azapropazone-7277 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the azapropazone-7277 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCA7 ATP-binding cassette, sub-family A (ABC1), member 7
ANKRA2 ankyrin repeat, family A (RFXANK-like), 2
ARAP2 ArfGAP with RhoGAP domain, ankyrin repeat and PH domain 2
ARMC9 armadillo repeat containing 9
ATP9B ATPase, class II, type 9B
ATXN3 ataxin 3
AVL9 AVL9 homolog (S. cerevisiase)
B3GNT2 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 2
BAIAP2 BAI1-associated protein 2
BBS7 Bardet-Biedl syndrome 7
BCL11A B-cell CLL/lymphoma 11A (zinc finger protein)
C10ORF88 chromosome 10 open reading frame 88
C9ORF156 chromosome 9 open reading frame 156
CDIP1 cell death-inducing p53 target 1
CFAP69 cilia and flagella associated protein 69
CLUHP3 clustered mitochondria (cluA/CLU1) homolog pseudogene 3
COPS8 COP9 signalosome subunit 8
COX15 cytochrome c oxidase assembly homolog 15 (yeast)
CSPP1 centrosome and spindle pole associated protein 1
CST6 cystatin E/M
CTBS chitobiase, di-N-acetyl-
DDX17 DEAD (Asp-Glu-Ala-Asp) box helicase 17
DDX3X DEAD (Asp-Glu-Ala-Asp) box helicase 3, X-linked
DHODH dihydroorotate dehydrogenase (quinone)
DNAJC8 DnaJ (Hsp40) homolog, subfamily C, member 8
DTX2 deltex 2, E3 ubiquitin ligase
EIF5B eukaryotic translation initiation factor 5B
FAM131B family with sequence similarity 131, member B
FAM188A family with sequence similarity 188, member A
FCGR2A Fc fragment of IgG, low affinity IIa, receptor (CD32)
FGF13 fibroblast growth factor 13
GOLGA1 golgin A1
GRK5 G protein-coupled receptor kinase 5
GSAP gamma-secretase activating protein
HNRNPH1 heterogeneous nuclear ribonucleoprotein H1 (H)
HOMER2 homer scaffolding protein 2
HOMER3 homer scaffolding protein 3
IL1R2 interleukin 1 receptor, type II
ING1 inhibitor of growth family, member 1
INTS6 integrator complex subunit 6
KCNAB1 potassium channel, voltage gated subfamily A regulatory beta subunit 1
KCNJ2 potassium channel, inwardly rectifying subfamily J, member 2
LDB1 LIM domain binding 1
LGR5 leucine-rich repeat containing G protein-coupled receptor 5
LOC730101 uncharacterized LOC730101
LRRFIP1 leucine rich repeat (in FLII) interacting protein 1
MAP7 microtubule-associated protein 7
MAPK7 mitogen-activated protein kinase 7
MARS methionyl-tRNA synthetase
MBD3 methyl-CpG binding domain protein 3
MBTPS2 membrane-bound transcription factor peptidase, site 2
MGMT O-6-methylguanine-DNA methyltransferase
MUM1 melanoma associated antigen (mutated) 1
MYO9B myosin IXB
NCKIPSD NCK interacting protein with SH3 domain
PDE1C phosphodiesterase 1C, calmodulin-dependent 70kDa
PEX7 peroxisomal biogenesis factor 7
PHF2 PHD finger protein 2
PKP2 plakophilin 2
PLEKHG6 pleckstrin homology domain containing, family G (with RhoGef domain) member 6
PRKAB2 protein kinase, AMP-activated, beta 2 non-catalytic subunit
PRKACG protein kinase, cAMP-dependent, catalytic, gamma
PTHLH parathyroid hormone-like hormone
PTPRF protein tyrosine phosphatase, receptor type, F
PTPRN2 protein tyrosine phosphatase, receptor type, N polypeptide 2
R3HDM4 R3H domain containing 4
RABGAP1 RAB GTPase activating protein 1
RAD52 RAD52 homolog (S. cerevisiae)
RDH11 retinol dehydrogenase 11 (all-trans/9-cis/11-cis)
RGS4 regulator of G-protein signaling 4
RGS5 regulator of G-protein signaling 5
RNF19B ring finger protein 19B
RNF216 ring finger protein 216
RPS6KB1 ribosomal protein S6 kinase, 70kDa, polypeptide 1
RUSC2 RUN and SH3 domain containing 2
S100A11 S100 calcium binding protein A11
SEC14L2 SEC14-like 2 (S. cerevisiae)
SLC12A4 solute carrier family 12 (potassium/chloride transporter), member 4
SLC14A1 solute carrier family 14 (urea transporter), member 1 (Kidd blood group)
SLC25A16 solute carrier family 25 (mitochondrial carrier), member 16
SLC26A6 solute carrier family 26 (anion exchanger), member 6
SLITRK5 SLIT and NTRK-like family, member 5
SOGA1 suppressor of glucose, autophagy associated 1
SPATA2L spermatogenesis associated 2-like
SPSB3 splA/ryanodine receptor domain and SOCS box containing 3
SPTAN1 spectrin, alpha, non-erythrocytic 1
SSBP2 single-stranded DNA binding protein 2
STK16 serine/threonine kinase 16
STK4 serine/threonine kinase 4
TAZ tafazzin
TGOLN2 trans-golgi network protein 2
TMEM254 transmembrane protein 254
WNT7A wingless-type MMTV integration site family, member 7A
WWC1 WW and C2 domain containing 1
ZC3H7B zinc finger CCCH-type containing 7B
ZEB1 zinc finger E-box binding homeobox 1
ZNF165 zinc finger protein 165
ZNF426 zinc finger protein 426
ZNF688 zinc finger protein 688

decreased expression

Symbol Name
ACADSB acyl-CoA dehydrogenase, short/branched chain
ACTR3B ARP3 actin-related protein 3 homolog B (yeast)
AEN apoptosis enhancing nuclease
AKR1B10 aldo-keto reductase family 1, member B10 (aldose reductase)
ANKFY1 ankyrin repeat and FYVE domain containing 1
AP4M1 adaptor-related protein complex 4, mu 1 subunit
ASB6 ankyrin repeat and SOCS box containing 6
ATP7B ATPase, Cu++ transporting, beta polypeptide
AXIN1 axin 1
C11ORF80 chromosome 11 open reading frame 80
C17ORF80 chromosome 17 open reading frame 80
C4ORF19 chromosome 4 open reading frame 19
C7ORF43 chromosome 7 open reading frame 43
CARD8 caspase recruitment domain family, member 8
CCNA1 cyclin A1
CCNO cyclin O
CDK3 cyclin-dependent kinase 3
CEP131 centrosomal protein 131kDa
CLEC10A C-type lectin domain family 10, member A
CNGB3 cyclic nucleotide gated channel beta 3
CNKSR1 connector enhancer of kinase suppressor of Ras 1
COLGALT2 collagen beta(1-O)galactosyltransferase 2
CUL9 cullin 9
DEXI Dexi homolog (mouse)
DFFB DNA fragmentation factor, 40kDa, beta polypeptide (caspase-activated DNase)
DSPP dentin sialophosphoprotein
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
EFCAB2 EF-hand calcium binding domain 2
EFNA3 ephrin-A3
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM155A family with sequence similarity 155, member A
FARP2 FERM, RhoGEF and pleckstrin domain protein 2
FBXL15 F-box and leucine-rich repeat protein 15
FCHO1 FCH domain only 1
FXN frataxin
GAMT guanidinoacetate N-methyltransferase
GBX2 gastrulation brain homeobox 2
GDAP1 ganglioside induced differentiation associated protein 1
GLCE glucuronic acid epimerase
GRAMD4 GRAM domain containing 4
HHLA3 HERV-H LTR-associating 3
HIST1H2AM histone cluster 1, H2am
HIST1H4D histone cluster 1, H4d
HOXA4 homeobox A4
IFT54 intraflagellar transport 54
IQCG IQ motif containing G
KLK5 kallikrein-related peptidase 5
LPAR4 lysophosphatidic acid receptor 4
LYL1 lymphoblastic leukemia associated hematopoiesis regulator 1
ME3 malic enzyme 3, NADP(+)-dependent, mitochondrial
MRPL28 mitochondrial ribosomal protein L28
NAG18 NAG18 mRNA
NBEAL2 neurobeachin-like 2
NXPH4 neurexophilin 4
ODF2 outer dense fiber of sperm tails 2
OPLAH 5-oxoprolinase (ATP-hydrolysing)
OSBP2 oxysterol binding protein 2
PAFAH1B2 platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (30kDa)
PARD6A par-6 family cell polarity regulator alpha
PARG poly (ADP-ribose) glycohydrolase
PDE12 phosphodiesterase 12
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PPP1R3C protein phosphatase 1, regulatory subunit 3C
PRICKLE3 prickle homolog 3 (Drosophila)
QTRT1 queuine tRNA-ribosyltransferase 1
RCBTB2 regulator of chromosome condensation (RCC1) and BTB (POZ) domain containing protein 2
RGCC regulator of cell cycle
RIN1 Ras and Rab interactor 1
RNF126P1 ring finger protein 126 pseudogene 1
RPAP1 RNA polymerase II associated protein 1
RRAGB Ras-related GTP binding B
SCARA3 scavenger receptor class A, member 3
SLC2A6 solute carrier family 2 (facilitated glucose transporter), member 6
SMR3A submaxillary gland androgen regulated protein 3A
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2
TBC1D17 TBC1 domain family, member 17
TBX19 T-box 19
TMC5 transmembrane channel-like 5
TMEM132A transmembrane protein 132A
TMEM156 transmembrane protein 156
TMEM53 transmembrane protein 53
TMEM8A transmembrane protein 8A
TRABD TraB domain containing
TRPM4 transient receptor potential cation channel, subfamily M, member 4
USP18 ubiquitin specific peptidase 18
VCPIP1 valosin containing protein (p97)/p47 complex interacting protein 1
WDR18 WD repeat domain 18
WDR46 WD repeat domain 46
WNT10B wingless-type MMTV integration site family, member 10B
XAB2 XPA binding protein 2
ZDHHC14 zinc finger, DHHC-type containing 14
ZNF222 zinc finger protein 222
ZNF227 zinc finger protein 227
ZNF230 zinc finger protein 230
ZNF254 zinc finger protein 254
ZNF324 zinc finger protein 324
ZNF862 zinc finger protein 862