diltiazem-1532 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

193 genes differentially expressed following the diltiazem-1532 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AIRE autoimmune regulator
ANKRD12 ankyrin repeat domain 12
ARL4C ADP-ribosylation factor-like 4C
B9D2 B9 protein domain 2
BAZ2A bromodomain adjacent to zinc finger domain, 2A
CA5A carbonic anhydrase VA, mitochondrial
CDC14B cell division cycle 14B
CDRT1 CMT1A duplicated region transcript 1
CEACAM5 carcinoembryonic antigen-related cell adhesion molecule 5
CEP97 centrosomal protein 97kDa
CHST5 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 5
CNTN1 contactin 1
CNTNAP2 contactin associated protein-like 2
COL3A1 collagen, type III, alpha 1
CYP2B7P cytochrome P450, family 2, subfamily B, polypeptide 7, pseudogene
DEPDC5 DEP domain containing 5
DHRS2 dehydrogenase/reductase (SDR family) member 2
DHX34 DEAH (Asp-Glu-Ala-His) box polypeptide 34
DOK2 docking protein 2, 56kDa
EFNB3 ephrin-B3
EMID1 EMI domain containing 1
ENTPD4 ectonucleoside triphosphate diphosphohydrolase 4
EPS8L1 EPS8-like 1
ETV5 ets variant 5
EVI5 ecotropic viral integration site 5
FAM46C family with sequence similarity 46, member C
FOXG1 forkhead box G1
GNA14 guanine nucleotide binding protein (G protein), alpha 14
GPD2 glycerol-3-phosphate dehydrogenase 2 (mitochondrial)
GTPBP1 GTP binding protein 1
HIST1H2AL histone cluster 1, H2al
HSD17B6 hydroxysteroid (17-beta) dehydrogenase 6
ICAM1 intercellular adhesion molecule 1
ICAM4 intercellular adhesion molecule 4 (Landsteiner-Wiener blood group)
IDUA iduronidase, alpha-L-
IMPG2 interphotoreceptor matrix proteoglycan 2
INHBE inhibin, beta E
INPP5B inositol polyphosphate-5-phosphatase, 75kDa
KRT17 keratin 17, type I
LILRA5 leukocyte immunoglobulin-like receptor, subfamily A (with TM domain), member 5
LPXN leupaxin
LYZL6 lysozyme-like 6
MAP2K5 mitogen-activated protein kinase kinase 5
MED16 mediator complex subunit 16
MED25 mediator complex subunit 25
MFGE8 milk fat globule-EGF factor 8 protein
MPPE1 metallophosphoesterase 1
MTSS1L metastasis suppressor 1-like
MYL4 myosin, light chain 4, alkali; atrial, embryonic
MYOM2 myomesin 2
NFATC1 nuclear factor of activated T-cells, cytoplasmic, calcineurin-dependent 1
NPHP1 nephronophthisis 1 (juvenile)
NR3C1 nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)
OLFML2A olfactomedin-like 2A
OR1G1 olfactory receptor, family 1, subfamily G, member 1
PARD6B par-6 family cell polarity regulator beta
PBX2 pre-B-cell leukemia homeobox 2
PCDH9 protocadherin 9
POFUT1 protein O-fucosyltransferase 1
POPDC3 popeye domain containing 3
PRKCQ protein kinase C, theta
PTCRA pre T-cell antigen receptor alpha
PVR poliovirus receptor
RALGAPA1 Ral GTPase activating protein, alpha subunit 1 (catalytic)
RSU1 Ras suppressor protein 1
SCAI suppressor of cancer cell invasion
SCUBE3 signal peptide, CUB domain, EGF-like 3
SEC61A2 Sec61 alpha 2 subunit (S. cerevisiae)
SFTPD surfactant protein D
SLC24A2 solute carrier family 24 (sodium/potassium/calcium exchanger), member 2
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC2A9 solute carrier family 2 (facilitated glucose transporter), member 9
SLC46A3 solute carrier family 46, member 3
SLC7A9 solute carrier family 7 (amino acid transporter light chain, bo,+ system), member 9
SPRY1 sprouty homolog 1, antagonist of FGF signaling (Drosophila)
SPTBN1 spectrin, beta, non-erythrocytic 1
SYT5 synaptotagmin V
TAB1 TGF-beta activated kinase 1/MAP3K7 binding protein 1
TDRKH tudor and KH domain containing
TMEM206 transmembrane protein 206
TNFAIP3 tumor necrosis factor, alpha-induced protein 3
TUBA3C tubulin, alpha 3c
UBE3A ubiquitin protein ligase E3A
USB1 U6 snRNA biogenesis 1
USP36 ubiquitin specific peptidase 36
VIPR1 vasoactive intestinal peptide receptor 1
WSCD1 WSC domain containing 1
YY2 YY2 transcription factor
ZBTB43 zinc finger and BTB domain containing 43
ZCCHC14 zinc finger, CCHC domain containing 14
ZFYVE9 zinc finger, FYVE domain containing 9
ZNF442 zinc finger protein 442
ZNF518A zinc finger protein 518A
ZNF532 zinc finger protein 532
ZNF747 zinc finger protein 747
ZNF79 zinc finger protein 79

decreased expression

Symbol Name
ABHD4 abhydrolase domain containing 4
ACTR3B ARP3 actin-related protein 3 homolog B (yeast)
AHDC1 AT hook, DNA binding motif, containing 1
ARHGDIG Rho GDP dissociation inhibitor (GDI) gamma
ARMC6 armadillo repeat containing 6
ATAD3A ATPase family, AAA domain containing 3A
ATG2A autophagy related 2A
BAGE B melanoma antigen
BBS7 Bardet-Biedl syndrome 7
C1ORF105 chromosome 1 open reading frame 105
C7ORF43 chromosome 7 open reading frame 43
CBX4 chromobox homolog 4
CD3EAP CD3e molecule, epsilon associated protein
CHKB choline kinase beta
CLCF1 cardiotrophin-like cytokine factor 1
CLCN5 chloride channel, voltage-sensitive 5
CLN6 ceroid-lipofuscinosis, neuronal 6, late infantile, variant
DENND4A DENN/MADD domain containing 4A
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha
EDEM1 ER degradation enhancer, mannosidase alpha-like 1
ERCC4 excision repair cross-complementation group 4
F2R coagulation factor II (thrombin) receptor
FAM189A2 family with sequence similarity 189, member A2
FAM86C1 family with sequence similarity 86, member C1
FBXL6 F-box and leucine-rich repeat protein 6
FER fer (fps/fes related) tyrosine kinase
FOSL1 FOS-like antigen 1
GPR87 G protein-coupled receptor 87
GSTA4 glutathione S-transferase alpha 4
GTPBP2 GTP binding protein 2
HIST1H2AE histone cluster 1, H2ae
HIST1H2AJ histone cluster 1, H2aj
ICK intestinal cell (MAK-like) kinase
IL17RA interleukin 17 receptor A
IRF2BP1 interferon regulatory factor 2 binding protein 1
KLC2 kinesin light chain 2
KLHL25 kelch-like family member 25
KRI1 KRI1 homolog (S. cerevisiae)
LGALS4 lectin, galactoside-binding, soluble, 4
LIME1 Lck interacting transmembrane adaptor 1
LNPEP leucyl/cystinyl aminopeptidase
LOC257152 uncharacterized LOC257152
LOC642236 FSHD region gene 1 pseudogene
LRFN3 leucine rich repeat and fibronectin type III domain containing 3
MAN2C1 mannosidase, alpha, class 2C, member 1
MAP1S microtubule-associated protein 1S
MBTD1 mbt domain containing 1
MCMBP minichromosome maintenance complex binding protein
MCOLN3 mucolipin 3
MVP major vault protein
MYO19 myosin XIX
NACAP1 nascent-polypeptide-associated complex alpha polypeptide pseudogene 1
NDE1 nudE neurodevelopment protein 1
NEK11 NIMA-related kinase 11
NPIPB3 nuclear pore complex interacting protein family, member B3
NPL N-acetylneuraminate pyruvate lyase (dihydrodipicolinate synthase)
NT5C 5', 3'-nucleotidase, cytosolic
OLFML3 olfactomedin-like 3
PAFAH2 platelet-activating factor acetylhydrolase 2, 40kDa
PARP16 poly (ADP-ribose) polymerase family, member 16
PDPR pyruvate dehydrogenase phosphatase regulatory subunit
PIM1 Pim-1 proto-oncogene, serine/threonine kinase
PIP5K1C phosphatidylinositol-4-phosphate 5-kinase, type I, gamma
PITPNM1 phosphatidylinositol transfer protein, membrane-associated 1
PLCXD1 phosphatidylinositol-specific phospholipase C, X domain containing 1
PLXNA3 plexin A3
PODXL2 podocalyxin-like 2
PTTG3P pituitary tumor-transforming 3, pseudogene
PYCRL pyrroline-5-carboxylate reductase-like
RAB30 RAB30, member RAS oncogene family
RHBDD3 rhomboid domain containing 3
RNF31 ring finger protein 31
SKA1 spindle and kinetochore associated complex subunit 1
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SLC41A3 solute carrier family 41, member 3
SP1 Sp1 transcription factor
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5
TFF2 trefoil factor 2
THRAP3 thyroid hormone receptor associated protein 3
TMPRSS2 transmembrane protease, serine 2
TMSB15A thymosin beta 15a
TNFRSF11A tumor necrosis factor receptor superfamily, member 11a, NFKB activator
TOM1 target of myb1 (chicken)
TRABD TraB domain containing
TRAPPC13 trafficking protein particle complex 13
VEGFB vascular endothelial growth factor B
VPS54 vacuolar protein sorting 54 homolog (S. cerevisiae)
XAB2 XPA binding protein 2
XPNPEP3 X-prolyl aminopeptidase 3, mitochondrial
ZBTB22 zinc finger and BTB domain containing 22
ZCWPW1 zinc finger, CW type with PWWP domain 1
ZNF227 zinc finger protein 227
ZNF280D zinc finger protein 280D
ZNF480 zinc finger protein 480
ZNF768 zinc finger protein 768
ZNF816 zinc finger protein 816