Prestwick-692-4424 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
Similar Terms
Downloads & Tools

Genes

195 genes differentially expressed following the Prestwick-692-4424 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADAM22 ADAM metallopeptidase domain 22
ASIC1 acid sensing (proton gated) ion channel 1
ASPN asporin
ATP11A ATPase, class VI, type 11A
ATP8A2 ATPase, aminophospholipid transporter, class I, type 8A, member 2
BAIAP3 BAI1-associated protein 3
BCAN brevican
C1QTNF1 C1q and tumor necrosis factor related protein 1
CALB2 calbindin 2
CASP2 caspase 2, apoptosis-related cysteine peptidase
CCDC85B coiled-coil domain containing 85B
CEBPD CCAAT/enhancer binding protein (C/EBP), delta
CELF2 CUGBP, Elav-like family member 2
CEP41 centrosomal protein 41kDa
CHRNA4 cholinergic receptor, nicotinic, alpha 4 (neuronal)
CHRNB2 cholinergic receptor, nicotinic, beta 2 (neuronal)
CLCN1 chloride channel, voltage-sensitive 1
CLTB clathrin, light chain B
CRISP2 cysteine-rich secretory protein 2
CRMP1 collapsin response mediator protein 1
CTNS cystinosin, lysosomal cystine transporter
DOPEY2 dopey family member 2
E2F5 E2F transcription factor 5, p130-binding
ECEL1 endothelin converting enzyme-like 1
FRMD1 FERM domain containing 1
FYN FYN proto-oncogene, Src family tyrosine kinase
GABARAPL1 GABA(A) receptor-associated protein like 1
GABRD gamma-aminobutyric acid (GABA) A receptor, delta
GDPD2 glycerophosphodiester phosphodiesterase domain containing 2
GGT1 gamma-glutamyltransferase 1
GJA4 gap junction protein, alpha 4, 37kDa
GM2A GM2 ganglioside activator
HEY2 hes-related family bHLH transcription factor with YRPW motif 2
HLA-DQB2 major histocompatibility complex, class II, DQ beta 2
HOXA4 homeobox A4
HTR1B 5-hydroxytryptamine (serotonin) receptor 1B, G protein-coupled
HTR2A 5-hydroxytryptamine (serotonin) receptor 2A, G protein-coupled
IGFBP5 insulin-like growth factor binding protein 5
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
IL1R1 interleukin 1 receptor, type I
ITPR3 inositol 1,4,5-trisphosphate receptor, type 3
KLK13 kallikrein-related peptidase 13
LEF1 lymphoid enhancer-binding factor 1
LIM2 lens intrinsic membrane protein 2, 19kDa
LYL1 lymphoblastic leukemia associated hematopoiesis regulator 1
MAPK14 mitogen-activated protein kinase 14
MIER2 mesoderm induction early response 1, family member 2
MIR622 microRNA 622
MMP24 matrix metallopeptidase 24 (membrane-inserted)
MYO7A myosin VIIA
NUP188 nucleoporin 188kDa
OR1E1 olfactory receptor, family 1, subfamily E, member 1
PAPPA2 pappalysin 2
PCDHB11 protocadherin beta 11
PCNX pecanex homolog (Drosophila)
PDE1C phosphodiesterase 1C, calmodulin-dependent 70kDa
PEG10 paternally expressed 10
PML promyelocytic leukemia
POLM polymerase (DNA directed), mu
POU2F2 POU class 2 homeobox 2
PPP2R5B protein phosphatase 2, regulatory subunit B', beta
PRDX2 peroxiredoxin 2
PRKACA protein kinase, cAMP-dependent, catalytic, alpha
RARA retinoic acid receptor, alpha
RQCD1 RCD1 required for cell differentiation1 homolog (S. pombe)
SAMD4A sterile alpha motif domain containing 4A
SAYSD1 SAYSVFN motif domain containing 1
SCUBE3 signal peptide, CUB domain, EGF-like 3
SDS serine dehydratase
SEC24A SEC24 family member A
SEC24D SEC24 family member D
SECTM1 secreted and transmembrane 1
SEMA4F sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4F
SH3GL3 SH3-domain GRB2-like 3
SLC12A4 solute carrier family 12 (potassium/chloride transporter), member 4
SLC16A4 solute carrier family 16, member 4
SLCO2A1 solute carrier organic anion transporter family, member 2A1
SOCS7 suppressor of cytokine signaling 7
SORBS2 sorbin and SH3 domain containing 2
SPAG8 sperm associated antigen 8
SRRM2 serine/arginine repetitive matrix 2
ST3GAL4 ST3 beta-galactoside alpha-2,3-sialyltransferase 4
SVIL supervillin
SYNE1 spectrin repeat containing, nuclear envelope 1
TBC1D22B TBC1 domain family, member 22B
TBRG4 transforming growth factor beta regulator 4
TCF12 transcription factor 12
TFR2 transferrin receptor 2
THY1 Thy-1 cell surface antigen
TM4SF4 transmembrane 4 L six family member 4
TMEM80 transmembrane protein 80
TROVE2 TROVE domain family, member 2
TYRP1 tyrosinase-related protein 1
URB1 URB1 ribosome biogenesis 1 homolog (S. cerevisiae)
WSB1 WD repeat and SOCS box containing 1
ZDHHC8P1 zinc finger, DHHC-type containing 8 pseudogene 1
ZNF362 zinc finger protein 362
ZNF507 zinc finger protein 507

decreased expression

Symbol Name
ACBD4 acyl-CoA binding domain containing 4
ADAM2 ADAM metallopeptidase domain 2
ADM adrenomedullin
AGMAT agmatine ureohydrolase (agmatinase)
AP1S1 adaptor-related protein complex 1, sigma 1 subunit
ARC activity-regulated cytoskeleton-associated protein
ARHGEF17 Rho guanine nucleotide exchange factor (GEF) 17
ARMC4 armadillo repeat containing 4
ARPIN actin-related protein 2/3 complex inhibitor
ARR3 arrestin 3, retinal (X-arrestin)
B3GALT4 UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 4
BAX BCL2-associated X protein
BTF3P11 basic transcription factor 3 pseudogene 11
BTF3P12 basic transcription factor 3 pseudogene 12
C11ORF30 chromosome 11 open reading frame 30
C1ORF105 chromosome 1 open reading frame 105
CDK6 cyclin-dependent kinase 6
CLGN calmegin
CORT cortistatin
CRLF1 cytokine receptor-like factor 1
CYP4F11 cytochrome P450, family 4, subfamily F, polypeptide 11
CYP7B1 cytochrome P450, family 7, subfamily B, polypeptide 1
DBF4B DBF4 zinc finger B
DGKQ diacylglycerol kinase, theta 110kDa
DUSP8 dual specificity phosphatase 8
ERCC2 excision repair cross-complementation group 2
FBXL2 F-box and leucine-rich repeat protein 2
GPC3 glypican 3
GPR143 G protein-coupled receptor 143
GPR157 G protein-coupled receptor 157
GPR3 G protein-coupled receptor 3
HIRA histone cell cycle regulator
HIST1H3F histone cluster 1, H3f
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
HNRNPA3P1 heterogeneous nuclear ribonucleoprotein A3 pseudogene 1
HS3ST3A1 heparan sulfate (glucosamine) 3-O-sulfotransferase 3A1
HTR1E 5-hydroxytryptamine (serotonin) receptor 1E, G protein-coupled
HYAL3 hyaluronoglucosaminidase 3
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IL12RB1 interleukin 12 receptor, beta 1
IL1RAPL2 interleukin 1 receptor accessory protein-like 2
ITGA10 integrin, alpha 10
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor)
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNIP1 Kv channel interacting protein 1
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KCNN1 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 1
KCNQ3 potassium channel, voltage gated KQT-like subfamily Q, member 3
KHDRBS3 KH domain containing, RNA binding, signal transduction associated 3
KLHL29 kelch-like family member 29
KLK5 kallikrein-related peptidase 5
KREMEN2 kringle containing transmembrane protein 2
LHX6 LIM homeobox 6
LMNB1 lamin B1
LOXL3 lysyl oxidase-like 3
MAPK10 mitogen-activated protein kinase 10
MCTP2 multiple C2 domains, transmembrane 2
MLLT4-AS1 MLLT4 antisense RNA 1 (head to head)
MTHFD2L methylenetetrahydrofolate dehydrogenase (NADP+ dependent) 2-like
NEUROD1 neuronal differentiation 1
NKX2-5 NK2 homeobox 5
NPY1R neuropeptide Y receptor Y1
NPY4R neuropeptide Y receptor Y4
OCLM oculomedin
OR2F1 olfactory receptor, family 2, subfamily F, member 1 (gene/pseudogene)
PCDH17 protocadherin 17
PDE8B phosphodiesterase 8B
PDZD2 PDZ domain containing 2
PIK3R5 phosphoinositide-3-kinase, regulatory subunit 5
PLAC1 placenta-specific 1
POPDC3 popeye domain containing 3
PRKCE protein kinase C, epsilon
RBFOX1 RNA binding protein, fox-1 homolog (C. elegans) 1
RNF2 ring finger protein 2
ROBO3 roundabout, axon guidance receptor, homolog 3 (Drosophila)
RORC RAR-related orphan receptor C
RUSC2 RUN and SH3 domain containing 2
SCHIP1 schwannomin interacting protein 1
SEC14L5 SEC14-like 5 (S. cerevisiae)
SLC12A6 solute carrier family 12 (potassium/chloride transporter), member 6
SLC9A8 solute carrier family 9, subfamily A (NHE8, cation proton antiporter 8), member 8
SMIM14 small integral membrane protein 14
SPINK2 serine peptidase inhibitor, Kazal type 2 (acrosin-trypsin inhibitor)
SPRR2B small proline-rich protein 2B
STARD5 StAR-related lipid transfer (START) domain containing 5
STIM1 stromal interaction molecule 1
TAS2R10 taste receptor, type 2, member 10
THRB thyroid hormone receptor, beta
TMA16 translation machinery associated 16 homolog (S. cerevisiae)
TMEM158 transmembrane protein 158 (gene/pseudogene)
TRPV1 transient receptor potential cation channel, subfamily V, member 1
TUBA3C tubulin, alpha 3c
VASH2 vasohibin 2
ZNF197 zinc finger protein 197
ZNF250 zinc finger protein 250
ZNF750 zinc finger protein 750
ZNF76 zinc finger protein 76