cinchonine-2133 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

200 genes differentially expressed following the cinchonine-2133 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABHD2 abhydrolase domain containing 2
ABHD6 abhydrolase domain containing 6
ADGRL1 adhesion G protein-coupled receptor L1
AGGF1 angiogenic factor with G patch and FHA domains 1
ALDH5A1 aldehyde dehydrogenase 5 family, member A1
AP1M2 adaptor-related protein complex 1, mu 2 subunit
APAF1 apoptotic peptidase activating factor 1
ARMC4 armadillo repeat containing 4
ATF7IP activating transcription factor 7 interacting protein
ATP2A1 ATPase, Ca++ transporting, cardiac muscle, fast twitch 1
ATP9A ATPase, class II, type 9A
BCL6 B-cell CLL/lymphoma 6
BEND5 BEN domain containing 5
BTN3A1 butyrophilin, subfamily 3, member A1
CACNA1I calcium channel, voltage-dependent, T type, alpha 1I subunit
CAMSAP1 calmodulin regulated spectrin-associated protein 1
CD47 CD47 molecule
CDH8 cadherin 8, type 2
CLGN calmegin
COLQ collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase
CREM cAMP responsive element modulator
CSF2RA colony stimulating factor 2 receptor, alpha, low-affinity (granulocyte-macrophage)
CYP3A5 cytochrome P450, family 3, subfamily A, polypeptide 5
CYTH1 cytohesin 1
DCHS1 dachsous cadherin-related 1
DDR1-AS1 DDR1 antisense RNA 1 (head to head)
DDX51 DEAD (Asp-Glu-Ala-Asp) box polypeptide 51
DEPDC1 DEP domain containing 1
DGCR8 DGCR8 microprocessor complex subunit
DUS2 dihydrouridine synthase 2
EFNA4 ephrin-A4
EIF1 eukaryotic translation initiation factor 1
EMP1 epithelial membrane protein 1
ENTPD7 ectonucleoside triphosphate diphosphohydrolase 7
EPHA1 EPH receptor A1
EXTL3 exostosin-like glycosyltransferase 3
FAM127B family with sequence similarity 127, member B
FAM49A family with sequence similarity 49, member A
FLOT1 flotillin 1
FOXG1 forkhead box G1
GABBR2 gamma-aminobutyric acid (GABA) B receptor, 2
GCLM glutamate-cysteine ligase, modifier subunit
GNRH1 gonadotropin-releasing hormone 1 (luteinizing-releasing hormone)
HEYL hes-related family bHLH transcription factor with YRPW motif-like
HIF3A hypoxia inducible factor 3, alpha subunit
HMOX1 heme oxygenase 1
HOXA1 homeobox A1
HOXA10 homeobox A10
HTRA1 HtrA serine peptidase 1
IL18RAP interleukin 18 receptor accessory protein
IQCK IQ motif containing K
ITGA2B integrin, alpha 2b (platelet glycoprotein IIb of IIb/IIIa complex, antigen CD41)
IZUMO4 IZUMO family member 4
KCTD17 potassium channel tetramerization domain containing 17
KIF1A kinesin family member 1A
KIT v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog
KRAS Kirsten rat sarcoma viral oncogene homolog
LAD1 ladinin 1
LOC100286895 cell division cycle 27 homolog pseudogene
MAP7 microtubule-associated protein 7
MARC1 mitochondrial amidoxime reducing component 1
MCAM melanoma cell adhesion molecule
MORN1 MORN repeat containing 1
NPEPL1 aminopeptidase-like 1
NPTXR neuronal pentraxin receptor
NRF1 nuclear respiratory factor 1
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
NUMA1 nuclear mitotic apparatus protein 1
NXPE3 neurexophilin and PC-esterase domain family, member 3
ORAI2 ORAI calcium release-activated calcium modulator 2
PDK4 pyruvate dehydrogenase kinase, isozyme 4
PHC3 polyhomeotic homolog 3 (Drosophila)
PLSCR3 phospholipid scramblase 3
POU2F2 POU class 2 homeobox 2
PPARD peroxisome proliferator-activated receptor delta
PPP1R12B protein phosphatase 1, regulatory subunit 12B
PRDM1 PR domain containing 1, with ZNF domain
PRKAR2A protein kinase, cAMP-dependent, regulatory, type II, alpha
PRRG2 proline rich Gla (G-carboxyglutamic acid) 2
PVR poliovirus receptor
RPL13P5 ribosomal protein L13 pseudogene 5
RPS2 ribosomal protein S2
RUNX1 runt-related transcription factor 1
SLC1A7 solute carrier family 1 (glutamate transporter), member 7
SLC24A1 solute carrier family 24 (sodium/potassium/calcium exchanger), member 1
SLMO1 slowmo homolog 1 (Drosophila)
SOX10 SRY (sex determining region Y)-box 10
SRC SRC proto-oncogene, non-receptor tyrosine kinase
STAB2 stabilin 2
TAPBPL TAP binding protein-like
TAPT1 transmembrane anterior posterior transformation 1
TBX5 T-box 5
TNFSF14 tumor necrosis factor (ligand) superfamily, member 14
TSC22D2 TSC22 domain family, member 2
UPF3A UPF3 regulator of nonsense transcripts homolog A (yeast)
WNT16 wingless-type MMTV integration site family, member 16
XPNPEP2 X-prolyl aminopeptidase (aminopeptidase P) 2, membrane-bound
ZER1 zyg-11 related, cell cycle regulator
ZMAT5 zinc finger, matrin-type 5
ZNF277 zinc finger protein 277

decreased expression

Symbol Name
ACADS acyl-CoA dehydrogenase, C-2 to C-3 short chain
ACP6 acid phosphatase 6, lysophosphatidic
ALKBH4 alkB, alkylation repair homolog 4 (E. coli)
AOAH acyloxyacyl hydrolase (neutrophil)
AP5S1 adaptor-related protein complex 5, sigma 1 subunit
APOBEC2 apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 2
APOBEC3C apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3C
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BAHD1 bromo adjacent homology domain containing 1
BAX BCL2-associated X protein
BSPRY B-box and SPRY domain containing
C1ORF159 chromosome 1 open reading frame 159
C1ORF21 chromosome 1 open reading frame 21
C1ORF56 chromosome 1 open reading frame 56
C22ORF29 chromosome 22 open reading frame 29
C5 complement component 5
CA11 carbonic anhydrase XI
CCDC176 coiled-coil domain containing 176
CD320 CD320 molecule
CD69 CD69 molecule
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CFP complement factor properdin
CHPF chondroitin polymerizing factor
CILP cartilage intermediate layer protein, nucleotide pyrophosphohydrolase
DENND4C DENN/MADD domain containing 4C
DVL1 dishevelled segment polarity protein 1
EDAR ectodysplasin A receptor
EFNA3 ephrin-A3
ELMO3 engulfment and cell motility 3
ENO3 enolase 3 (beta, muscle)
EXOSC1 exosome component 1
FCGRT Fc fragment of IgG, receptor, transporter, alpha
FMOD fibromodulin
FOSB FBJ murine osteosarcoma viral oncogene homolog B
FOSL1 FOS-like antigen 1
FTO fat mass and obesity associated
GATAD2A GATA zinc finger domain containing 2A
GLTSCR1 glioma tumor suppressor candidate region gene 1
GPR85 G protein-coupled receptor 85
GRIP2 glutamate receptor interacting protein 2
HCAR3 hydroxycarboxylic acid receptor 3
HIRA histone cell cycle regulator
HIST1H1T histone cluster 1, H1t
HNRNPA3P1 heterogeneous nuclear ribonucleoprotein A3 pseudogene 1
HYAL2 hyaluronoglucosaminidase 2
IFT81 intraflagellar transport 81
IGF2BP2 insulin-like growth factor 2 mRNA binding protein 2
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
IL11RA interleukin 11 receptor, alpha
INO80D INO80 complex subunit D
JMJD4 jumonji domain containing 4
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KIFC1 kinesin family member C1
LY6G6C lymphocyte antigen 6 complex, locus G6C
MTHFSD methenyltetrahydrofolate synthetase domain containing
MYBBP1A MYB binding protein (P160) 1a
N6AMT1 N-6 adenine-specific DNA methyltransferase 1 (putative)
NABP1 nucleic acid binding protein 1
NAT6 N-acetyltransferase 6 (GCN5-related)
NEDD9 neural precursor cell expressed, developmentally down-regulated 9
NLK nemo-like kinase
NTSR1 neurotensin receptor 1 (high affinity)
OLR1 oxidized low density lipoprotein (lectin-like) receptor 1
PARP12 poly (ADP-ribose) polymerase family, member 12
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
PPT2 palmitoyl-protein thioesterase 2
PRICKLE3 prickle homolog 3 (Drosophila)
PTCD1 pentatricopeptide repeat domain 1
RAB13 RAB13, member RAS oncogene family
RAC3 ras-related C3 botulinum toxin substrate 3 (rho family, small GTP binding protein Rac3)
RGS13 regulator of G-protein signaling 13
RGS16 regulator of G-protein signaling 16
RNF122 ring finger protein 122
RNF39 ring finger protein 39
RRAS related RAS viral (r-ras) oncogene homolog
SALL2 spalt-like transcription factor 2
SEMA3G sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3G
SERGEF secretion regulating guanine nucleotide exchange factor
SERPINE2 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 2
SGTA small glutamine-rich tetratricopeptide repeat (TPR)-containing, alpha
SIRAL2 SIR2 antiphage like 2
SLC25A22 solute carrier family 25 (mitochondrial carrier: glutamate), member 22
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SNX29P2 sorting nexin 29 pseudogene 2
SOX12 SRY (sex determining region Y)-box 12
SPR sepiapterin reductase (7,8-dihydrobiopterin:NADP+ oxidoreductase)
SULT1B1 sulfotransferase family, cytosolic, 1B, member 1
TAF15 TAF15 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 68kDa
THBS3 thrombospondin 3
THRAP3 thyroid hormone receptor associated protein 3
TMEM180 transmembrane protein 180
TMEM212 transmembrane protein 212
TRIM45 tripartite motif containing 45
TSPAN32 tetraspanin 32
UPP1 uridine phosphorylase 1
WT1-AS WT1 antisense RNA
ZC3H12A zinc finger CCCH-type containing 12A
ZNF185 zinc finger protein 185 (LIM domain)
ZNF215 zinc finger protein 215
ZNF749 zinc finger protein 749