felodipine-6695 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the felodipine-6695 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADD2 adducin 2 (beta)
ADGRF5 adhesion G protein-coupled receptor F5
ADH6 alcohol dehydrogenase 6 (class V)
AIM2 absent in melanoma 2
AP2B1 adaptor-related protein complex 2, beta 1 subunit
APAF1 apoptotic peptidase activating factor 1
APC adenomatous polyposis coli
ASTN1 astrotactin 1
ATF6B activating transcription factor 6 beta
ATF7IP activating transcription factor 7 interacting protein
BHMT2 betaine--homocysteine S-methyltransferase 2
BICC1 BicC family RNA binding protein 1
BTF3P11 basic transcription factor 3 pseudogene 11
C10ORF12 chromosome 10 open reading frame 12
CBS cystathionine-beta-synthase
CD209 CD209 molecule
CEBPA CCAAT/enhancer binding protein (C/EBP), alpha
CEBPD CCAAT/enhancer binding protein (C/EBP), delta
CISH cytokine inducible SH2-containing protein
CLCN4 chloride channel, voltage-sensitive 4
CNGB3 cyclic nucleotide gated channel beta 3
CREBZF CREB/ATF bZIP transcription factor
CRTC1 CREB regulated transcription coactivator 1
CSTF2T cleavage stimulation factor, 3' pre-RNA, subunit 2, 64kDa, tau variant
CTSZ cathepsin Z
CXCR4 chemokine (C-X-C motif) receptor 4
DCSTAMP dendrocyte expressed seven transmembrane protein
DDIT4 DNA-damage-inducible transcript 4
DLK2 delta-like 2 homolog (Drosophila)
DOPEY2 dopey family member 2
EFNA3 ephrin-A3
ELAC1 elaC ribonuclease Z 1
ENPP2 ectonucleotide pyrophosphatase/phosphodiesterase 2
EYA4 EYA transcriptional coactivator and phosphatase 4
FGFR1 fibroblast growth factor receptor 1
GFI1 growth factor independent 1 transcription repressor
GPR135 G protein-coupled receptor 135
GRM4 glutamate receptor, metabotropic 4
GRM8 glutamate receptor, metabotropic 8
GTF2A1 general transcription factor IIA, 1, 19/37kDa
GULP1 GULP, engulfment adaptor PTB domain containing 1
HAPLN1 hyaluronan and proteoglycan link protein 1
HESX1 HESX homeobox 1
HIC2 hypermethylated in cancer 2
HMOX1 heme oxygenase 1
IFIT2 interferon-induced protein with tetratricopeptide repeats 2
IMPG2 interphotoreceptor matrix proteoglycan 2
ITGB3 integrin, beta 3 (platelet glycoprotein IIIa, antigen CD61)
KHDRBS1 KH domain containing, RNA binding, signal transduction associated 1
KIAA1467 KIAA1467
KLF4 Kruppel-like factor 4 (gut)
LDB3 LIM domain binding 3
LMX1B LIM homeobox transcription factor 1, beta
MCPH1 microcephalin 1
MORC1 MORC family CW-type zinc finger 1
NBEAL2 neurobeachin-like 2
NBR2 neighbor of BRCA1 gene 2 (non-protein coding)
NIPAL3 NIPA-like domain containing 3
NTF3 neurotrophin 3
NTRK2 neurotrophic tyrosine kinase, receptor, type 2
NUP88 nucleoporin 88kDa
NUPR1 nuclear protein, transcriptional regulator, 1
OASL 2'-5'-oligoadenylate synthetase-like
PACRG PARK2 co-regulated
PCDH9 protocadherin 9
PCDHB3 protocadherin beta 3
PDE10A phosphodiesterase 10A
PDE7B phosphodiesterase 7B
PDZRN3 PDZ domain containing ring finger 3
PHF7 PHD finger protein 7
PIP5K1A phosphatidylinositol-4-phosphate 5-kinase, type I, alpha
PLXNB3 plexin B3
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
POU5F1B POU class 5 homeobox 1B
PPFIA4 protein tyrosine phosphatase, receptor type, f polypeptide (PTPRF), interacting protein (liprin), alpha 4
PPP3R1 protein phosphatase 3, regulatory subunit B, alpha
PRKCA protein kinase C, alpha
RBM3 RNA binding motif (RNP1, RRM) protein 3
RGR retinal G protein coupled receptor
RHOT2 ras homolog family member T2
RNF19B ring finger protein 19B
RPH3AL rabphilin 3A-like (without C2 domains)
RPS3A ribosomal protein S3A
SPTBN5 spectrin, beta, non-erythrocytic 5
STK16 serine/threonine kinase 16
SULT1E1 sulfotransferase family 1E, estrogen-preferring, member 1
SYCP1 synaptonemal complex protein 1
SYMPK symplekin
TADA2A transcriptional adaptor 2A
TCL6 T-cell leukemia/lymphoma 6 (non-protein coding)
TECTA tectorin alpha
THSD4 thrombospondin, type I, domain containing 4
TNKS2 tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase 2
TROVE2 TROVE domain family, member 2
UBR2 ubiquitin protein ligase E3 component n-recognin 2
UPK1B uroplakin 1B
WDR55 WD repeat domain 55
ZNF550 zinc finger protein 550
ZNF639 zinc finger protein 639

decreased expression

Symbol Name
AAAS achalasia, adrenocortical insufficiency, alacrimia
ABCC2 ATP-binding cassette, sub-family C (CFTR/MRP), member 2
ALPK1 alpha-kinase 1
ANKRD1 ankyrin repeat domain 1 (cardiac muscle)
AURKC aurora kinase C
B3GALT4 UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 4
BAG4 BCL2-associated athanogene 4
BEX1 brain expressed, X-linked 1
C11ORF63 chromosome 11 open reading frame 63
C19ORF54 chromosome 19 open reading frame 54
CAND2 cullin-associated and neddylation-dissociated 2 (putative)
CASP5 caspase 5, apoptosis-related cysteine peptidase
CCP110 centriolar coiled coil protein 110kDa
CD79A CD79a molecule, immunoglobulin-associated alpha
CEL carboxyl ester lipase
CEMIP cell migration inducing protein, hyaluronan binding
CENPO centromere protein O
CHRDL1 chordin-like 1
CHRNB1 cholinergic receptor, nicotinic, beta 1 (muscle)
CIDEC cell death-inducing DFFA-like effector c
CNTLN centlein, centrosomal protein
CNTNAP3B contactin associated protein-like 3B
CYBRD1 cytochrome b reductase 1
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1
CYP39A1 cytochrome P450, family 39, subfamily A, polypeptide 1
CYP7B1 cytochrome P450, family 7, subfamily B, polypeptide 1
E2F8 E2F transcription factor 8
ETAA1 Ewing tumor-associated antigen 1
FAM184A family with sequence similarity 184, member A
FAM186A family with sequence similarity 186, member A
FAM50B family with sequence similarity 50, member B
FBXL7 F-box and leucine-rich repeat protein 7
FGFBP1 fibroblast growth factor binding protein 1
GSTA3 glutathione S-transferase alpha 3
HIST1H2AM histone cluster 1, H2am
HOXA1 homeobox A1
HOXA7 homeobox A7
HOXC5 homeobox C5
IER3IP1 immediate early response 3 interacting protein 1
IFNAR1 interferon (alpha, beta and omega) receptor 1
IFT22 intraflagellar transport 22
IFT54 intraflagellar transport 54
IL1B interleukin 1, beta
IL2 interleukin 2
IL36RN interleukin 36 receptor antagonist
ISYNA1 inositol-3-phosphate synthase 1
KCNS3 potassium voltage-gated channel, modifier subfamily S, member 3
KRT9 keratin 9, type I
LINC00115 long intergenic non-protein coding RNA 115
LINC00472 long intergenic non-protein coding RNA 472
LRRC61 leucine rich repeat containing 61
MANSC1 MANSC domain containing 1
MRPL41 mitochondrial ribosomal protein L41
MRPL44 mitochondrial ribosomal protein L44
MRPL46 mitochondrial ribosomal protein L46
MRPL52 mitochondrial ribosomal protein L52
NKX3-2 NK3 homeobox 2
NRTN neurturin
OR2F1 olfactory receptor, family 2, subfamily F, member 1 (gene/pseudogene)
OSR2 odd-skipped related transciption factor 2
PDE6B phosphodiesterase 6B, cGMP-specific, rod, beta
PDK4 pyruvate dehydrogenase kinase, isozyme 4
PLEKHA2 pleckstrin homology domain containing, family A (phosphoinositide binding specific) member 2
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PLEKHF1 pleckstrin homology domain containing, family F (with FYVE domain) member 1
POLL polymerase (DNA directed), lambda
POM121 POM121 transmembrane nucleoporin
PRR15L proline rich 15-like
RBL1 retinoblastoma-like 1
RUNDC3B RUN domain containing 3B
SCARA3 scavenger receptor class A, member 3
SCUBE3 signal peptide, CUB domain, EGF-like 3
SERPINB2 serpin peptidase inhibitor, clade B (ovalbumin), member 2
SH2D2A SH2 domain containing 2A
SKI SKI proto-oncogene
SLC12A8 solute carrier family 12, member 8
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC35F6 solute carrier family 35, member F6
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SLITRK5 SLIT and NTRK-like family, member 5
STAG3L4 stromal antigen 3-like 4 (pseudogene)
SYNGR3 synaptogyrin 3
THOP1 thimet oligopeptidase 1
TIPARP TCDD-inducible poly(ADP-ribose) polymerase
TMEM121 transmembrane protein 121
TMSB15A thymosin beta 15a
TRIM25 tripartite motif containing 25
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TTC30A tetratricopeptide repeat domain 30A
TTLL1 tubulin tyrosine ligase-like family member 1
ZBTB22 zinc finger and BTB domain containing 22
ZC2HC1C zinc finger, C2HC-type containing 1C
ZNF197 zinc finger protein 197
ZNF276 zinc finger protein 276
ZNF350 zinc finger protein 350
ZNF492 zinc finger protein 492
ZNF770 zinc finger protein 770