cyproheptadine-5340 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the cyproheptadine-5340 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADM adrenomedullin
AHI1 Abelson helper integration site 1
APOE apolipoprotein E
ARC activity-regulated cytoskeleton-associated protein
ARTN artemin
ATF3 activating transcription factor 3
BCL7A B-cell CLL/lymphoma 7A
BMP4 bone morphogenetic protein 4
CACTIN cactin, spliceosome C complex subunit
CALU calumenin
CGA glycoprotein hormones, alpha polypeptide
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CNNM2 cyclin and CBS domain divalent metal cation transport mediator 2
CTBS chitobiase, di-N-acetyl-
DDIT3 DNA-damage-inducible transcript 3
DDIT4 DNA-damage-inducible transcript 4
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
DUSP1 dual specificity phosphatase 1
DUSP10 dual specificity phosphatase 10
DUSP4 dual specificity phosphatase 4
DXO decapping exoribonuclease
EAF2 ELL associated factor 2
EGR1 early growth response 1
ELF4 E74-like factor 4 (ets domain transcription factor)
ELOVL5 ELOVL fatty acid elongase 5
EPOR erythropoietin receptor
ERO1LB ERO1-like beta (S. cerevisiae)
ESR1 estrogen receptor 1
F11R F11 receptor
FKBP5 FK506 binding protein 5
FOS FBJ murine osteosarcoma viral oncogene homolog
GADD45A growth arrest and DNA-damage-inducible, alpha
GAS2 growth arrest-specific 2
GDPD5 glycerophosphodiester phosphodiesterase domain containing 5
GEM GTP binding protein overexpressed in skeletal muscle
GLYR1 glyoxylate reductase 1 homolog (Arabidopsis)
HLA-J major histocompatibility complex, class I, J (pseudogene)
HMGCS1 3-hydroxy-3-methylglutaryl-CoA synthase 1 (soluble)
HMOX1 heme oxygenase 1
HN1L hematological and neurological expressed 1-like
HSPA6 heat shock 70kDa protein 6 (HSP70B')
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IFIT2 interferon-induced protein with tetratricopeptide repeats 2
IGLJ3 immunoglobulin lambda joining 3
ISG20 interferon stimulated exonuclease gene 20kDa
ITFG2 integrin alpha FG-GAP repeat containing 2
JUN jun proto-oncogene
KAZALD1 Kazal-type serine peptidase inhibitor domain 1
KLF4 Kruppel-like factor 4 (gut)
KLF6 Kruppel-like factor 6
KLHL24 kelch-like family member 24
LMF2 lipase maturation factor 2
LMNB1 lamin B1
MAFF v-maf avian musculoaponeurotic fibrosarcoma oncogene homolog F
MAOB monoamine oxidase B
MTF1 metal-regulatory transcription factor 1
NF2 neurofibromin 2 (merlin)
NFRKB nuclear factor related to kappaB binding protein
NKX3-1 NK3 homeobox 1
NR4A1 nuclear receptor subfamily 4, group A, member 1
NR4A2 nuclear receptor subfamily 4, group A, member 2
OASL 2'-5'-oligoadenylate synthetase-like
ONECUT2 one cut homeobox 2
PAWR PRKC, apoptosis, WT1, regulator
PDE4DIP phosphodiesterase 4D interacting protein
PDLIM7 PDZ and LIM domain 7 (enigma)
PHLDA1 pleckstrin homology-like domain, family A, member 1
PLAUR plasminogen activator, urokinase receptor
PLEKHF1 pleckstrin homology domain containing, family F (with FYVE domain) member 1
PLK3 polo-like kinase 3
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
PPP1R15A protein phosphatase 1, regulatory subunit 15A
RGS2 regulator of G-protein signaling 2
RNF39 ring finger protein 39
SAT1 spermidine/spermine N1-acetyltransferase 1
SLC39A7 solute carrier family 39 (zinc transporter), member 7
SLC6A8 solute carrier family 6 (neurotransmitter transporter), member 8
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SLCO4C1 solute carrier organic anion transporter family, member 4C1
SMAD3 SMAD family member 3
SMG7 SMG7 nonsense mediated mRNA decay factor
SNAPC2 small nuclear RNA activating complex, polypeptide 2, 45kDa
SOGA1 suppressor of glucose, autophagy associated 1
SPRY2 sprouty homolog 2 (Drosophila)
TAP1 transporter 1, ATP-binding cassette, sub-family B (MDR/TAP)
TMED7 transmembrane emp24 protein transport domain containing 7
TNFAIP3 tumor necrosis factor, alpha-induced protein 3
TNFRSF11B tumor necrosis factor receptor superfamily, member 11b
TRIM25 tripartite motif containing 25
TTLL3 tubulin tyrosine ligase-like family member 3
TTLL5 tubulin tyrosine ligase-like family member 5
ULBP2 UL16 binding protein 2
ZBTB48 zinc finger and BTB domain containing 48
ZHX3 zinc fingers and homeoboxes 3
ZNF16 zinc finger protein 16
ZNF37BP zinc finger protein 37B, pseudogene
ZNF428 zinc finger protein 428
ZNF573 zinc finger protein 573
ZNF589 zinc finger protein 589

decreased expression

Symbol Name
ABCB7 ATP-binding cassette, sub-family B (MDR/TAP), member 7
ABCC6 ATP-binding cassette, sub-family C (CFTR/MRP), member 6
ABLIM3 actin binding LIM protein family, member 3
ADCK3 aarF domain containing kinase 3
ANKEF1 ankyrin repeat and EF-hand domain containing 1
ANKZF1 ankyrin repeat and zinc finger domain containing 1
ANXA2P3 annexin A2 pseudogene 3
ASB8 ankyrin repeat and SOCS box containing 8
B4GALT2 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 2
BCKDHA branched chain keto acid dehydrogenase E1, alpha polypeptide
BCKDK branched chain ketoacid dehydrogenase kinase
BDH1 3-hydroxybutyrate dehydrogenase, type 1
BTF3P12 basic transcription factor 3 pseudogene 12
C10ORF2 chromosome 10 open reading frame 2
C9ORF40 chromosome 9 open reading frame 40
CA2 carbonic anhydrase II
CAMKMT calmodulin-lysine N-methyltransferase
CCNJ cyclin J
CDK5RAP2 CDK5 regulatory subunit associated protein 2
CDR2L cerebellar degeneration-related protein 2-like
CEBPA CCAAT/enhancer binding protein (C/EBP), alpha
CMTR1 cap methyltransferase 1
CPT2 carnitine palmitoyltransferase 2
DCUN1D2 DCN1, defective in cullin neddylation 1, domain containing 2
DDX31 DEAD (Asp-Glu-Ala-Asp) box polypeptide 31
DNAJC24 DnaJ (Hsp40) homolog, subfamily C, member 24
DYNC2H1 dynein, cytoplasmic 2, heavy chain 1
EFHD2 EF-hand domain family, member D2
EHHADH enoyl-CoA, hydratase/3-hydroxyacyl CoA dehydrogenase
ETAA1 Ewing tumor-associated antigen 1
EVL Enah/Vasp-like
EYA2 EYA transcriptional coactivator and phosphatase 2
FAM155B family with sequence similarity 155, member B
FAM50B family with sequence similarity 50, member B
GFOD2 glucose-fructose oxidoreductase domain containing 2
GLI3 GLI family zinc finger 3
GPR19 G protein-coupled receptor 19
GRAMD4 GRAM domain containing 4
GTF2H3 general transcription factor IIH, polypeptide 3, 34kDa
GUSBP3 glucuronidase, beta pseudogene 3
HMGCL 3-hydroxymethyl-3-methylglutaryl-CoA lyase
IFI6 interferon, alpha-inducible protein 6
IFITM1 interferon induced transmembrane protein 1
IGFLR1 IGF-like family receptor 1
ITPKC inositol-trisphosphate 3-kinase C
KATNBL1 katanin p80 subunit B-like 1
KLHL36 kelch-like family member 36
LIAS lipoic acid synthetase
LIG1 ligase I, DNA, ATP-dependent
LYPLA2P1 lysophospholipase II pseudogene 1
LZTR1 leucine-zipper-like transcription regulator 1
MAMLD1 mastermind-like domain containing 1
MAPK12 mitogen-activated protein kinase 12
MBOAT2 membrane bound O-acyltransferase domain containing 2
MCM3AP-AS1 MCM3AP antisense RNA 1
MED15 mediator complex subunit 15
MFSD11 major facilitator superfamily domain containing 11
MPPED2 metallophosphoesterase domain containing 2
MTG1 mitochondrial ribosome-associated GTPase 1
MYBBP1A MYB binding protein (P160) 1a
NDE1 nudE neurodevelopment protein 1
NLK nemo-like kinase
NPFFR1 neuropeptide FF receptor 1
OGDH oxoglutarate (alpha-ketoglutarate) dehydrogenase (lipoamide)
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PCSK7 proprotein convertase subtilisin/kexin type 7
PCYOX1L prenylcysteine oxidase 1 like
PFKM phosphofructokinase, muscle
PILRB paired immunoglobin-like type 2 receptor beta
POLR3F polymerase (RNA) III (DNA directed) polypeptide F, 39 kDa
POMGNT1 protein O-linked mannose N-acetylglucosaminyltransferase 1 (beta 1,2-)
POP1 processing of precursor 1, ribonuclease P/MRP subunit (S. cerevisiae)
PRRG1 proline rich Gla (G-carboxyglutamic acid) 1
PTCD2 pentatricopeptide repeat domain 2
PTPRU protein tyrosine phosphatase, receptor type, U
RASSF1 Ras association (RalGDS/AF-6) domain family member 1
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RNF121 ring finger protein 121
RNF31 ring finger protein 31
SEC61A2 Sec61 alpha 2 subunit (S. cerevisiae)
SECISBP2 SECIS binding protein 2
SH3BGR SH3 domain binding glutamate-rich protein
SLC22A18 solute carrier family 22, member 18
SUOX sulfite oxidase
SUSD6 sushi domain containing 6
TARS2 threonyl-tRNA synthetase 2, mitochondrial (putative)
THAP1 THAP domain containing, apoptosis associated protein 1
THBS3 thrombospondin 3
TRAF5 TNF receptor-associated factor 5
TTF2 transcription termination factor, RNA polymerase II
TYK2 tyrosine kinase 2
YRDC yrdC N(6)-threonylcarbamoyltransferase domain containing
ZBED1 zinc finger, BED-type containing 1
ZNF180 zinc finger protein 180
ZNF219 zinc finger protein 219
ZNF227 zinc finger protein 227
ZNF408 zinc finger protein 408
ZNF721 zinc finger protein 721
ZNF787 zinc finger protein 787
ZNF839 zinc finger protein 839