cimetidine-4063 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the cimetidine-4063 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACOX3 acyl-CoA oxidase 3, pristanoyl
ACSS3 acyl-CoA synthetase short-chain family member 3
ADGB androglobin
ADGRB3 adhesion G protein-coupled receptor B3
ALDH3B2 aldehyde dehydrogenase 3 family, member B2
APOBEC3G apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3G
ASIC4 acid sensing (proton gated) ion channel family member 4
ATF7 activating transcription factor 7
ATP2B4 ATPase, Ca++ transporting, plasma membrane 4
C10ORF12 chromosome 10 open reading frame 12
C2CD2L C2CD2-like
CAMK2B calcium/calmodulin-dependent protein kinase II beta
CCND2 cyclin D2
CLCN6 chloride channel, voltage-sensitive 6
CLDN16 claudin 16
CLUL1 clusterin-like 1 (retinal)
CNTN5 contactin 5
COL3A1 collagen, type III, alpha 1
COL9A3 collagen, type IX, alpha 3
COMMD4 COMM domain containing 4
CTSS cathepsin S
CYP2B7P cytochrome P450, family 2, subfamily B, polypeptide 7, pseudogene
DHODH dihydroorotate dehydrogenase (quinone)
ELSPBP1 epididymal sperm binding protein 1
EPHB1 EPH receptor B1
FAXDC2 fatty acid hydroxylase domain containing 2
G3BP1 GTPase activating protein (SH3 domain) binding protein 1
GLP1R glucagon-like peptide 1 receptor
GNRHR gonadotropin-releasing hormone receptor
GRIP2 glutamate receptor interacting protein 2
HIF3A hypoxia inducible factor 3, alpha subunit
HOXD13 homeobox D13
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HTR6 5-hydroxytryptamine (serotonin) receptor 6, G protein-coupled
ING4 inhibitor of growth family, member 4
INSR insulin receptor
KALRN kalirin, RhoGEF kinase
KCNAB1 potassium channel, voltage gated subfamily A regulatory beta subunit 1
KIF1C kinesin family member 1C
KLK1 kallikrein 1
LILRA5 leukocyte immunoglobulin-like receptor, subfamily A (with TM domain), member 5
LSS lanosterol synthase (2,3-oxidosqualene-lanosterol cyclase)
MAPK8 mitogen-activated protein kinase 8
MAPK8IP3 mitogen-activated protein kinase 8 interacting protein 3
MEP1B meprin A, beta
MS4A1 membrane-spanning 4-domains, subfamily A, member 1
MST1L macrophage stimulating 1-like
NCAPH2 non-SMC condensin II complex, subunit H2
NR0B1 nuclear receptor subfamily 0, group B, member 1
NTRK1 neurotrophic tyrosine kinase, receptor, type 1
OGG1 8-oxoguanine DNA glycosylase
OSGIN2 oxidative stress induced growth inhibitor family member 2
P2RY4 pyrimidinergic receptor P2Y, G-protein coupled, 4
PAOX polyamine oxidase (exo-N4-amino)
PDE7B phosphodiesterase 7B
PDGFRA platelet-derived growth factor receptor, alpha polypeptide
PDX1 pancreatic and duodenal homeobox 1
PHF8 PHD finger protein 8
PKD1 polycystic kidney disease 1 (autosomal dominant)
PLCG2 phospholipase C, gamma 2 (phosphatidylinositol-specific)
PLK4 polo-like kinase 4
POU5F1P3 POU class 5 homeobox 1 pseudogene 3
PPBP pro-platelet basic protein (chemokine (C-X-C motif) ligand 7)
PRDM14 PR domain containing 14
PRKACG protein kinase, cAMP-dependent, catalytic, gamma
PSG11 pregnancy specific beta-1-glycoprotein 11
PTAFR platelet-activating factor receptor
PTCRA pre T-cell antigen receptor alpha
PTGDS prostaglandin D2 synthase 21kDa (brain)
PTPN12 protein tyrosine phosphatase, non-receptor type 12
RAP1GAP RAP1 GTPase activating protein
REN renin
RIF1 replication timing regulatory factor 1
RNF126P1 ring finger protein 126 pseudogene 1
RPH3A rabphilin 3A
SAMD4A sterile alpha motif domain containing 4A
SCGB1A1 secretoglobin, family 1A, member 1 (uteroglobin)
SCN4A sodium channel, voltage gated, type IV alpha subunit
SCNN1B sodium channel, non voltage gated 1 beta subunit
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SIGLEC8 sialic acid binding Ig-like lectin 8
SLC25A30 solute carrier family 25, member 30
SMG6 SMG6 nonsense mediated mRNA decay factor
SNAP25 synaptosomal-associated protein, 25kDa
SNTB1 syntrophin, beta 1 (dystrophin-associated protein A1, 59kDa, basic component 1)
SNX13 sorting nexin 13
SPAG6 sperm associated antigen 6
SPATA1 spermatogenesis associated 1
ST8SIA4 ST8 alpha-N-acetyl-neuraminide alpha-2,8-sialyltransferase 4
SYT5 synaptotagmin V
TAOK2 TAO kinase 2
TBXA2R thromboxane A2 receptor
TCF3 transcription factor 3
TTC30A tetratricopeptide repeat domain 30A
ULBP1 UL16 binding protein 1
USP53 ubiquitin specific peptidase 53
VAV2 vav 2 guanine nucleotide exchange factor
VPS16 vacuolar protein sorting 16 homolog (S. cerevisiae)
XRCC6 X-ray repair complementing defective repair in Chinese hamster cells 6
ZNF573 zinc finger protein 573

decreased expression

Symbol Name
ABCB8 ATP-binding cassette, sub-family B (MDR/TAP), member 8
ACADSB acyl-CoA dehydrogenase, short/branched chain
AMDHD2 amidohydrolase domain containing 2
ANKFY1 ankyrin repeat and FYVE domain containing 1
ANKRD36 ankyrin repeat domain 36
ANP32A-IT1 ANP32A intronic transcript 1
ANXA2P1 annexin A2 pseudogene 1
ARHGEF38 Rho guanine nucleotide exchange factor (GEF) 38
ATG16L1 autophagy related 16-like 1 (S. cerevisiae)
BTF3P12 basic transcription factor 3 pseudogene 12
C1RL complement component 1, r subcomponent-like
CAMKMT calmodulin-lysine N-methyltransferase
CLCA1 chloride channel accessory 1
CRELD1 cysteine-rich with EGF-like domains 1
CRMP1 collapsin response mediator protein 1
CUZD1 CUB and zona pellucida-like domains 1
CYB5R2 cytochrome b5 reductase 2
CYP26B1 cytochrome P450, family 26, subfamily B, polypeptide 1
CYP39A1 cytochrome P450, family 39, subfamily A, polypeptide 1
DEPTOR DEP domain containing MTOR-interacting protein
DFNB31 deafness, autosomal recessive 31
DLK2 delta-like 2 homolog (Drosophila)
DPYS dihydropyrimidinase
DTX2 deltex 2, E3 ubiquitin ligase
ERMAP erythroblast membrane-associated protein (Scianna blood group)
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM53B family with sequence similarity 53, member B
FBXO22 F-box protein 22
FBXO31 F-box protein 31
FGL1 fibrinogen-like 1
FURIN furin (paired basic amino acid cleaving enzyme)
GAN gigaxonin
GPC3 glypican 3
GPRIN2 G protein regulated inducer of neurite outgrowth 2
GTF2H2B general transcription factor IIH, polypeptide 2B (pseudogene)
HIST1H1E histone cluster 1, H1e
HIST1H3A histone cluster 1, H3a
HIST1H4C histone cluster 1, H4c
HOOK1 hook microtubule-tethering protein 1
HOXA2 homeobox A2
HOXC5 homeobox C5
HSPA1L heat shock 70kDa protein 1-like
IFT140 intraflagellar transport 140
INO80D INO80 complex subunit D
IRAK4 interleukin-1 receptor-associated kinase 4
KCNS1 potassium voltage-gated channel, modifier subfamily S, member 1
KIF13B kinesin family member 13B
KRT86 keratin 86, type II
LINC00260 long intergenic non-protein coding RNA 260
LPPR4 lipid phosphate phosphatase-related protein type 4
MFHAS1 malignant fibrous histiocytoma amplified sequence 1
MYBBP1A MYB binding protein (P160) 1a
NECAB3 N-terminal EF-hand calcium binding protein 3
NFKBIL1 nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor-like 1
NGF nerve growth factor (beta polypeptide)
NINJ1 ninjurin 1
NPFFR1 neuropeptide FF receptor 1
NT5M 5',3'-nucleotidase, mitochondrial
OR1D2 olfactory receptor, family 1, subfamily D, member 2
P2RY1 purinergic receptor P2Y, G-protein coupled, 1
PAIP2B poly(A) binding protein interacting protein 2B
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
PITPNM1 phosphatidylinositol transfer protein, membrane-associated 1
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PREX2 phosphatidylinositol-3,4,5-trisphosphate-dependent Rac exchange factor 2
PRKAA2 protein kinase, AMP-activated, alpha 2 catalytic subunit
PRR14L proline rich 14-like
RABEP1 rabaptin, RAB GTPase binding effector protein 1
SAYSD1 SAYSVFN motif domain containing 1
SCD5 stearoyl-CoA desaturase 5
SDC3 syndecan 3
SETD8 SET domain containing (lysine methyltransferase) 8
SLC16A6 solute carrier family 16, member 6
SLC6A20 solute carrier family 6 (proline IMINO transporter), member 20
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SMR3A submaxillary gland androgen regulated protein 3A
SSTR4 somatostatin receptor 4
STEAP4 STEAP family member 4
TAOK1 TAO kinase 1
TINAGL1 tubulointerstitial nephritis antigen-like 1
TNFSF12 tumor necrosis factor (ligand) superfamily, member 12
TRAF2 TNF receptor-associated factor 2
TRPV6 transient receptor potential cation channel, subfamily V, member 6
TUBA3C tubulin, alpha 3c
UGT8 UDP glycosyltransferase 8
VASP vasodilator-stimulated phosphoprotein
VEZT vezatin, adherens junctions transmembrane protein
VGF VGF nerve growth factor inducible
WDR25 WD repeat domain 25
WDR62 WD repeat domain 62
ZMAT5 zinc finger, matrin-type 5
ZNF415 zinc finger protein 415
ZNF669 zinc finger protein 669
ZNF747 zinc finger protein 747
ZNF749 zinc finger protein 749
ZNF76 zinc finger protein 76
ZNF768 zinc finger protein 768
ZNF816 zinc finger protein 816
ZSCAN2 zinc finger and SCAN domain containing 2