bufexamac-5515 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the bufexamac-5515 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADH1B alcohol dehydrogenase 1B (class I), beta polypeptide
AFF2 AF4/FMR2 family, member 2
AHI1 Abelson helper integration site 1
AMH anti-Mullerian hormone
ANTXR1 anthrax toxin receptor 1
APBA2 amyloid beta (A4) precursor protein-binding, family A, member 2
APOL6 apolipoprotein L, 6
ARHGAP26 Rho GTPase activating protein 26
ARL4C ADP-ribosylation factor-like 4C
ARR3 arrestin 3, retinal (X-arrestin)
ATG16L1 autophagy related 16-like 1 (S. cerevisiae)
B3GNT4 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 4
BCL11B B-cell CLL/lymphoma 11B (zinc finger protein)
CAPN9 calpain 9
CCDC33 coiled-coil domain containing 33
CCDC88A coiled-coil domain containing 88A
CD34 CD34 molecule
CDC14B cell division cycle 14B
CDC25C cell division cycle 25C
CDK3 cyclin-dependent kinase 3
CELSR1 cadherin, EGF LAG seven-pass G-type receptor 1
CEP164 centrosomal protein 164kDa
CFAP69 cilia and flagella associated protein 69
CHRNE cholinergic receptor, nicotinic, epsilon (muscle)
CHST11 carbohydrate (chondroitin 4) sulfotransferase 11
DOCK9 dedicator of cytokinesis 9
EDNRB endothelin receptor type B
EDRF1 erythroid differentiation regulatory factor 1
EFNB3 ephrin-B3
ESR1 estrogen receptor 1
EVPL envoplakin
FAM182B family with sequence similarity 182, member B
FHL1 four and a half LIM domains 1
FLJ22184
FYB FYN binding protein
GPR137 G protein-coupled receptor 137
GRIP2 glutamate receptor interacting protein 2
HECW1 HECT, C2 and WW domain containing E3 ubiquitin protein ligase 1
HFE hemochromatosis
HLA-DOA major histocompatibility complex, class II, DO alpha
HOXB9 homeobox B9
HSPA12A heat shock 70kDa protein 12A
IBSP integrin-binding sialoprotein
IRS2 insulin receptor substrate 2
JAM3 junctional adhesion molecule 3
KCNC1 potassium channel, voltage gated Shaw related subfamily C, member 1
KCND3 potassium channel, voltage gated Shal related subfamily D, member 3
KCNH2 potassium channel, voltage gated eag related subfamily H, member 2
KCNN1 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 1
KIAA0754 KIAA0754
KLHL25 kelch-like family member 25
LAG3 lymphocyte-activation gene 3
LAMC2 laminin, gamma 2
LMX1B LIM homeobox transcription factor 1, beta
LPPR2 lipid phosphate phosphatase-related protein type 2
LTC4S leukotriene C4 synthase
MAPK14 mitogen-activated protein kinase 14
MC2R melanocortin 2 receptor (adrenocorticotropic hormone)
MED15 mediator complex subunit 15
MN1 meningioma (disrupted in balanced translocation) 1
MTA1 metastasis associated 1
MYO9B myosin IXB
NDUFAF5 NADH dehydrogenase (ubiquinone) complex I, assembly factor 5
NR3C1 nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)
PDE3B phosphodiesterase 3B, cGMP-inhibited
PPARA peroxisome proliferator-activated receptor alpha
PPFIBP2 PTPRF interacting protein, binding protein 2 (liprin beta 2)
PRB1 proline-rich protein BstNI subfamily 1
QTRT1 queuine tRNA-ribosyltransferase 1
RAD54L2 RAD54-like 2 (S. cerevisiae)
RASGRF1 Ras protein-specific guanine nucleotide-releasing factor 1
REC8 REC8 meiotic recombination protein
RELN reelin
RGS7 regulator of G-protein signaling 7
SH3GL3 SH3-domain GRB2-like 3
SIPA1L1 signal-induced proliferation-associated 1 like 1
SIRT5 sirtuin 5
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC24A3 solute carrier family 24 (sodium/potassium/calcium exchanger), member 3
SLC43A3 solute carrier family 43, member 3
SLCO3A1 solute carrier organic anion transporter family, member 3A1
SPTBN1 spectrin, beta, non-erythrocytic 1
SYNJ1 synaptojanin 1
T T, brachyury homolog (mouse)
TAGLN3 transgelin 3
TBC1D13 TBC1 domain family, member 13
TMEM158 transmembrane protein 158 (gene/pseudogene)
TMEM259 transmembrane protein 259
TRIP11 thyroid hormone receptor interactor 11
TRPC5 transient receptor potential cation channel, subfamily C, member 5
TSPAN9 tetraspanin 9
TTLL3 tubulin tyrosine ligase-like family member 3
UNC119 unc-119 homolog (C. elegans)
VAC14 Vac14 homolog (S. cerevisiae)
ZDHHC14 zinc finger, DHHC-type containing 14
ZFPL1 zinc finger protein-like 1
ZNF235 zinc finger protein 235
ZNF324 zinc finger protein 324

decreased expression

Symbol Name
ADRA2C adrenoceptor alpha 2C
AKR1C3 aldo-keto reductase family 1, member C3
ANKEF1 ankyrin repeat and EF-hand domain containing 1
AP1B1 adaptor-related protein complex 1, beta 1 subunit
APBB3 amyloid beta (A4) precursor protein-binding, family B, member 3
APOBEC3B apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3B
ARHGEF16 Rho guanine nucleotide exchange factor (GEF) 16
BCAR3 breast cancer anti-estrogen resistance 3
CAPN15 calpain 15
CCDC85C coiled-coil domain containing 85C
CHST8 carbohydrate (N-acetylgalactosamine 4-0) sulfotransferase 8
CIT citron rho-interacting serine/threonine kinase
CPPED1 calcineurin-like phosphoesterase domain containing 1
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
DCAF10 DDB1 and CUL4 associated factor 10
DNMBP dynamin binding protein
DZANK1 double zinc ribbon and ankyrin repeat domains 1
EHD3 EH-domain containing 3
ELP3 elongator acetyltransferase complex subunit 3
EPPK1 epiplakin 1
FAM160B2 family with sequence similarity 160, member B2
FKBPL FK506 binding protein like
GUSBP3 glucuronidase, beta pseudogene 3
HIRA histone cell cycle regulator
HIST1H1D histone cluster 1, H1d
HIST1H2AJ histone cluster 1, H2aj
HIST1H2BC histone cluster 1, H2bc
HMOX1 heme oxygenase 1
HSD17B1 hydroxysteroid (17-beta) dehydrogenase 1
HSPA2 heat shock 70kDa protein 2
IFNGR2 interferon gamma receptor 2 (interferon gamma transducer 1)
INTS9 integrator complex subunit 9
IRAK4 interleukin-1 receptor-associated kinase 4
IREB2 iron-responsive element binding protein 2
KCTD7 potassium channel tetramerization domain containing 7
KLHL26 kelch-like family member 26
LAMA3 laminin, alpha 3
LINC00339 long intergenic non-protein coding RNA 339
LOC202181 SUMO-interacting motifs containing 1 pseudogene
LOXL1 lysyl oxidase-like 1
LRP2 low density lipoprotein receptor-related protein 2
LRRC8E leucine rich repeat containing 8 family, member E
LSM14B LSM14B, SCD6 homolog B (S. cerevisiae)
LY6D lymphocyte antigen 6 complex, locus D
MANEA mannosidase, endo-alpha
MAP1S microtubule-associated protein 1S
MBNL3 muscleblind-like splicing regulator 3
MECR mitochondrial trans-2-enoyl-CoA reductase
MGC12488
MOCS3 molybdenum cofactor synthesis 3
MSANTD2 Myb/SANT-like DNA-binding domain containing 2
NAV2 neuron navigator 2
NIP7 NIP7, nucleolar pre-rRNA processing protein
NME6 NME/NM23 nucleoside diphosphate kinase 6
OBFC1 oligonucleotide/oligosaccharide-binding fold containing 1
ONECUT2 one cut homeobox 2
OR7E156P olfactory receptor, family 7, subfamily E, member 156 pseudogene
OXTR oxytocin receptor
PCNXL4 pecanex-like 4 (Drosophila)
PHACTR4 phosphatase and actin regulator 4
PIGH phosphatidylinositol glycan anchor biosynthesis, class H
PIM1 Pim-1 proto-oncogene, serine/threonine kinase
PLA2G3 phospholipase A2, group III
POLD1 polymerase (DNA directed), delta 1, catalytic subunit
POLR1B polymerase (RNA) I polypeptide B, 128kDa
PTK6 protein tyrosine kinase 6
PTPN13 protein tyrosine phosphatase, non-receptor type 13 (APO-1/CD95 (Fas)-associated phosphatase)
RAB17 RAB17, member RAS oncogene family
RAB3A RAB3A, member RAS oncogene family
REEP4 receptor accessory protein 4
RFTN1 raftlin, lipid raft linker 1
RNF2 ring finger protein 2
RWDD3 RWD domain containing 3
SERPINA3 serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 3
SHARPIN SHANK-associated RH domain interactor
SHB Src homology 2 domain containing adaptor protein B
SIRT6 sirtuin 6
SLC25A21 solute carrier family 25 (mitochondrial oxoadipate carrier), member 21
SLC9A2 solute carrier family 9, subfamily A (NHE2, cation proton antiporter 2), member 2
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SNORA21 small nucleolar RNA, H/ACA box 21
ST3GAL1 ST3 beta-galactoside alpha-2,3-sialyltransferase 1
SYTL2 synaptotagmin-like 2
TEAD1 TEA domain family member 1 (SV40 transcriptional enhancer factor)
TM6SF1 transmembrane 6 superfamily member 1
TMEM180 transmembrane protein 180
TMEM2 transmembrane protein 2
TMPRSS3 transmembrane protease, serine 3
TNKS2 tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase 2
TRAF2 TNF receptor-associated factor 2
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TSPAN15 tetraspanin 15
TUBA3D tubulin, alpha 3d
USP6NL USP6 N-terminal like
ZBED1 zinc finger, BED-type containing 1
ZFAND3 zinc finger, AN1-type domain 3
ZNF282 zinc finger protein 282
ZNF652 zinc finger protein 652
ZXDC ZXD family zinc finger C