dropropizine-2398 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the dropropizine-2398 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCG4 ATP-binding cassette, sub-family G (WHITE), member 4
ABHD17B abhydrolase domain containing 17B
ADAMTS8 ADAM metallopeptidase with thrombospondin type 1 motif, 8
ADAMTS9 ADAM metallopeptidase with thrombospondin type 1 motif, 9
ADGRL1 adhesion G protein-coupled receptor L1
AKR1C1 aldo-keto reductase family 1, member C1
ALDH4A1 aldehyde dehydrogenase 4 family, member A1
AMACR alpha-methylacyl-CoA racemase
AP4S1 adaptor-related protein complex 4, sigma 1 subunit
APAF1 apoptotic peptidase activating factor 1
APCS amyloid P component, serum
APOBEC3C apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3C
AVL9 AVL9 homolog (S. cerevisiase)
BTN2A2 butyrophilin, subfamily 2, member A2
C11ORF30 chromosome 11 open reading frame 30
CASP10 caspase 10, apoptosis-related cysteine peptidase
CCDC106 coiled-coil domain containing 106
CD200 CD200 molecule
CDC42BPA CDC42 binding protein kinase alpha (DMPK-like)
CDX1 caudal type homeobox 1
CEACAM6 carcinoembryonic antigen-related cell adhesion molecule 6 (non-specific cross reacting antigen)
CHGB chromogranin B
CTSF cathepsin F
CXXC4 CXXC finger protein 4
DDX17 DEAD (Asp-Glu-Ala-Asp) box helicase 17
DEFA4 defensin, alpha 4, corticostatin
DHRS9 dehydrogenase/reductase (SDR family) member 9
DNAJC1 DnaJ (Hsp40) homolog, subfamily C, member 1
EIF1 eukaryotic translation initiation factor 1
EMC3 ER membrane protein complex subunit 3
ENTPD5 ectonucleoside triphosphate diphosphohydrolase 5
EXPH5 exophilin 5
FERMT1 fermitin family member 1
FLJ11292
FOXO4 forkhead box O4
GABARAPL1 GABA(A) receptor-associated protein like 1
GLB1L galactosidase, beta 1-like
HDAC6 histone deacetylase 6
HSD17B6 hydroxysteroid (17-beta) dehydrogenase 6
HTR4 5-hydroxytryptamine (serotonin) receptor 4, G protein-coupled
IFNA14 interferon, alpha 14
INHBA inhibin, beta A
KCNIP1 Kv channel interacting protein 1
KIF1C kinesin family member 1C
L3MBTL1 l(3)mbt-like 1 (Drosophila)
LAD1 ladinin 1
LBX1 ladybird homeobox 1
LINC00652 long intergenic non-protein coding RNA 652
LRP1 low density lipoprotein receptor-related protein 1
MAGEA5 melanoma antigen family A5
MAP7 microtubule-associated protein 7
MST1 macrophage stimulating 1
MYCNOS MYCN opposite strand
N4BP2L2-IT2 N4BPL2 intronic transcript 2
NMT2 N-myristoyltransferase 2
NR2F1 nuclear receptor subfamily 2, group F, member 1
NR4A1 nuclear receptor subfamily 4, group A, member 1
NRF1 nuclear respiratory factor 1
NRL neural retina leucine zipper
NUP188 nucleoporin 188kDa
OSBPL7 oxysterol binding protein-like 7
PAX9 paired box 9
PCGF3 polycomb group ring finger 3
PDE3B phosphodiesterase 3B, cGMP-inhibited
PDE8B phosphodiesterase 8B
PDLIM2 PDZ and LIM domain 2 (mystique)
PGAP3 post-GPI attachment to proteins 3
PLK4 polo-like kinase 4
POU6F2 POU class 6 homeobox 2
PPP2R2B protein phosphatase 2, regulatory subunit B, beta
QSER1 glutamine and serine rich 1
RPL13P5 ribosomal protein L13 pseudogene 5
RUNX1T1 runt-related transcription factor 1; translocated to, 1 (cyclin D-related)
SERPINB3 serpin peptidase inhibitor, clade B (ovalbumin), member 3
SFI1 Sfi1 homolog, spindle assembly associated (yeast)
SLC4A4 solute carrier family 4 (sodium bicarbonate cotransporter), member 4
SNAPC5 small nuclear RNA activating complex, polypeptide 5, 19kDa
SNPH syntaphilin
SOS2 son of sevenless homolog 2 (Drosophila)
SPRR1B small proline-rich protein 1B
SS18 synovial sarcoma translocation, chromosome 18
STBD1 starch binding domain 1
STS steroid sulfatase (microsomal), isozyme S
STYK1 serine/threonine/tyrosine kinase 1
TBC1D17 TBC1 domain family, member 17
TBC1D9 TBC1 domain family, member 9 (with GRAM domain)
TBX2 T-box 2
TGFB1I1 transforming growth factor beta 1 induced transcript 1
TGFBR2 transforming growth factor, beta receptor II (70/80kDa)
TNNT2 troponin T type 2 (cardiac)
TTC38 tetratricopeptide repeat domain 38
UBOX5 U-box domain containing 5
UBXN1 UBX domain protein 1
USP2 ubiquitin specific peptidase 2
VEZT vezatin, adherens junctions transmembrane protein
ZC3H7B zinc finger CCCH-type containing 7B
ZNF177 zinc finger protein 177
ZNF185 zinc finger protein 185 (LIM domain)
ZNF34 zinc finger protein 34

decreased expression

Symbol Name
ACVR1 activin A receptor, type I
AEN apoptosis enhancing nuclease
AGO4 argonaute RISC catalytic component 4
AHR aryl hydrocarbon receptor
ANAPC2 anaphase promoting complex subunit 2
ARSB arylsulfatase B
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
AXIN1 axin 1
BACE1 beta-site APP-cleaving enzyme 1
BHLHE41 basic helix-loop-helix family, member e41
BRIX1 BRX1, biogenesis of ribosomes
CA11 carbonic anhydrase XI
CAPN1 calpain 1, (mu/I) large subunit
CAPN5 calpain 5
CCS copper chaperone for superoxide dismutase
CDR2L cerebellar degeneration-related protein 2-like
CECR1 cat eye syndrome chromosome region, candidate 1
CEP97 centrosomal protein 97kDa
CHMP1A charged multivesicular body protein 1A
CLCF1 cardiotrophin-like cytokine factor 1
COL4A3BP collagen, type IV, alpha 3 (Goodpasture antigen) binding protein
CST3 cystatin C
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1
DDN dendrin
DENND2D DENN/MADD domain containing 2D
DGCR11 DiGeorge syndrome critical region gene 11 (non-protein coding)
DKK2 dickkopf WNT signaling pathway inhibitor 2
ERCC4 excision repair cross-complementation group 4
ERN2 endoplasmic reticulum to nucleus signaling 2
ETAA1 Ewing tumor-associated antigen 1
FAM163A family with sequence similarity 163, member A
FAM184A family with sequence similarity 184, member A
GLTSCR1 glioma tumor suppressor candidate region gene 1
GSTCD glutathione S-transferase, C-terminal domain containing
GSTZ1 glutathione S-transferase zeta 1
HDAC5 histone deacetylase 5
HIST1H4J histone cluster 1, H4j
HOPX HOP homeobox
IER3 immediate early response 3
IFT88 intraflagellar transport 88
ITGB7 integrin, beta 7
JUNB jun B proto-oncogene
L2HGDH L-2-hydroxyglutarate dehydrogenase
LAIR2 leukocyte-associated immunoglobulin-like receptor 2
LPPR3 lipid phosphate phosphatase-related protein type 3
LRP2 low density lipoprotein receptor-related protein 2
LRP5 low density lipoprotein receptor-related protein 5
LRRK1 leucine-rich repeat kinase 1
MANSC1 MANSC domain containing 1
MAP1S microtubule-associated protein 1S
METTL21B methyltransferase like 21B
MKS1 Meckel syndrome, type 1
MTA2 metastasis associated 1 family, member 2
NCS1 neuronal calcium sensor 1
NPFFR1 neuropeptide FF receptor 1
NR1H2 nuclear receptor subfamily 1, group H, member 2
OCEL1 occludin/ELL domain containing 1
PADI1 peptidyl arginine deiminase, type I
PITPNM1 phosphatidylinositol transfer protein, membrane-associated 1
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
POLM polymerase (DNA directed), mu
POMZP3 POM121 and ZP3 fusion
PRKG2 protein kinase, cGMP-dependent, type II
PYCR1 pyrroline-5-carboxylate reductase 1
RAB33B RAB33B, member RAS oncogene family
RARS arginyl-tRNA synthetase
RBM42 RNA binding motif protein 42
RELB v-rel avian reticuloendotheliosis viral oncogene homolog B
RNF121 ring finger protein 121
RNF126P1 ring finger protein 126 pseudogene 1
RPA4 replication protein A4, 30kDa
SCAI suppressor of cancer cell invasion
SCML1 sex comb on midleg-like 1 (Drosophila)
SETD1A SET domain containing 1A
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SLITRK5 SLIT and NTRK-like family, member 5
SLPI secretory leukocyte peptidase inhibitor
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SMYD5 SMYD family member 5
SPATA2L spermatogenesis associated 2-like
SULT1B1 sulfotransferase family, cytosolic, 1B, member 1
TASP1 taspase, threonine aspartase, 1
TEC tec protein tyrosine kinase
TET3 tet methylcytosine dioxygenase 3
TSPAN32 tetraspanin 32
TUBA3C tubulin, alpha 3c
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
UBXN6 UBX domain protein 6
USP19 ubiquitin specific peptidase 19
VPS37B vacuolar protein sorting 37 homolog B (S. cerevisiae)
YY2 YY2 transcription factor
ZBTB39 zinc finger and BTB domain containing 39
ZHX2 zinc fingers and homeoboxes 2
ZKSCAN3 zinc finger with KRAB and SCAN domains 3
ZNF493 zinc finger protein 493
ZNF665 zinc finger protein 665
ZNF710 zinc finger protein 710
ZNF747 zinc finger protein 747