dacarbazine-6816 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the dacarbazine-6816 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAK1 AP2 associated kinase 1
ADAMTS5 ADAM metallopeptidase with thrombospondin type 1 motif, 5
ADGRB3 adhesion G protein-coupled receptor B3
ADRBK1 adrenergic, beta, receptor kinase 1
ALDH1L1 aldehyde dehydrogenase 1 family, member L1
AMT aminomethyltransferase
ANGPTL2 angiopoietin-like 2
ARVCF armadillo repeat gene deleted in velocardiofacial syndrome
ATG10 autophagy related 10
CACNA1A calcium channel, voltage-dependent, P/Q type, alpha 1A subunit
CARD10 caspase recruitment domain family, member 10
CARD14 caspase recruitment domain family, member 14
CASP10 caspase 10, apoptosis-related cysteine peptidase
CCL16 chemokine (C-C motif) ligand 16
CDK18 cyclin-dependent kinase 18
CPN2 carboxypeptidase N, polypeptide 2
CPNE7 copine VII
CPQ carboxypeptidase Q
CYB5R2 cytochrome b5 reductase 2
DAGLA diacylglycerol lipase, alpha
DCN decorin
DOCK6 dedicator of cytokinesis 6
DPYS dihydropyrimidinase
DSC3 desmocollin 3
EDAR ectodysplasin A receptor
EHD2 EH-domain containing 2
ENPP2 ectonucleotide pyrophosphatase/phosphodiesterase 2
ERCC2 excision repair cross-complementation group 2
FARP2 FERM, RhoGEF and pleckstrin domain protein 2
FGF13 fibroblast growth factor 13
FLJ11292
FN1 fibronectin 1
FUT7 fucosyltransferase 7 (alpha (1,3) fucosyltransferase)
GNA15 guanine nucleotide binding protein (G protein), alpha 15 (Gq class)
GPR137 G protein-coupled receptor 137
GRM1 glutamate receptor, metabotropic 1
HAP1 huntingtin-associated protein 1
HEMK1 HemK methyltransferase family member 1
HESX1 HESX homeobox 1
HLA-DMB major histocompatibility complex, class II, DM beta
ICA1 islet cell autoantigen 1, 69kDa
IL1RAP interleukin 1 receptor accessory protein
IL1RN interleukin 1 receptor antagonist
INO80B INO80 complex subunit B
INPP5J inositol polyphosphate-5-phosphatase J
KAT6A K(lysine) acetyltransferase 6A
KCND3 potassium channel, voltage gated Shal related subfamily D, member 3
KHSRP KH-type splicing regulatory protein
KIAA1109 KIAA1109
KIAA1462 KIAA1462
KIF25-AS1 KIF25 antisense RNA 1
MBNL3 muscleblind-like splicing regulator 3
MST1R macrophage stimulating 1 receptor
MUC8 mucin 8
MYBPC3 myosin binding protein C, cardiac
MYH14 myosin, heavy chain 14, non-muscle
MYL4 myosin, light chain 4, alkali; atrial, embryonic
NAAA N-acylethanolamine acid amidase
NAG18 NAG18 mRNA
NEDD4L neural precursor cell expressed, developmentally down-regulated 4-like, E3 ubiquitin protein ligase
ONECUT2 one cut homeobox 2
PAOX polyamine oxidase (exo-N4-amino)
PER1 period circadian clock 1
PFKFB2 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 2
PIP prolactin-induced protein
PIP5K1A phosphatidylinositol-4-phosphate 5-kinase, type I, alpha
PKD1 polycystic kidney disease 1 (autosomal dominant)
PPP2R1B protein phosphatase 2, regulatory subunit A, beta
PRKCE protein kinase C, epsilon
PTGER3 prostaglandin E receptor 3 (subtype EP3)
PVR poliovirus receptor
PXDC1 PX domain containing 1
RABGAP1L RAB GTPase activating protein 1-like
REEP2 receptor accessory protein 2
RELB v-rel avian reticuloendotheliosis viral oncogene homolog B
RNF125 ring finger protein 125, E3 ubiquitin protein ligase
RNF208 ring finger protein 208
RUNDC3A RUN domain containing 3A
SCLY selenocysteine lyase
SH3GL3 SH3-domain GRB2-like 3
SIK3 SIK family kinase 3
SIT1 signaling threshold regulating transmembrane adaptor 1
SIX3 SIX homeobox 3
SLC35D1 solute carrier family 35 (UDP-GlcA/UDP-GalNAc transporter), member D1
SOX9 SRY (sex determining region Y)-box 9
SPRR1A small proline-rich protein 1A
SPRR2B small proline-rich protein 2B
TAT tyrosine aminotransferase
TBKBP1 TBK1 binding protein 1
TBL2 transducin (beta)-like 2
TFAP2B transcription factor AP-2 beta (activating enhancer binding protein 2 beta)
TFF2 trefoil factor 2
TGFB1 transforming growth factor, beta 1
TMPRSS4 transmembrane protease, serine 4
TNFSF18 tumor necrosis factor (ligand) superfamily, member 18
TUBA4B tubulin, alpha 4b
XYLB xylulokinase homolog (H. influenzae)
ZCCHC24 zinc finger, CCHC domain containing 24
ZNF862 zinc finger protein 862

decreased expression

Symbol Name
ALS2CL ALS2 C-terminal like
ANP32A-IT1 ANP32A intronic transcript 1
ARHGDIG Rho GDP dissociation inhibitor (GDI) gamma
B3GNT3 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 3
BAG4 BCL2-associated athanogene 4
BTF3P12 basic transcription factor 3 pseudogene 12
C1ORF105 chromosome 1 open reading frame 105
CAMKMT calmodulin-lysine N-methyltransferase
CAPG capping protein (actin filament), gelsolin-like
CBX8 chromobox homolog 8
CCNO cyclin O
CD302 CD302 molecule
CD82 CD82 molecule
CDK3 cyclin-dependent kinase 3
CLCN5 chloride channel, voltage-sensitive 5
CLCN6 chloride channel, voltage-sensitive 6
CRY2 cryptochrome circadian clock 2
CTBS chitobiase, di-N-acetyl-
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
DGAT1 diacylglycerol O-acyltransferase 1
DHX8 DEAH (Asp-Glu-Ala-His) box polypeptide 8
DNAL4 dynein, axonemal, light chain 4
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha
DOC2A double C2-like domains, alpha
DUSP2 dual specificity phosphatase 2
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3
EDC4 enhancer of mRNA decapping 4
ELOVL4 ELOVL fatty acid elongase 4
F2R coagulation factor II (thrombin) receptor
F8 coagulation factor VIII, procoagulant component
FAM204A family with sequence similarity 204, member A
FAM63A family with sequence similarity 63, member A
FBXW12 F-box and WD repeat domain containing 12
GBP2 guanylate binding protein 2, interferon-inducible
GPATCH3 G patch domain containing 3
HIST1H2AJ histone cluster 1, H2aj
HMHA1 histocompatibility (minor) HA-1
HOXC8 homeobox C8
IFI27 interferon, alpha-inducible protein 27
IFI6 interferon, alpha-inducible protein 6
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IL4R interleukin 4 receptor
IMPACT impact RWD domain protein
KAT2A K(lysine) acetyltransferase 2A
LINC00115 long intergenic non-protein coding RNA 115
MAP9 microtubule-associated protein 9
MAST3 microtubule associated serine/threonine kinase 3
MUL1 mitochondrial E3 ubiquitin protein ligase 1
MVP major vault protein
MYO1D myosin ID
NDRG1 N-myc downstream regulated 1
NEK11 NIMA-related kinase 11
NFKBIE nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, epsilon
NRSN2 neurensin 2
OR7E47P olfactory receptor, family 7, subfamily E, member 47 pseudogene
PADI3 peptidyl arginine deiminase, type III
PIK3R2 phosphoinositide-3-kinase, regulatory subunit 2 (beta)
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PIP5K1C phosphatidylinositol-4-phosphate 5-kinase, type I, gamma
PLCXD1 phosphatidylinositol-specific phospholipase C, X domain containing 1
PLEKHM2 pleckstrin homology domain containing, family M (with RUN domain) member 2
PNPLA6 patatin-like phospholipase domain containing 6
PPT2 palmitoyl-protein thioesterase 2
PRRG1 proline rich Gla (G-carboxyglutamic acid) 1
PTTG3P pituitary tumor-transforming 3, pseudogene
RAD54L2 RAD54-like 2 (S. cerevisiae)
RAMP1 receptor (G protein-coupled) activity modifying protein 1
RFTN1 raftlin, lipid raft linker 1
RUFY2 RUN and FYVE domain containing 2
SCD5 stearoyl-CoA desaturase 5
SETD8 SET domain containing (lysine methyltransferase) 8
SIGIRR single immunoglobulin and toll-interleukin 1 receptor (TIR) domain
SLC31A2 solute carrier family 31 (copper transporter), member 2
SLC39A7 solute carrier family 39 (zinc transporter), member 7
SLC44A1 solute carrier family 44 (choline transporter), member 1
SLC8B1 solute carrier family 8 (sodium/lithium/calcium exchanger), member B1
SYNGR3 synaptogyrin 3
TAF4B TAF4b RNA polymerase II, TATA box binding protein (TBP)-associated factor, 105kDa
TH tyrosine hydroxylase
THBS3 thrombospondin 3
THNSL1 threonine synthase-like 1 (S. cerevisiae)
TMA16 translation machinery associated 16 homolog (S. cerevisiae)
TRABD TraB domain containing
TRMU tRNA 5-methylaminomethyl-2-thiouridylate methyltransferase
TUBA3C tubulin, alpha 3c
TUBGCP5 tubulin, gamma complex associated protein 5
UNC119 unc-119 homolog (C. elegans)
VASH1 vasohibin 1
WDR4 WD repeat domain 4
WLS wntless Wnt ligand secretion mediator
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZCWPW1 zinc finger, CW type with PWWP domain 1
ZNF219 zinc finger protein 219
ZNF268 zinc finger protein 268
ZNF282 zinc finger protein 282
ZNF324 zinc finger protein 324
ZNF516 zinc finger protein 516
ZNF571 zinc finger protein 571
ZNF675 zinc finger protein 675