azathioprine-2028 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the azathioprine-2028 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCD4 ATP-binding cassette, sub-family D (ALD), member 4
ABHD2 abhydrolase domain containing 2
ABL2 ABL proto-oncogene 2, non-receptor tyrosine kinase
ADAMTS1 ADAM metallopeptidase with thrombospondin type 1 motif, 1
ALDH3B1 aldehyde dehydrogenase 3 family, member B1
ASPH aspartate beta-hydroxylase
ATR ATR serine/threonine kinase
BAX BCL2-associated X protein
BCL2 B-cell CLL/lymphoma 2
C21ORF91 chromosome 21 open reading frame 91
C2ORF27A chromosome 2 open reading frame 27A
C5ORF30 chromosome 5 open reading frame 30
C6 complement component 6
CA12 carbonic anhydrase XII
CA5BP1 carbonic anhydrase VB pseudogene 1
CHMP6 charged multivesicular body protein 6
CHST5 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 5
CLCN6 chloride channel, voltage-sensitive 6
CLPB ClpB homolog, mitochondrial AAA ATPase chaperonin
CLSPN claspin
CNPY3 canopy FGF signaling regulator 3
CNTN1 contactin 1
CTRC chymotrypsin C (caldecrin)
CTRL chymotrypsin-like
DBN1 drebrin 1
DRD5 dopamine receptor D5
EPHB2 EPH receptor B2
EPOR erythropoietin receptor
ERCC6 excision repair cross-complementation group 6
FAS Fas cell surface death receptor
FBXW11 F-box and WD repeat domain containing 11
FCGR2C Fc fragment of IgG, low affinity IIc, receptor for (CD32) (gene/pseudogene)
FKBP4 FK506 binding protein 4, 59kDa
FLNC filamin C, gamma
FRY furry homolog (Drosophila)
FYB FYN binding protein
GATA2 GATA binding protein 2
GCKR glucokinase (hexokinase 4) regulator
GNB1L guanine nucleotide binding protein (G protein), beta polypeptide 1-like
GOSR2 golgi SNAP receptor complex member 2
GOT2 glutamic-oxaloacetic transaminase 2, mitochondrial
IDH3G isocitrate dehydrogenase 3 (NAD+) gamma
IFNA17 interferon, alpha 17
IL22RA1 interleukin 22 receptor, alpha 1
INHA inhibin, alpha
INPP4A inositol polyphosphate-4-phosphatase, type I, 107kDa
ITIH2 inter-alpha-trypsin inhibitor heavy chain 2
KRI1 KRI1 homolog (S. cerevisiae)
LENEP lens epithelial protein
LMTK1 lemur tail kinase 1
MAP3K2 mitogen-activated protein kinase kinase kinase 2
MAZ MYC-associated zinc finger protein (purine-binding transcription factor)
MBTPS2 membrane-bound transcription factor peptidase, site 2
MFSD11 major facilitator superfamily domain containing 11
MICA MHC class I polypeptide-related sequence A
MLC1 megalencephalic leukoencephalopathy with subcortical cysts 1
MPZ myelin protein zero
MUC5AC mucin 5AC, oligomeric mucus/gel-forming
MYL10 myosin, light chain 10, regulatory
MYO9B myosin IXB
N4BP1 NEDD4 binding protein 1
NINJ2 ninjurin 2
NUDT2 nudix (nucleoside diphosphate linked moiety X)-type motif 2
OCRL oculocerebrorenal syndrome of Lowe
OS9 osteosarcoma amplified 9, endoplasmic reticulum lectin
PDCD4 programmed cell death 4 (neoplastic transformation inhibitor)
POLD4 polymerase (DNA-directed), delta 4, accessory subunit
POLR3G polymerase (RNA) III (DNA directed) polypeptide G (32kD)
RBBP5 retinoblastoma binding protein 5
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
SEMA3G sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3G
SFTPB surfactant protein B
SH3BP5 SH3-domain binding protein 5 (BTK-associated)
SHARPIN SHANK-associated RH domain interactor
SLC2A5 solute carrier family 2 (facilitated glucose/fructose transporter), member 5
SMIM8 small integral membrane protein 8
SNX19 sorting nexin 19
SOX4 SRY (sex determining region Y)-box 4
SPG7 spastic paraplegia 7 (pure and complicated autosomal recessive)
SPN sialophorin
SPTLC1 serine palmitoyltransferase, long chain base subunit 1
SRBD1 S1 RNA binding domain 1
SRCAP Snf2-related CREBBP activator protein
STARD13 StAR-related lipid transfer (START) domain containing 13
TAC3 tachykinin 3
TBC1D4 TBC1 domain family, member 4
TBCD tubulin folding cofactor D
TES testin LIM domain protein
THG1L tRNA-histidine guanylyltransferase 1-like (S. cerevisiae)
TMEM62 transmembrane protein 62
TPRA1 transmembrane protein, adipocyte asscociated 1
TRABD TraB domain containing
TRIP11 thyroid hormone receptor interactor 11
TTLL4 tubulin tyrosine ligase-like family member 4
YIF1B Yip1 interacting factor homolog B (S. cerevisiae)
YLPM1 YLP motif containing 1
ZC4H2 zinc finger, C4H2 domain containing
ZNF787 zinc finger protein 787
ZNF816 zinc finger protein 816
ZNHIT2 zinc finger, HIT-type containing 2

decreased expression

Symbol Name
ABHD3 abhydrolase domain containing 3
AGL amylo-alpha-1, 6-glucosidase, 4-alpha-glucanotransferase
ANKRD40 ankyrin repeat domain 40
ARMC7 armadillo repeat containing 7
ASAP1 ArfGAP with SH3 domain, ankyrin repeat and PH domain 1
ATAD2B ATPase family, AAA domain containing 2B
BAP1 BRCA1 associated protein-1 (ubiquitin carboxy-terminal hydrolase)
C1GALT1C1 C1GALT1-specific chaperone 1
CCDC130 coiled-coil domain containing 130
CD2AP CD2-associated protein
CDC42SE1 CDC42 small effector 1
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CENPQ centromere protein Q
CHST4 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 4
CNP 2',3'-cyclic nucleotide 3' phosphodiesterase
CPOX coproporphyrinogen oxidase
DCAF6 DDB1 and CUL4 associated factor 6
DCK deoxycytidine kinase
DNAJB14 DnaJ (Hsp40) homolog, subfamily B, member 14
DNAJC12 DnaJ (Hsp40) homolog, subfamily C, member 12
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3
DPYD dihydropyrimidine dehydrogenase
EGLN1 egl-9 family hypoxia-inducible factor 1
ERCC3 excision repair cross-complementation group 3
FABP5 fatty acid binding protein 5 (psoriasis-associated)
FANCL Fanconi anemia, complementation group L
FBXL4 F-box and leucine-rich repeat protein 4
FCGR2B Fc fragment of IgG, low affinity IIb, receptor (CD32)
FTH1P5 ferritin, heavy polypeptide 1 pseudogene 5
GAB2 GRB2-associated binding protein 2
GGH gamma-glutamyl hydrolase (conjugase, folylpolygammaglutamyl hydrolase)
GIMAP6 GTPase, IMAP family member 6
GNG10 guanine nucleotide binding protein (G protein), gamma 10
GOLPH3L golgi phosphoprotein 3-like
GPR27 G protein-coupled receptor 27
HIST2H2BE histone cluster 2, H2be
HMGB3P1 high mobility group box 3 pseudogene 1
KLF2 Kruppel-like factor 2
LINC00339 long intergenic non-protein coding RNA 339
MAPKBP1 mitogen-activated protein kinase binding protein 1
MED23 mediator complex subunit 23
METTL18 methyltransferase like 18
MORC3 MORC family CW-type zinc finger 3
MPDU1 mannose-P-dolichol utilization defect 1
MRPL16 mitochondrial ribosomal protein L16
MRPL19 mitochondrial ribosomal protein L19
MT1HL1 metallothionein 1H-like 1
MXRA8 matrix-remodelling associated 8
NRIP3 nuclear receptor interacting protein 3
PAQR3 progestin and adipoQ receptor family member III
PEMT phosphatidylethanolamine N-methyltransferase
PITPNM1 phosphatidylinositol transfer protein, membrane-associated 1
PJA1 praja ring finger 1, E3 ubiquitin protein ligase
PKN1 protein kinase N1
PLGRKT plasminogen receptor, C-terminal lysine transmembrane protein
PPIP5K2 diphosphoinositol pentakisphosphate kinase 2
PRPF39 pre-mRNA processing factor 39
PTTG3P pituitary tumor-transforming 3, pseudogene
RAB4B RAB4B, member RAS oncogene family
RAD51AP1 RAD51 associated protein 1
RAP1A RAP1A, member of RAS oncogene family
RAPGEF6 Rap guanine nucleotide exchange factor (GEF) 6
RBM15B RNA binding motif protein 15B
RNF122 ring finger protein 122
RRN3 RRN3 RNA polymerase I transcription factor homolog (S. cerevisiae)
RWDD3 RWD domain containing 3
S1PR4 sphingosine-1-phosphate receptor 4
SEC61B Sec61 beta subunit
SELP selectin P (granule membrane protein 140kDa, antigen CD62)
SERINC1 serine incorporator 1
SKI SKI proto-oncogene
SLC10A1 solute carrier family 10 (sodium/bile acid cotransporter), member 1
SLC35C2 solute carrier family 35 (GDP-fucose transporter), member C2
SLC39A1 solute carrier family 39 (zinc transporter), member 1
SMARCAL1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a-like 1
SP3 Sp3 transcription factor
STXBP3 syntaxin binding protein 3
TAOK3 TAO kinase 3
TFB2M transcription factor B2, mitochondrial
THAP1 THAP domain containing, apoptosis associated protein 1
TM7SF3 transmembrane 7 superfamily member 3
TMEM14A transmembrane protein 14A
TMEM168 transmembrane protein 168
TMEM184C transmembrane protein 184C
TNFRSF1B tumor necrosis factor receptor superfamily, member 1B
TOB1 transducer of ERBB2, 1
TRAPPC11 trafficking protein particle complex 11
TRMT12 tRNA methyltransferase 12 homolog (S. cerevisiae)
TRMT61B tRNA methyltransferase 61B
TUBA1A tubulin, alpha 1a
UBXN2B UBX domain protein 2B
VCPKMT valosin containing protein lysine (K) methyltransferase
WDR82 WD repeat domain 82
ZCCHC8 zinc finger, CCHC domain containing 8
ZDHHC13 zinc finger, DHHC-type containing 13
ZNF217 zinc finger protein 217
ZNF32 zinc finger protein 32
ZNF652 zinc finger protein 652
ZNF804A zinc finger protein 804A