ampyrone-1402 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the ampyrone-1402 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADGRB2 adhesion G protein-coupled receptor B2
ADK adenosine kinase
AGPAT2 1-acylglycerol-3-phosphate O-acyltransferase 2
ALX3 ALX homeobox 3
ANKRD12 ankyrin repeat domain 12
APH1B APH1B gamma secretase subunit
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BAMBI BMP and activin membrane-bound inhibitor
BIRC7 baculoviral IAP repeat containing 7
BMP2K BMP2 inducible kinase
C2ORF54 chromosome 2 open reading frame 54
C7ORF43 chromosome 7 open reading frame 43
CACNA1A calcium channel, voltage-dependent, P/Q type, alpha 1A subunit
CALB2 calbindin 2
CAMKV CaM kinase-like vesicle-associated
CC2D1A coiled-coil and C2 domain containing 1A
CDH6 cadherin 6, type 2, K-cadherin (fetal kidney)
CHRNA2 cholinergic receptor, nicotinic, alpha 2 (neuronal)
CIITA class II, major histocompatibility complex, transactivator
CLTA clathrin, light chain A
COMT catechol-O-methyltransferase
CORT cortistatin
CPM carboxypeptidase M
CPTP ceramide-1-phosphate transfer protein
CROT carnitine O-octanoyltransferase
CYP27A1 cytochrome P450, family 27, subfamily A, polypeptide 1
DGCR11 DiGeorge syndrome critical region gene 11 (non-protein coding)
DIP2C DIP2 disco-interacting protein 2 homolog C (Drosophila)
DUSP26 dual specificity phosphatase 26 (putative)
EFNB3 ephrin-B3
EFR3B EFR3 homolog B (S. cerevisiae)
EIF4E eukaryotic translation initiation factor 4E
ERN2 endoplasmic reticulum to nucleus signaling 2
FBRS fibrosin
FGF6 fibroblast growth factor 6
FGFR1 fibroblast growth factor receptor 1
GAP43 growth associated protein 43
GIT1 G protein-coupled receptor kinase interacting ArfGAP 1
GNL1 guanine nucleotide binding protein-like 1
GPX3 glutathione peroxidase 3
H6PD hexose-6-phosphate dehydrogenase (glucose 1-dehydrogenase)
HAMP hepcidin antimicrobial peptide
IBSP integrin-binding sialoprotein
IGHA1 immunoglobulin heavy constant alpha 1
KCNF1 potassium channel, voltage gated modifier subfamily F, member 1
LAMA2 laminin, alpha 2
LILRA4 leukocyte immunoglobulin-like receptor, subfamily A (with TM domain), member 4
LILRB3 leukocyte immunoglobulin-like receptor, subfamily B (with TM and ITIM domains), member 3
LIMS2 LIM and senescent cell antigen-like domains 2
MAP1A microtubule-associated protein 1A
MAP1B microtubule-associated protein 1B
MFSD11 major facilitator superfamily domain containing 11
MIIP migration and invasion inhibitory protein
MMP25 matrix metallopeptidase 25
MOB3B MOB kinase activator 3B
MT3 metallothionein 3
MUC5AC mucin 5AC, oligomeric mucus/gel-forming
MYF6 myogenic factor 6 (herculin)
NPEPL1 aminopeptidase-like 1
OR10H1 olfactory receptor, family 10, subfamily H, member 1
PDE8B phosphodiesterase 8B
PELP1 proline, glutamate and leucine rich protein 1
PFKFB2 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 2
PHF3 PHD finger protein 3
PLCG1 phospholipase C, gamma 1
POMT2 protein-O-mannosyltransferase 2
POU5F1B POU class 5 homeobox 1B
PPARA peroxisome proliferator-activated receptor alpha
PRB1 proline-rich protein BstNI subfamily 1
PRB3 proline-rich protein BstNI subfamily 3
RAB2A RAB2A, member RAS oncogene family
RAB40B RAB40B, member RAS oncogene family
RAMP1 receptor (G protein-coupled) activity modifying protein 1
RARA retinoic acid receptor, alpha
ROBO4 roundabout, axon guidance receptor, homolog 4 (Drosophila)
RPL7 ribosomal protein L7
SAMD14 sterile alpha motif domain containing 14
SCN5A sodium channel, voltage gated, type V alpha subunit
SCNN1A sodium channel, non voltage gated 1 alpha subunit
SH2B1 SH2B adaptor protein 1
SLC12A4 solute carrier family 12 (potassium/chloride transporter), member 4
SLC22A18AS solute carrier family 22 (organic cation transporter), member 18 antisense
SLC6A11 solute carrier family 6 (neurotransmitter transporter), member 11
SNAP25 synaptosomal-associated protein, 25kDa
SPATA2L spermatogenesis associated 2-like
SPDEF SAM pointed domain containing ETS transcription factor
TMCC2 transmembrane and coiled-coil domain family 2
TTF2 transcription termination factor, RNA polymerase II
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
UBQLN4 ubiquilin 4
UBTD1 ubiquitin domain containing 1
VDR vitamin D (1,25- dihydroxyvitamin D3) receptor
VGF VGF nerve growth factor inducible
VIPR2 vasoactive intestinal peptide receptor 2
ZC3H7B zinc finger CCCH-type containing 7B
ZFHX2 zinc finger homeobox 2
ZNF688 zinc finger protein 688

decreased expression

Symbol Name
ACACA acetyl-CoA carboxylase alpha
ADAM15 ADAM metallopeptidase domain 15
AKT1 v-akt murine thymoma viral oncogene homolog 1
APOC2 apolipoprotein C-II
ARL4A ADP-ribosylation factor-like 4A
AVEN apoptosis, caspase activation inhibitor
BABAM1 BRISC and BRCA1 A complex member 1
BSG basigin (Ok blood group)
BST1 bone marrow stromal cell antigen 1
C11ORF49 chromosome 11 open reading frame 49
CA7 carbonic anhydrase VII
CCDC53 coiled-coil domain containing 53
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
COMMD9 COMM domain containing 9
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
DHRS7B dehydrogenase/reductase (SDR family) member 7B
DHX8 DEAH (Asp-Glu-Ala-His) box polypeptide 8
DOLK dolichol kinase
DPF2 D4, zinc and double PHD fingers family 2
EMC9 ER membrane protein complex subunit 9
ENTPD6 ectonucleoside triphosphate diphosphohydrolase 6 (putative)
ERCC2 excision repair cross-complementation group 2
ERI3 ERI1 exoribonuclease family member 3
ETFB electron-transfer-flavoprotein, beta polypeptide
FAM168B family with sequence similarity 168, member B
FAM63A family with sequence similarity 63, member A
FBXL6 F-box and leucine-rich repeat protein 6
FES FES proto-oncogene, tyrosine kinase
FZD2 frizzled class receptor 2
GAB2 GRB2-associated binding protein 2
GALNS galactosamine (N-acetyl)-6-sulfatase
GBAP1 glucosidase, beta, acid pseudogene 1
GEMIN4 gem (nuclear organelle) associated protein 4
GTPBP2 GTP binding protein 2
H1FX H1 histone family, member X
HMHA1 histocompatibility (minor) HA-1
HYAL2 hyaluronoglucosaminidase 2
IFITM3 interferon induced transmembrane protein 3
IP6K1 inositol hexakisphosphate kinase 1
ISG15 ISG15 ubiquitin-like modifier
JMJD4 jumonji domain containing 4
KEAP1 kelch-like ECH-associated protein 1
KLF13 Kruppel-like factor 13
KLHL21 kelch-like family member 21
LIG1 ligase I, DNA, ATP-dependent
LMTK1 lemur tail kinase 1
MGMT O-6-methylguanine-DNA methyltransferase
MPG N-methylpurine-DNA glycosylase
MPV17 MpV17 mitochondrial inner membrane protein
MYO9A myosin IXA
NADSYN1 NAD synthetase 1
NCAPH non-SMC condensin I complex, subunit H
NCF1C neutrophil cytosolic factor 1C pseudogene
NDUFC1 NADH dehydrogenase (ubiquinone) 1, subcomplex unknown, 1, 6kDa
NFE2 nuclear factor, erythroid 2
NRBP1 nuclear receptor binding protein 1
NSUN5P1 NOP2/Sun domain family, member 5 pseudogene 1
OBFC1 oligonucleotide/oligosaccharide-binding fold containing 1
OGDH oxoglutarate (alpha-ketoglutarate) dehydrogenase (lipoamide)
ORC1 origin recognition complex, subunit 1
PAGR1 PAXIP1 associated glutamate-rich protein 1
PCBD1 pterin-4 alpha-carbinolamine dehydratase/dimerization cofactor of hepatocyte nuclear factor 1 alpha
PCTP phosphatidylcholine transfer protein
PKN1 protein kinase N1
PLEKHM2 pleckstrin homology domain containing, family M (with RUN domain) member 2
POP7 processing of precursor 7, ribonuclease P/MRP subunit (S. cerevisiae)
PPIEL peptidylprolyl isomerase E-like pseudogene
PPP4C protein phosphatase 4, catalytic subunit
PTOV1 prostate tumor overexpressed 1
PTPN9 protein tyrosine phosphatase, non-receptor type 9
PTPRCAP protein tyrosine phosphatase, receptor type, C-associated protein
QPRT quinolinate phosphoribosyltransferase
RAB4B RAB4B, member RAS oncogene family
RASSF1 Ras association (RalGDS/AF-6) domain family member 1
RBM10 RNA binding motif protein 10
RNF123 ring finger protein 123
SAC3D1 SAC3 domain containing 1
SARS2 seryl-tRNA synthetase 2, mitochondrial
SLC35C2 solute carrier family 35 (GDP-fucose transporter), member C2
SMG9 SMG9 nonsense mediated mRNA decay factor
SNX6 sorting nexin 6
STARD3 StAR-related lipid transfer (START) domain containing 3
SUPT3H suppressor of Ty 3 homolog (S. cerevisiae)
TGFBRAP1 transforming growth factor, beta receptor associated protein 1
TMEM109 transmembrane protein 109
TRAIP TRAF interacting protein
TST thiosulfate sulfurtransferase (rhodanese)
TTPAL tocopherol (alpha) transfer protein-like
UFD1L ubiquitin fusion degradation 1 like (yeast)
USP5 ubiquitin specific peptidase 5 (isopeptidase T)
VILL villin-like
VPS28 vacuolar protein sorting 28 homolog (S. cerevisiae)
VPS52 vacuolar protein sorting 52 homolog (S. cerevisiae)
WDR19 WD repeat domain 19
WDR6 WD repeat domain 6
YIPF1 Yip1 domain family, member 1
ZC3H3 zinc finger CCCH-type containing 3
ZNF408 zinc finger protein 408
ZNHIT2 zinc finger, HIT-type containing 2