benzocaine-2167 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the benzocaine-2167 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACTA2 actin, alpha 2, smooth muscle, aorta
ADGRB1 adhesion G protein-coupled receptor B1
ADGRL1 adhesion G protein-coupled receptor L1
AGFG1 ArfGAP with FG repeats 1
ALDH6A1 aldehyde dehydrogenase 6 family, member A1
ALDH7A1 aldehyde dehydrogenase 7 family, member A1
AMELX amelogenin, X-linked
ANKRD6 ankyrin repeat domain 6
APOH apolipoprotein H (beta-2-glycoprotein I)
ARNT aryl hydrocarbon receptor nuclear translocator
ATG10 autophagy related 10
BNC1 basonuclin 1
BTN3A1 butyrophilin, subfamily 3, member A1
BUB1 BUB1 mitotic checkpoint serine/threonine kinase
C3ORF18 chromosome 3 open reading frame 18
CAMK4 calcium/calmodulin-dependent protein kinase IV
CD177 CD177 molecule
CD59 CD59 molecule, complement regulatory protein
CDH6 cadherin 6, type 2, K-cadherin (fetal kidney)
CEP170B centrosomal protein 170B
CMAHP cytidine monophospho-N-acetylneuraminic acid hydroxylase, pseudogene
COBLL1 cordon-bleu WH2 repeat protein-like 1
CPTP ceramide-1-phosphate transfer protein
CREM cAMP responsive element modulator
DFNA5 deafness, autosomal dominant 5
DNAJC1 DnaJ (Hsp40) homolog, subfamily C, member 1
ENPP1 ectonucleotide pyrophosphatase/phosphodiesterase 1
EXO5 exonuclease 5
EXOSC2 exosome component 2
FAM65A family with sequence similarity 65, member A
FGF22 fibroblast growth factor 22
FUBP1 far upstream element (FUSE) binding protein 1
GALNT10 polypeptide N-acetylgalactosaminyltransferase 10
GJA4 gap junction protein, alpha 4, 37kDa
GLE1 GLE1 RNA export mediator
GPR19 G protein-coupled receptor 19
GPR35 G protein-coupled receptor 35
HEXIM1 hexamethylene bis-acetamide inducible 1
HIC2 hypermethylated in cancer 2
HYAL1 hyaluronoglucosaminidase 1
IDS iduronate 2-sulfatase
IQCK IQ motif containing K
ISG20 interferon stimulated exonuclease gene 20kDa
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KDM8 lysine (K)-specific demethylase 8
KIF3A kinesin family member 3A
L3MBTL1 l(3)mbt-like 1 (Drosophila)
LGR5 leucine-rich repeat containing G protein-coupled receptor 5
LILRB2 leukocyte immunoglobulin-like receptor, subfamily B (with TM and ITIM domains), member 2
LOC100286895 cell division cycle 27 homolog pseudogene
LRRC23 leucine rich repeat containing 23
MAOA monoamine oxidase A
MAP4 microtubule-associated protein 4
MTA2 metastasis associated 1 family, member 2
MTCP1 mature T-cell proliferation 1
MUC8 mucin 8
N4BP2L2-IT2 N4BPL2 intronic transcript 2
NDUFA2 NADH dehydrogenase (ubiquinone) 1 alpha subcomplex, 2, 8kDa
NEK11 NIMA-related kinase 11
NEK9 NIMA-related kinase 9
NNAT neuronatin
NR4A2 nuclear receptor subfamily 4, group A, member 2
PDE4DIP phosphodiesterase 4D interacting protein
PDK4 pyruvate dehydrogenase kinase, isozyme 4
PDLIM7 PDZ and LIM domain 7 (enigma)
PGAM2 phosphoglycerate mutase 2 (muscle)
PHC1 polyhomeotic homolog 1 (Drosophila)
PML promyelocytic leukemia
POLR2L polymerase (RNA) II (DNA directed) polypeptide L, 7.6kDa
POU2F2 POU class 2 homeobox 2
PTBP3 polypyrimidine tract binding protein 3
PTPRN2 protein tyrosine phosphatase, receptor type, N polypeptide 2
PYCRL pyrroline-5-carboxylate reductase-like
PYGB phosphorylase, glycogen; brain
RFPL3 ret finger protein-like 3
SAMD4A sterile alpha motif domain containing 4A
SLC19A1 solute carrier family 19 (folate transporter), member 1
SNRNP200 small nuclear ribonucleoprotein 200kDa (U5)
SOX4 SRY (sex determining region Y)-box 4
SP140 SP140 nuclear body protein
SS18 synovial sarcoma translocation, chromosome 18
TACR1 tachykinin receptor 1
TCAF1 TRPM8 channel-associated factor 1
TCP11L1 t-complex 11, testis-specific-like 1
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
THTPA thiamine triphosphatase
TMC7 transmembrane channel-like 7
TMEM43 transmembrane protein 43
TNFSF14 tumor necrosis factor (ligand) superfamily, member 14
TNK1 tyrosine kinase, non-receptor, 1
TUBB2A tubulin, beta 2A class IIa
VPRBP Vpr (HIV-1) binding protein
WIF1 WNT inhibitory factor 1
ZC3H7B zinc finger CCCH-type containing 7B
ZFPL1 zinc finger protein-like 1
ZNF134 zinc finger protein 134
ZNF177 zinc finger protein 177
ZNF768 zinc finger protein 768
ZNF862 zinc finger protein 862

decreased expression

Symbol Name
A1CF APOBEC1 complementation factor
ADTRP androgen-dependent TFPI-regulating protein
AOAH acyloxyacyl hydrolase (neutrophil)
APOBEC3C apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3C
ATAT1 alpha tubulin acetyltransferase 1
BNC2 basonuclin 2
C16ORF45 chromosome 16 open reading frame 45
C16ORF59 chromosome 16 open reading frame 59
CBY1 chibby homolog 1 (Drosophila)
CCDC85C coiled-coil domain containing 85C
CD34 CD34 molecule
CDH10 cadherin 10, type 2 (T2-cadherin)
CDK3 cyclin-dependent kinase 3
CLEC4E C-type lectin domain family 4, member E
CYP2W1 cytochrome P450, family 2, subfamily W, polypeptide 1
DDX6 DEAD (Asp-Glu-Ala-Asp) box helicase 6
DNMT3B DNA (cytosine-5-)-methyltransferase 3 beta
DOC2A double C2-like domains, alpha
EFNA3 ephrin-A3
ELP6 elongator acetyltransferase complex subunit 6
FAM206A family with sequence similarity 206, member A
FAM50B family with sequence similarity 50, member B
FAM53B family with sequence similarity 53, member B
FAM63A family with sequence similarity 63, member A
FAM86C1 family with sequence similarity 86, member C1
FMOD fibromodulin
FRMD1 FERM domain containing 1
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GALK1 galactokinase 1
GDAP1 ganglioside induced differentiation associated protein 1
GJA1 gap junction protein, alpha 1, 43kDa
GNL3LP1 guanine nucleotide binding protein-like 3 (nucleolar)-like pseudogene 1
GRIP2 glutamate receptor interacting protein 2
GSTA3 glutathione S-transferase alpha 3
GSTM2 glutathione S-transferase mu 2 (muscle)
GSTT1 glutathione S-transferase theta 1
HIST1H2AM histone cluster 1, H2am
HOXC8 homeobox C8
IFIT3 interferon-induced protein with tetratricopeptide repeats 3
INA internexin neuronal intermediate filament protein, alpha
INO80D INO80 complex subunit D
KLHL21 kelch-like family member 21
KLHL3 kelch-like family member 3
KLK5 kallikrein-related peptidase 5
LOC729164 hCG1732469
LTBP2 latent transforming growth factor beta binding protein 2
MCOLN1 mucolipin 1
MTMR12 myotubularin related protein 12
MX1 MX dynamin-like GTPase 1
NOL6 nucleolar protein 6 (RNA-associated)
NTSR1 neurotensin receptor 1 (high affinity)
OR12D2 olfactory receptor, family 12, subfamily D, member 2 (gene/pseudogene)
OR7E156P olfactory receptor, family 7, subfamily E, member 156 pseudogene
OVGP1 oviductal glycoprotein 1, 120kDa
PARG poly (ADP-ribose) glycohydrolase
PIK3R2 phosphoinositide-3-kinase, regulatory subunit 2 (beta)
PITPNM1 phosphatidylinositol transfer protein, membrane-associated 1
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma
PPDPF pancreatic progenitor cell differentiation and proliferation factor
PREX2 phosphatidylinositol-3,4,5-trisphosphate-dependent Rac exchange factor 2
PTGES2 prostaglandin E synthase 2
PTTG3P pituitary tumor-transforming 3, pseudogene
RAB11FIP5 RAB11 family interacting protein 5 (class I)
RAB13 RAB13, member RAS oncogene family
RAC3 ras-related C3 botulinum toxin substrate 3 (rho family, small GTP binding protein Rac3)
RASAL1 RAS protein activator like 1 (GAP1 like)
RIPK1 receptor (TNFRSF)-interacting serine-threonine kinase 1
RNF2 ring finger protein 2
SALL2 spalt-like transcription factor 2
SCD5 stearoyl-CoA desaturase 5
SCGB2A2 secretoglobin, family 2A, member 2
SCUBE3 signal peptide, CUB domain, EGF-like 3
SERINC5 serine incorporator 5
SIGLEC15 sialic acid binding Ig-like lectin 15
SLC12A8 solute carrier family 12, member 8
SLC12A9 solute carrier family 12, member 9
SOCS7 suppressor of cytokine signaling 7
SP4 Sp4 transcription factor
SPAG4 sperm associated antigen 4
SULT1B1 sulfotransferase family, cytosolic, 1B, member 1
SYCP2 synaptonemal complex protein 2
TCN1 transcobalamin I (vitamin B12 binding protein, R binder family)
TEC tec protein tyrosine kinase
TGFBR1 transforming growth factor, beta receptor 1
THBS3 thrombospondin 3
TMEM187 transmembrane protein 187
TRAIP TRAF interacting protein
TSC22D4 TSC22 domain family, member 4
WASF3 WAS protein family, member 3
WDR78 WD repeat domain 78
YPEL1 yippee-like 1 (Drosophila)
ZBTB39 zinc finger and BTB domain containing 39
ZC3H3 zinc finger CCCH-type containing 3
ZIM2 zinc finger, imprinted 2
ZNF185 zinc finger protein 185 (LIM domain)
ZNF219 zinc finger protein 219
ZNF528 zinc finger protein 528
ZNF695 zinc finger protein 695
ZNF749 zinc finger protein 749