estropipate-2506 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the estropipate-2506 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCA12 ATP-binding cassette, sub-family A (ABC1), member 12
ADGRE1 adhesion G protein-coupled receptor E1
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2
B3GALNT1 beta-1,3-N-acetylgalactosaminyltransferase 1 (globoside blood group)
BTC betacellulin
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
CCR4 chemokine (C-C motif) receptor 4
CD24 CD24 molecule
CD28 CD28 molecule
CD6 CD6 molecule
CFAP45 cilia and flagella associated protein 45
CHRNA9 cholinergic receptor, nicotinic, alpha 9 (neuronal)
CNKSR2 connector enhancer of kinase suppressor of Ras 2
COQ7 coenzyme Q7 homolog, ubiquinone (yeast)
CSHL1 chorionic somatomammotropin hormone-like 1
DAPK2 death-associated protein kinase 2
DMTN dematin actin binding protein
DNAH2 dynein, axonemal, heavy chain 2
DNAH7 dynein, axonemal, heavy chain 7
DRD1 dopamine receptor D1
DSTYK dual serine/threonine and tyrosine protein kinase
ESR1 estrogen receptor 1
FCER1A Fc fragment of IgE, high affinity I, receptor for; alpha polypeptide
FGB fibrinogen beta chain
FGF5 fibroblast growth factor 5
FGG fibrinogen gamma chain
FLJ11292
GABARAPL3 GABA(A) receptors associated protein like 3, pseudogene
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GLP1R glucagon-like peptide 1 receptor
GNAO1 guanine nucleotide binding protein (G protein), alpha activating activity polypeptide O
GRIN2C glutamate receptor, ionotropic, N-methyl D-aspartate 2C
GULP1 GULP, engulfment adaptor PTB domain containing 1
HDAC11 histone deacetylase 11
HPCAL4 hippocalcin like 4
HS6ST1 heparan sulfate 6-O-sulfotransferase 1
HTR3A 5-hydroxytryptamine (serotonin) receptor 3A, ionotropic
IQCK IQ motif containing K
ITGB5 integrin, beta 5
ITIH1 inter-alpha-trypsin inhibitor heavy chain 1
JAG1 jagged 1
KCNIP2 Kv channel interacting protein 2
KCNJ8 potassium channel, inwardly rectifying subfamily J, member 8
KRT24 keratin 24, type I
LGR5 leucine-rich repeat containing G protein-coupled receptor 5
LILRB2 leukocyte immunoglobulin-like receptor, subfamily B (with TM and ITIM domains), member 2
LINC00216 long intergenic non-protein coding RNA 216
LINC00652 long intergenic non-protein coding RNA 652
MAG myelin associated glycoprotein
MBL1P mannose-binding lectin (protein A) 1, pseudogene
MCAM melanoma cell adhesion molecule
MEG3 maternally expressed 3 (non-protein coding)
METTL7A methyltransferase like 7A
NF2 neurofibromin 2 (merlin)
NMRK2 nicotinamide riboside kinase 2
NPHS2 nephrosis 2, idiopathic, steroid-resistant (podocin)
NR2E3 nuclear receptor subfamily 2, group E, member 3
NRCAM neuronal cell adhesion molecule
NTRK1 neurotrophic tyrosine kinase, receptor, type 1
NUDT11 nudix (nucleoside diphosphate linked moiety X)-type motif 11
PADI1 peptidyl arginine deiminase, type I
PAFAH2 platelet-activating factor acetylhydrolase 2, 40kDa
PCDH11X protocadherin 11 X-linked
PHKG1 phosphorylase kinase, gamma 1 (muscle)
PML promyelocytic leukemia
PPP1R3A protein phosphatase 1, regulatory subunit 3A
PRF1 perforin 1 (pore forming protein)
PRKAR1B protein kinase, cAMP-dependent, regulatory, type I, beta
RAB40A RAB40A, member RAS oncogene family
RHOD ras homolog family member D
RIC3 RIC3 acetylcholine receptor chaperone
SCN1B sodium channel, voltage gated, type I beta subunit
SCN2B sodium channel, voltage gated, type II beta subunit
SETD1A SET domain containing 1A
SIGLEC8 sialic acid binding Ig-like lectin 8
SIX2 SIX homeobox 2
SLCO1B1 solute carrier organic anion transporter family, member 1B1
SLCO2A1 solute carrier organic anion transporter family, member 2A1
SLCO3A1 solute carrier organic anion transporter family, member 3A1
SNED1 sushi, nidogen and EGF-like domains 1
SPINK1 serine peptidase inhibitor, Kazal type 1
SPINK5 serine peptidase inhibitor, Kazal type 5
ST8SIA3 ST8 alpha-N-acetyl-neuraminide alpha-2,8-sialyltransferase 3
TCF7L2 transcription factor 7-like 2 (T-cell specific, HMG-box)
TEAD3 TEA domain family member 3
TFAP2B transcription factor AP-2 beta (activating enhancer binding protein 2 beta)
TGFB1 transforming growth factor, beta 1
TIAM1 T-cell lymphoma invasion and metastasis 1
TJP3 tight junction protein 3
TK2 thymidine kinase 2, mitochondrial
TMEM51 transmembrane protein 51
TRIM31 tripartite motif containing 31
TTC12 tetratricopeptide repeat domain 12
UCP3 uncoupling protein 3 (mitochondrial, proton carrier)
ZER1 zyg-11 related, cell cycle regulator
ZNF235 zinc finger protein 235
ZNF259P1 zinc finger protein 259 pseudogene 1
ZNF280B zinc finger protein 280B

decreased expression

Symbol Name
ADAP2 ArfGAP with dual PH domains 2
ARAP3 ArfGAP with RhoGAP domain, ankyrin repeat and PH domain 3
ARFGAP1 ADP-ribosylation factor GTPase activating protein 1
ARNTL2 aryl hydrocarbon receptor nuclear translocator-like 2
ASAP1-IT1 ASAP1 intronic transcript 1
AXIN1 axin 1
B3GNT1
BAG4 BCL2-associated athanogene 4
BBS1 Bardet-Biedl syndrome 1
BBS10 Bardet-Biedl syndrome 10
C10ORF88 chromosome 10 open reading frame 88
C11ORF71 chromosome 11 open reading frame 71
C1GALT1C1 C1GALT1-specific chaperone 1
C1ORF54 chromosome 1 open reading frame 54
CCDC47 coiled-coil domain containing 47
CDT1 chromatin licensing and DNA replication factor 1
CEP85 centrosomal protein 85kDa
CHMP6 charged multivesicular body protein 6
CLPB ClpB homolog, mitochondrial AAA ATPase chaperonin
CSF1R colony stimulating factor 1 receptor
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
DDN dendrin
DDX58 DEAD (Asp-Glu-Ala-Asp) box polypeptide 58
DDX60 DEAD (Asp-Glu-Ala-Asp) box polypeptide 60
DENND4C DENN/MADD domain containing 4C
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DPY19L4 dpy-19-like 4 (C. elegans)
ECSIT ECSIT signalling integrator
ERF Ets2 repressor factor
ERMAP erythroblast membrane-associated protein (Scianna blood group)
ETV4 ets variant 4
EXOC2 exocyst complex component 2
F8 coagulation factor VIII, procoagulant component
FAM188A family with sequence similarity 188, member A
FICD FIC domain containing
FPGS folylpolyglutamate synthase
GATC glutamyl-tRNA(Gln) amidotransferase, subunit C
GNG11 guanine nucleotide binding protein (G protein), gamma 11
HAL histidine ammonia-lyase
HPSE heparanase
HSPA1L heat shock 70kDa protein 1-like
HYAL3 hyaluronoglucosaminidase 3
IFT57 intraflagellar transport 57
ITPKB inositol-trisphosphate 3-kinase B
KIAA0753 KIAA0753
KIFC1 kinesin family member C1
KPNA4 karyopherin alpha 4 (importin alpha 3)
LIN7A lin-7 homolog A (C. elegans)
LMNB1 lamin B1
MAN2C1 mannosidase, alpha, class 2C, member 1
MAP3K2 mitogen-activated protein kinase kinase kinase 2
MATK megakaryocyte-associated tyrosine kinase
MFSD11 major facilitator superfamily domain containing 11
MLYCD malonyl-CoA decarboxylase
MTERF4 mitochondrial transcription termination factor 4
MXD3 MAX dimerization protein 3
NDST2 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 2
NMD3 NMD3 ribosome export adaptor
NUBPL nucleotide binding protein-like
OPA3 optic atrophy 3 (autosomal recessive, with chorea and spastic paraplegia)
PEX13 peroxisomal biogenesis factor 13
PLA2G15 phospholipase A2, group XV
PLEKHJ1 pleckstrin homology domain containing, family J member 1
PLS1 plastin 1
PPIP5K1 diphosphoinositol pentakisphosphate kinase 1
PRKAR2B protein kinase, cAMP-dependent, regulatory, type II, beta
PROSER1 proline and serine rich 1
RFX7 regulatory factor X, 7
RINT1 RAD50 interactor 1
RPP25 ribonuclease P/MRP 25kDa subunit
RRAS related RAS viral (r-ras) oncogene homolog
S1PR4 sphingosine-1-phosphate receptor 4
SAR1B secretion associated, Ras related GTPase 1B
SENP2 SUMO1/sentrin/SMT3 specific peptidase 2
SERINC5 serine incorporator 5
SERPINB6 serpin peptidase inhibitor, clade B (ovalbumin), member 6
SETD8 SET domain containing (lysine methyltransferase) 8
SLC15A3 solute carrier family 15 (oligopeptide transporter), member 3
SLC9A8 solute carrier family 9, subfamily A (NHE8, cation proton antiporter 8), member 8
SPATA7 spermatogenesis associated 7
THBS4 thrombospondin 4
TMEM115 transmembrane protein 115
TMEM183A transmembrane protein 183A
TMEM254 transmembrane protein 254
TRAC T cell receptor alpha constant
TRAIP TRAF interacting protein
TRIM26 tripartite motif containing 26
TSPAN32 tetraspanin 32
UBE2NL ubiquitin-conjugating enzyme E2N-like (gene/pseudogene)
UGGT1 UDP-glucose glycoprotein glucosyltransferase 1
ULK1 unc-51 like autophagy activating kinase 1
WDR37 WD repeat domain 37
WDR44 WD repeat domain 44
WDR5B WD repeat domain 5B
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZBTB10 zinc finger and BTB domain containing 10
ZMAT5 zinc finger, matrin-type 5
ZNF273 zinc finger protein 273
ZNF32 zinc finger protein 32
ZNF37BP zinc finger protein 37B, pseudogene