estradiol-1299 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

200 genes differentially expressed following the estradiol-1299 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCA1 ATP-binding cassette, sub-family A (ABC1), member 1
ADAM28 ADAM metallopeptidase domain 28
AP4S1 adaptor-related protein complex 4, sigma 1 subunit
ARHGDIA Rho GDP dissociation inhibitor (GDI) alpha
ARL1 ADP-ribosylation factor-like 1
ATP13A3 ATPase type 13A3
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BCAT1 branched chain amino-acid transaminase 1, cytosolic
BTN3A1 butyrophilin, subfamily 3, member A1
CASP2 caspase 2, apoptosis-related cysteine peptidase
CASP8 caspase 8, apoptosis-related cysteine peptidase
CDC14A cell division cycle 14A
CDK2AP2 cyclin-dependent kinase 2 associated protein 2
CEP72 centrosomal protein 72kDa
CLCN7 chloride channel, voltage-sensitive 7
COPA coatomer protein complex, subunit alpha
CR1 complement component (3b/4b) receptor 1 (Knops blood group)
CRISPLD2 cysteine-rich secretory protein LCCL domain containing 2
CRKL v-crk avian sarcoma virus CT10 oncogene homolog-like
CSF2RA colony stimulating factor 2 receptor, alpha, low-affinity (granulocyte-macrophage)
CTAGE5 CTAGE family, member 5
CUL4B cullin 4B
DDX3X DEAD (Asp-Glu-Ala-Asp) box helicase 3, X-linked
DNAJB12 DnaJ (Hsp40) homolog, subfamily B, member 12
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
DSCR3 Down syndrome critical region 3
EWSR1 EWS RNA-binding protein 1
FEZ2 fasciculation and elongation protein zeta 2 (zygin II)
FKBP8 FK506 binding protein 8, 38kDa
FLOT1 flotillin 1
FNDC3A fibronectin type III domain containing 3A
FOSL2 FOS-like antigen 2
GLE1 GLE1 RNA export mediator
GLG1 golgi glycoprotein 1
GTF2I general transcription factor IIi
HCRP1 hepatocellular carcinoma-related HCRP1
HIST1H2BG histone cluster 1, H2bg
HOXA5 homeobox A5
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1
ICAM4 intercellular adhesion molecule 4 (Landsteiner-Wiener blood group)
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
INF2 inverted formin, FH2 and WH2 domain containing
ING4 inhibitor of growth family, member 4
JAG1 jagged 1
LINC00094 long intergenic non-protein coding RNA 94
LMAN1 lectin, mannose-binding, 1
MAP4 microtubule-associated protein 4
MCL1 myeloid cell leukemia 1
MED20 mediator complex subunit 20
MFN2 mitofusin 2
MLH3 mutL homolog 3
MLLT10 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 10
MT1E metallothionein 1E
MT1F metallothionein 1F
MT1G metallothionein 1G
MT1H metallothionein 1H
MT1HL1 metallothionein 1H-like 1
MT1X metallothionein 1X
MT2A metallothionein 2A
MYDGF myeloid-derived growth factor
N6AMT1 N-6 adenine-specific DNA methyltransferase 1 (putative)
NAB1 NGFI-A binding protein 1 (EGR1 binding protein 1)
NEK1 NIMA-related kinase 1
NFYA nuclear transcription factor Y, alpha
NIPSNAP3B nipsnap homolog 3B (C. elegans)
NRP1 neuropilin 1
NUP160 nucleoporin 160kDa
NUS1P3 nuclear undecaprenyl pyrophosphate synthase 1 homolog (S. cerevisiae) pseudogene 3
NXT2 nuclear transport factor 2-like export factor 2
PCM1 pericentriolar material 1
PDE4B phosphodiesterase 4B, cAMP-specific
PEX1 peroxisomal biogenesis factor 1
PGM3 phosphoglucomutase 3
PIP5K1A phosphatidylinositol-4-phosphate 5-kinase, type I, alpha
PRKAR1A protein kinase, cAMP-dependent, regulatory, type I, alpha
PRNP prion protein
PTAFR platelet-activating factor receptor
RAB23 RAB23, member RAS oncogene family
RBKS ribokinase
RNF6 ring finger protein (C3H2C3 type) 6
RNGTT RNA guanylyltransferase and 5'-phosphatase
RPL7 ribosomal protein L7
RRN3P1 RNA polymerase I transcription factor homolog (S. cerevisiae) pseudogene 1
RUNX1 runt-related transcription factor 1
SCARB2 scavenger receptor class B, member 2
SH3BP2 SH3-domain binding protein 2
SIRT5 sirtuin 5
SMEK1 SMEK homolog 1, suppressor of mek1 (Dictyostelium)
SNAI1 snail family zinc finger 1
SRSF1 serine/arginine-rich splicing factor 1
THBS1 thrombospondin 1
TMED2 transmembrane emp24 domain trafficking protein 2
TNFRSF12A tumor necrosis factor receptor superfamily, member 12A
TNFSF14 tumor necrosis factor (ligand) superfamily, member 14
TRAM1 translocation associated membrane protein 1
TRIM36 tripartite motif containing 36
VAMP2 vesicle-associated membrane protein 2 (synaptobrevin 2)
WIPI2 WD repeat domain, phosphoinositide interacting 2
YKT6 YKT6 v-SNARE homolog (S. cerevisiae)
ZNF675 zinc finger protein 675

decreased expression

Symbol Name
ACVR2B activin A receptor, type IIB
AES amino-terminal enhancer of split
AGBL5 ATP/GTP binding protein-like 5
ALPK1 alpha-kinase 1
AMPD2 adenosine monophosphate deaminase 2
ARHGEF1 Rho guanine nucleotide exchange factor (GEF) 1
ASB13 ankyrin repeat and SOCS box containing 13
ATG9A autophagy related 9A
BAHD1 bromo adjacent homology domain containing 1
BBC3 BCL2 binding component 3
BRPF1 bromodomain and PHD finger containing, 1
BTBD18 BTB (POZ) domain containing 18
C3 complement component 3
C5AR1 complement component 5a receptor 1
C5ORF45 chromosome 5 open reading frame 45
C6ORF47 chromosome 6 open reading frame 47
CHD8 chromodomain helicase DNA binding protein 8
CHMP7 charged multivesicular body protein 7
CNP 2',3'-cyclic nucleotide 3' phosphodiesterase
CPSF7 cleavage and polyadenylation specific factor 7, 59kDa
DEAF1 DEAF1 transcription factor
DENND1C DENN/MADD domain containing 1C
DIP2A DIP2 disco-interacting protein 2 homolog A (Drosophila)
EOGT EGF domain-specific O-linked N-acetylglucosamine (GlcNAc) transferase
ETAA1 Ewing tumor-associated antigen 1
FAM189B family with sequence similarity 189, member B
GNL1 guanine nucleotide binding protein-like 1
GRAMD4 GRAM domain containing 4
GRINA glutamate receptor, ionotropic, N-methyl D-aspartate-associated protein 1 (glutamate binding)
GRWD1 glutamate-rich WD repeat containing 1
GSDMD gasdermin D
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
INPP4B inositol polyphosphate-4-phosphatase, type II, 105kDa
IRF8 interferon regulatory factor 8
KAT2A K(lysine) acetyltransferase 2A
KDM5C lysine (K)-specific demethylase 5C
KEAP1 kelch-like ECH-associated protein 1
LAMP5 lysosomal-associated membrane protein family, member 5
LMNB1 lamin B1
LMNB2 lamin B2
MATK megakaryocyte-associated tyrosine kinase
MBIP MAP3K12 binding inhibitory protein 1
MBTD1 mbt domain containing 1
MCMBP minichromosome maintenance complex binding protein
MGMT O-6-methylguanine-DNA methyltransferase
MRM1 mitochondrial rRNA methyltransferase 1 homolog (S. cerevisiae)
MRPL4 mitochondrial ribosomal protein L4
MTHFS 5,10-methenyltetrahydrofolate synthetase (5-formyltetrahydrofolate cyclo-ligase)
NAT6 N-acetyltransferase 6 (GCN5-related)
NBEAL2 neurobeachin-like 2
NSD1 nuclear receptor binding SET domain protein 1
PCBD1 pterin-4 alpha-carbinolamine dehydratase/dimerization cofactor of hepatocyte nuclear factor 1 alpha
PDLIM2 PDZ and LIM domain 2 (mystique)
PELP1 proline, glutamate and leucine rich protein 1
PHLPP1 PH domain and leucine rich repeat protein phosphatase 1
PIGT phosphatidylinositol glycan anchor biosynthesis, class T
PITRM1 pitrilysin metallopeptidase 1
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PNPLA6 patatin-like phospholipase domain containing 6
POMGNT1 protein O-linked mannose N-acetylglucosaminyltransferase 1 (beta 1,2-)
POMZP3 POM121 and ZP3 fusion
POTEKP POTE ankyrin domain family, member K, pseudogene
PPFIA4 protein tyrosine phosphatase, receptor type, f polypeptide (PTPRF), interacting protein (liprin), alpha 4
PRKD2 protein kinase D2
PTDSS2 phosphatidylserine synthase 2
QPRT quinolinate phosphoribosyltransferase
RGP1 RGP1 retrograde golgi transport homolog (S. cerevisiae)
RHBDF1 rhomboid 5 homolog 1 (Drosophila)
RNASEL ribonuclease L (2',5'-oligoisoadenylate synthetase-dependent)
RPP25 ribonuclease P/MRP 25kDa subunit
S100A6 S100 calcium binding protein A6
SEC31B SEC31 homolog B (S. cerevisiae)
SLC2A6 solute carrier family 2 (facilitated glucose transporter), member 6
SLC39A4 solute carrier family 39 (zinc transporter), member 4
SLC39A7 solute carrier family 39 (zinc transporter), member 7
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SLC9A3R1 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3 regulator 1
STIM1 stromal interaction molecule 1
SYNGR2 synaptogyrin 2
TAOK1 TAO kinase 1
TERT telomerase reverse transcriptase
THEM6 thioesterase superfamily member 6
TIMM50 translocase of inner mitochondrial membrane 50 homolog (S. cerevisiae)
TM7SF3 transmembrane 7 superfamily member 3
TMEM159 transmembrane protein 159
TMUB2 transmembrane and ubiquitin-like domain containing 2
TNFSF13 tumor necrosis factor (ligand) superfamily, member 13
TNNT1 troponin T type 1 (skeletal, slow)
USB1 U6 snRNA biogenesis 1
USP20 ubiquitin specific peptidase 20
VAT1 vesicle amine transport 1
VSIG4 V-set and immunoglobulin domain containing 4
WBP2 WW domain binding protein 2
WBSCR16 Williams-Beuren syndrome chromosome region 16
WDR6 WD repeat domain 6
ZBED1 zinc finger, BED-type containing 1
ZC3H12A zinc finger CCCH-type containing 12A
ZNF223 zinc finger protein 223
ZNF408 zinc finger protein 408
ZNF606 zinc finger protein 606