ethisterone-3783 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the ethisterone-3783 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADAM8 ADAM metallopeptidase domain 8
AFF1 AF4/FMR2 family, member 1
ANKH ANKH inorganic pyrophosphate transport regulator
APAF1 apoptotic peptidase activating factor 1
APBA1 amyloid beta (A4) precursor protein-binding, family A, member 1
AR androgen receptor
BMP10 bone morphogenetic protein 10
C3AR1 complement component 3a receptor 1
CACNG4 calcium channel, voltage-dependent, gamma subunit 4
CD5 CD5 molecule
CDH7 cadherin 7, type 2
CLCN6 chloride channel, voltage-sensitive 6
COL1A1 collagen, type I, alpha 1
COL4A4 collagen, type IV, alpha 4
CREBZF CREB/ATF bZIP transcription factor
CRTC1 CREB regulated transcription coactivator 1
CWH43 cell wall biogenesis 43 C-terminal homolog (S. cerevisiae)
CYP2A6 cytochrome P450, family 2, subfamily A, polypeptide 6
CYP2A7 cytochrome P450, family 2, subfamily A, polypeptide 7
DNASE2B deoxyribonuclease II beta
DUOX2 dual oxidase 2
ESR1 estrogen receptor 1
FAM182A family with sequence similarity 182, member A
FRMD4B FERM domain containing 4B
FZD1 frizzled class receptor 1
GADD45GIP1 growth arrest and DNA-damage-inducible, gamma interacting protein 1
GHRHR growth hormone releasing hormone receptor
GNG3 guanine nucleotide binding protein (G protein), gamma 3
GOLGA8A golgin A8 family, member A
GP5 glycoprotein V (platelet)
GPR135 G protein-coupled receptor 135
HERC4 HECT and RLD domain containing E3 ubiquitin protein ligase 4
HFE hemochromatosis
HIST1H2BB histone cluster 1, H2bb
HIST1H3A histone cluster 1, H3a
IFI27 interferon, alpha-inducible protein 27
IFI6 interferon, alpha-inducible protein 6
IFITM1 interferon induced transmembrane protein 1
INHBC inhibin, beta C
KAT8 K(lysine) acetyltransferase 8
KIF25-AS1 KIF25 antisense RNA 1
KLHL25 kelch-like family member 25
LILRB2 leukocyte immunoglobulin-like receptor, subfamily B (with TM and ITIM domains), member 2
LRRK1 leucine-rich repeat kinase 1
MAP7D3 MAP7 domain containing 3
MAPK8IP3 mitogen-activated protein kinase 8 interacting protein 3
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase
MIER2 mesoderm induction early response 1, family member 2
MOBP myelin-associated oligodendrocyte basic protein
NF1 neurofibromin 1
NPPA natriuretic peptide A
NUMA1 nuclear mitotic apparatus protein 1
OAS1 2'-5'-oligoadenylate synthetase 1, 40/46kDa
OASL 2'-5'-oligoadenylate synthetase-like
OSBPL7 oxysterol binding protein-like 7
P2RY11 purinergic receptor P2Y, G-protein coupled, 11
PGAP3 post-GPI attachment to proteins 3
PHF3 PHD finger protein 3
PIK3R4 phosphoinositide-3-kinase, regulatory subunit 4
PKNOX2 PBX/knotted 1 homeobox 2
PKP4 plakophilin 4
PMCHL1 pro-melanin-concentrating hormone-like 1, pseudogene
PSG4 pregnancy specific beta-1-glycoprotein 4
PTGDS prostaglandin D2 synthase 21kDa (brain)
PYY peptide YY
R3HDM1 R3H domain containing 1
RAB40AL RAB40A, member RAS oncogene family-like
RAB6B RAB6B, member RAS oncogene family
RAPGEF5 Rap guanine nucleotide exchange factor (GEF) 5
RARRES2 retinoic acid receptor responder (tazarotene induced) 2
RASL12 RAS-like, family 12
RASSF9 Ras association (RalGDS/AF-6) domain family (N-terminal) member 9
RNF208 ring finger protein 208
RNGTT RNA guanylyltransferase and 5'-phosphatase
SAPCD1 suppressor APC domain containing 1
SEMA4F sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4F
SH3BP1 SH3-domain binding protein 1
SLAMF7 SLAM family member 7
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC16A5 solute carrier family 16 (monocarboxylate transporter), member 5
SMO smoothened, frizzled class receptor
SOX21 SRY (sex determining region Y)-box 21
SP110 SP110 nuclear body protein
SRPK3 SRSF protein kinase 3
STAT2 signal transducer and activator of transcription 2, 113kDa
SYNGR3 synaptogyrin 3
TAAR5 trace amine associated receptor 5
TBCD tubulin folding cofactor D
TCF15 transcription factor 15 (basic helix-loop-helix)
TEF thyrotrophic embryonic factor
TLK1 tousled-like kinase 1
TM4SF5 transmembrane 4 L six family member 5
TNFRSF4 tumor necrosis factor receptor superfamily, member 4
TNNT2 troponin T type 2 (cardiac)
TSC22D2 TSC22 domain family, member 2
TSGA10 testis specific, 10
VAMP1 vesicle-associated membrane protein 1 (synaptobrevin 1)
ZC2HC1C zinc finger, C2HC-type containing 1C

decreased expression

Symbol Name
ABCG2 ATP-binding cassette, sub-family G (WHITE), member 2 (Junior blood group)
ACBD4 acyl-CoA binding domain containing 4
ACSS3 acyl-CoA synthetase short-chain family member 3
ADGRB2 adhesion G protein-coupled receptor B2
APOH apolipoprotein H (beta-2-glycoprotein I)
ARHGEF38 Rho guanine nucleotide exchange factor (GEF) 38
ARMC6 armadillo repeat containing 6
C16ORF59 chromosome 16 open reading frame 59
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
CACNG1 calcium channel, voltage-dependent, gamma subunit 1
CCDC132 coiled-coil domain containing 132
CCDC134 coiled-coil domain containing 134
CCDC186 coiled-coil domain containing 186
CD79B CD79b molecule, immunoglobulin-associated beta
CDH10 cadherin 10, type 2 (T2-cadherin)
CEP85 centrosomal protein 85kDa
CFAP45 cilia and flagella associated protein 45
CFHR2 complement factor H-related 2
CGREF1 cell growth regulator with EF-hand domain 1
CHRNG cholinergic receptor, nicotinic, gamma (muscle)
CNR2 cannabinoid receptor 2 (macrophage)
CSN3 casein kappa
CUZD1 CUB and zona pellucida-like domains 1
CYP2J2 cytochrome P450, family 2, subfamily J, polypeptide 2
CYP7B1 cytochrome P450, family 7, subfamily B, polypeptide 1
DCAF4 DDB1 and CUL4 associated factor 4
DDN dendrin
DHRS9 dehydrogenase/reductase (SDR family) member 9
ERF Ets2 repressor factor
FMOD fibromodulin
FOXO4 forkhead box O4
GLB1L galactosidase, beta 1-like
GLS2 glutaminase 2 (liver, mitochondrial)
GNA14 guanine nucleotide binding protein (G protein), alpha 14
GSTM5 glutathione S-transferase mu 5
HAAO 3-hydroxyanthranilate 3,4-dioxygenase
HDAC5 histone deacetylase 5
HIST1H2AB histone cluster 1, H2ab
HIST1H2BM histone cluster 1, H2bm
HIST1H4A histone cluster 1, H4a
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
IFNA17 interferon, alpha 17
IFNAR1 interferon (alpha, beta and omega) receptor 1
IL2RG interleukin 2 receptor, gamma
INPP5J inositol polyphosphate-5-phosphatase J
IPO8 importin 8
IQCC IQ motif containing C
KCNS1 potassium voltage-gated channel, modifier subfamily S, member 1
KLHL28 kelch-like family member 28
KRT37 keratin 37, type I
LIME1 Lck interacting transmembrane adaptor 1
LRRC2 leucine rich repeat containing 2
LRRC61 leucine rich repeat containing 61
LTC4S leukotriene C4 synthase
MBL1P mannose-binding lectin (protein A) 1, pseudogene
NDOR1 NADPH dependent diflavin oxidoreductase 1
NEK11 NIMA-related kinase 11
NELL2 NEL-like 2 (chicken)
NEO1 neogenin 1
NEURL1 neuralized E3 ubiquitin protein ligase 1
NEUROD4 neuronal differentiation 4
NTF3 neurotrophin 3
OGDHL oxoglutarate dehydrogenase-like
OR1D2 olfactory receptor, family 1, subfamily D, member 2
OR2F1 olfactory receptor, family 2, subfamily F, member 1 (gene/pseudogene)
PADI1 peptidyl arginine deiminase, type I
PCBP3 poly(rC) binding protein 3
PGLYRP1 peptidoglycan recognition protein 1
PHACTR4 phosphatase and actin regulator 4
PLD2 phospholipase D2
PLEKHO1 pleckstrin homology domain containing, family O member 1
PLXNB3 plexin B3
PPARA peroxisome proliferator-activated receptor alpha
PQLC2 PQ loop repeat containing 2
PROL1 proline rich, lacrimal 1
PRPH peripherin
RFX2 regulatory factor X, 2 (influences HLA class II expression)
SASH3 SAM and SH3 domain containing 3
SERGEF secretion regulating guanine nucleotide exchange factor
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SLC6A9 solute carrier family 6 (neurotransmitter transporter, glycine), member 9
SLITRK5 SLIT and NTRK-like family, member 5
STAG3 stromal antigen 3
SUSD4 sushi domain containing 4
TAGLN3 transgelin 3
TNFSF15 tumor necrosis factor (ligand) superfamily, member 15
TRIM45 tripartite motif containing 45
TRPM4 transient receptor potential cation channel, subfamily M, member 4
TSPAN32 tetraspanin 32
VASH1 vasohibin 1
VGF VGF nerve growth factor inducible
VN1R1 vomeronasal 1 receptor 1
WDR76 WD repeat domain 76
ZNF141 zinc finger protein 141
ZNF324 zinc finger protein 324
ZNF334 zinc finger protein 334
ZNF480 zinc finger protein 480
ZNF695 zinc finger protein 695