bromocriptine-5665 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

194 genes differentially expressed following the bromocriptine-5665 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADAM22 ADAM metallopeptidase domain 22
ADGRB3 adhesion G protein-coupled receptor B3
AHNAK2 AHNAK nucleoprotein 2
ALPK1 alpha-kinase 1
APBA2 amyloid beta (A4) precursor protein-binding, family A, member 2
B3GALT4 UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 4
BAAT bile acid CoA:amino acid N-acyltransferase
BHMT2 betaine--homocysteine S-methyltransferase 2
BTN3A1 butyrophilin, subfamily 3, member A1
C10ORF95 chromosome 10 open reading frame 95
C5ORF42 chromosome 5 open reading frame 42
C8A complement component 8, alpha polypeptide
CACNA1I calcium channel, voltage-dependent, T type, alpha 1I subunit
CACNA2D2 calcium channel, voltage-dependent, alpha 2/delta subunit 2
CACNG2 calcium channel, voltage-dependent, gamma subunit 2
CAMK1D calcium/calmodulin-dependent protein kinase ID
CCT8 chaperonin containing TCP1, subunit 8 (theta)
CHRNA10 cholinergic receptor, nicotinic, alpha 10 (neuronal)
CLDN15 claudin 15
CSPG4 chondroitin sulfate proteoglycan 4
CXCR4 chemokine (C-X-C motif) receptor 4
CYP4B1 cytochrome P450, family 4, subfamily B, polypeptide 1
DCT dopachrome tautomerase
DGCR8 DGCR8 microprocessor complex subunit
DOK1 docking protein 1, 62kDa (downstream of tyrosine kinase 1)
DSCAM Down syndrome cell adhesion molecule
DUOX1 dual oxidase 1
ECE1 endothelin converting enzyme 1
ECM2 extracellular matrix protein 2, female organ and adipocyte specific
ETV6 ets variant 6
FAM53B family with sequence similarity 53, member B
FGFR1 fibroblast growth factor receptor 1
FPR1 formyl peptide receptor 1
FSHB follicle stimulating hormone, beta polypeptide
FUT6 fucosyltransferase 6 (alpha (1,3) fucosyltransferase)
GABARAPL1 GABA(A) receptor-associated protein like 1
GNA15 guanine nucleotide binding protein (G protein), alpha 15 (Gq class)
GUK1 guanylate kinase 1
HFE hemochromatosis
HIPK2 homeodomain interacting protein kinase 2
HLCS holocarboxylase synthetase (biotin-(proprionyl-CoA-carboxylase (ATP-hydrolysing)) ligase)
HOXB5 homeobox B5
INPP4A inositol polyphosphate-4-phosphatase, type I, 107kDa
ITGB8 integrin, beta 8
KCNH2 potassium channel, voltage gated eag related subfamily H, member 2
KCNIP2 Kv channel interacting protein 2
KLHDC8A kelch domain containing 8A
KRT38 keratin 38, type I
KRTAP5-9 keratin associated protein 5-9
LPCAT4 lysophosphatidylcholine acyltransferase 4
LPIN1 lipin 1
LTBP4 latent transforming growth factor beta binding protein 4
MARS methionyl-tRNA synthetase
MED16 mediator complex subunit 16
MEF2C myocyte enhancer factor 2C
MEG3 maternally expressed 3 (non-protein coding)
MEGF6 multiple EGF-like-domains 6
MIA2 melanoma inhibitory activity 2
MUC5AC mucin 5AC, oligomeric mucus/gel-forming
MYBPC1 myosin binding protein C, slow type
MYLPF myosin light chain, phosphorylatable, fast skeletal muscle
NDRG2 NDRG family member 2
NKX2-1 NK2 homeobox 1
NUPR1 nuclear protein, transcriptional regulator, 1
OASL 2'-5'-oligoadenylate synthetase-like
OR2B6 olfactory receptor, family 2, subfamily B, member 6
OR7A10 olfactory receptor, family 7, subfamily A, member 10
P2RY1 purinergic receptor P2Y, G-protein coupled, 1
PAK6 p21 protein (Cdc42/Rac)-activated kinase 6
PBXIP1 pre-B-cell leukemia homeobox interacting protein 1
PCDH11Y protocadherin 11 Y-linked
PDGFRA platelet-derived growth factor receptor, alpha polypeptide
PFKFB2 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 2
RAI2 retinoic acid induced 2
RARA retinoic acid receptor, alpha
RNF208 ring finger protein 208
RNF43 ring finger protein 43
RPL23AP32 ribosomal protein L23a pseudogene 32
SH3BP2 SH3-domain binding protein 2
SIM2 single-minded family bHLH transcription factor 2
SLC12A4 solute carrier family 12 (potassium/chloride transporter), member 4
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMC1A structural maintenance of chromosomes 1A
SPAG11A sperm associated antigen 11A
TCF25 transcription factor 25 (basic helix-loop-helix)
THBS3 thrombospondin 3
TMBIM1 transmembrane BAX inhibitor motif containing 1
TREM2 triggering receptor expressed on myeloid cells 2
TRIM3 tripartite motif containing 3
TRPV1 transient receptor potential cation channel, subfamily V, member 1
TUBA4B tubulin, alpha 4b
TXNRD3 thioredoxin reductase 3
UBXN1 UBX domain protein 1
UGT2B15 UDP glucuronosyltransferase 2 family, polypeptide B15
VLDLR very low density lipoprotein receptor
VPS45 vacuolar protein sorting 45 homolog (S. cerevisiae)
ZC4H2 zinc finger, C4H2 domain containing
ZNF76 zinc finger protein 76

decreased expression

Symbol Name
ACAD10 acyl-CoA dehydrogenase family, member 10
ADGRE5 adhesion G protein-coupled receptor E5
AIM2 absent in melanoma 2
ALS2CL ALS2 C-terminal like
AP4M1 adaptor-related protein complex 4, mu 1 subunit
APLP1 amyloid beta (A4) precursor-like protein 1
ARMCX2 armadillo repeat containing, X-linked 2
ARRB1 arrestin, beta 1
ATAD5 ATPase family, AAA domain containing 5
ATP10D ATPase, class V, type 10D
BMP15 bone morphogenetic protein 15
C16ORF45 chromosome 16 open reading frame 45
CBX8 chromobox homolog 8
CCBL1 cysteine conjugate-beta lyase, cytoplasmic
CCDC121 coiled-coil domain containing 121
CCZ1B CCZ1 vacuolar protein trafficking and biogenesis associated homolog B (S. cerevisiae)
CD70 CD70 molecule
CD82 CD82 molecule
CDADC1 cytidine and dCMP deaminase domain containing 1
CDHR2 cadherin-related family member 2
CHST2 carbohydrate (N-acetylglucosamine-6-O) sulfotransferase 2
CIDEB cell death-inducing DFFA-like effector b
CRABP1 cellular retinoic acid binding protein 1
CXORF21 chromosome X open reading frame 21
CYP26A1 cytochrome P450, family 26, subfamily A, polypeptide 1
CYP2B7P cytochrome P450, family 2, subfamily B, polypeptide 7, pseudogene
DDX58 DEAD (Asp-Glu-Ala-Asp) box polypeptide 58
DUSP2 dual specificity phosphatase 2
EPB41L5 erythrocyte membrane protein band 4.1 like 5
EXOC6B exocyst complex component 6B
FBRS fibrosin
FBXW7 F-box and WD repeat domain containing 7, E3 ubiquitin protein ligase
FLVCR2 feline leukemia virus subgroup C cellular receptor family, member 2
GPR3 G protein-coupled receptor 3
HERC6 HECT and RLD domain containing E3 ubiquitin protein ligase family member 6
HIST1H4D histone cluster 1, H4d
HOXA4 homeobox A4
HS3ST3A1 heparan sulfate (glucosamine) 3-O-sulfotransferase 3A1
HSPA1L heat shock 70kDa protein 1-like
HTR1E 5-hydroxytryptamine (serotonin) receptor 1E, G protein-coupled
IFI27 interferon, alpha-inducible protein 27
IFI35 interferon-induced protein 35
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
KCNF1 potassium channel, voltage gated modifier subfamily F, member 1
KCTD7 potassium channel tetramerization domain containing 7
KLF7 Kruppel-like factor 7 (ubiquitous)
LIME1 Lck interacting transmembrane adaptor 1
LONRF3 LON peptidase N-terminal domain and ring finger 3
LRRC37A3 leucine rich repeat containing 37, member A3
LZTR1 leucine-zipper-like transcription regulator 1
MAP3K6 mitogen-activated protein kinase kinase kinase 6
NDRG1 N-myc downstream regulated 1
NPM3 nucleophosmin/nucleoplasmin 3
OR7E47P olfactory receptor, family 7, subfamily E, member 47 pseudogene
OTUD3 OTU deubiquitinase 3
PACS1 phosphofurin acidic cluster sorting protein 1
PDK1 pyruvate dehydrogenase kinase, isozyme 1
PGR progesterone receptor
PIGL phosphatidylinositol glycan anchor biosynthesis, class L
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PLCXD1 phosphatidylinositol-specific phospholipase C, X domain containing 1
POM121 POM121 transmembrane nucleoporin
PPP1R3C protein phosphatase 1, regulatory subunit 3C
PROL1 proline rich, lacrimal 1
RFPL3 ret finger protein-like 3
RGP1 RGP1 retrograde golgi transport homolog (S. cerevisiae)
RNF125 ring finger protein 125, E3 ubiquitin protein ligase
S100A2 S100 calcium binding protein A2
SCN10A sodium channel, voltage gated, type X alpha subunit
SLC12A5 solute carrier family 12 (potassium/chloride transporter), member 5
SLC9A8 solute carrier family 9, subfamily A (NHE8, cation proton antiporter 8), member 8
SP1 Sp1 transcription factor
TDRD12 tudor domain containing 12
TGFBR3 transforming growth factor, beta receptor III
TIMM50 translocase of inner mitochondrial membrane 50 homolog (S. cerevisiae)
TMEM19 transmembrane protein 19
TNFRSF11A tumor necrosis factor receptor superfamily, member 11a, NFKB activator
TSC22D4 TSC22 domain family, member 4
TWISTNB TWIST neighbor
VIM vimentin
VWA1 von Willebrand factor A domain containing 1
WDR33 WD repeat domain 33
WDR91 WD repeat domain 91
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZBTB39 zinc finger and BTB domain containing 39
ZMAT5 zinc finger, matrin-type 5
ZNF428 zinc finger protein 428
ZNF506 zinc finger protein 506
ZNF516 zinc finger protein 516
ZNF586 zinc finger protein 586
ZNF696 zinc finger protein 696
ZNF747 zinc finger protein 747
ZNF750 zinc finger protein 750
ZNF770 zinc finger protein 770
ZNF8 zinc finger protein 8
ZSCAN26 zinc finger and SCAN domain containing 26