TAK-715 Gene Set

Dataset LINCS KinomeScan Kinase Inhibitor Targets
Category physical interactions
Type small molecule
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Genes

22 kinases inhibited by the TAK-715 small molecule from the KinomeScan Kinase Inhibitor Targets dataset.

Symbol Name Standardized Value
CSNK1E casein kinase 1, epsilon 1.36211
ADCK3 aarF domain containing kinase 3 1.35325
CIT citron rho-interacting serine/threonine kinase 1.32726
MAP4K4 mitogen-activated protein kinase kinase kinase kinase 4 1.28583
RIPK2 receptor-interacting serine-threonine kinase 2 1.26991
CSNK1A1L casein kinase 1, alpha 1-like 1.26209
TGFBR1 transforming growth factor, beta receptor 1 1.22432
CSNK1D casein kinase 1, delta 1.20983
ADCK4 aarF domain containing kinase 4 1.19568
ERBB4 erb-b2 receptor tyrosine kinase 4 1.15523
DDR1 discoidin domain receptor tyrosine kinase 1 1.15523
EGFR epidermal growth factor receptor 1.09415
NLK nemo-like kinase 1.08283
GAK cyclin G associated kinase 1.06105
ACVR1B activin A receptor, type IB 1.05057
STK36 serine/threonine kinase 36 1.04035
TNIK TRAF2 and NCK interacting kinase 1.00664
YES1 YES proto-oncogene 1, Src family tyrosine kinase 1.00208
STK32B serine/threonine kinase 32B 0.944052
MINK1 misshapen-like kinase 1 0.895762
ZAK sterile alpha motif and leucine zipper containing kinase AZK 0.866209
ACVR1 activin A receptor, type I 0.860727