Prestwick-864-2994 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the Prestwick-864-2994 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAMDC adipogenesis associated, Mth938 domain containing
ABAT 4-aminobutyrate aminotransferase
ABHD6 abhydrolase domain containing 6
ALDH3A1 aldehyde dehydrogenase 3 family, member A1
APPBP2 amyloid beta precursor protein (cytoplasmic tail) binding protein 2
ART4 ADP-ribosyltransferase 4 (Dombrock blood group)
ASAP3 ArfGAP with SH3 domain, ankyrin repeat and PH domain 3
ATP2A3 ATPase, Ca++ transporting, ubiquitous
ATP2B3 ATPase, Ca++ transporting, plasma membrane 3
BAAT bile acid CoA:amino acid N-acyltransferase
BCL2L1 BCL2-like 1
BMP7 bone morphogenetic protein 7
C11ORF1 chromosome 11 open reading frame 1
CACNG2 calcium channel, voltage-dependent, gamma subunit 2
CCDC81 coiled-coil domain containing 81
CEACAM3 carcinoembryonic antigen-related cell adhesion molecule 3
CEACAM7 carcinoembryonic antigen-related cell adhesion molecule 7
CHST7 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 7
CMAHP cytidine monophospho-N-acetylneuraminic acid hydroxylase, pseudogene
CNNM1 cyclin and CBS domain divalent metal cation transport mediator 1
COL2A1 collagen, type II, alpha 1
CYP4F11 cytochrome P450, family 4, subfamily F, polypeptide 11
DCBLD2 discoidin, CUB and LCCL domain containing 2
DCTN2 dynactin 2 (p50)
DDR1 discoidin domain receptor tyrosine kinase 1
DGCR5 DiGeorge syndrome critical region gene 5 (non-protein coding)
DRD2 dopamine receptor D2
DSCR4 Down syndrome critical region 4
DSTYK dual serine/threonine and tyrosine protein kinase
EFNB3 ephrin-B3
ENPP1 ectonucleotide pyrophosphatase/phosphodiesterase 1
EPHB2 EPH receptor B2
EXOG endo/exonuclease (5'-3'), endonuclease G-like
FGFR2 fibroblast growth factor receptor 2
FZD3 frizzled class receptor 3
FZD9 frizzled class receptor 9
GHRH growth hormone releasing hormone
GIF gastric intrinsic factor (vitamin B synthesis)
GJA8 gap junction protein, alpha 8, 50kDa
GNB1L guanine nucleotide binding protein (G protein), beta polypeptide 1-like
GOLGA2P5 golgin A2 pseudogene 5
GSPT2 G1 to S phase transition 2
GULP1 GULP, engulfment adaptor PTB domain containing 1
HEMK1 HemK methyltransferase family member 1
HOXA4 homeobox A4
HOXB3 homeobox B3
IGFBP3 insulin-like growth factor binding protein 3
KLHL18 kelch-like family member 18
KRT14 keratin 14, type I
LAMP1 lysosomal-associated membrane protein 1
LIMD1 LIM domains containing 1
LINC01587 long intergenic non-protein coding RNA 1587
LZTS1 leucine zipper, putative tumor suppressor 1
MAP9 microtubule-associated protein 9
MARC1 mitochondrial amidoxime reducing component 1
MCAM melanoma cell adhesion molecule
MS4A5 membrane-spanning 4-domains, subfamily A, member 5
MYOD1 myogenic differentiation 1
MYOM1 myomesin 1
NCOR2 nuclear receptor corepressor 2
NDUFA2 NADH dehydrogenase (ubiquinone) 1 alpha subcomplex, 2, 8kDa
NFKB2 nuclear factor of kappa light polypeptide gene enhancer in B-cells 2 (p49/p100)
ONECUT2 one cut homeobox 2
PACRG PARK2 co-regulated
PALLD palladin, cytoskeletal associated protein
PAWR PRKC, apoptosis, WT1, regulator
PCDHA5 protocadherin alpha 5
PITPNM3 PITPNM family member 3
PLA2G5 phospholipase A2, group V
PMEPA1 prostate transmembrane protein, androgen induced 1
PODNL1 podocan-like 1
PPP1R3A protein phosphatase 1, regulatory subunit 3A
PTGER3 prostaglandin E receptor 3 (subtype EP3)
PVR poliovirus receptor
RAB11B RAB11B, member RAS oncogene family
RENBP renin binding protein
RFPL1 ret finger protein-like 1
RFX2 regulatory factor X, 2 (influences HLA class II expression)
ROR1 receptor tyrosine kinase-like orphan receptor 1
SH3BP1 SH3-domain binding protein 1
SLAMF7 SLAM family member 7
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC1A7 solute carrier family 1 (glutamate transporter), member 7
SLC6A20 solute carrier family 6 (proline IMINO transporter), member 20
SNRNP200 small nuclear ribonucleoprotein 200kDa (U5)
STXBP6 syntaxin binding protein 6 (amisyn)
TMEM242 transmembrane protein 242
TMPRSS4 transmembrane protease, serine 4
TNFRSF25 tumor necrosis factor receptor superfamily, member 25
TPMT thiopurine S-methyltransferase
TRPC7 transient receptor potential cation channel, subfamily C, member 7
TSKS testis-specific serine kinase substrate
TSPAN2 tetraspanin 2
ZBTB17 zinc finger and BTB domain containing 17
ZNF133 zinc finger protein 133
ZNF442 zinc finger protein 442
ZNF688 zinc finger protein 688
ZNF783 zinc finger family member 783
ZNF814 zinc finger protein 814

decreased expression

Symbol Name
ABL2 ABL proto-oncogene 2, non-receptor tyrosine kinase
ADGRD2 adhesion G protein-coupled receptor D2
ALDOAP2 aldolase A, fructose-bisphosphate pseudogene 2
AP5S1 adaptor-related protein complex 5, sigma 1 subunit
APOBEC3C apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3C
BIRC3 baculoviral IAP repeat containing 3
CACNB4 calcium channel, voltage-dependent, beta 4 subunit
CAMKMT calmodulin-lysine N-methyltransferase
CCDC33 coiled-coil domain containing 33
CCDC71 coiled-coil domain containing 71
CFAP69 cilia and flagella associated protein 69
CLGN calmegin
COPG2IT1 COPG2 imprinted transcript 1 (non-protein coding)
CROT carnitine O-octanoyltransferase
CTAGE9 CTAGE family, member 9
CYP2W1 cytochrome P450, family 2, subfamily W, polypeptide 1
DDX58 DEAD (Asp-Glu-Ala-Asp) box polypeptide 58
DHRS3 dehydrogenase/reductase (SDR family) member 3
EHD3 EH-domain containing 3
FAM86C1 family with sequence similarity 86, member C1
FBXL7 F-box and leucine-rich repeat protein 7
FBXO40 F-box protein 40
FBXW4P1 F-box and WD repeat domain containing 4 pseudogene 1
FCGR1A Fc fragment of IgG, high affinity Ia, receptor (CD64)
FRMPD1 FERM and PDZ domain containing 1
GABRA4 gamma-aminobutyric acid (GABA) A receptor, alpha 4
GABRP gamma-aminobutyric acid (GABA) A receptor, pi
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GID4 GID complex subunit 4
GNRH1 gonadotropin-releasing hormone 1 (luteinizing-releasing hormone)
GPR35 G protein-coupled receptor 35
HDAC7 histone deacetylase 7
HIST1H1T histone cluster 1, H1t
HOXA6 homeobox A6
HOXD10 homeobox D10
IBSP integrin-binding sialoprotein
IFT140 intraflagellar transport 140
IFT54 intraflagellar transport 54
IL12B interleukin 12B
INO80D INO80 complex subunit D
ITGA10 integrin, alpha 10
KCNA6 potassium channel, voltage gated shaker related subfamily A, member 6
KCNK12 potassium channel, two pore domain subfamily K, member 12
LIME1 Lck interacting transmembrane adaptor 1
LIN7A lin-7 homolog A (C. elegans)
MAGEH1 melanoma antigen family H1
MAP3K14 mitogen-activated protein kinase kinase kinase 14
MAP3K8 mitogen-activated protein kinase kinase kinase 8
MAP6D1 MAP6 domain containing 1
MUC2 mucin 2, oligomeric mucus/gel-forming
MUC6 mucin 6, oligomeric mucus/gel-forming
NME8 NME/NM23 family member 8
NMUR1 neuromedin U receptor 1
NPFFR1 neuropeptide FF receptor 1
PARP11 poly (ADP-ribose) polymerase family, member 11
PDE12 phosphodiesterase 12
PDLIM2 PDZ and LIM domain 2 (mystique)
PIP prolactin-induced protein
PITX2 paired-like homeodomain 2
PLA2G3 phospholipase A2, group III
PLAT plasminogen activator, tissue
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PRDM12 PR domain containing 12
PROX1 prospero homeobox 1
RAB33A RAB33A, member RAS oncogene family
RAB40A RAB40A, member RAS oncogene family
RABL6 RAB, member RAS oncogene family-like 6
RAC3 ras-related C3 botulinum toxin substrate 3 (rho family, small GTP binding protein Rac3)
RBFOX1 RNA binding protein, fox-1 homolog (C. elegans) 1
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RPL23AP32 ribosomal protein L23a pseudogene 32
SCRT1 scratch family zinc finger 1
SETD1A SET domain containing 1A
SGCE sarcoglycan, epsilon
SGPP1 sphingosine-1-phosphate phosphatase 1
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SLFN12 schlafen family member 12
SLITRK5 SLIT and NTRK-like family, member 5
SNAI1 snail family zinc finger 1
SRPX sushi-repeat containing protein, X-linked
STARD13 StAR-related lipid transfer (START) domain containing 13
SYNJ2BP synaptojanin 2 binding protein
TFDP3 transcription factor Dp family, member 3
TIAM2 T-cell lymphoma invasion and metastasis 2
TMEM140 transmembrane protein 140
TMEM206 transmembrane protein 206
TTC30A tetratricopeptide repeat domain 30A
UNKL unkempt family zinc finger-like
UPK3A uroplakin 3A
USP27X ubiquitin specific peptidase 27, X-linked
YY2 YY2 transcription factor
ZC3H3 zinc finger CCCH-type containing 3
ZFHX3 zinc finger homeobox 3
ZNF155 zinc finger protein 155
ZNF345 zinc finger protein 345
ZNF711 zinc finger protein 711
ZNF747 zinc finger protein 747
ZNF816 zinc finger protein 816