrial)
GPATCH3 G patch domain containing 3
GPR22 G protein-coupled receptor 22
GSTTP1 glutathione S-transferase theta pseudogene 1
HIST1H2BO histone cluster 1, H2bo
HIST2H2AA3 histone cluster 2, H2aa3
HPN hepsin
IDI2-AS1 IDI2 antisense RNA 1
INPP1 inositol polyphosphate-1-phosphatase
INPP5J inositol polyphosphate-5-phosphatase J
KAT2A K(lysine) acetyltransferase 2A
KCNK5 potassium channel, two pore domain subfamily K, member 5
KPNA5 karyopherin alpha 5 (importin alpha 6)
LY6D lymphocyte antigen 6 complex, locus D
LY6G6C lymphocyte antigen 6 complex, locus G6C
MGC12488
MOBP myelin-associated oligodendrocyte basic protein
MOSPD3 motile sperm domain containing 3
MX1 MX dynamin-like GTPase 1
MYL12A myosin, light chain 12A, regulatory, non-sarcomeric
MYO1F myosin IF
MYOZ3 myozenin 3
NEAT1 nuclear paraspeckle assembly transcript 1 (non-protein coding)
NME5 NME/NM23 family member 5
NPFFR1 neuropeptide FF receptor 1
NPTX1 neuronal pentraxin I
PCDHA6 protocadherin alpha 6
PDK1 pyruvate dehydrogenase kinase, isozyme 1
PHLPP1 PH domain and leucine rich repeat protein phosphatase 1
PLA2G10 phospholipase A2, group X
PLA2G3 phospholipase A2, group III
PNRC1 proline-rich nuclear receptor coactivator 1
POLL polymerase (DNA directed), lambda
PRRG2 proline rich Gla (G-carboxyglutamic acid) 2
PRRG4 proline rich Gla (G-carboxyglutamic acid) 4 (transmembrane)
PTDSS2 phosphatidylserine synthase 2
QSER1 glutamine and serine rich 1
RASSF8 Ras association (RalGDS/AF-6) domain family (N-terminal) member 8
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RHOBTB2 Rho-related BTB domain containing 2
RIN1 Ras and Rab interactor 1
RNF122 ring finger protein 122
RNF125 ring finger protein 125, E3 ubiquitin protein ligase
RPL10L ribosomal protein L10-like
RPL23AP32 ribosomal protein L23a pseudogene 32
RPS6KA4 ribosomal protein S6 kinase, 90kDa, polypeptide 4
SAYSD1 SAYSVFN motif domain containing 1
SLC44A1 solute carrier family 44 (choline transporter), member 1
SLC46A3 solute carrier family 46, member 3
SNAI2 snail family zinc finger 2
SPINK4 serine peptidase inhibitor, Kazal type 4
STON1 stonin 1
STX1A syntaxin 1A (brain)
SYCP2 synaptonemal complex protein 2
TEP1 telomerase-associated protein 1
TGFBR3 transforming growth factor, beta receptor III
TMEM19 transmembrane protein 19
TNS2 tensin 2
TRDMT1 tRNA aspartic acid methyltransferase 1
TUBA3C tubulin, alpha 3c
TWISTNB TWIST neighbor
ZBTB22 zinc finger and BTB domain containing 22
ZFP37 ZFP37 zinc finger protein
ZNF329 zinc finger protein 329
ZNF516 zinc finger protein 516
ZNF552 zinc finger protein 552
ZNF701 zinc finger protein 701
ZNF750 zinc finger protein 750
ZNF770 zinc finger protein 770