articaine-3138 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

200 genes differentially expressed following the articaine-3138 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADORA1 adenosine A1 receptor
ALDH4A1 aldehyde dehydrogenase 4 family, member A1
ALDOAP2 aldolase A, fructose-bisphosphate pseudogene 2
ALG12 ALG12, alpha-1,6-mannosyltransferase
ARHGEF11 Rho guanine nucleotide exchange factor (GEF) 11
BCAS3 breast carcinoma amplified sequence 3
BMPR2 bone morphogenetic protein receptor, type II (serine/threonine kinase)
CAMKMT calmodulin-lysine N-methyltransferase
CCDC181 coiled-coil domain containing 181
CD2 CD2 molecule
CD247 CD247 molecule
CDHR1 cadherin-related family member 1
CORO1B coronin, actin binding protein, 1B
CPN2 carboxypeptidase N, polypeptide 2
CREBBP CREB binding protein
CXXC4 CXXC finger protein 4
CYP19A1 cytochrome P450, family 19, subfamily A, polypeptide 1
DCT dopachrome tautomerase
DEPTOR DEP domain containing MTOR-interacting protein
DGAT1 diacylglycerol O-acyltransferase 1
DLGAP4 discs, large (Drosophila) homolog-associated protein 4
DZANK1 double zinc ribbon and ankyrin repeat domains 1
EDA ectodysplasin A
ELK4 ELK4, ETS-domain protein (SRF accessory protein 1)
ELN elastin
EXOC7 exocyst complex component 7
FAM65A family with sequence similarity 65, member A
FAP fibroblast activation protein, alpha
FBXO31 F-box protein 31
FGFR3 fibroblast growth factor receptor 3
FLT3LG fms-related tyrosine kinase 3 ligand
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GCNT4 glucosaminyl (N-acetyl) transferase 4, core 2
GLDC glycine dehydrogenase (decarboxylating)
GNA11 guanine nucleotide binding protein (G protein), alpha 11 (Gq class)
GPR12 G protein-coupled receptor 12
GPR132 G protein-coupled receptor 132
GPR153 G protein-coupled receptor 153
GSPT1 G1 to S phase transition 1
GUCY1A2 guanylate cyclase 1, soluble, alpha 2
HNF4A hepatocyte nuclear factor 4, alpha
HOXA3 homeobox A3
ICAM1 intercellular adhesion molecule 1
IL12RB1 interleukin 12 receptor, beta 1
IL22RA1 interleukin 22 receptor, alpha 1
JAM3 junctional adhesion molecule 3
KIAA1024 KIAA1024
KLF12 Kruppel-like factor 12
KRT81 keratin 81, type II
LRRC31 leucine rich repeat containing 31
LRRC48 leucine rich repeat containing 48
MAP6D1 MAP6 domain containing 1
MBD2 methyl-CpG binding domain protein 2
MBOAT2 membrane bound O-acyltransferase domain containing 2
MCM3AP minichromosome maintenance complex component 3 associated protein
MUC1 mucin 1, cell surface associated
MYO15A myosin XVA
NDST1 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 1
NEK9 NIMA-related kinase 9
NPHP1 nephronophthisis 1 (juvenile)
NR2F1 nuclear receptor subfamily 2, group F, member 1
NRCAM neuronal cell adhesion molecule
NUP188 nucleoporin 188kDa
OLFML2A olfactomedin-like 2A
OR1E1 olfactory receptor, family 1, subfamily E, member 1
PDE6B phosphodiesterase 6B, cGMP-specific, rod, beta
PRAMEF11 PRAME family member 11
PTCRA pre T-cell antigen receptor alpha
RCN3 reticulocalbin 3, EF-hand calcium binding domain
RDH5 retinol dehydrogenase 5 (11-cis/9-cis)
RGS11 regulator of G-protein signaling 11
RGS12 regulator of G-protein signaling 12
SLC17A2 solute carrier family 17, member 2
SLC48A1 solute carrier family 48 (heme transporter), member 1
SNAI2 snail family zinc finger 2
SNN stannin
SORBS3 sorbin and SH3 domain containing 3
SPDEF SAM pointed domain containing ETS transcription factor
ST8SIA3 ST8 alpha-N-acetyl-neuraminide alpha-2,8-sialyltransferase 3
STAG3L4 stromal antigen 3-like 4 (pseudogene)
STATH statherin
STK3 serine/threonine kinase 3
SYNE2 spectrin repeat containing, nuclear envelope 2
TEF thyrotrophic embryonic factor
TICAM1 toll-like receptor adaptor molecule 1
TJAP1 tight junction associated protein 1 (peripheral)
TM4SF5 transmembrane 4 L six family member 5
TNKS tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase
TNNT3 troponin T type 3 (skeletal, fast)
TRIM2 tripartite motif containing 2
TSC2 tuberous sclerosis 2
TTLL7 tubulin tyrosine ligase-like family member 7
UNC119 unc-119 homolog (C. elegans)
WNT2B wingless-type MMTV integration site family, member 2B
ZC3H7B zinc finger CCCH-type containing 7B
ZER1 zyg-11 related, cell cycle regulator
ZNF407 zinc finger protein 407
ZNF471 zinc finger protein 471
ZNF639 zinc finger protein 639
ZNF710 zinc finger protein 710

decreased expression

Symbol Name
ABCA7 ATP-binding cassette, sub-family A (ABC1), member 7
ACPP acid phosphatase, prostate
ACVR2B activin A receptor, type IIB
ADAM15 ADAM metallopeptidase domain 15
ASPN asporin
ASPSCR1 alveolar soft part sarcoma chromosome region, candidate 1
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
B3GNT1
BAHCC1 BAH domain and coiled-coil containing 1
BCL7C B-cell CLL/lymphoma 7C
BEST1 bestrophin 1
BTBD18 BTB (POZ) domain containing 18
C7ORF43 chromosome 7 open reading frame 43
CCDC186 coiled-coil domain containing 186
CDCP1 CUB domain containing protein 1
CDK3 cyclin-dependent kinase 3
CNR2 cannabinoid receptor 2 (macrophage)
COQ6 coenzyme Q6 monooxygenase
CROT carnitine O-octanoyltransferase
CTNNBIP1 catenin, beta interacting protein 1
CUL9 cullin 9
CX3CR1 chemokine (C-X3-C motif) receptor 1
CYP17A1 cytochrome P450, family 17, subfamily A, polypeptide 1
CYP27B1 cytochrome P450, family 27, subfamily B, polypeptide 1
DCAF13 DDB1 and CUL4 associated factor 13
DCAF17 DDB1 and CUL4 associated factor 17
DDX60 DEAD (Asp-Glu-Ala-Asp) box polypeptide 60
DGKG diacylglycerol kinase, gamma 90kDa
ECM1 extracellular matrix protein 1
ENTPD7 ectonucleoside triphosphate diphosphohydrolase 7
EPHX1 epoxide hydrolase 1, microsomal (xenobiotic)
ERMAP erythroblast membrane-associated protein (Scianna blood group)
ERN2 endoplasmic reticulum to nucleus signaling 2
EXD3 exonuclease 3'-5' domain containing 3
FER fer (fps/fes related) tyrosine kinase
FGF22 fibroblast growth factor 22
FOXO4 forkhead box O4
GABRA4 gamma-aminobutyric acid (GABA) A receptor, alpha 4
GPATCH2L G patch domain containing 2-like
GPATCH3 G patch domain containing 3
IDI2-AS1 IDI2 antisense RNA 1
INF2 inverted formin, FH2 and WH2 domain containing
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
LAIR2 leukocyte-associated immunoglobulin-like receptor 2
LIMD2 LIM domain containing 2
LNPEP leucyl/cystinyl aminopeptidase
LOC100286895 cell division cycle 27 homolog pseudogene
LRRK1 leucine-rich repeat kinase 1
LSM14B LSM14B, SCD6 homolog B (S. cerevisiae)
MAK male germ cell-associated kinase
MANSC1 MANSC domain containing 1
MAST3 microtubule associated serine/threonine kinase 3
MECR mitochondrial trans-2-enoyl-CoA reductase
MKL2 MKL/myocardin-like 2
MMP2 matrix metallopeptidase 2
MTMR12 myotubularin related protein 12
MX1 MX dynamin-like GTPase 1
MYH15 myosin, heavy chain 15
NABP2 nucleic acid binding protein 2
NFE2L3 nuclear factor, erythroid 2-like 3
NINJ2 ninjurin 2
NLRX1 NLR family member X1
NOD2 nucleotide-binding oligomerization domain containing 2
NOL10 nucleolar protein 10
NT5C 5', 3'-nucleotidase, cytosolic
OSGEPL1 O-sialoglycoprotein endopeptidase-like 1
PARP16 poly (ADP-ribose) polymerase family, member 16
PDPR pyruvate dehydrogenase phosphatase regulatory subunit
PECR peroxisomal trans-2-enoyl-CoA reductase
PIPOX pipecolic acid oxidase
PMFBP1 polyamine modulated factor 1 binding protein 1
PMP22 peripheral myelin protein 22
POM121L2 POM121 transmembrane nucleoporin-like 2
POMGNT1 protein O-linked mannose N-acetylglucosaminyltransferase 1 (beta 1,2-)
PPDPF pancreatic progenitor cell differentiation and proliferation factor
PRDM1 PR domain containing 1, with ZNF domain
PSKH1 protein serine kinase H1
QSER1 glutamine and serine rich 1
SCML2 sex comb on midleg-like 2 (Drosophila)
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC9A3R1 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3 regulator 1
SMR3A submaxillary gland androgen regulated protein 3A
SPATA20 spermatogenesis associated 20
TAB1 TGF-beta activated kinase 1/MAP3K7 binding protein 1
TERT telomerase reverse transcriptase
TET3 tet methylcytosine dioxygenase 3
TMA16 translation machinery associated 16 homolog (S. cerevisiae)
TMEM115 transmembrane protein 115
TMEM39B transmembrane protein 39B
TNFSF13 tumor necrosis factor (ligand) superfamily, member 13
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TSPAN13 tetraspanin 13
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
ZCWPW1 zinc finger, CW type with PWWP domain 1
ZDHHC24 zinc finger, DHHC-type containing 24
ZNF408 zinc finger protein 408
ZNF552 zinc finger protein 552
ZNF804A zinc finger protein 804A