Prestwick-860-3040 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the Prestwick-860-3040 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADGRB1 adhesion G protein-coupled receptor B1
AGFG1 ArfGAP with FG repeats 1
AIM1L absent in melanoma 1-like
ALDH6A1 aldehyde dehydrogenase 6 family, member A1
ANKRD2 ankyrin repeat domain 2 (stretch responsive muscle)
APC2 adenomatosis polyposis coli 2
ARHGEF10 Rho guanine nucleotide exchange factor (GEF) 10
ARHGEF16 Rho guanine nucleotide exchange factor (GEF) 16
BCAS3 breast carcinoma amplified sequence 3
CALCR calcitonin receptor
CAMK2A calcium/calmodulin-dependent protein kinase II alpha
CEP170B centrosomal protein 170B
CHD5 chromodomain helicase DNA binding protein 5
COL10A1 collagen, type X, alpha 1
CSF2 colony stimulating factor 2 (granulocyte-macrophage)
CSN2 casein beta
DCBLD2 discoidin, CUB and LCCL domain containing 2
DDAH2 dimethylarginine dimethylaminohydrolase 2
DGCR5 DiGeorge syndrome critical region gene 5 (non-protein coding)
DOT1L DOT1-like histone H3K79 methyltransferase
DZIP3 DAZ interacting zinc finger protein 3
EFR3B EFR3 homolog B (S. cerevisiae)
EHD2 EH-domain containing 2
EPS8L3 EPS8-like 3
EVX1 even-skipped homeobox 1
EXT1 exostosin glycosyltransferase 1
FCGBP Fc fragment of IgG binding protein
FCN2 ficolin (collagen/fibrinogen domain containing lectin) 2
FZD4 frizzled class receptor 4
GAS1 growth arrest-specific 1
GATA6 GATA binding protein 6
GPRC5B G protein-coupled receptor, class C, group 5, member B
GRK4 G protein-coupled receptor kinase 4
GSTT1 glutathione S-transferase theta 1
GUCY1A3 guanylate cyclase 1, soluble, alpha 3
HNF4A hepatocyte nuclear factor 4, alpha
HNRNPDL heterogeneous nuclear ribonucleoprotein D-like
HPSE2 heparanase 2 (inactive)
HR hair growth associated
IGFBP5 insulin-like growth factor binding protein 5
IGLL1 immunoglobulin lambda-like polypeptide 1
KCNK1 potassium channel, two pore domain subfamily K, member 1
KIR2DS4 killer cell immunoglobulin-like receptor, two domains, short cytoplasmic tail, 4
KIT v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog
KLK7 kallikrein-related peptidase 7
KRT17 keratin 17, type I
LARGE like-glycosyltransferase
LPPR1 lipid phosphate phosphatase-related protein type 1
MAGI2 membrane associated guanylate kinase, WW and PDZ domain containing 2
MAP9 microtubule-associated protein 9
MC3R melanocortin 3 receptor
MDK midkine (neurite growth-promoting factor 2)
MFAP3L microfibrillar-associated protein 3-like
MMP24 matrix metallopeptidase 24 (membrane-inserted)
MPPE1 metallophosphoesterase 1
MSTN myostatin
MUSK muscle, skeletal, receptor tyrosine kinase
NFKBIB nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, beta
NRAP nebulin-related anchoring protein
PARVA parvin, alpha
PCP4 Purkinje cell protein 4
PLN phospholamban
POU1F1 POU class 1 homeobox 1
PPP1R1A protein phosphatase 1, regulatory (inhibitor) subunit 1A
PPP2CB protein phosphatase 2, catalytic subunit, beta isozyme
PRSS2 protease, serine, 2 (trypsin 2)
PSG11 pregnancy specific beta-1-glycoprotein 11
RAD51B RAD51 paralog B
RDH8 retinol dehydrogenase 8 (all-trans)
RELN reelin
RTEL1 regulator of telomere elongation helicase 1
RUNDC3A RUN domain containing 3A
SEMA3C sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3C
SH3BP1 SH3-domain binding protein 1
SIGLEC8 sialic acid binding Ig-like lectin 8
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC22A7 solute carrier family 22 (organic anion transporter), member 7
SLC9A3 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3
SNTB2 syntrophin, beta 2 (dystrophin-associated protein A1, 59kDa, basic component 2)
SRPX2 sushi-repeat containing protein, X-linked 2
ST3GAL2 ST3 beta-galactoside alpha-2,3-sialyltransferase 2
SVIL supervillin
SYNM synemin, intermediate filament protein
TAAR5 trace amine associated receptor 5
TACSTD2 tumor-associated calcium signal transducer 2
THSD7A thrombospondin, type I, domain containing 7A
TMEM140 transmembrane protein 140
TNFSF11 tumor necrosis factor (ligand) superfamily, member 11
TNP2 transition protein 2 (during histone to protamine replacement)
TOX thymocyte selection-associated high mobility group box
TRBC1 T cell receptor beta constant 1
TSKU tsukushi, small leucine rich proteoglycan
TSR3 TSR3, 20S rRNA accumulation, homolog (S. cerevisiae)
TYMP thymidine phosphorylase
UGT2B17 UDP glucuronosyltransferase 2 family, polypeptide B17
UNC119 unc-119 homolog (C. elegans)
ZCCHC14 zinc finger, CCHC domain containing 14
ZNF287 zinc finger protein 287
ZNF407 zinc finger protein 407
ZZEF1 zinc finger, ZZ-type with EF-hand domain 1

decreased expression

Symbol Name
ACAD10 acyl-CoA dehydrogenase family, member 10
ACPP acid phosphatase, prostate
ACTR8 ARP8 actin-related protein 8 homolog (yeast)
ALDOAP2 aldolase A, fructose-bisphosphate pseudogene 2
AP1G2 adaptor-related protein complex 1, gamma 2 subunit
BAG4 BCL2-associated athanogene 4
BAHD1 bromo adjacent homology domain containing 1
BSPRY B-box and SPRY domain containing
C17ORF53 chromosome 17 open reading frame 53
CCDC106 coiled-coil domain containing 106
CCDC186 coiled-coil domain containing 186
CCL20 chemokine (C-C motif) ligand 20
CD82 CD82 molecule
CDKL1 cyclin-dependent kinase-like 1 (CDC2-related kinase)
CHPF chondroitin polymerizing factor
CWF19L1 CWF19-like 1, cell cycle control (S. pombe)
DDX31 DEAD (Asp-Glu-Ala-Asp) box polypeptide 31
DENND1A DENN/MADD domain containing 1A
DEPDC5 DEP domain containing 5
DHRS11 dehydrogenase/reductase (SDR family) member 11
DOLK dolichol kinase
DTX2 deltex 2, E3 ubiquitin ligase
EDAR ectodysplasin A receptor
FCGR1A Fc fragment of IgG, high affinity Ia, receptor (CD64)
FCHO1 FCH domain only 1
FLJ21369 uncharacterized protein FLJ21369
GALK1 galactokinase 1
GALNT12 polypeptide N-acetylgalactosaminyltransferase 12
GBP2 guanylate binding protein 2, interferon-inducible
GJA1 gap junction protein, alpha 1, 43kDa
GPATCH2L G patch domain containing 2-like
GSDMD gasdermin D
HERC4 HECT and RLD domain containing E3 ubiquitin protein ligase 4
HIST1H1B histone cluster 1, H1b
HIST1H2AJ histone cluster 1, H2aj
HIST1H3G histone cluster 1, H3g
HNRNPA3P1 heterogeneous nuclear ribonucleoprotein A3 pseudogene 1
HOXB9 homeobox B9
HYOU1 hypoxia up-regulated 1
KLF2 Kruppel-like factor 2
KPNA5 karyopherin alpha 5 (importin alpha 6)
LOC100286895 cell division cycle 27 homolog pseudogene
LOC100287590 uncharacterized LOC100287590
LRRC20 leucine rich repeat containing 20
MAGEH1 melanoma antigen family H1
MCPH1 microcephalin 1
MPZ myelin protein zero
MRPL44 mitochondrial ribosomal protein L44
MX2 MX dynamin-like GTPase 2
MXD3 MAX dimerization protein 3
NAT6 N-acetyltransferase 6 (GCN5-related)
NFE2L3 nuclear factor, erythroid 2-like 3
NIPAL2 NIPA-like domain containing 2
NSUN6 NOP2/Sun domain family, member 6
OTUD3 OTU deubiquitinase 3
PDE6B phosphodiesterase 6B, cGMP-specific, rod, beta
PGGT1B protein geranylgeranyltransferase type I, beta subunit
PHC1 polyhomeotic homolog 1 (Drosophila)
PLA2G7 phospholipase A2, group VII (platelet-activating factor acetylhydrolase, plasma)
PMFBP1 polyamine modulated factor 1 binding protein 1
PTCD1 pentatricopeptide repeat domain 1
RAB33A RAB33A, member RAS oncogene family
RAPGEFL1 Rap guanine nucleotide exchange factor (GEF)-like 1
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RIC8B RIC8 guanine nucleotide exchange factor B
RPL23AP32 ribosomal protein L23a pseudogene 32
SKA1 spindle and kinetochore associated complex subunit 1
SLC15A3 solute carrier family 15 (oligopeptide transporter), member 3
SLC17A2 solute carrier family 17, member 2
SLC35F5 solute carrier family 35, member F5
SP1 Sp1 transcription factor
SPATA20 spermatogenesis associated 20
SPATA2L spermatogenesis associated 2-like
SREBF1 sterol regulatory element binding transcription factor 1
ST8SIA4 ST8 alpha-N-acetyl-neuraminide alpha-2,8-sialyltransferase 4
STAG3L4 stromal antigen 3-like 4 (pseudogene)
SYNC syncoilin, intermediate filament protein
TAF13 TAF13 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 18kDa
TEC tec protein tyrosine kinase
TMEM209 transmembrane protein 209
TMEM8A transmembrane protein 8A
TNFRSF14 tumor necrosis factor receptor superfamily, member 14
TOM1 target of myb1 (chicken)
TRAF2 TNF receptor-associated factor 2
TRIM36 tripartite motif containing 36
TRPC5 transient receptor potential cation channel, subfamily C, member 5
TSC22D4 TSC22 domain family, member 4
TSPYL2 TSPY-like 2
YIPF1 Yip1 domain family, member 1
YY2 YY2 transcription factor
ZNF10 zinc finger protein 10
ZNF225 zinc finger protein 225
ZNF286A zinc finger protein 286A
ZNF428 zinc finger protein 428
ZNF574 zinc finger protein 574
ZNF668 zinc finger protein 668
ZNF675 zinc finger protein 675
ZNF862 zinc finger protein 862