Rimonabant_COLO 205 Gene Set

Dataset Tahoe Therapeutics Tahoe 100M Perturbation Atlas
Category transcriptomics
Type cell type
Description Rimonabant perturbation in COLO 205 cell line (Tahoe Therapeutics)
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Genes

200 genes differentially expressed following the Rimonabant_COLO 205 drug perturbation from the Tahoe Therapeutics Tahoe 100M Perturbation Atlas dataset.

increased expression

Symbol Name Standardized Value
SMAD3 SMAD family member 3 0.0895886
STS steroid sulfatase (microsomal), isozyme S 0.089024
DNAJC15 DnaJ (Hsp40) homolog, subfamily C, member 15 0.0839894
CHST11 carbohydrate (chondroitin 4) sulfotransferase 11 0.0763597
EXT1 exostosin glycosyltransferase 1 0.0727262
LMO7 LIM domain 7 0.0692886
GMDS GDP-mannose 4,6-dehydratase 0.0637777
CYP3A5 cytochrome P450, family 3, subfamily A, polypeptide 5 0.0612545
RNF213 ring finger protein 213 0.0554452
ARHGAP26 Rho GTPase activating protein 26 0.0542994
VCL vinculin 0.0508969
SHB Src homology 2 domain containing adaptor protein B 0.0505035
CEMIP cell migration inducing protein, hyaluronan binding 0.0504014
AKAP13 A kinase (PRKA) anchor protein 13 0.0473751
ABCA1 ATP-binding cassette, sub-family A (ABC1), member 1 0.0467934
MX2 MX dynamin-like GTPase 2 0.0463162
BCL2L1 BCL2-like 1 0.0458666
HCN1 hyperpolarization activated cyclic nucleotide gated potassium channel 1 0.0436001
ITGA6 integrin, alpha 6 0.0433927
ANXA2 annexin A2 0.0426482
TNFRSF21 tumor necrosis factor receptor superfamily, member 21 0.0417469
TSHZ2 teashirt zinc finger homeobox 2 0.0415327
SNTB1 syntrophin, beta 1 (dystrophin-associated protein A1, 59kDa, basic component 1) 0.0411694
MSI2 musashi RNA-binding protein 2 0.0410415
MYH9 myosin, heavy chain 9, non-muscle 0.0409157
MX1 MX dynamin-like GTPase 1 0.0407877
LRCH1 leucine-rich repeats and calponin homology (CH) domain containing 1 0.039008
MLPH melanophilin 0.0384438
SIPA1L2 signal-induced proliferation-associated 1 like 2 0.0383806
C6ORF132 chromosome 6 open reading frame 132 0.0368349
NFAT5 nuclear factor of activated T-cells 5, tonicity-responsive 0.0363376
CTBP2 C-terminal binding protein 2 0.0352723
EPB41L1 erythrocyte membrane protein band 4.1-like 1 0.035145
SLC2A1 solute carrier family 2 (facilitated glucose transporter), member 1 0.0338755
CATSPERB catsper channel auxiliary subunit beta 0.0334229
IGF1R insulin-like growth factor 1 receptor 0.0332362
ERBIN erbb2 interacting protein 0.0329313
RSAD2 radical S-adenosyl methionine domain containing 2 0.0326736
LCN2 lipocalin 2 0.0320441
MYO1E myosin IE 0.0315292
EPHB2 EPH receptor B2 0.0309408
IMMP2L IMP2 inner mitochondrial membrane peptidase-like (S. cerevisiae) 0.0308358
MYH14 myosin, heavy chain 14, non-muscle 0.0307947
BAIAP2L1 BAI1-associated protein 2-like 1 0.0304619
ETV6 ets variant 6 0.0301975
SPATA13 spermatogenesis associated 13 0.0298932
MYO5B myosin VB 0.0296154
ATP10B ATPase, class V, type 10B 0.0295622
ABCC3 ATP-binding cassette, sub-family C (CFTR/MRP), member 3 0.0294899
ACTN4 actinin, alpha 4 0.0294763
SLC12A2 solute carrier family 12 (sodium/potassium/chloride transporter), member 2 0.0294495
INTS6 integrator complex subunit 6 0.0290458
CTNNA1 catenin (cadherin-associated protein), alpha 1, 102kDa 0.0280748
NIBAN2 niban apoptosis regulator 2 0.0279512
IFIT2 interferon-induced protein with tetratricopeptide repeats 2 0.0278332
TM4SF19 transmembrane 4 L six family member 19 0.0275951
MAML2 mastermind-like 2 (Drosophila) 0.0273516
LPP LIM domain containing preferred translocation partner in lipoma 0.0269466
DDX60 DEAD (Asp-Glu-Ala-Asp) box polypeptide 60 0.0266613
ZHX2 zinc fingers and homeoboxes 2 0.0263793
ITGA2 integrin, alpha 2 (CD49B, alpha 2 subunit of VLA-2 receptor) 0.0261851
SEPTIN9 septin 9 0.0260161
PITPNC1 phosphatidylinositol transfer protein, cytoplasmic 1 0.0257601
GAREM1 GRB2 associated regulator of MAPK1 subtype 1 0.0256844
EFNB2 ephrin-B2 0.0249778
NKD1 naked cuticle homolog 1 (Drosophila) 0.0244871
FHIT fragile histidine triad 0.0240911
IFIT1 interferon-induced protein with tetratricopeptide repeats 1 0.0236552
OAS1 2'-5'-oligoadenylate synthetase 1, 40/46kDa 0.0230787
HNRNPA2B1 heterogeneous nuclear ribonucleoprotein A2/B1 0.0230703
RIGI RNA sensor RIG-I 0.0229608
KYNU kynureninase 0.0229105
SP100 SP100 nuclear antigen 0.0225073
DIAPH1 diaphanous-related formin 1 0.0218915
ARHGAP27 Rho GTPase activating protein 27 0.0217698
LURAP1L leucine rich adaptor protein 1-like 0.02172
IGFBP3 insulin-like growth factor binding protein 3 0.0215793
PRSS3 protease, serine, 3 0.0212396
VPS37B vacuolar protein sorting 37 homolog B (S. cerevisiae) 0.0211986
FAT1 FAT atypical cadherin 1 0.0211084
AREG amphiregulin 0.0206085
ANKRD10 ankyrin repeat domain 10 0.0202128
AFAP1L2 actin filament associated protein 1-like 2 0.0201411
FHL2 four and a half LIM domains 2 0.0201316
NCEH1 neutral cholesterol ester hydrolase 1 0.0199451
PLSCR2 phospholipid scramblase 2 0.0199217
EPHA2 EPH receptor A2 0.0195154
SLK STE20-like kinase 0.0194858
SH3PXD2A SH3 and PX domains 2A 0.0193887
WWOX WW domain containing oxidoreductase 0.0192867
DIP2B DIP2 disco-interacting protein 2 homolog B (Drosophila) 0.0190378
SIPA1L1 signal-induced proliferation-associated 1 like 1 0.019006
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor) 0.0188127
TNS4 tensin 4 0.0186688
HDAC4 histone deacetylase 4 0.0185941
PPP1R15A protein phosphatase 1, regulatory subunit 15A 0.0185726
SAMD9 sterile alpha motif domain containing 9 0.0184362
ANXA11 annexin A11 0.0184304
DDX60L DEAD (Asp-Glu-Ala-Asp) box polypeptide 60-like 0.0183358
DUSP10 dual specificity phosphatase 10 0.0182839

decreased expression

Symbol Name Standardized Value
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1 -0.269723
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) -0.138693
TPT1 tumor protein, translationally-controlled 1 -0.123875
MBNL2 muscleblind-like splicing regulator 2 -0.120088
B2M beta-2-microglobulin -0.11946
UBR2 ubiquitin protein ligase E3 component n-recognin 2 -0.107215
PDIA3 protein disulfide isomerase family A, member 3 -0.0983146
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3 -0.0965049
P4HA1 prolyl 4-hydroxylase, alpha polypeptide I -0.089987
AHI1 Abelson helper integration site 1 -0.0873765
GOLGB1 golgin B1 -0.0862492
CANX calnexin -0.0832494
FNDC3A fibronectin type III domain containing 3A -0.0704431
BTBD9 BTB (POZ) domain containing 9 -0.0693681
GFPT1 glutamine--fructose-6-phosphate transaminase 1 -0.0662284
TTC3 tetratricopeptide repeat domain 3 -0.0650321
EIF1 eukaryotic translation initiation factor 1 -0.0643866
P4HB prolyl 4-hydroxylase, beta polypeptide -0.0636101
PTMA prothymosin, alpha -0.062105
SEC31A SEC31 homolog A (S. cerevisiae) -0.0607519
ANKHD1 ankyrin repeat and KH domain containing 1 -0.0579529
TXNIP thioredoxin interacting protein -0.05775
TM9SF2 transmembrane 9 superfamily member 2 -0.0574001
NCKAP5 NCK-associated protein 5 -0.0563555
BCLAF1 BCL2-associated transcription factor 1 -0.0562237
GAPDH glyceraldehyde-3-phosphate dehydrogenase -0.0560653
RPS6 ribosomal protein S6 -0.0551801
PABPC1 poly(A) binding protein, cytoplasmic 1 -0.0532111
RBM39 RNA binding motif protein 39 -0.05121
PERP PERP, TP53 apoptosis effector -0.0510006
IFNGR1 interferon gamma receptor 1 -0.0507918
TOP2A topoisomerase (DNA) II alpha 170kDa -0.0500788
ARL6IP1 ADP-ribosylation factor-like 6 interacting protein 1 -0.0490727
GOLGA4 golgin A4 -0.0490252
AKAP9 A kinase (PRKA) anchor protein 9 -0.0486175
EPCAM epithelial cell adhesion molecule -0.048012
PTBP3 polypyrimidine tract binding protein 3 -0.0469607
COG6 component of oligomeric golgi complex 6 -0.0469459
RHOBTB3 Rho-related BTB domain containing 3 -0.0462563
SEC24D SEC24 family member D -0.0459719
DIS3 DIS3 exosome endoribonuclease and 3'-5' exoribonuclease -0.0443791
N4BP2L2 NEDD4 binding protein 2-like 2 -0.0442056
CLTC clathrin, heavy chain (Hc) -0.0441217
RRBP1 ribosome binding protein 1 -0.0429439
PIBF1 progesterone immunomodulatory binding factor 1 -0.0425342
ATP1B1 ATPase, Na+/K+ transporting, beta 1 polypeptide -0.0424644
WSB1 WD repeat and SOCS box containing 1 -0.042369
HLA-B major histocompatibility complex, class I, B -0.0423278
RAB1A RAB1A, member RAS oncogene family -0.0415577
DSCAM Down syndrome cell adhesion molecule -0.0415231
SUCO SUN domain containing ossification factor -0.0410548
ACBD3 acyl-CoA binding domain containing 3 -0.0405943
ZMYM2 zinc finger, MYM-type 2 -0.0402721
DSTN destrin (actin depolymerizing factor) -0.0397449
CPEB4 cytoplasmic polyadenylation element binding protein 4 -0.0394726
ARID4B AT rich interactive domain 4B (RBP1-like) -0.0394501
PIK3C2A phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 alpha -0.0391927
CEP350 centrosomal protein 350kDa -0.0384722
SBF2 SET binding factor 2 -0.0379709
HM13 histocompatibility (minor) 13 -0.0375129
AP3B1 adaptor-related protein complex 3, beta 1 subunit -0.0372091
DHRS3 dehydrogenase/reductase (SDR family) member 3 -0.0366231
CALR calreticulin -0.0363693
ZNF292 zinc finger protein 292 -0.0362037
COPA coatomer protein complex, subunit alpha -0.0361942
ZKSCAN1 zinc finger with KRAB and SCAN domains 1 -0.0361248
MORF4L2 mortality factor 4 like 2 -0.0358837
DIAPH3 diaphanous-related formin 3 -0.0354893
CALU calumenin -0.0351371
COPB1 coatomer protein complex, subunit beta 1 -0.0350074
KMT2C lysine (K)-specific methyltransferase 2C -0.0349766
PDIA4 protein disulfide isomerase family A, member 4 -0.0347513
UBC ubiquitin C -0.0342868
PATJ PATJ crumbs cell polarity complex component -0.0341445
KMT2E lysine (K)-specific methyltransferase 2E -0.0337391
IRF1 interferon regulatory factor 1 -0.0334717
ASH1L ash1 (absent, small, or homeotic)-like (Drosophila) -0.0327746
FNIP1 folliculin interacting protein 1 -0.0327585
PTEN phosphatase and tensin homolog -0.0321311
PHF3 PHD finger protein 3 -0.0320063
NUFIP2 nuclear fragile X mental retardation protein interacting protein 2 -0.0319304
TMEM263 transmembrane protein 263 -0.0319045
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3 -0.0317615
SSR1 signal sequence receptor, alpha -0.0316383
SEC24A SEC24 family member A -0.0314565
GCC2 GRIP and coiled-coil domain containing 2 -0.0312403
MON2 MON2 homolog (S. cerevisiae) -0.0311582
UFM1 ubiquitin-fold modifier 1 -0.031108
PRRC1 proline-rich coiled-coil 1 -0.0310472
CCNL1 cyclin L1 -0.0309585
COPB2 coatomer protein complex, subunit beta 2 (beta prime) -0.0307334
BPTF bromodomain PHD finger transcription factor -0.0307262
NUCB2 nucleobindin 2 -0.0307018
MEIS2 Meis homeobox 2 -0.0305711
SREBF2 sterol regulatory element binding transcription factor 2 -0.0305571
NF1 neurofibromin 1 -0.0303626
GOLPH3L golgi phosphoprotein 3-like -0.030358
MINDY2 MINDY lysine 48 deubiquitinase 2 -0.0303262
RPL12 ribosomal protein L12 -0.0301604
ERC2 ELKS/RAB6-interacting/CAST family member 2 -0.0298157